cp 93129 has been researched along with pyrroles in 102 studies
Studies (cp 93129) | Trials (cp 93129) | Recent Studies (post-2010) (cp 93129) | Studies (pyrroles) | Trials (pyrroles) | Recent Studies (post-2010) (pyrroles) |
---|---|---|---|---|---|
109 | 0 | 11 | 26,129 | 2,815 | 12,100 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 36 (35.29) | 18.2507 |
2000's | 55 (53.92) | 29.6817 |
2010's | 11 (10.78) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Boccalini, P; Moskowitz, MA; Nozaki, K | 1 |
Fox, CB; Johnson, C; Koe, BK; Lebel, LA; Macor, JE; Zorn, SH | 1 |
Byun, B; Matsubara, T; Moskowitz, MA | 1 |
Hjorth, S; Tao, R | 1 |
Burkhart, CA; Heym, JH; Ives, JL; Lebel, LA; Macor, JE; Newman, ME; Nielsen, JA; Ryan, K; Schulz, DW; Torgersen, LK | 1 |
Buhot, MC; Naïli, S | 1 |
Brain, SD; Gupta, P; Kajekar, R; Shepperson, NB | 1 |
Alvarez Sanz, MC; Kunimoto, K; Levy, AD; Li, Q; Rittenhouse, PA; Van de Kar, LD; Yracheta, JM | 1 |
Hjorth, S; Sharp, T | 1 |
Bruinvels, AT; Hoyer, D; Landwehrmeyer, B; Palacios, JM; Probst, A | 1 |
Galloway, MP; Hjorth, S; Keegan, MJ; Suchowski, CS | 1 |
Byun, B; Huang, Z; Matsubara, T; Moskowitz, MA | 1 |
Buhot, MC; Naïli, S; Patra, SK | 1 |
Castanon, N; Chauveau, J; Chaveau, J; Hen, R; Macor, JE; Moskowitz, MA; Scearce, K; Waeber, C; Yu, XJ | 1 |
Arnaboldi, S; Baldi, G; Consolo, S; Ladinsky, H; Nannini, L; Ramponi, S | 1 |
Cassel, JC; Jackisch, R; Jeltsch, H; Lauth, D; Neufang, B; Szabo, B | 1 |
Auerbach, SB; Hjorth, S | 1 |
Fillion, G; Seguin, L; Seznec, JC | 1 |
Davidson, C; Stamford, JA | 2 |
Hotta, H; Messlinger, K; Pawlak, M; Schmidt, RF | 1 |
Anmella, MC; Gardier, AM; Hen, R; Jacquot, C; Malagié, I; Pons, D; Scearce, K; Trillat, AC | 1 |
Gjerstad, J; Hole, K; Tjølsen, A | 1 |
Fillion, G; Guezennec, Y; Liscia, P; Seguin, L | 1 |
Aloyo, VJ; Fluharty, SJ; Lee, MD; Simansky, KJ | 1 |
Allain, H; Bentué-Ferrer, D; Bourin, M; Fillion, G; Massot, O; Reymann, JM; Rousselle, JC | 1 |
Koob, GF; Parsons, LH; Weiss, F | 1 |
Branchek, TA; Zgombick, JM | 1 |
Cumberbatch, MJ; Hargreaves, RJ; Hill, RG | 1 |
Ebersberger, A; Messlinger, K; Schaible, HG | 1 |
Centurión, D; Rabelo, G; Sánchez-López, A; Villalón, CM | 1 |
Cloëz-Tayarani, I; Fillion, G; Fillion, MP; Massot, O; Sarhan, H | 1 |
Fletcher, PJ; Korth, KM | 1 |
Bakker, MH; Bonaventure, P; Cras, P; Langlois, X; Leysen, JE; Luyten, WH; Megens, AA; Serneels, L; Umans, L; Van Leuven, F | 1 |
Alper, RH; Mize, AL | 1 |
Balse, E; Cassel, JC; Haaf, A; Jackisch, R; Kelche, C; Suhr, R | 1 |
Fillion, G; Sarhan, H | 1 |
Fillion, G; Grimaldi, B; Hen, R; Sarhan, H | 1 |
Bailly, JM; Deschamps, F; Fillion, G; Grimaldi, B; Kochanek, M; Lambrozo, J; Massot, O | 1 |
Bonnin, A; Chennaoui, M; Drogou, C; Fillion, G; Fillion, MP; Grimaldi, B; Guezennec, CY | 1 |
Béïque, J; Blier, P; de Montigny, C; Debonnel, G | 1 |
Atack, J; Chadha, A; Duty, S; Sur, C | 1 |
Hopwood, SE; Stamford, JA | 1 |
Yan, QS; Yan, SE | 2 |
Goto, F; Ishizaki, K; Obata, H; Sasaki, M | 1 |
Adell, A; Artigas, F; Celada, P | 1 |
Banes, AK; Watts, SW | 2 |
Blier, P; Hen, R; Richer, M | 1 |
Cases, O; Gaspar, P; Goaillard, JM; Laurent, A; Lebrand, C; Ropert, N | 1 |
Geyer, MA; Martinez-Price, DL | 1 |
Nicklous, DM; Simansky, KJ | 1 |
Azampanah, A; Fletcher, PJ; Korth, KM | 1 |
De Groote, L; Olivier, B; Westenberg, HG | 3 |
Filip, M; Jungersmith, K; Nowak, E; Papla, I; Przegaliński, E | 1 |
Filip, M; Papla, I; Przegaliński, E; Siwanowicz, J | 2 |
Czepiel, K; Filip, M; Papla, I; Przegaliński, E | 1 |
Berger, AJ; Huynh, P | 1 |
Birthelmer, A; Cassel, JC; Jackisch, R; Jeltsch, H; Schweizer, T | 1 |
Amtage, F; Birthelmer, A; Cassel, JC; Ehret, A; Förster, S; Jackisch, R; Jeltsch, H; Lehmann, O | 1 |
Gibert-Rahola, J; Micó, JA; Ortega-Alvaro, A; Roca-Vinardell, A | 1 |
Birthelmer, A; Cassel, JC; Jackisch, R; Stemmelin, J | 1 |
Birthelmer, A; Cassel, JC; Jackisch, R; Lazaris, A; Schweizer, T | 1 |
Averbeck, B; Reeh, WP; Zimmermann, K | 1 |
Pini, LA; Sandrini, M; Vitale, G | 1 |
Arulmani, U; Centurión, D; Sánchez-López, A; Saxena, PR; Vázquez, E; Villalón, CM | 1 |
Adell, A; Amargós-Bosch, M; Artigas, F; Bortolozzi, A; Toth, M | 1 |
Akasu, T; Hasuo, H; Matsuoka, T | 1 |
Yan, QS; Yan, SE; Zheng, SZ | 1 |
Castro, ME; Mostany, R; Pazos, A | 1 |
Diksic, M; Hasegawa, S; Nguyen, KQ; Nishi, K; Watanabe, A | 1 |
Bramley, JR; Dudek, FE; Pickard, GE; Sollars, PJ | 1 |
Höglund, AU; Kommalage, M | 1 |
Berrocoso, E; Micó, JA; Rojas-Corrales, MO | 1 |
Buhot, MC; Cassel, JC; Jackisch, R; Riegert, C; Rothmaier, AK; Rutz, S | 1 |
Hurley, LM | 1 |
