Page last updated: 2024-09-03

cp 65,526 and colchicine

cp 65,526 has been researched along with colchicine in 6 studies

Compound Research Comparison

Studies
(cp 65,526)
Trials
(cp 65,526)
Recent Studies (post-2010)
(cp 65,526)
Studies
(colchicine)
Trials
(colchicine)
Recent Studies (post-2010) (colchicine)
651515,4724042,974

Protein Interaction Comparison

ProteinTaxonomycp 65,526 (IC50)colchicine (IC50)
Tubulin alpha-1A chainSus scrofa (pig)3.7639
Tubulin beta chainSus scrofa (pig)3.8663
Tubulin beta-4A chainHomo sapiens (human)2.4334
Tubulin beta chainHomo sapiens (human)2.7244
Tubulin alpha-3C chainHomo sapiens (human)2.4334
Serine/threonine-protein kinase pim-1Homo sapiens (human)4.3
Tubulin alpha-1B chainHomo sapiens (human)2.4334
Tubulin alpha-4A chainHomo sapiens (human)2.4334
Tubulin beta-4B chainHomo sapiens (human)2.4334
Vesicular acetylcholine transporterTetronarce californica (Pacific electric ray)2.62
Tubulin beta-3 chainHomo sapiens (human)2.4334
Tubulin beta-2A chainHomo sapiens (human)2.4334
Tubulin beta-8 chainHomo sapiens (human)2.4334
Tubulin beta-2B chainBos taurus (cattle)2.8255
Tubulin alpha-3E chainHomo sapiens (human)2.4334
Tubulin alpha-1A chainHomo sapiens (human)2.4334
Similar to alpha-tubulin isoform 1 Bos taurus (cattle)3.0611
Similar to alpha-tubulin isoform 1 Bos taurus (cattle)3.1553
Tubulin alpha-1C chainHomo sapiens (human)2.4334
Tubulin beta-6 chainHomo sapiens (human)2.4334
Tubulin beta-2B chainHomo sapiens (human)2.4334
Tubulin beta-1 chainHomo sapiens (human)2.4334

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's6 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Agresti, M; Mehta, ND; Safa, AR; Tamai, I; Vahabi, S1
Croop, JM; Kronauge, JF; Piwnica-Worms, D; Rao, VV1
Agresti, M; Grizzuti, K; Gros, P; Kajiji, S; Safa, AR; Talbot, F; Van Dyke-Phillips, V1
Collins, KI; Greenberger, LM; Zhang, X1
Beaudet, L; Gros, P; Urbatsch, IL1
Gottesman, MM; Hrycyna, CA; Pastan, I; Ramachandra, M1

Other Studies

6 other study(ies) available for cp 65,526 and colchicine

ArticleYear
The alpha 1-adrenergic photoaffinity probe [125I]arylazidoprazosin binds to a specific peptide of P-glycoprotein in multidrug-resistant cells.
    Biochemical and biophysical research communications, 1990, Jan-15, Volume: 166, Issue:1

    Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Line; Colchicine; Cricetinae; Cricetulus; Dactinomycin; Drug Resistance; Electrophoresis, Polyacrylamide Gel; Iodine Radioisotopes; Kinetics; Membrane Glycoproteins; Neoplasm Proteins; Peptide Mapping; Prazosin; Quinazolines; Vinca Alkaloids; Vincristine

1990
Characterization of multidrug resistance P-glycoprotein transport function with an organotechnetium cation.
    Biochemistry, 1995, Sep-26, Volume: 34, Issue:38

    Topics: Adenosine Triphosphate; Allosteric Regulation; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Transport; Cations; Cell Survival; Cells, Cultured; Colchicine; Cricetinae; Dose-Response Relationship, Drug; Doxorubicin; Humans; Kinetics; Lipid Bilayers; Pharmaceutical Preparations; Phloretin; Prazosin; Quinidine; Technetium Tc 99m Sestamibi; Tetraphenylborate

1995
Functional analysis of P-glycoprotein mutants identifies predicted transmembrane domain 11 as a putative drug binding site.
    Biochemistry, 1993, Apr-27, Volume: 32, Issue:16

    Topics: Affinity Labels; Amino Acid Sequence; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Biological Transport; Cell Membrane; CHO Cells; Cloning, Molecular; Colchicine; Cricetinae; Dactinomycin; Doxorubicin; Drug Resistance; Gramicidin; Iodine Radioisotopes; Kinetics; Membrane Glycoproteins; Mice; Mutagenesis, Site-Directed; Phenylalanine; Prazosin; Serine; Transfection; Vinblastine

1993
Functional evidence that transmembrane 12 and the loop between transmembrane 11 and 12 form part of the drug-binding domain in P-glycoprotein encoded by MDR1.
    The Journal of biological chemistry, 1995, Mar-10, Volume: 270, Issue:10

    Topics: Affinity Labels; Amino Acid Sequence; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Cell Line; Cisplatin; Colchicine; Dactinomycin; Doxorubicin; Drug Resistance, Multiple; Humans; Iodine Radioisotopes; Melanoma; Molecular Sequence Data; Phenotype; Prazosin; Protein Structure, Secondary; Recombinant Fusion Proteins; Sequence Homology, Amino Acid; Transfection; Tumor Cells, Cultured; Vincristine

1995
High-level expression of mouse Mdr3 P-glycoprotein in yeast Pichia pastoris and characterization of ATPase activity.
    Methods in enzymology, 1998, Volume: 292

    Topics: Adenosine Triphosphatases; Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Azides; Binding, Competitive; Cell Fractionation; Cell Membrane; Cloning, Molecular; Colchicine; Doxorubicin; Drug Resistance, Multiple; Iodine Radioisotopes; Kinetics; Mice; Pichia; Plasmids; Prazosin; Recombinant Proteins; Time Factors; Transformation, Genetic; Valinomycin; Vinblastine

1998
Functional expression of human P-glycoprotein from plasmids using vaccinia virus-bacteriophage T7 RNA polymerase system.
    Methods in enzymology, 1998, Volume: 292

    Topics: Adenosine Triphosphatases; Affinity Labels; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Membrane; Cloning, Molecular; Colchicine; Daunorubicin; Dihydropyridines; DNA-Directed RNA Polymerases; Drug Resistance, Multiple; Electrophoresis, Polyacrylamide Gel; Escherichia coli; HeLa Cells; Humans; Indicators and Reagents; Iodine Radioisotopes; Osteosarcoma; Plasmids; Polymerase Chain Reaction; Prazosin; Recombinant Proteins; Restriction Mapping; Transfection; Tritium; Tumor Cells, Cultured; Vaccinia virus; Vinblastine; Viral Proteins

1998