Page last updated: 2024-09-03

cp 93129 and 5-carboxamidotryptamine

cp 93129 has been researched along with 5-carboxamidotryptamine in 7 studies

Compound Research Comparison

Studies
(cp 93129)
Trials
(cp 93129)
Recent Studies (post-2010)
(cp 93129)
Studies
(5-carboxamidotryptamine)
Trials
(5-carboxamidotryptamine)
Recent Studies (post-2010) (5-carboxamidotryptamine)
109011392136

Protein Interaction Comparison

ProteinTaxonomycp 93129 (IC50)5-carboxamidotryptamine (IC50)
5-hydroxytryptamine receptor 1DSus scrofa (pig)0.004

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (85.71)18.2507
2000's0 (0.00)29.6817
2010's1 (14.29)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Audinot-Bouchez, V; Chaput, C; Conte, C; Lavielle, G; Lochon, S; Millan, MJ; Newman-Tancredi, A; Verrièle, L1
Bruinvels, AT; Hoyer, D; Landwehrmeyer, B; Palacios, JM; Probst, A1
Castanon, N; Chauveau, J; Chaveau, J; Hen, R; Macor, JE; Moskowitz, MA; Scearce, K; Waeber, C; Yu, XJ1
Fletcher, PJ; Korth, KM1
Bakker, MH; Bonaventure, P; Cras, P; Langlois, X; Leysen, JE; Luyten, WH; Megens, AA; Serneels, L; Umans, L; Van Leuven, F1
Alper, RH; Mize, AL1
Barman, SM; Burnett, R; Darios, ES; Davis, RP; Morrison, SF; Orer, HS; Seitz, BM; Watts, SW1

Other Studies

7 other study(ies) available for cp 93129 and 5-carboxamidotryptamine

ArticleYear
Agonist activity of antimigraine drugs at recombinant human 5-HT1A receptors: potential implications for prophylactic and acute therapy.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 355, Issue:6

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Benzopyrans; Binding, Competitive; Cell Membrane; Cricetinae; Dihydroergotamine; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Humans; In Vitro Techniques; Indoles; Lisuride; Methysergide; Migraine Disorders; Piperazines; Piperidines; Pizotyline; Propranolol; Propylamines; Protein Binding; Pyridines; Pyrimidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Recombinant Proteins; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sumatriptan; Tryptamines

1997
A comparative autoradiographic study of 5-HT1D binding sites in human and guinea-pig brain using different radioligands.
    Brain research. Molecular brain research, 1994, Volume: 21, Issue:1-2

    Topics: Aged; Animals; Autoradiography; Binding Sites; Binding, Competitive; Brain; Dipeptides; Female; Guinea Pigs; Humans; Iodine Radioisotopes; Kinetics; Ligands; Male; Organ Specificity; Pyridines; Pyrroles; Receptors, Serotonin; Serotonin; Species Specificity; Sumatriptan; Tritium; Yohimbine

1994
5-Carboxamido-tryptamine, CP-122,288 and dihydroergotamine but not sumatriptan, CP-93,129, and serotonin-5-O-carboxymethyl-glycyl -tyrosinamide block dural plasma protein extravasation in knockout mice that lack 5-hydroxytryptamine1B receptors.
    Molecular pharmacology, 1996, Volume: 49, Issue:5

    Topics: Animals; Capillary Permeability; Dihydroergotamine; Dipeptides; Mice; Mice, Knockout; Pyridines; Pyrroles; Pyrrolidines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Sumatriptan; Trigeminal Ganglion

1996
Activation of 5-HT1B receptors in the nucleus accumbens reduces amphetamine-induced enhancement of responding for conditioned reward.
    Psychopharmacology, 1999, Volume: 142, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Amphetamine; Animals; Conditioning, Psychological; Indoles; Male; Nucleus Accumbens; Pyridines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Reward; Serotonin; Serotonin Receptor Agonists; Water

1999
Humanization of mouse 5-hydroxytryptamine1B receptor gene by homologous recombination: in vitro and in vivo characterization.
    Molecular pharmacology, 1999, Volume: 56, Issue:1

    Topics: Animals; Benzamides; Benzopyrans; Binding Sites; Brain; Gene Expression; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hypothermia; In Situ Hybridization; Indoles; Mice; Mice, Transgenic; Motor Activity; Piperidones; Propylamines; Pyridines; Pyrimidines; Pyrroles; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Recombination, Genetic; RNA, Messenger; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Spiro Compounds; Tritium

1999
Serotonin 5-HT(1B/1D) agonist-stimulated [(35)S]GTPgammaS binding in rat and guinea pig striatal membranes.
    Brain research, 1999, Jul-31, Volume: 836, Issue:1-2

    Topics: Animals; Corpus Striatum; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Male; Membranes; Oxadiazoles; Pyridines; Pyrroles; Radioligand Assay; Rats; Serotonin; Serotonin Receptor Agonists; Stimulation, Chemical; Sulfur Radioisotopes; Tryptamines

1999
5-Hydroxytryptamine does not reduce sympathetic nerve activity or neuroeffector function in the splanchnic circulation.
    European journal of pharmacology, 2015, May-05, Volume: 754

    Topics: Animals; Blood Pressure; Dose-Response Relationship, Drug; Electric Stimulation; Ganglia, Sympathetic; Male; Mesenteric Artery, Superior; Pyridines; Pyrroles; Rats; Serotonin; Serotonin Receptor Agonists; Splanchnic Circulation; Splanchnic Nerves; Sympathetic Nervous System; Vasoconstriction

2015