Page last updated: 2024-09-03

cp 93129 and 8-hydroxy-2-(di-n-propylamino)tetralin

cp 93129 has been researched along with 8-hydroxy-2-(di-n-propylamino)tetralin in 21 studies

Compound Research Comparison

Studies
(cp 93129)
Trials
(cp 93129)
Recent Studies (post-2010)
(cp 93129)
Studies
(8-hydroxy-2-(di-n-propylamino)tetralin)
Trials
(8-hydroxy-2-(di-n-propylamino)tetralin)
Recent Studies (post-2010) (8-hydroxy-2-(di-n-propylamino)tetralin)
1090113,5307389

Protein Interaction Comparison

ProteinTaxonomycp 93129 (IC50)8-hydroxy-2-(di-n-propylamino)tetralin (IC50)
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.0012
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0032
Alpha-2B adrenergic receptorRattus norvegicus (Norway rat)0.81
D(2) dopamine receptorBos taurus (cattle)0.8
Alpha-2C adrenergic receptorRattus norvegicus (Norway rat)0.81
Alpha-2A adrenergic receptorRattus norvegicus (Norway rat)0.81
D(2) dopamine receptorRattus norvegicus (Norway rat)2.8959
Lysosomal alpha-glucosidaseBos taurus (cattle)0.0021

Research

Studies (21)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's8 (38.10)18.2507
2000's10 (47.62)29.6817
2010's3 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Buhot, MC; Naïli, S1
Hjorth, S; Sharp, T1
Buhot, MC; Naïli, S; Patra, SK1
Cassel, JC; Jackisch, R; Jeltsch, H; Lauth, D; Neufang, B; Szabo, B1
Koob, GF; Parsons, LH; Weiss, F1
Cumberbatch, MJ; Hargreaves, RJ; Hill, RG1
Fletcher, PJ; Korth, KM1
Balse, E; Cassel, JC; Haaf, A; Jackisch, R; Kelche, C; Suhr, R1
Hopwood, SE; Stamford, JA1
Goto, F; Ishizaki, K; Obata, H; Sasaki, M1
Yan, QS; Yan, SE1
Geyer, MA; Martinez-Price, DL1
Azampanah, A; Fletcher, PJ; Korth, KM1
Gibert-Rahola, J; Micó, JA; Ortega-Alvaro, A; Roca-Vinardell, A1
Adell, A; Amargós-Bosch, M; Artigas, F; Bortolozzi, A; Toth, M1
Höglund, AU; Kommalage, M1
Hurley, LM1
Fujita, S; Hatanaka, H; Kiguchi, M; Koshikawa, N; Lee, J; Suga, K; Terakado, M1
da Veiga, CP; de Almeida, RM; Lucion, AB; Miczek, KA1
Ding, S; Li, L; Zhou, FM1
Cruz-Martínez, AM; Escartín-Pérez, RE; Florán-Garduño, B; López-Alonso, VE; Mancilla-Díaz, JM; Tejas-Juárez, JG1

Other Studies

21 other study(ies) available for cp 93129 and 8-hydroxy-2-(di-n-propylamino)tetralin

ArticleYear
Changes in exploratory activity following stimulation of hippocampal 5-HT1A and 5-HT1B receptors in the rat.
    Hippocampus, 1995, Volume: 5, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Exploratory Behavior; Habituation, Psychophysiologic; Hippocampus; Male; Motor Activity; Pyridines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Serotonin; Scopolamine; Serotonin Receptor Agonists; Space Perception; Stimulation, Chemical

1995
In vivo microdialysis evidence for central serotonin1A and serotonin1B autoreceptor blocking properties of the beta adrenoceptor antagonist (-)penbutolol.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 265, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adrenergic beta-Antagonists; Animals; Citalopram; Dialysis; Hippocampus; Male; Metoprolol; Penbutolol; Perfusion; Pindolol; Propanolamines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Stereoisomerism

1993
Spatial memory deficits following stimulation of hippocampal 5-HT1B receptors in the rat.
    European journal of pharmacology, 1995, Oct-24, Volume: 285, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Handling, Psychological; Hippocampus; Injections; Male; Maze Learning; Memory Disorders; Memory, Short-Term; Muscarinic Antagonists; Pyridines; Pyrroles; Rats; Receptors, Serotonin; Scopolamine; Serotonin Receptor Agonists; Space Perception