Hori, T; Mizutani, H; Takahashi, T | 1 |
Jeggo, RD; Jordan, D; Ramage, AG; Wang, Y | 1 |
Jackisch, R; Riegert, C; Rothmaier, AK; Rutz, S | 1 |
Fink, AE; Gray, EE; O'dell, TJ; Sariñana, J | 1 |
Bannai, M; Faccidomo, S; Fish, EW; Miczek, KA | 1 |
Birthelmer, A; Ehret, A; Jackisch, R; Riegert, C; Rothmaier, AK; Rutz, S | 1 |
Almeida, RM; Lucion, AB; Miczek, KA; Veiga, CP | 1 |
Bohorquez, A; Hurley, LM; Tracy, JA | 1 |
Centenaro, LA; de Almeida, RM; Lucion, AB; Miczek, KA; Vieira, K; Zimmermann, N | 1 |
Fujita, S; Hatanaka, H; Kiguchi, M; Koshikawa, N; Lee, J; Suga, K; Terakado, M | 1 |
Murano, M; Saitow, F; Suzuki, H | 1 |
Centurión, D; González-Hernández, A; Lozano-Cuenca, J; Muñoz-Islas, E; Ramírez-Rosas, MB; Ramírez-San Juan, E; Sánchez-López, A; Villalón, CM | 1 |
Guptarak, J; Hiegel, C; Uphouse, L | 1 |
da Veiga, CP; de Almeida, RM; Lucion, AB; Miczek, KA | 1 |
Agius, L; Arden, C; Hampson, LJ; Kieswich, J; Malcomson, F; Petrie, JL; Potts, L; Tudhope, SJ; Wang, CC; Yaqoob, MM | 1 |
Faccidomo, S; Fish, EW; Miczek, KA; Quadros, IM; Takahashi, A | 1 |
An, CH; Cho, JH; Choi, IS; Choi, JK; Hur, YK; Jang, IS; Jung, JK | 1 |
Ding, S; Li, L; Zhou, FM | 1 |
Chen, L; Chen, WF; Chen, XY; Wang, H; Wei, L; Xue, Y | 1 |
Lee, LJ; Liao, CC | 1 |
Barman, SM; Burnett, R; Darios, ES; Davis, RP; Morrison, SF; Orer, HS; Seitz, BM; Watts, SW | 1 |
Cruz-Martínez, AM; Escartín-Pérez, RE; Florán-Garduño, B; López-Alonso, VE; Mancilla-Díaz, JM; Tejas-Juárez, JG | 1 |
102 other study(ies) available for cp 93129 and pyrroles
Article | Year |
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CP-93,129, sumatriptan, dihydroergotamine block c-fos expression within rat trigeminal nucleus caudalis caused by chemical stimulation of the meninges.
Topics: Animals; Animals, Newborn; Capsaicin; Carrageenan; Dihydroergotamine; Formaldehyde; Gene Expression Regulation, Neoplastic; Guinea Pigs; Immunohistochemistry; In Vitro Techniques; Indoles; Meninges; Nasal Mucosa; Proto-Oncogene Proteins c-fos; Pyridines; Pyrroles; Rats; Sulfonamides; Sumatriptan | 1992 |
1-(2-Aminoethyl)-3-methyl-8,9-dihydropyrano[3,2-e]indole: a rotationally restricted phenolic analog of the neurotransmitter serotonin and agonist selective for serotonin (5-HT2-type) receptors.
Topics: Animals; Indoles; Pyridines; Pyrroles; Rats; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Structure-Activity Relationship | 1992 |
CP-93,129, a potent and selective 5-HT1B receptor agonist blocks neurogenic plasma extravasation within rat but not guinea-pig dura mater.
Topics: Animals; Blood Pressure; Capsaicin; Dura Mater; Electric Stimulation; Guinea Pigs; Indoles; Ligands; Male; Plasma; Proteins; Pyridines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serum Albumin, Radio-Iodinated; Sulfonamides; Sumatriptan; Trigeminal Ganglion; Vasoconstrictor Agents | 1991 |
The putative 5-HT1B receptor agonist CP-93,129 suppresses rat hippocampal 5-HT release in vivo: comparison with RU 24969.
Topics: Animals; Brain Chemistry; Citalopram; Dialysis; Hippocampus; Indoles; Male; Methiothepin; Pyridines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin | 1991 |
3-(1,2,5,6-Tetrahydropyrid-4-yl)pyrrolo[3,2-b]pyrid-5-one: a potent and selective serotonin (5-HT1B) agonist and rotationally restricted phenolic analogue of 5-methoxy-3-(1,2,5,6-tetrahydropyrid-4-yl)indole.
Topics: Adenylyl Cyclase Inhibitors; Animals; Chemical Phenomena; Chemistry; Colforsin; Cyclization; Eating; Guinea Pigs; Hippocampus; Indoles; Molecular Structure; Paraventricular Hypothalamic Nucleus; Pyridines; Pyrroles; Rats; Receptors, Serotonin; Serotonin; Substantia Nigra | 1990 |
Changes in exploratory activity following stimulation of hippocampal 5-HT1A and 5-HT1B receptors in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Exploratory Behavior; Habituation, Psychophysiologic; Hippocampus; Male; Motor Activity; Pyridines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Serotonin; Scopolamine; Serotonin Receptor Agonists; Space Perception; Stimulation, Chemical | 1995 |
Effect of a 5-HT1 receptor agonist, CP-122,288, on oedema formation induced by stimulation of the rat saphenous nerve.
Topics: Analysis of Variance; Animals; Edema; Electric Stimulation; Male; Neuritis; Neurons, Afferent; Pyridines; Pyrroles; Pyrrolidines; Rats; Rats, Wistar; Serotonin Receptor Agonists; Sumatriptan | 1995 |
ICV injection of the serotonin 5-HT1B agonist CP-93,129 increases the secretion of ACTH, prolactin, and renin and increases blood pressure by nonserotonergic mechanisms.
