Page last updated: 2024-09-03

cp 93129 and citalopram

cp 93129 has been researched along with citalopram in 4 studies

Compound Research Comparison

Studies
(cp 93129)
Trials
(cp 93129)
Recent Studies (post-2010)
(cp 93129)
Studies
(citalopram)
Trials
(citalopram)
Recent Studies (post-2010) (citalopram)
1090115,3481,4242,350

Protein Interaction Comparison

ProteinTaxonomycp 93129 (IC50)citalopram (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.297
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)2.196
AromataseRattus norvegicus (Norway rat)0.0018
Sodium-dependent noradrenaline transporter Homo sapiens (human)2.196
Alpha-1D adrenergic receptorHomo sapiens (human)3.289
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.297
Sodium-dependent serotonin transporterHomo sapiens (human)0.0227
Sodium-dependent serotonin transporterRattus norvegicus (Norway rat)0.0027
Histamine H1 receptorHomo sapiens (human)3.194
5-hydroxytryptamine receptor 2BHomo sapiens (human)1.839
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)3.1869
Sigma non-opioid intracellular receptor 1Homo sapiens (human)0.398
TransporterRattus norvegicus (Norway rat)8.8

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (75.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hjorth, S; Tao, R1
Hjorth, S; Sharp, T1
Auerbach, SB; Hjorth, S1
Höglund, AU; Kommalage, M1

Other Studies

4 other study(ies) available for cp 93129 and citalopram

ArticleYear
The putative 5-HT1B receptor agonist CP-93,129 suppresses rat hippocampal 5-HT release in vivo: comparison with RU 24969.
    European journal of pharmacology, 1991, Dec-17, Volume: 209, Issue:3

    Topics: Animals; Brain Chemistry; Citalopram; Dialysis; Hippocampus; Indoles; Male; Methiothepin; Pyridines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin

1991
In vivo microdialysis evidence for central serotonin1A and serotonin1B autoreceptor blocking properties of the beta adrenoceptor antagonist (-)penbutolol.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Citalopram; Dialysis; Hippocampus; Male; Metoprolol; Penbutolol; Perfusion; Pindolol; Propanolamines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stereoisomerism

1993
Effect of chronic administration of the selective serotonin (5-HT) uptake inhibitor citalopram on extracellular 5-HT and apparent autoreceptor sensitivity in rat forebrain in vivo.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:6

    Topics: Analysis of Variance; Animals; Antidepressive Agents; Autoreceptors; Citalopram; Dialysis; Drug Tolerance; Indoles; Infusions, Intravenous; Male; Prosencephalon; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Receptor Agonists

1995
Involvement of spinal serotonin receptors in the regulation of intraspinal acetylcholine release.
    European journal of pharmacology, 2005, Feb-21, Volume: 509, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Amphetamines; Animals; Biguanides; Citalopram; Dose-Response Relationship, Drug; Ketanserin; Male; Microdialysis; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Time Factors

2005