1995
Downregulation of muscarinic- and 5-HT1B-mediated modulation of [3H]acetylcholine release in hippocampal slices of rats with fimbria-fornix lesions and intrahippocampal grafts of septal origin.
    Brain research, 1995, Dec-18, Volume: 704, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Atropine; Brain Tissue Transplantation; Choline; Choline O-Acetyltransferase; Cholinergic Fibers; Cholinesterase Inhibitors; Diffusion Chambers, Culture; Down-Regulation; Electric Stimulation; Female; Hippocampus; Hydroxyindoleacetic Acid; Mecamylamine; Methiothepin; Muscarinic Agonists; Muscarinic Antagonists; Neurons; Nicotinic Antagonists; Norepinephrine; Oxotremorine; Physostigmine; Pyridines; Pyrroles; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Receptors, Serotonin; Septal Nuclei; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tritium

1995
Serotonin1B receptor stimulation enhances cocaine reinforcement.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Dec-01, Volume: 18, Issue:23

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminopyridines; Animals; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Indoles; Injections, Intraventricular; Male; Oxadiazoles; Piperazines; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Self Administration; Serotonin Antagonists; Serotonin Receptor Agonists

1998
The effects of 5-HT1A, 5-HT1B and 5-HT1D receptor agonists on trigeminal nociceptive neurotransmission in anaesthetized rats.
    European journal of pharmacology, 1998, Nov-27, Volume: 362, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Analgesics; Animals; Electric Stimulation; Male; Migraine Disorders; Oxazoles; Oxazolidinones; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin Receptor Agonists; Trigeminal Caudal Nucleus; Tryptamines

1998
Activation of 5-HT1B receptors in the nucleus accumbens reduces amphetamine-induced enhancement of responding for conditioned reward.
    Psychopharmacology, 1999, Volume: 142, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamine; Animals; Conditioning, Psychological; Indoles; Male; Nucleus Accumbens; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Reward; Serotonin; Serotonin Receptor Agonists; Water

1999
Modulation of acetylcholine and 5-hydroxytryptamine release in hippocampal slices of rats with fimbria-fornix lesions and intrahippocampal grafts containing cholinergic and/or serotonergic neurons.
    Brain research bulletin, 1999, Sep-01, Volume: 50, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Biological Transport; Brain Tissue Transplantation; Choline; Choline O-Acetyltransferase; Diagonal Band of Broca; Electric Stimulation; Female; Fornix, Brain; Hippocampus; Muscarinic Agonists; Neurons; Organ Culture Techniques; Oxotremorine; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Long-Evans; Receptor, Serotonin, 5-HT1B; Receptors, Muscarinic; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Septal Nuclei; Serotonin; Serotonin Receptor Agonists; Tritium

1999
Multiple 5-HT(1) autoreceptor subtypes govern serotonin release in dorsal and median raphé nuclei.
    Neuropharmacology, 2001, Volume: 40, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Autoreceptors; Benzamides; Biphenyl Compounds; Drug Synergism; Electric Stimulation; In Vitro Techniques; Male; Oxadiazoles; Piperazines; Protein Isoforms; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Time Factors

2001
Effects of 5-HT2 and 5-HT3 receptors on the modulation of nociceptive transmission in rat spinal cord according to the formalin test.
    European journal of pharmacology, 2001, Jul-13, Volume: 424, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Dose-Response Relationship, Drug; Formaldehyde; Injections, Spinal; Male; Nociceptors; Pain; Pain Measurement; Pyridines; Pyrroles; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Synaptic Transmission; Tropanes

2001
Serotonin-1B receptor-mediated inhibition of [(3)H]GABA release from rat ventral tegmental area slices.
    Journal of neurochemistry, 2001, Volume: 79, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzamides; Electrophysiology; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Indoles; Male; Oxadiazoles; Pindolol; Piperazines; Potassium; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Ventral Tegmental Area

2001
Subthalamic 5-HT(1A) and 5-HT(1B) receptor modulation of RU 24969-induced behavioral profile in rats.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 71, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Behavior, Animal; Drug Interactions; Exploratory Behavior; Indoles; Male; Microinjections; Motor Activity; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Receptor Agonists; Substantia Nigra; Subthalamus