Topics: Adrenocorticotropic Hormone; Animals; Blood Pressure; Injections, Intra-Arterial; Injections, Intraperitoneal; Injections, Intraventricular; Male; Metergoline; Prolactin; Propranolol; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Renin; Serotonin; Serotonin Receptor Agonists | 1994 |
In vivo microdialysis evidence for central serotonin1A and serotonin1B autoreceptor blocking properties of the beta adrenoceptor antagonist (-)penbutolol.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Citalopram; Dialysis; Hippocampus; Male; Metoprolol; Penbutolol; Perfusion; Pindolol; Propanolamines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stereoisomerism | 1993 |
A comparative autoradiographic study of 5-HT1D binding sites in human and guinea-pig brain using different radioligands.
Topics: Aged; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Dipeptides; Female; Guinea Pigs; Humans; Iodine Radioisotopes; Kinetics; Ligands; Male; Organ Specificity; Pyridines; Pyrroles; Receptors, Serotonin; Serotonin; Species Specificity; Sumatriptan; Tritium; Yohimbine | 1994 |
Local infusion of the selective 5HT-1b agonist CP-93,129 facilitates striatal dopamine release in vivo.
Topics: Animals; Corpus Striatum; Dopamine; In Vitro Techniques; Infusions, Parenteral; Male; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists | 1993 |
Time-dependent blockade of neurogenic plasma extravasation in dura mater by 5-HT1B/D agonists and endopeptidase 24.11.
Topics: Animals; Capsaicin; Disease Models, Animal; Dura Mater; Electric Stimulation; Extravasation of Diagnostic and Therapeutic Materials; Guinea Pigs; Indoles; Male; Neprilysin; Neuropeptides; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Serotonin Receptor Agonists; Sulfonamides; Sumatriptan; Time Factors; Trigeminal Ganglion | 1993 |
Spatial memory deficits following stimulation of hippocampal 5-HT1B receptors in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Handling, Psychological; Hippocampus; Injections; Male; Maze Learning; Memory Disorders; Memory, Short-Term; Muscarinic Antagonists; Pyridines; Pyrroles; Rats; Receptors, Serotonin; Scopolamine; Serotonin Receptor Agonists; Space Perception | 1995 |
5-Carboxamido-tryptamine, CP-122,288 and dihydroergotamine but not sumatriptan, CP-93,129, and serotonin-5-O-carboxymethyl-glycyl -tyrosinamide block dural plasma protein extravasation in knockout mice that lack 5-hydroxytryptamine1B receptors.
Topics: Animals; Capillary Permeability; Dihydroergotamine; Dipeptides; Mice; Mice, Knockout; Pyridines; Pyrroles; Pyrrolidines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Sumatriptan; Trigeminal Ganglion | 1996 |
Endogenous serotonin facilitates in vivo acetylcholine release in rat frontal cortex through 5-HT 1B receptors.
Topics: Acetylcholine; Animals; Dose-Response Relationship, Drug; Female; Frontal Lobe; Indoles; Norfenfluramine; Pyridines; Pyrroles; Rats; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Sulfonamides; Tetrodotoxin | 1996 |
Downregulation of muscarinic- and 5-HT1B-mediated modulation of [3H]acetylcholine release in hippocampal slices of rats with fimbria-fornix lesions and intrahippocampal grafts of septal origin.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Atropine; Brain Tissue Transplantation; Choline; Choline O-Acetyltransferase; Cholinergic Fibers; Cholinesterase Inhibitors; Diffusion Chambers, Culture; Down-Regulation; Electric Stimulation; Female; Hippocampus; Hydroxyindoleacetic Acid; Mecamylamine; Methiothepin; Muscarinic Agonists; Muscarinic Antagonists; Neurons; Nicotinic Antagonists; Norepinephrine; Oxotremorine; Physostigmine; Pyridines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Receptors, Serotonin; Septal Nuclei; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium | 1995 |
Effect of chronic administration of the selective serotonin (5-HT) uptake inhibitor citalopram on extracellular 5-HT and apparent autoreceptor sensitivity in rat forebrain in vivo.
Topics: Analysis of Variance; Animals; Antidepressive Agents; Autoreceptors; Citalopram; Dialysis; Drug Tolerance; Indoles; Infusions, Intravenous; Male; Prosencephalon; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists | 1995 |
The endogenous cerebral tetrapeptide 5-HT-moduline reduces in vivo the functional activity of central 5-HT1B receptors in the rat.
Topics: Animals; Brain; Dose-Response Relationship, Drug; Male; Neuropeptides; Oligopeptides; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptors, Serotonin | 1997 |
Chronic paroxetine desensitises 5-HT1D but not 5-HT1B autoreceptors in rat lateral geniculate nucleus.
Topics: Animals; Autoreceptors; Geniculate Bodies; Male; Paroxetine; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Receptor Agonists; Sumatriptan; Time Factors | 1997 |
Effects of the 5-HT1 receptor agonists, sumatriptan and CP 93,129, on dural arterial flow in the rat.
Topics: Animals; Cerebrovascular Circulation; Dura Mater; Male; Meningeal Arteries; Pyridines; Pyrroles; Rats; Rats, Wistar; Serotonin Receptor Agonists; Sumatriptan; Trigeminal Ganglion | 1997 |
Regulation of serotonin release in the frontal cortex and ventral hippocampus of homozygous mice lacking 5-HT1B receptors: in vivo microdialysis studies.
Topics: Animals; Frontal Lobe; Hippocampus; Homozygote; Male; Mice; Mice, Knockout; Mice, Transgenic; Microdialysis; Nerve Endings; Potassium; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Sumatriptan | 1997 |
A dual effect of 5-HT1B receptor stimulation on nociceptive dorsal horn neurones in rats.
Topics: Action Potentials; Animals; Drug Interactions; Electric Stimulation; Female; Neurons; Pain; Pindolol; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission | 1997 |
Effects of moderate and intensive training on functional activity of central 5-HT1B receptors in the rat substantia nigra.
Topics: Adenylyl Cyclases; Animals; Colforsin; Enzyme Induction; Male; Physical Conditioning, Animal; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Restraint, Physical; Serotonin Receptor Agonists; Substantia Nigra | 1998 |
Infusion of the serotonin1B (5-HT1B) agonist CP-93,129 into the parabrachial nucleus potently and selectively reduces food intake in rats.
