Page last updated: 2024-09-03

cp 93129 and pindolol

cp 93129 has been researched along with pindolol in 6 studies

Compound Research Comparison

Studies
(cp 93129)
Trials
(cp 93129)
Recent Studies (post-2010)
(cp 93129)
Studies
(pindolol)
Trials
(pindolol)
Recent Studies (post-2010) (pindolol)
1090113,71866292

Protein Interaction Comparison

ProteinTaxonomycp 93129 (IC50)pindolol (IC50)
Beta-2 adrenergic receptorHomo sapiens (human)0.0005
Beta-1 adrenergic receptorHomo sapiens (human)0.0009
Beta-3 adrenergic receptorHomo sapiens (human)0.088
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.048
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.048

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (66.67)18.2507
2000's2 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hjorth, S; Sharp, T1
Gjerstad, J; Hole, K; Tjølsen, A1
Branchek, TA; Zgombick, JM1
Centurión, D; Rabelo, G; Sánchez-López, A; Villalón, CM1
Yan, QS; Yan, SE2

Other Studies

6 other study(ies) available for cp 93129 and pindolol

ArticleYear
In vivo microdialysis evidence for central serotonin1A and serotonin1B autoreceptor blocking properties of the beta adrenoceptor antagonist (-)penbutolol.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Citalopram; Dialysis; Hippocampus; Male; Metoprolol; Penbutolol; Perfusion; Pindolol; Propanolamines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stereoisomerism

1993
A dual effect of 5-HT1B receptor stimulation on nociceptive dorsal horn neurones in rats.
    European journal of pharmacology, 1997, Sep-24, Volume: 335, Issue:2-3

    Topics: Action Potentials; Animals; Drug Interactions; Electric Stimulation; Female; Neurons; Pain; Pindolol; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission

1997
Native 5-HT1B receptors expressed in OK cells display dual coupling to elevation of intracellular calcium concentrations and inhibition of adenylate cyclase.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:5

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Calcium; Cell Line; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Kidney; Methiothepin; Opossums; Oxadiazoles; Pertussis Toxin; Pindolol; Piperazines; Pyridines; Pyrroles; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Virulence Factors, Bordetella

1998
Pharmacological profile of the prejunctional 5-HT1 receptors mediating inhibition of sympathetic vasopressor outflow in the pithed rat.
    Annals of the New York Academy of Sciences, 1998, Dec-15, Volume: 861

    Topics: 5-Methoxytryptamine; Animals; Blood Pressure; Central Nervous System; Oxadiazoles; Pindolol; Piperazines; Pyridines; Pyrroles; Rats; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Sympathetic Nervous System

1998
Activation of 5-HT(1B/1D) receptors in the mesolimbic dopamine system increases dopamine release from the nucleus accumbens: a microdialysis study.
    European journal of pharmacology, 2001, Apr-20, Volume: 418, Issue:1-2

    Topics: Animals; Dopamine; Male; Microdialysis; Nucleus Accumbens; Pindolol; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Time Factors; Ventral Tegmental Area

2001
Serotonin-1B receptor-mediated inhibition of [(3)H]GABA release from rat ventral tegmental area slices.
    Journal of neurochemistry, 2001, Volume: 79, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzamides; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Male; Oxadiazoles; Pindolol; Piperazines; Potassium; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Ventral Tegmental Area

2001