Page last updated: 2024-09-03

cp 93129 and colforsin

cp 93129 has been researched along with colforsin in 4 studies

Compound Research Comparison

Studies
(cp 93129)
Trials
(cp 93129)
Recent Studies (post-2010)
(cp 93129)
Studies
(colforsin)
Trials
(colforsin)
Recent Studies (post-2010) (colforsin)
10901113,460461,298

Protein Interaction Comparison

ProteinTaxonomycp 93129 (IC50)colforsin (IC50)
nuclear receptor subfamily 0 group B member 1Homo sapiens (human)1.729
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.041
Adenylate cyclase type 1Homo sapiens (human)0.0955

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (75.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Burkhart, CA; Heym, JH; Ives, JL; Lebel, LA; Macor, JE; Newman, ME; Nielsen, JA; Ryan, K; Schulz, DW; Torgersen, LK1
Fillion, G; Guezennec, Y; Liscia, P; Seguin, L1
Branchek, TA; Zgombick, JM1
Bailly, JM; Deschamps, F; Fillion, G; Grimaldi, B; Kochanek, M; Lambrozo, J; Massot, O1

Other Studies

4 other study(ies) available for cp 93129 and colforsin

ArticleYear
3-(1,2,5,6-Tetrahydropyrid-4-yl)pyrrolo[3,2-b]pyrid-5-one: a potent and selective serotonin (5-HT1B) agonist and rotationally restricted phenolic analogue of 5-methoxy-3-(1,2,5,6-tetrahydropyrid-4-yl)indole.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:8

    Topics: Adenylyl Cyclase Inhibitors; Animals; Chemical Phenomena; Chemistry; Colforsin; Cyclization; Eating; Guinea Pigs; Hippocampus; Indoles; Molecular Structure; Paraventricular Hypothalamic Nucleus; Pyridines; Pyrroles; Rats; Receptors, Serotonin; Serotonin; Substantia Nigra

1990
Effects of moderate and intensive training on functional activity of central 5-HT1B receptors in the rat substantia nigra.
    Acta physiologica Scandinavica, 1998, Volume: 162, Issue:1

    Topics: Adenylyl Cyclases; Animals; Colforsin; Enzyme Induction; Male; Physical Conditioning, Animal; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Restraint, Physical; Serotonin Receptor Agonists; Substantia Nigra

1998
Native 5-HT1B receptors expressed in OK cells display dual coupling to elevation of intracellular calcium concentrations and inhibition of adenylate cyclase.
    Naunyn-Schmiedeberg's archives of pharmacology, 1998, Volume: 358, Issue:5

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Calcium; Cell Line; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Kidney; Methiothepin; Opossums; Oxadiazoles; Pertussis Toxin; Pindolol; Piperazines; Pyridines; Pyrroles; Radioligand Assay; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Virulence Factors, Bordetella

1998
Magnetic field desensitizes 5-HT(1B) receptor in brain: pharmacological and functional studies.
    Brain research, 2000, Mar-06, Volume: 858, Issue:1

    Topics: Animals; Binding, Competitive; Cell Membrane; Cerebral Cortex; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Electromagnetic Fields; Guanosine Triphosphate; Guinea Pigs; Humans; In Vitro Techniques; Ligands; Protein Conformation; Pyridines; Pyrroles; Rats; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Synaptosomes; Temperature; Transfection

2000