Topics: Animals; Autoradiography; Depression, Chemical; Dose-Response Relationship, Drug; Eating; Injections; Male; Pons; Pyridines; Pyrroles; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Satiety Response; Serotonin Receptor Agonists | 1998 |
5-HT-moduline, a 5-HT(1B/1D) receptor endogenous modulator, interacts with dopamine release measured in vivo by microdialysis.
Topics: Animals; Brain; Dopamine; Drug Interactions; Male; Microdialysis; Neuropeptides; Oligopeptides; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Receptor Agonists | 1998 |
Serotonin1B receptor stimulation enhances cocaine reinforcement.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminopyridines; Animals; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Indoles; Injections, Intraventricular; Male; Oxadiazoles; Piperazines; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Self Administration; Serotonin Antagonists; Serotonin Receptor Agonists | 1998 |
Native 5-HT1B receptors expressed in OK cells display dual coupling to elevation of intracellular calcium concentrations and inhibition of adenylate cyclase.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Calcium; Cell Line; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Kidney; Methiothepin; Opossums; Oxadiazoles; Pertussis Toxin; Pindolol; Piperazines; Pyridines; Pyrroles; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Virulence Factors, Bordetella | 1998 |
The effects of 5-HT1A, 5-HT1B and 5-HT1D receptor agonists on trigeminal nociceptive neurotransmission in anaesthetized rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Analgesics; Animals; Electric Stimulation; Male; Migraine Disorders; Oxazoles; Oxazolidinones; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists; Trigeminal Caudal Nucleus; Tryptamines | 1998 |
Release of immunoreactive substance P in the brain stem upon stimulation of the cranial dura mater with low pH - inhibition by the serotonin (5-HT1) receptor agonist CP 93,129.
Topics: Animals; Brain; Brain Stem; Drug Administration Routes; Dura Mater; Hydrogen-Ion Concentration; Injections, Intravenous; Male; Pyridines; Pyrroles; Rats; Rats, Wistar; Serotonin Receptor Agonists; Substance P; Trigeminal Nuclei | 1998 |
Pharmacological profile of the prejunctional 5-HT1 receptors mediating inhibition of sympathetic vasopressor outflow in the pithed rat.
Topics: 5-Methoxytryptamine; Animals; Blood Pressure; Central Nervous System; Oxadiazoles; Pindolol; Piperazines; Pyridines; Pyrroles; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathetic Nervous System | 1998 |
5-HT1B receptors modulate release of [3H]dopamine from rat striatal synaptosomes.
Topics: Animals; Dopamine; Male; Neostriatum; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Receptor Agonists; Synaptosomes | 1999 |
Activation of 5-HT1B receptors in the nucleus accumbens reduces amphetamine-induced enhancement of responding for conditioned reward.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamine; Animals; Conditioning, Psychological; Indoles; Male; Nucleus Accumbens; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Reward; Serotonin; Serotonin Receptor Agonists; Water | 1999 |
Humanization of mouse 5-hydroxytryptamine1B receptor gene by homologous recombination: in vitro and in vivo characterization.
Topics: Animals; Benzamides; Benzopyrans; Binding Sites; Brain; Gene Expression; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hypothermia; In Situ Hybridization; Indoles; Mice; Mice, Transgenic; Motor Activity; Piperidones; Propylamines; Pyridines; Pyrimidines; Pyrroles; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Recombination, Genetic; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Tritium | 1999 |
Serotonin 5-HT(1B/1D) agonist-stimulated [(35)S]GTPgammaS binding in rat and guinea pig striatal membranes.
Topics: Animals; Corpus Striatum; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Male; Membranes; Oxadiazoles; Pyridines; Pyrroles; Radioligand Assay; Rats; Serotonin; Serotonin Receptor Agonists; Stimulation, Chemical; Sulfur Radioisotopes; Tryptamines | 1999 |
Modulation of acetylcholine and 5-hydroxytryptamine release in hippocampal slices of rats with fimbria-fornix lesions and intrahippocampal grafts containing cholinergic and/or serotonergic neurons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Biological Transport; Brain Tissue Transplantation; Choline; Choline O-Acetyltransferase; Diagonal Band of Broca; Electric Stimulation; Female; Fornix, Brain; Hippocampus; Muscarinic Agonists; Neurons; Organ Culture Techniques; Oxotremorine; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT1B; Receptors, Muscarinic; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Septal Nuclei; Serotonin; Serotonin Receptor Agonists; Tritium | 1999 |
Differential sensitivity of 5-HT1B auto and heteroreceptors.
Topics: Acetylcholine; Animals; Autoreceptors; Dopamine; Dose-Response Relationship, Drug; Hippocampus; Male; Neurotransmitter Agents; Potassium; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptosomes; Visual Cortex | 1999 |
5-HT1B receptors modulate release of [3H]dopamine from rat striatal synaptosomes: further evidence using 5-HT moduline, polyclonal 5-HT1B receptor antibodies and 5-HT1B receptor knock-out mice.
Topics: Amino Acid Sequence; Animals; Antibodies, Blocking; Antibody Specificity; Dopamine; In Vitro Techniques; Male; Mice; Mice, Knockout; Mice, Transgenic; Molecular Sequence Data; Neostriatum; Neuropeptides; Oligopeptides; Piperidones; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Synaptosomes | 2000 |
Effect of chronic paroxetine treatment on 5-HT1B and 5-HT1D autoreceptors in rat dorsal raphe nucleus.
Topics: Animals; Electric Stimulation; Male; Paroxetine; Piperazines; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan | 2000 |
Magnetic field desensitizes 5-HT(1B) receptor in brain: pharmacological and functional studies.
Topics: Animals; Binding, Competitive; Cell Membrane; Cerebral Cortex; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Electromagnetic Fields; Guanosine Triphosphate; Guinea Pigs; Humans; In Vitro Techniques; Ligands; Protein Conformation; Pyridines; Pyrroles; Rats; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Synaptosomes; Temperature; Transfection | 2000 |
Effects of physical training on functional activity of 5-HT1B receptors in rat central nervous system: role of 5-HT-moduline.
Topics: Animals; Guanosine 5'-O-(3-Thiotriphosphate); Hippocampus; Male; Neuropeptides; Oligopeptides; Physical Conditioning, Animal; Physical Exertion; Pyridines; Pyrroles; Radioligand Assay; Random Allocation; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Receptor Agonists; Substantia Nigra | 2000 |
Effects of sustained administration of the serotonin and norepinephrine reuptake inhibitor venlafaxine: II. In vitro studies in the rat.
