cp 93129 has been researched along with 8-hydroxy-2-(di-n-propylamino)tetralin in 21 studies
Studies (cp 93129) | Trials (cp 93129) | Recent Studies (post-2010) (cp 93129) | Studies (8-hydroxy-2-(di-n-propylamino)tetralin) | Trials (8-hydroxy-2-(di-n-propylamino)tetralin) | Recent Studies (post-2010) (8-hydroxy-2-(di-n-propylamino)tetralin) |
---|---|---|---|---|---|
109 | 0 | 11 | 3,530 | 7 | 389 |
Protein | Taxonomy | cp 93129 (IC50) | 8-hydroxy-2-(di-n-propylamino)tetralin (IC50) |
---|---|---|---|
5-hydroxytryptamine receptor 1A | Homo sapiens (human) | 0.0012 | |
5-hydroxytryptamine receptor 1A | Rattus norvegicus (Norway rat) | 0.0032 | |
Alpha-2B adrenergic receptor | Rattus norvegicus (Norway rat) | 0.81 | |
D(2) dopamine receptor | Bos taurus (cattle) | 0.8 | |
Alpha-2C adrenergic receptor | Rattus norvegicus (Norway rat) | 0.81 | |
Alpha-2A adrenergic receptor | Rattus norvegicus (Norway rat) | 0.81 | |
D(2) dopamine receptor | Rattus norvegicus (Norway rat) | 2.8959 | |
Lysosomal alpha-glucosidase | Bos taurus (cattle) | 0.0021 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 8 (38.10) | 18.2507 |
2000's | 10 (47.62) | 29.6817 |
2010's | 3 (14.29) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Buhot, MC; Naïli, S | 1 |
Hjorth, S; Sharp, T | 1 |
Buhot, MC; Naïli, S; Patra, SK | 1 |
Cassel, JC; Jackisch, R; Jeltsch, H; Lauth, D; Neufang, B; Szabo, B | 1 |
Koob, GF; Parsons, LH; Weiss, F | 1 |
Cumberbatch, MJ; Hargreaves, RJ; Hill, RG | 1 |
Fletcher, PJ; Korth, KM | 1 |
Balse, E; Cassel, JC; Haaf, A; Jackisch, R; Kelche, C; Suhr, R | 1 |
Hopwood, SE; Stamford, JA | 1 |
Goto, F; Ishizaki, K; Obata, H; Sasaki, M | 1 |
Yan, QS; Yan, SE | 1 |
Geyer, MA; Martinez-Price, DL | 1 |
Azampanah, A; Fletcher, PJ; Korth, KM | 1 |
Gibert-Rahola, J; Micó, JA; Ortega-Alvaro, A; Roca-Vinardell, A | 1 |
Adell, A; Amargós-Bosch, M; Artigas, F; Bortolozzi, A; Toth, M | 1 |
Höglund, AU; Kommalage, M | 1 |
Hurley, LM | 1 |
Fujita, S; Hatanaka, H; Kiguchi, M; Koshikawa, N; Lee, J; Suga, K; Terakado, M | 1 |
da Veiga, CP; de Almeida, RM; Lucion, AB; Miczek, KA | 1 |
Ding, S; Li, L; Zhou, FM | 1 |
Cruz-Martínez, AM; Escartín-Pérez, RE; Florán-Garduño, B; López-Alonso, VE; Mancilla-Díaz, JM; Tejas-Juárez, JG | 1 |
21 other study(ies) available for cp 93129 and 8-hydroxy-2-(di-n-propylamino)tetralin
Article | Year |
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Changes in exploratory activity following stimulation of hippocampal 5-HT1A and 5-HT1B receptors in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Exploratory Behavior; Habituation, Psychophysiologic; Hippocampus; Male; Motor Activity; Pyridines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Serotonin; Scopolamine; Serotonin Receptor Agonists; Space Perception; Stimulation, Chemical | 1995 |
In vivo microdialysis evidence for central serotonin1A and serotonin1B autoreceptor blocking properties of the beta adrenoceptor antagonist (-)penbutolol.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Citalopram; Dialysis; Hippocampus; Male; Metoprolol; Penbutolol; Perfusion; Pindolol; Propanolamines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stereoisomerism | 1993 |
Spatial memory deficits following stimulation of hippocampal 5-HT1B receptors in the rat.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Handling, Psychological; Hippocampus; Injections; Male; Maze Learning; Memory Disorders; Memory, Short-Term; Muscarinic Antagonists; Pyridines; Pyrroles; Rats; Receptors, Serotonin; Scopolamine; Serotonin Receptor Agonists; Space Perception | 1995 |
