cp 65,526 has been researched along with colchicine in 6 studies
Studies (cp 65,526) | Trials (cp 65,526) | Recent Studies (post-2010) (cp 65,526) | Studies (colchicine) | Trials (colchicine) | Recent Studies (post-2010) (colchicine) |
---|---|---|---|---|---|
65 | 1 | 5 | 15,472 | 404 | 2,974 |
Protein | Taxonomy | cp 65,526 (IC50) | colchicine (IC50) |
---|---|---|---|
Tubulin alpha-1A chain | Sus scrofa (pig) | 3.7639 | |
Tubulin beta chain | Sus scrofa (pig) | 3.8663 | |
Tubulin beta-4A chain | Homo sapiens (human) | 2.4334 | |
Tubulin beta chain | Homo sapiens (human) | 2.7244 | |
Tubulin alpha-3C chain | Homo sapiens (human) | 2.4334 | |
Serine/threonine-protein kinase pim-1 | Homo sapiens (human) | 4.3 | |
Tubulin alpha-1B chain | Homo sapiens (human) | 2.4334 | |
Tubulin alpha-4A chain | Homo sapiens (human) | 2.4334 | |
Tubulin beta-4B chain | Homo sapiens (human) | 2.4334 | |
Vesicular acetylcholine transporter | Tetronarce californica (Pacific electric ray) | 2.62 | |
Tubulin beta-3 chain | Homo sapiens (human) | 2.4334 | |
Tubulin beta-2A chain | Homo sapiens (human) | 2.4334 | |
Tubulin beta-8 chain | Homo sapiens (human) | 2.4334 | |
Tubulin beta-2B chain | Bos taurus (cattle) | 2.8255 | |
Tubulin alpha-3E chain | Homo sapiens (human) | 2.4334 | |
Tubulin alpha-1A chain | Homo sapiens (human) | 2.4334 | |
Similar to alpha-tubulin isoform 1 | Bos taurus (cattle) | 3.0611 | |
Similar to alpha-tubulin isoform 1 | Bos taurus (cattle) | 3.1553 | |
Tubulin alpha-1C chain | Homo sapiens (human) | 2.4334 | |
Tubulin beta-6 chain | Homo sapiens (human) | 2.4334 | |
Tubulin beta-2B chain | Homo sapiens (human) | 2.4334 | |
Tubulin beta-1 chain | Homo sapiens (human) | 2.4334 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 6 (100.00) | 18.2507 |
2000's | 0 (0.00) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Agresti, M; Mehta, ND; Safa, AR; Tamai, I; Vahabi, S | 1 |
Croop, JM; Kronauge, JF; Piwnica-Worms, D; Rao, VV | 1 |
Agresti, M; Grizzuti, K; Gros, P; Kajiji, S; Safa, AR; Talbot, F; Van Dyke-Phillips, V | 1 |
Collins, KI; Greenberger, LM; Zhang, X | 1 |
Beaudet, L; Gros, P; Urbatsch, IL | 1 |
Gottesman, MM; Hrycyna, CA; Pastan, I; Ramachandra, M | 1 |
6 other study(ies) available for cp 65,526 and colchicine
Article | Year |
---|---|
The alpha 1-adrenergic photoaffinity probe [125I]arylazidoprazosin binds to a specific peptide of P-glycoprotein in multidrug-resistant cells.
Topics: Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Line; Colchicine; Cricetinae; Cricetulus; Dactinomycin; Drug Resistance; Electrophoresis, Polyacrylamide Gel; Iodine Radioisotopes; Kinetics; Membrane Glycoproteins; Neoplasm Proteins; Peptide Mapping; Prazosin; Quinazolines; Vinca Alkaloids; Vincristine | 1990 |
Characterization of multidrug resistance P-glycoprotein transport function with an organotechnetium cation.
Topics: Adenosine Triphosphate; Allosteric Regulation; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Biological Transport; Cations; Cell Survival; Cells, Cultured; Colchicine; Cricetinae; Dose-Response Relationship, Drug; Doxorubicin; Humans; Kinetics; Lipid Bilayers; Pharmaceutical Preparations; Phloretin; Prazosin; Quinidine; Technetium Tc 99m Sestamibi; Tetraphenylborate | 1995 |
Functional analysis of P-glycoprotein mutants identifies predicted transmembrane domain 11 as a putative drug binding site.
Topics: Affinity Labels; Amino Acid Sequence; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Biological Transport; Cell Membrane; CHO Cells; Cloning, Molecular; Colchicine; Cricetinae; Dactinomycin; Doxorubicin; Drug Resistance; Gramicidin; Iodine Radioisotopes; Kinetics; Membrane Glycoproteins; Mice; Mutagenesis, Site-Directed; Phenylalanine; Prazosin; Serine; Transfection; Vinblastine | 1993 |
Functional evidence that transmembrane 12 and the loop between transmembrane 11 and 12 form part of the drug-binding domain in P-glycoprotein encoded by MDR1.
Topics: Affinity Labels; Amino Acid Sequence; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Binding Sites; Cell Line; Cisplatin; Colchicine; Dactinomycin; Doxorubicin; Drug Resistance, Multiple; Humans; Iodine Radioisotopes; Melanoma; Molecular Sequence Data; Phenotype; Prazosin; Protein Structure, Secondary; Recombinant Fusion Proteins; Sequence Homology, Amino Acid; Transfection; Tumor Cells, Cultured; Vincristine | 1995 |
High-level expression of mouse Mdr3 P-glycoprotein in yeast Pichia pastoris and characterization of ATPase activity.
Topics: Adenosine Triphosphatases; Affinity Labels; Animals; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; ATP-Binding Cassette Transporters; Azides; Binding, Competitive; Cell Fractionation; Cell Membrane; Cloning, Molecular; Colchicine; Doxorubicin; Drug Resistance, Multiple; Iodine Radioisotopes; Kinetics; Mice; Pichia; Plasmids; Prazosin; Recombinant Proteins; Time Factors; Transformation, Genetic; Valinomycin; Vinblastine | 1998 |
Functional expression of human P-glycoprotein from plasmids using vaccinia virus-bacteriophage T7 RNA polymerase system.
Topics: Adenosine Triphosphatases; Affinity Labels; ATP Binding Cassette Transporter, Subfamily B, Member 1; Azides; Cell Membrane; Cloning, Molecular; Colchicine; Daunorubicin; Dihydropyridines; DNA-Directed RNA Polymerases; Drug Resistance, Multiple; Electrophoresis, Polyacrylamide Gel; Escherichia coli; HeLa Cells; Humans; Indicators and Reagents; Iodine Radioisotopes; Osteosarcoma; Plasmids; Polymerase Chain Reaction; Prazosin; Recombinant Proteins; Restriction Mapping; Transfection; Tritium; Tumor Cells, Cultured; Vaccinia virus; Vinblastine; Viral Proteins | 1998 |