Topics: Adrenergic alpha-Agonists; Animals; Autoreceptors; Brimonidine Tartrate; Carrier Proteins; Cricetinae; Cyclohexanols; Dose-Response Relationship, Drug; Hippocampus; In Vitro Techniques; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Pyridines; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Adrenergic, alpha-2; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists; Symporters; Time Factors; Tritium; Venlafaxine Hydrochloride | 2000 |
The 5HT(1B) receptor agonist, CP-93129, inhibits [(3)H]-GABA release from rat globus pallidus slices and reverses akinesia following intrapallidal injection in the reserpine-treated rat.
Topics: Animals; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Globus Pallidus; In Vitro Techniques; Male; Movement Disorders; Propanolamines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Reserpine; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium | 2000 |
Multiple 5-HT(1) autoreceptor subtypes govern serotonin release in dorsal and median raphé nuclei.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoreceptors; Benzamides; Biphenyl Compounds; Drug Synergism; Electric Stimulation; In Vitro Techniques; Male; Oxadiazoles; Piperazines; Protein Isoforms; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Time Factors | 2001 |
Activation of 5-HT(1B/1D) receptors in the mesolimbic dopamine system increases dopamine release from the nucleus accumbens: a microdialysis study.
Topics: Animals; Dopamine; Male; Microdialysis; Nucleus Accumbens; Pindolol; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Time Factors; Ventral Tegmental Area | 2001 |
Effects of 5-HT2 and 5-HT3 receptors on the modulation of nociceptive transmission in rat spinal cord according to the formalin test.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Dose-Response Relationship, Drug; Formaldehyde; Injections, Spinal; Male; Nociceptors; Pain; Pain Measurement; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission; Tropanes | 2001 |
The role of 5-HT1B receptors in the regulation of serotonin cell firing and release in the rat brain.
Topics: Animals; Brain; Electrophysiology; Kinetics; Male; Piperazines; Piperidones; Prosencephalon; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds | 2001 |
Enhanced contraction to 5-hydroxytryptamine is not due to "unmasking" of 5-hydroxytryptamine(1b) receptors in the mesenteric artery of the deoxycorticosterone acetate-salt rat.
Topics: Animals; Benzamides; Blood Pressure; Desoxycorticosterone; Dose-Response Relationship, Drug; Hypertension; In Vitro Techniques; Ketanserin; Male; Mesenteric Arteries; Phenylephrine; Potassium Chloride; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Vasoconstriction; Vasoconstrictor Agents | 2001 |
Serotonin-1B receptor-mediated inhibition of [(3)H]GABA release from rat ventral tegmental area slices.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzamides; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Male; Oxadiazoles; Pindolol; Piperazines; Potassium; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Ventral Tegmental Area | 2001 |
Modification of serotonin neuron properties in mice lacking 5-HT1A receptors.
Topics: Animals; Autoreceptors; Brimonidine Tartrate; Hippocampus; In Vitro Techniques; Male; Mice; Neurons; Norepinephrine; Pyridines; Pyrroles; Quinoxalines; Raphe Nuclei; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Adrenergic, alpha-2; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Receptor Agonists; Sumatriptan; Tritium | 2002 |
Activity-dependent presynaptic effect of serotonin 1B receptors on the somatosensory thalamocortical transmission in neonatal mice.
Topics: Aging; Animals; Animals, Newborn; Electric Stimulation; Excitatory Postsynaptic Potentials; In Vitro Techniques; Mice; Mice, Inbred Strains; Mice, Knockout; Neural Inhibition; Neurons; Patch-Clamp Techniques; Presynaptic Terminals; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; RNA, Messenger; Serotonin; Serotonin Receptor Agonists; Somatosensory Cortex; Synaptic Transmission; Thalamus; Ventral Thalamic Nuclei | 2002 |
Subthalamic 5-HT(1A) and 5-HT(1B) receptor modulation of RU 24969-induced behavioral profile in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Drug Interactions; Exploratory Behavior; Indoles; Male; Microinjections; Motor Activity; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Substantia Nigra; Subthalamus | 2002 |
Parabrachial infusion of D-fenfluramine reduces food intake. Blockade by the 5-HT(1B) antagonist SB-216641.
Topics: Animals; Benzamides; Brachial Plexus; Dose-Response Relationship, Drug; Eating; Fenfluramine; Infusions, Intravenous; Male; Oxadiazoles; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists | 2002 |
Activation of 5-HT(1B) receptors in the nucleus accumbens reduces self-administration of amphetamine on a progressive ratio schedule.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamine; Amphetamines; Animals; Central Nervous System Stimulants; Conditioning, Operant; Dose-Response Relationship, Drug; Food; Male; Nucleus Accumbens; Oxadiazoles; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Reinforcement Schedule; Self Administration; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 2002 |
The effects of selective serotonin reuptake inhibitors on extracellular 5-HT levels in the hippocampus of 5-HT(1B) receptor knockout mice.
Topics: Animals; Dose-Response Relationship, Drug; Extracellular Space; Fluvoxamine; Genotype; Hippocampus; Injections, Intraperitoneal; Mice; Mice, Inbred Strains; Mice, Knockout; Microdialysis; Paroxetine; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists; Time Factors | 2002 |
Extracellular serotonin in the prefrontal cortex is limited through terminal 5-HT(1B) autoreceptors: a microdialysis study in knockout mice.
Topics: Analysis of Variance; Animals; Autoreceptors; Benzopyrans; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Drug Interactions; Extracellular Space; Fluvoxamine; Male; Mice; Mice, Knockout; Microdialysis; Morpholines; Prefrontal Cortex; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors | 2002 |
Effects of serotonin (5-HT)(1B) receptor ligands, microinjected into accumbens subregions, on cocaine discrimination in rats.
Topics: Animals; Behavior, Animal; Benzamides; Cocaine; Conditioning, Operant; Discrimination Learning; Dose-Response Relationship, Drug; Ligands; Male; Microinjections; Nucleus Accumbens; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 2002 |
Effects of 5-HT(1B) receptor ligands microinjected into the accumbal shell or core on the sensitization to cocaine in rats.
Topics: Analysis of Variance; Animals; Benzamides; Cocaine; Dose-Response Relationship, Drug; Drug Interactions; Male; Microinjections; Motor Activity; Nucleus Accumbens; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 2002 |
Effects of 5-HT1B receptor ligands microinjected into the accumbal shell or core on the cocaine-induced locomotor hyperactivity in rats.