Downregulation of muscarinic- and 5-HT1B-mediated modulation of [3H]acetylcholine release in hippocampal slices of rats with fimbria-fornix lesions and intrahippocampal grafts of septal origin.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Atropine; Brain Tissue Transplantation; Choline; Choline O-Acetyltransferase; Cholinergic Fibers; Cholinesterase Inhibitors; Diffusion Chambers, Culture; Down-Regulation; Electric Stimulation; Female; Hippocampus; Hydroxyindoleacetic Acid; Mecamylamine; Methiothepin; Muscarinic Agonists; Muscarinic Antagonists; Neurons; Nicotinic Antagonists; Norepinephrine; Oxotremorine; Physostigmine; Pyridines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Receptors, Serotonin; Septal Nuclei; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium | 1995 |
Serotonin1B receptor stimulation enhances cocaine reinforcement.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminopyridines; Animals; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Indoles; Injections, Intraventricular; Male; Oxadiazoles; Piperazines; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Self Administration; Serotonin Antagonists; Serotonin Receptor Agonists | 1998 |
The effects of 5-HT1A, 5-HT1B and 5-HT1D receptor agonists on trigeminal nociceptive neurotransmission in anaesthetized rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Analgesics; Animals; Electric Stimulation; Male; Migraine Disorders; Oxazoles; Oxazolidinones; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists; Trigeminal Caudal Nucleus; Tryptamines | 1998 |
Activation of 5-HT1B receptors in the nucleus accumbens reduces amphetamine-induced enhancement of responding for conditioned reward.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamine; Animals; Conditioning, Psychological; Indoles; Male; Nucleus Accumbens; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Reward; Serotonin; Serotonin Receptor Agonists; Water | 1999 |
Modulation of acetylcholine and 5-hydroxytryptamine release in hippocampal slices of rats with fimbria-fornix lesions and intrahippocampal grafts containing cholinergic and/or serotonergic neurons.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Biological Transport; Brain Tissue Transplantation; Choline; Choline O-Acetyltransferase; Diagonal Band of Broca; Electric Stimulation; Female; Fornix, Brain; Hippocampus; Muscarinic Agonists; Neurons; Organ Culture Techniques; Oxotremorine; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT1B; Receptors, Muscarinic; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Septal Nuclei; Serotonin; Serotonin Receptor Agonists; Tritium | 1999 |
Multiple 5-HT(1) autoreceptor subtypes govern serotonin release in dorsal and median raphé nuclei.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoreceptors; Benzamides; Biphenyl Compounds; Drug Synergism; Electric Stimulation; In Vitro Techniques; Male; Oxadiazoles; Piperazines; Protein Isoforms; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Time Factors | 2001 |
Effects of 5-HT2 and 5-HT3 receptors on the modulation of nociceptive transmission in rat spinal cord according to the formalin test.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Dose-Response Relationship, Drug; Formaldehyde; Injections, Spinal; Male; Nociceptors; Pain; Pain Measurement; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission; Tropanes | 2001 |
Serotonin-1B receptor-mediated inhibition of [(3)H]GABA release from rat ventral tegmental area slices.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzamides; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Male; Oxadiazoles; Pindolol; Piperazines; Potassium; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Ventral Tegmental Area | 2001 |
Subthalamic 5-HT(1A) and 5-HT(1B) receptor modulation of RU 24969-induced behavioral profile in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Drug Interactions; Exploratory Behavior; Indoles; Male; Microinjections; Motor Activity; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Substantia Nigra; Subthalamus | 2002 |
