Page last updated: 2024-09-03

cp 65,526 and sdz psc 833

cp 65,526 has been researched along with sdz psc 833 in 4 studies

Compound Research Comparison

Studies
(cp 65,526)
Trials
(cp 65,526)
Recent Studies (post-2010)
(cp 65,526)
Studies
(sdz psc 833)
Trials
(sdz psc 833)
Recent Studies (post-2010) (sdz psc 833)
65154555566

Protein Interaction Comparison

ProteinTaxonomycp 65,526 (IC50)sdz psc 833 (IC50)
ATP-dependent translocase ABCB1Homo sapiens (human)0.3969

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's3 (75.00)18.2507
2000's1 (25.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beliveau, R; Jetté, L; Leclerc, JM; Murphy, GF1
Beaulieu, E; Béliveau, R; Jetté, L; Leclerc, JM1
Béliveau, R; Jetté, L; Murphy, GF1
Ambudkar, SV; Barnett, D; Bates, SE; Finley, EM; Fojo, T; Oldham, RK; Robey, RW; Shukla, S1

Trials

1 trial(s) available for cp 65,526 and sdz psc 833

ArticleYear
Inhibition of P-glycoprotein (ABCB1)- and multidrug resistance-associated protein 1 (ABCC1)-mediated transport by the orally administered inhibitor, CBT-1((R)).
    Biochemical pharmacology, 2008, Mar-15, Volume: 75, Issue:6

    Topics: Adenosine Triphosphatases; Alkaloids; Animals; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Factors; Biological Transport; Cell Line; Cell Line, Tumor; Cyclosporins; Depsipeptides; Fluorescent Dyes; Fluorouracil; Humans; Insecta; Multidrug Resistance-Associated Proteins; Neoplasms; Paclitaxel; Prazosin; Quinolines; Rhodamine 123; Verapamil; Vinblastine

2008

Other Studies

3 other study(ies) available for cp 65,526 and sdz psc 833

ArticleYear
Interaction of drugs with P-glycoprotein in brain capillaries.
    Biochemical pharmacology, 1995, Nov-09, Volume: 50, Issue:10

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blood-Brain Barrier; Brain; Capillaries; Cyclosporine; Cyclosporins; Drug Interactions; Glycerol; In Vitro Techniques; Iodine Radioisotopes; Male; Prazosin; Rats; Rats, Sprague-Dawley; Time Factors; Tritium

1995
Cyclosporin A treatment induces overexpression of P-glycoprotein in the kidney and other tissues.
    The American journal of physiology, 1996, Volume: 270, Issue:5 Pt 2

    Topics: Administration, Oral; Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cyclosporine; Cyclosporins; Immunosuppressive Agents; Injections, Subcutaneous; Kidney; Male; Microvilli; Prazosin; Rats; Rats, Sprague-Dawley; Time Factors

1996
Drug binding to P-glycoprotein is inhibited in normal tissues following SDZ-PSC 833 treatment.
    International journal of cancer, 1998, May-29, Volume: 76, Issue:5

    Topics: Administration, Oral; Animals; Antineoplastic Agents, Phytogenic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Blotting, Western; Brain; Calcium Channel Blockers; Capillaries; Cyclosporine; Cyclosporins; Drug Interactions; Fluorescent Dyes; Injections, Subcutaneous; Iodine Radioisotopes; Kidney; Liver; Male; Microvilli; Photoaffinity Labels; Prazosin; Rats; Rats, Sprague-Dawley; Rhodamine 123; Rhodamines; Verapamil; Vinblastine

1998