2002
Activation of 5-HT(1B) receptors in the nucleus accumbens reduces self-administration of amphetamine on a progressive ratio schedule.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 71, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamine; Amphetamines; Animals; Central Nervous System Stimulants; Conditioning, Operant; Dose-Response Relationship, Drug; Food; Male; Nucleus Accumbens; Oxadiazoles; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Reinforcement Schedule; Self Administration; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2002
The role of 5-HT1A/B autoreceptors in the antinociceptive effect of systemic administration of acetaminophen.
    Anesthesiology, 2003, Volume: 98, Issue:3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetaminophen; Analgesics, Non-Narcotic; Animals; Autoreceptors; Benzamides; Male; Mice; Oxadiazoles; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Receptors, Serotonin, 5-HT1

2003
In vivo efflux of serotonin in the dorsal raphe nucleus of 5-HT1A receptor knockout mice.
    Journal of neurochemistry, 2004, Volume: 88, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Dose-Response Relationship, Drug; Extracellular Fluid; Fluoxetine; Handling, Psychological; Male; Mice; Mice, Knockout; Microdialysis; Pyridines; Pyrroles; Raphe Nuclei; Receptor, Serotonin, 5-HT1A; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists; Sodium Chloride; Stress, Physiological

2004
Involvement of spinal serotonin receptors in the regulation of intraspinal acetylcholine release.
    European journal of pharmacology, 2005, Feb-21, Volume: 509, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Amphetamines; Animals; Biguanides; Citalopram; Dose-Response Relationship, Drug; Ketanserin; Male; Microdialysis; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spinal Cord; Time Factors

2005
Different serotonin receptor agonists have distinct effects on sound-evoked responses in inferior colliculus.
    Journal of neurophysiology, 2006, Volume: 96, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acoustic Stimulation; Animals; Chiroptera; Dose-Response Relationship, Drug; Electrodes; Electrophysiology; Evoked Potentials, Auditory; Extracellular Space; gamma-Aminobutyric Acid; Glutamic Acid; Inferior Colliculi; Iontophoresis; Male; Pyrazines; Pyridines; Pyrroles; Receptor, Serotonin, 5-HT1A; Serotonin; Serotonin Receptor Agonists

2006
5-HT(1A) and 5-HT(1B) receptors in the ventrolateral striatum differentially modulate apomorphine-induced jaw movements in rats.
    Journal of oral science, 2008, Volume: 50, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Apomorphine; Benzamides; Corpus Striatum; Dopamine Agonists; Dose-Response Relationship, Drug; Electromyography; Magnetics; Male; Mandible; Masseter Muscle; Microinjections; Movement; Neck Muscles; Piperazines; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Serotonin Receptor Agonists

2008
Social instigation and aggression in postpartum female rats: role of 5-Ht1A and 5-Ht1B receptors in the dorsal raphé nucleus and prefrontal cortex.
    Psychopharmacology, 2011, Volume: 213, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aggression; Animals; Female; Postpartum Period; Prefrontal Cortex; Pyridines; Pyrroles; Raphe Nuclei; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptor, Serotonin, 5-HT1B; Serotonin Antagonists; Serotonin Receptor Agonists

2011
Presynaptic serotonergic gating of the subthalamonigral glutamatergic projection.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Mar-13, Volume: 33, Issue:11

    Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; 8-Hydroxy-2-(di-n-propylamino)tetralin; Action Potentials; Analysis of Variance; Animals; Benzopyrans; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Female; GABAergic Neurons; Glutamates; In Vitro Techniques; Ion Channel Gating; Male; Mice; Morpholines; Neural Pathways; Patch-Clamp Techniques; Presynaptic Terminals; Pyridines; Pyrroles; Serotonin; Serotonin Antagonists; Serotonin Plasma Membrane Transport Proteins; Serotonin Receptor Agonists; Sodium Channel Blockers; Substantia Nigra; Subthalamic Nucleus; Tetrodotoxin; Valine

2013
CB1 receptors in the paraventricular nucleus of the hypothalamus modulate the release of 5-HT and GABA to stimulate food intake in rats.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2018, Volume: 28, Issue:11

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamines; Animals; Arachidonic Acids; Cyproheptadine; Drug Interactions; Eating; gamma-Aminobutyric Acid; Male; Microinjections; Paraventricular Hypothalamic Nucleus; Piperazines; Piperidines; Piperidones; Pyrazoles; Pyridines; Pyrroles; Rats; Receptor, Cannabinoid, CB1; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Tritium

2018