Topics: Animals; Benzamides; Cocaine; Hyperkinesis; Ligands; Male; Microinjections; Motor Activity; Nucleus Accumbens; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 2002 |
Activation of 5HT1B receptors inhibits glycinergic synaptic inputs to mammalian motoneurons during postnatal development.
Topics: Animals; Animals, Newborn; Dose-Response Relationship, Drug; Glycine; Glycine Agents; Hypoglossal Nerve; Motor Neurons; Neural Inhibition; Patch-Clamp Techniques; Pyridines; Pyrroles; Rats; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin Receptor Agonists; Strychnine; Synaptic Transmission | 2002 |
5,7-Dihydroxytryptamine lesions enhance and serotonergic grafts normalize the evoked overflow of acetylcholine in rat hippocampal slices.
Topics: 5,7-Dihydroxytryptamine; Acetylcholine; Animals; Choline; Chromatography, High Pressure Liquid; Hippocampus; Injections, Intraventricular; Male; Methiothepin; Neurons; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium | 2002 |
Neurotransmitter release and its presynaptic modulation in the rat hippocampus after selective damage to cholinergic or/and serotonergic afferents.
Topics: 5,7-Dihydroxytryptamine; Acetylcholine; Adrenergic alpha-Agonists; Animals; Antibodies, Monoclonal; Biogenic Monoamines; Brimonidine Tartrate; Choline O-Acetyltransferase; Cholinergic Agents; Cholinergic Fibers; Electric Stimulation; Hippocampus; Immunotoxins; Male; N-Glycosyl Hydrolases; Neurons, Afferent; Neurotoxins; Nicotine; Nicotinic Agonists; Norepinephrine; Organ Culture Techniques; Pyridines; Pyrroles; Quinoxalines; Rats; Rats, Long-Evans; Ribosome Inactivating Proteins, Type 1; Saporins; Serotonin; Serotonin Agents; Serotonin Receptor Agonists | 2003 |
The role of 5-HT1A/B autoreceptors in the antinociceptive effect of systemic administration of acetaminophen.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetaminophen; Analgesics, Non-Narcotic; Animals; Autoreceptors; Benzamides; Male; Mice; Oxadiazoles; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1 | 2003 |
Presynaptic modulation of acetylcholine, noradrenaline, and serotonin release in the hippocampus of aged rats with various levels of memory impairments.
Topics: Acetylcholine; Acetylcholinesterase; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Analysis of Variance; Animals; Behavior, Animal; Brimonidine Tartrate; Choline O-Acetyltransferase; Female; Hippocampus; Idazoxan; In Vitro Techniques; Maze Learning; Memory Disorders; Methiothepin; Muscarinic Agonists; Norepinephrine; Oxotremorine; Presynaptic Terminals; Pyridines; Pyrroles; Quinoxalines; Rats; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming; Tritium | 2003 |
Presynaptic regulation of neurotransmitter release in the cortex of aged rats with differential memory impairments.
Topics: Acetylcholine; Acetylcholinesterase; Adrenergic alpha-Agonists; Aging; Animals; Brimonidine Tartrate; Cerebral Cortex; Choline; Choline O-Acetyltransferase; Chromatography, High Pressure Liquid; Electric Stimulation; Female; Maze Learning; Memory Disorders; Muscarinic Agonists; Neurotransmitter Agents; Norepinephrine; Oxotremorine; Pyridines; Pyrroles; Quinoxalines; Rats; Rats, Long-Evans; Receptors, Presynaptic; Serotonin; Serotonin Receptor Agonists | 2003 |
S+ -flurbiprofen but not 5-HT1 agonists suppress basal and stimulated CGRP and PGE2 release from isolated rat dura mater.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Calcitonin Gene-Related Peptide; Culture Media, Conditioned; Dinoprostone; Drug Interactions; Dura Mater; Flurbiprofen; Immunoassay; In Vitro Techniques; Indoles; Inflammation Mediators; Male; Piperidines; Pyridines; Pyrroles; Rats; Rats, Wistar; Serotonin Receptor Agonists; Time Factors; Tryptamines | 2003 |
Role of 5-HT1B receptors in the regulation of extracellular serotonin and dopamine in the dorsal striatum of mice.
Topics: Animals; Chromatography, High Pressure Liquid; Corpus Striatum; Dopamine; Electrochemistry; Extracellular Fluid; Genotype; Male; Mice; Mice, Knockout; Microdialysis; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Receptor Agonists; Time Factors | 2003 |
Arterial expression of 5-HT2B and 5-HT1B receptors during development of DOCA-salt hypertension.
Topics: Animals; Arteries; Desoxycorticosterone; Female; Gene Expression; Hypertension; Indoles; Male; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2B; Serotonin Antagonists; Serotonin Receptor Agonists; Sodium Chloride; Thiophenes; Vasoconstriction | 2003 |
Differential involvement of central 5-HT1B and 5-HT3 receptor subtypes in the antinociceptive effect of paracetamol.
Topics: Acetaminophen; Analgesics, Non-Narcotic; Animals; Binding Sites; Brain; Male; Ondansetron; Pain Measurement; Protein Binding; Protein Isoforms; Pyridines; Pyrroles; Random Allocation; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin, 5-HT3; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT3 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2003 |
Further characterization of the 5-HT1 receptors mediating cardiac sympatho-inhibition in pithed rats: pharmacological correlation with the 5-HT1B and 5-HT1D subtypes.
Topics: Animals; Biphenyl Compounds; Decerebrate State; Male; Norepinephrine; Oxadiazoles; Piperazines; Piperidones; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Spiro Compounds; Sumatriptan; Sympathomimetics; Tachycardia | 2004 |
In vivo efflux of serotonin in the dorsal raphe nucleus of 5-HT1A receptor knockout mice.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dose-Response Relationship, Drug; Extracellular Fluid; Fluoxetine; Handling, Psychological; Male; Mice; Mice, Knockout; Microdialysis; Pyridines; Pyrroles; Raphe Nuclei; Receptor, Serotonin, 5-HT1A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists; Sodium Chloride; Stress, Physiological | 2004 |
Effects of 5-HT1B receptor ligands microinjected into the ventral tegmental area on the locomotor and sensitizating effects of cocaine in rats.
Topics: Analysis of Variance; Anesthetics, Local; Animals; Behavior, Animal; Benzamides; Cocaine; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Hyperkinesis; Male; Microinjections; Motor Activity; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Agents; Ventral Tegmental Area | 2004 |
5-Hydroxytryptamine 1B receptors mediate presynaptic inhibition of monosynaptic IPSC in the rat dorsolateral septal nucleus.