Activation of 5-HT(1B) receptors in the nucleus accumbens reduces self-administration of amphetamine on a progressive ratio schedule.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamine; Amphetamines; Animals; Central Nervous System Stimulants; Conditioning, Operant; Dose-Response Relationship, Drug; Food; Male; Nucleus Accumbens; Oxadiazoles; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Reinforcement Schedule; Self Administration; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists | 2002 |
The role of 5-HT1A/B autoreceptors in the antinociceptive effect of systemic administration of acetaminophen.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetaminophen; Analgesics, Non-Narcotic; Animals; Autoreceptors; Benzamides; Male; Mice; Oxadiazoles; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1 | 2003 |
In vivo efflux of serotonin in the dorsal raphe nucleus of 5-HT1A receptor knockout mice.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dose-Response Relationship, Drug; Extracellular Fluid; Fluoxetine; Handling, Psychological; Male; Mice; Mice, Knockout; Microdialysis; Pyridines; Pyrroles; Raphe Nuclei; Receptor, Serotonin, 5-HT1A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists; Sodium Chloride; Stress, Physiological | 2004 |
Involvement of spinal serotonin receptors in the regulation of intraspinal acetylcholine release.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Amphetamines; Animals; Biguanides; Citalopram; Dose-Response Relationship, Drug; Ketanserin; Male; Microdialysis; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Time Factors | 2005 |
Different serotonin receptor agonists have distinct effects on sound-evoked responses in inferior colliculus.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acoustic Stimulation; Animals; Chiroptera; Dose-Response Relationship, Drug; Electrodes; Electrophysiology; Evoked Potentials, Auditory; Extracellular Space; gamma-Aminobutyric Acid; Glutamic Acid; Inferior Colliculi; Iontophoresis; Male; Pyrazines; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1A; Serotonin; Serotonin Receptor Agonists | 2006 |
5-HT(1A) and 5-HT(1B) receptors in the ventrolateral striatum differentially modulate apomorphine-induced jaw movements in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Benzamides; Corpus Striatum; Dopamine Agonists; Dose-Response Relationship, Drug; Electromyography; Magnetics; Male; Mandible; Masseter Muscle; Microinjections; Movement; Neck Muscles; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists | 2008 |
Social instigation and aggression in postpartum female rats: role of 5-Ht1A and 5-Ht1B receptors in the dorsal raphé nucleus and prefrontal cortex.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aggression; Animals; Female; Postpartum Period; Prefrontal Cortex; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Serotonin Antagonists; Serotonin Receptor Agonists | 2011 |
Presynaptic serotonergic gating of the subthalamonigral glutamatergic projection.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Analysis of Variance; Animals; Benzopyrans; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABAergic Neurons; Glutamates; In Vitro Techniques; Ion Channel Gating; Male; Mice; Morpholines; Neural Pathways; Patch-Clamp Techniques; Presynaptic Terminals; Pyridines; Pyrroles; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists; Sodium Channel Blockers; Substantia Nigra; Subthalamic Nucleus; Tetrodotoxin; Valine | 2013 |
CB1 receptors in the paraventricular nucleus of the hypothalamus modulate the release of 5-HT and GABA to stimulate food intake in rats.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Arachidonic Acids; Cyproheptadine; Drug Interactions; Eating; gamma-Aminobutyric Acid; Male; Microinjections; Paraventricular Hypothalamic Nucleus; Piperazines; Piperidines; Piperidones; Pyrazoles; Pyridines; Pyrroles; Rats; Receptor, Cannabinoid, CB1; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Tritium | 2018 |