Page last updated: 2024-09-03

cp 122288 and gr 127935

cp 122288 has been researched along with gr 127935 in 1 studies

Compound Research Comparison

Studies
(cp 122288)
Trials
(cp 122288)
Recent Studies (post-2010)
(cp 122288)
Studies
(gr 127935)
Trials
(gr 127935)
Recent Studies (post-2010) (gr 127935)
1710221028

Protein Interaction Comparison

ProteinTaxonomycp 122288 (IC50)gr 127935 (IC50)
5-hydroxytryptamine receptor 1DHomo sapiens (human)0.052
Sodium-dependent serotonin transporterHomo sapiens (human)1

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cutrer, FM; Moskowitz, MA; Waeber, C; Yu, XJ1

Other Studies

1 other study(ies) available for cp 122288 and gr 127935

ArticleYear
The 5-HT1D receptor antagonist GR-127,935 prevents inhibitory effects of sumatriptan but not CP-122,288 and 5-CT on neurogenic plasma extravasation within guinea pig dura mater.
    Neuropharmacology, 1997, Volume: 36, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Dura Mater; Electric Stimulation; Female; Guinea Pigs; Male; Oxadiazoles; Pertussis Toxin; Piperazines; Prosencephalon; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sumatriptan; Trigeminal Nerve; Virulence Factors, Bordetella

1997