Topics: Analysis of Variance; Animals; Benzamides; Biphenyl Compounds; Calcium Channel Blockers; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Muscimol; Neural Inhibition; Neurons; omega-Agatoxin IVA; omega-Conotoxin GVIA; Oxadiazoles; Patch-Clamp Techniques; Pertussis Toxin; Phosphinic Acids; Piperazines; Presynaptic Terminals; Propanolamines; Pyridines; Pyrroles; Quinoxalines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Septal Nuclei; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission | 2004 |
Involvement of 5-HT1B receptors within the ventral tegmental area in regulation of mesolimbic dopaminergic neuronal activity via GABA mechanisms: a study with dual-probe microdialysis.
Topics: Animals; Baclofen; Benzamides; Biphenyl Compounds; Dopamine; GABA Agonists; gamma-Aminobutyric Acid; Male; Microdialysis; Neural Pathways; Neurons; Nucleus Accumbens; Oxadiazoles; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Serotonin Antagonists; Serotonin Receptor Agonists; Ventral Tegmental Area | 2004 |
Autoradiographic characterisation of [35S]GTPgammaS binding stimulation mediated by 5-HT1B receptor in postmortem human brain.
Topics: Aged; Autoradiography; Binding, Competitive; Biphenyl Compounds; Brain; Dipeptides; Drug Interactions; Female; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Male; Middle Aged; Oxadiazoles; Piperazines; Piperidones; Postmortem Changes; Protein Binding; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Sulfur Isotopes | 2005 |
Selective 5-HT1B receptor agonist reduces serotonin synthesis following acute, and not chronic, drug administration: results of an autoradiographic study.
Topics: Animals; Autoradiography; Brain Chemistry; Capillaries; Infusion Pumps, Implantable; Kinetics; Male; Neural Pathways; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Receptor Agonists; Time Factors; Tryptophan | 2005 |
5-HT1B receptor-mediated presynaptic inhibition of GABA release in the suprachiasmatic nucleus.
Topics: Animals; Bicuculline; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Potentials; Mice; Mice, Knockout; Neural Inhibition; Neurons; Patch-Clamp Techniques; Presynaptic Terminals; Pyridines; Pyrroles; Quinoxalines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Serotonin Receptor Agonists; Suprachiasmatic Nucleus; Tetrodotoxin; Time Factors; Valine | 2005 |
Involvement of spinal serotonin receptors in the regulation of intraspinal acetylcholine release.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Amphetamines; Animals; Biguanides; Citalopram; Dose-Response Relationship, Drug; Ketanserin; Male; Microdialysis; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Time Factors | 2005 |
Role of 5-HT1A and 5-HT1B receptors in the antinociceptive effect of tramadol.
Topics: Analgesics, Opioid; Animals; Benzamides; Dose-Response Relationship, Drug; Male; Mice; Oxadiazoles; Pain Threshold; Piperazines; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Serotonin Antagonists; Serotonin Receptor Agonists; Tramadol | 2005 |
Presynaptic serotonergic modulation of 5-HT and acetylcholine release in the hippocampus and the cortex of 5-HT1B-receptor knockout mice.
Topics: Acetylcholine; Analysis of Variance; Animals; Cerebral Cortex; Choline; Dose-Response Relationship, Drug; Electric Stimulation; Hippocampus; Male; Mice; Mice, Knockout; Presynaptic Terminals; Pyridines; Pyrroles; Quipazine; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium | 2006 |
Different serotonin receptor agonists have distinct effects on sound-evoked responses in inferior colliculus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acoustic Stimulation; Animals; Chiroptera; Dose-Response Relationship, Drug; Electrodes; Electrophysiology; Evoked Potentials, Auditory; Extracellular Space; gamma-Aminobutyric Acid; Glutamic Acid; Inferior Colliculi; Iontophoresis; Male; Pyrazines; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1A; Serotonin; Serotonin Receptor Agonists | 2006 |
5-HT1B receptor-mediated presynaptic inhibition at the calyx of Held of immature rats.
Topics: Age Factors; Animals; Animals, Newborn; Baclofen; Benzopyrans; Brain Stem; Calcium; Drug Interactions; Egtazic Acid; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Agonists; In Vitro Techniques; Morpholines; Neural Inhibition; Neurons; Patch-Clamp Techniques; Presynaptic Terminals; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Time Factors | 2006 |
Activation of 5-HT1B and 5-HT1D receptors in the rat nucleus tractus solitarius: opposing action on neurones that receive an excitatory vagal C-fibre afferent input.
Topics: Action Potentials; Animals; Benzamides; Drug Synergism; Electric Stimulation; Iontophoresis; Ketanserin; Male; Neural Inhibition; Neurons; Neurons, Afferent; Patch-Clamp Techniques; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists; Solitary Nucleus; Sumatriptan; Time Factors; Vagus Nerve | 2007 |
Presynaptic modulation of 5-HT release in the rat septal region.
Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Adrenergic alpha-Agonists; Analgesics, Non-Narcotic; Animals; Brimonidine Tartrate; Calcium; Dose-Response Relationship, Drug; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; In Vitro Techniques; Male; Neurons; Presynaptic Terminals; Pyridines; Pyrroles; Quinoxalines; Quipazine; Rats; Rats, Wistar; Septum of Brain; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 2007 |
Activity-dependent depression of local excitatory connections in the CA1 region of mouse hippocampus.
Topics: Animals; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Postsynaptic Potentials; GABA Antagonists; Hippocampus; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Nerve Net; Neural Inhibition; Patch-Clamp Techniques; Picrotoxin; Pyramidal Cells; Pyridines; Pyrroles; Serotonin Receptor Agonists; Xanthines | 2007 |
Anti-aggressive effects of agonists at 5-HT1B receptors in the dorsal raphe nucleus of mice.
Topics: Aggression; Animals; Behavior, Animal; Conditioning, Operant; Dose-Response Relationship, Drug; Male; Mice; Oxadiazoles; Piperazines; Pyridines; Pyrroles; Raphe Nuclei; Serotonin 5-HT1 Receptor Agonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2007 |
Agonist-mediated regulation of presynaptic receptor function during development of rat septal neurons in culture.
Topics: Acetylcholine; Animals; Cells, Cultured; Coculture Techniques; Dose-Response Relationship, Drug; Electric Stimulation; Embryo, Mammalian; Gene Expression Regulation, Developmental; Muscarinic Agonists; Neurons; Oxotremorine; Pyridines; Pyrroles; Rats; Receptors, Muscarinic; Receptors, Presynaptic; Septum of Brain; Serotonin; Serotonin Receptor Agonists; Time Factors; Tritium; Tryptophan Hydroxylase; Vesicular Acetylcholine Transport Proteins | 2007 |
Effect of 5-HT1B receptor agonists injected into the prefrontal cortex on maternal aggression in rats.
