Page last updated: 2024-09-03

cp 122288 and metergoline

cp 122288 has been researched along with metergoline in 1 studies

Compound Research Comparison

Studies
(cp 122288)
Trials
(cp 122288)
Recent Studies (post-2010)
(cp 122288)
Studies
(metergoline)
Trials
(metergoline)
Recent Studies (post-2010) (metergoline)
17106563744

Protein Interaction Comparison

ProteinTaxonomycp 122288 (IC50)metergoline (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.0007
Bile salt export pumpHomo sapiens (human)10
Aldo-keto reductase family 1 member B1Rattus norvegicus (Norway rat)0.366
5-hydroxytryptamine receptor 1AHomo sapiens (human)0.0041
Alpha-2A adrenergic receptorHomo sapiens (human)0.058
Cytochrome P450 2D6Homo sapiens (human)0.2
D(2) dopamine receptorHomo sapiens (human)0.063
Alpha-2B adrenergic receptorHomo sapiens (human)0.016
Alpha-2C adrenergic receptorHomo sapiens (human)0.189
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0062
Substance-K receptorHomo sapiens (human)4.071
D(1A) dopamine receptorHomo sapiens (human)0.074
AcetylcholinesteraseHomo sapiens (human)1.344
Sodium-dependent noradrenaline transporter Homo sapiens (human)0.366
Histamine H2 receptorHomo sapiens (human)0.975
Alpha-1D adrenergic receptorHomo sapiens (human)0.136
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.0004
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.0007
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.0062
Sodium-dependent serotonin transporterHomo sapiens (human)0.59
Histamine H1 receptorHomo sapiens (human)4.133
D(3) dopamine receptorHomo sapiens (human)0.0077
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0004
5-hydroxytryptamine receptor 6Homo sapiens (human)0.028
Sodium-dependent dopamine transporter Homo sapiens (human)0.063

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beleta, J; Doménech, T; Palacios, JM1

Other Studies

1 other study(ies) available for cp 122288 and metergoline

ArticleYear
Characterization of human serotonin 1D and 1B receptors using [3H]-GR-125743, a novel radiolabelled serotonin 5HT1D/1B receptor antagonist.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:3

    Topics: Benzamides; Binding, Competitive; Gene Expression; HeLa Cells; Humans; Kinetics; Ligands; Pyridines; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Substantia Nigra; Tritium

1997