Topics: Aggression; Animals; Behavior, Animal; Female; Male; Maternal Behavior; Microinjections; Prefrontal Cortex; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Serotonin Receptor Agonists | 2007 |
Serotonin 1B receptor modulates frequency response curves and spectral integration in the inferior colliculus by reducing GABAergic inhibition.
Topics: Action Potentials; Animals; Bicuculline; Drug Interactions; GABA Antagonists; gamma-Aminobutyric Acid; Inferior Colliculi; Male; Mice; Mice, Inbred CBA; Neural Inhibition; Neurons; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Serotonin Receptor Agonists | 2008 |
Social instigation and aggressive behavior in mice: role of 5-HT1A and 5-HT1B receptors in the prefrontal cortex.
Topics: Aggression; Analysis of Variance; Animals; Behavior, Animal; Bites and Stings; Dose-Response Relationship, Drug; Grooming; Male; Mice; Photomicrography; Piperazines; Piperidones; Prefrontal Cortex; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Serotonin 5-HT1 Receptor Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Walking | 2008 |
5-HT(1A) and 5-HT(1B) receptors in the ventrolateral striatum differentially modulate apomorphine-induced jaw movements in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Benzamides; Corpus Striatum; Dopamine Agonists; Dose-Response Relationship, Drug; Electromyography; Magnetics; Male; Mandible; Masseter Muscle; Microinjections; Movement; Neck Muscles; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2008 |
Modulatory effects of serotonin on GABAergic synaptic transmission and membrane properties in the deep cerebellar nuclei.
Topics: Animals; Animals, Newborn; Biophysical Phenomena; Biophysics; Cerebellar Nuclei; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; GABA Agents; gamma-Aminobutyric Acid; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Membrane Potentials; Neural Inhibition; Neurons; Patch-Clamp Techniques; Pyridines; Pyrroles; Rats; Rats, Wistar; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptic Transmission; Time Factors | 2009 |
Activation of 5-HT1B receptors inhibits the vasodepressor sensory CGRPergic outflow in pithed rats.
Topics: Animals; Blood Pressure; Calcitonin Gene-Related Peptide; Disease Models, Animal; Dose-Response Relationship, Drug; Electric Stimulation; Heart Rate; Hexamethonium; Infusions, Intravenous; Male; Methoxamine; Piperidones; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists; Sodium Chloride; Spinal Cord; Spiro Compounds; Time Factors; Vasoconstrictor Agents | 2010 |
Progesterone reduces the inhibitory effect of a serotonin 1B receptor agonist on lordosis behavior.
Topics: Animals; Estradiol; Female; Handling, Psychological; Microinjections; Ovariectomy; Posture; Progesterone; Pyridines; Pyrroles; Rats; Rats, Inbred F344; Receptor, Serotonin, 5-HT1B; Serotonin Receptor Agonists; Sexual Behavior, Animal; Ventromedial Hypothalamic Nucleus | 2010 |
Social instigation and aggression in postpartum female rats: role of 5-Ht1A and 5-Ht1B receptors in the dorsal raphé nucleus and prefrontal cortex.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aggression; Animals; Female; Postpartum Period; Prefrontal Cortex; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Serotonin Antagonists; Serotonin Receptor Agonists | 2011 |
A novel mechanism for regulating hepatic glycogen synthesis involving serotonin and cyclin-dependent kinase-5.
Topics: Animals; Cells, Cultured; Cyclin-Dependent Kinase 5; Hepatocytes; Indoles; Liver; Liver Glycogen; Male; Metabolic Networks and Pathways; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrahydronaphthalenes | 2012 |
Infralimbic and dorsal raphé microinjection of the 5-HT(1B) receptor agonist CP-93,129: attenuation of aggressive behavior in CFW male mice.
Topics: Aggression; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Ethanol; Male; Mice; Microinjections; Motor Activity; Prefrontal Cortex; Pyridines; Pyrroles; Raphe Nuclei; Receptor, Serotonin, 5-HT1B; Reinforcement Schedule; Self Administration; Serotonin 5-HT1 Receptor Agonists | 2012 |
5-HT(1B) receptors inhibit glutamate release from primary afferent terminals in rat medullary dorsal horn neurons.
Topics: Action Potentials; Afferent Pathways; Animals; Electrophysiological Phenomena; Glutamic Acid; Posterior Horn Cells; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B | 2012 |
Presynaptic serotonergic gating of the subthalamonigral glutamatergic projection.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Analysis of Variance; Animals; Benzopyrans; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABAergic Neurons; Glutamates; In Vitro Techniques; Ion Channel Gating; Male; Mice; Morpholines; Neural Pathways; Patch-Clamp Techniques; Presynaptic Terminals; Pyridines; Pyrroles; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists; Sodium Channel Blockers; Substantia Nigra; Subthalamic Nucleus; Tetrodotoxin; Valine | 2013 |
Anticataleptic effects of 5-HT(1B) receptors in the globus pallidus.
Topics: Animals; Catalepsy; Globus Pallidus; Haloperidol; Locomotion; Male; Neurons; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists | 2013 |
Presynaptic 5-HT1B receptor-mediated synaptic suppression to the subplate neurons in the somatosensory cortex of neonatal rats.
Topics: Animals; Animals, Newborn; Dose-Response Relationship, Drug; Excitatory Postsynaptic Potentials; Male; Neurons; Piperidones; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Somatosensory Cortex; Spiro Compounds | 2014 |
5-Hydroxytryptamine does not reduce sympathetic nerve activity or neuroeffector function in the splanchnic circulation.
Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Electric Stimulation; Ganglia, Sympathetic; Male; Mesenteric Artery, Superior; Pyridines; Pyrroles; Rats; Serotonin; Serotonin Receptor Agonists; Splanchnic Circulation; Splanchnic Nerves; Sympathetic Nervous System; Vasoconstriction | 2015 |
CB1 receptors in the paraventricular nucleus of the hypothalamus modulate the release of 5-HT and GABA to stimulate food intake in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Arachidonic Acids; Cyproheptadine; Drug Interactions; Eating; gamma-Aminobutyric Acid; Male; Microinjections; Paraventricular Hypothalamic Nucleus; Piperazines; Piperidines; Piperidones; Pyrazoles; Pyridines; Pyrroles; Rats; Receptor, Cannabinoid, CB1; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Tritium | 2018 |