Page last updated: 2024-09-03

cp 122288 and dihydroergotamine

cp 122288 has been researched along with dihydroergotamine in 2 studies

Compound Research Comparison

Studies
(cp 122288)
Trials
(cp 122288)
Recent Studies (post-2010)
(cp 122288)
Studies
(dihydroergotamine)
Trials
(dihydroergotamine)
Recent Studies (post-2010) (dihydroergotamine)
17101,450241116

Protein Interaction Comparison

ProteinTaxonomycp 122288 (IC50)dihydroergotamine (IC50)
5-hydroxytryptamine receptor 4Cavia porcellus (domestic guinea pig)0.09
Cytochrome P450 3A4Homo sapiens (human)3.9996
Alpha-2A adrenergic receptorHomo sapiens (human)0.001
D(2) dopamine receptorHomo sapiens (human)0.0089
Alpha-2B adrenergic receptorHomo sapiens (human)0.0039
Alpha-2C adrenergic receptorHomo sapiens (human)0.01
5-hydroxytryptamine receptor 1ARattus norvegicus (Norway rat)0.0007
D(1A) dopamine receptorHomo sapiens (human)2.395
Alpha-1D adrenergic receptorHomo sapiens (human)0.029
5-hydroxytryptamine receptor 2AHomo sapiens (human)0.008
5-hydroxytryptamine receptor 2CHomo sapiens (human)0.09
5-hydroxytryptamine receptor 1BRattus norvegicus (Norway rat)0.0007
D(3) dopamine receptorHomo sapiens (human)0.0053
5-hydroxytryptamine receptor 2BHomo sapiens (human)0.0068
5-hydroxytryptamine receptor 6Homo sapiens (human)0.0032
Multidrug and toxin extrusion protein 1Homo sapiens (human)2.8

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (50.00)18.2507
2000's1 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Castanon, N; Chauveau, J; Chaveau, J; Hen, R; Macor, JE; Moskowitz, MA; Scearce, K; Waeber, C; Yu, XJ1
Hargreaves, RJ; Williamson, DJ1

Reviews

1 review(s) available for cp 122288 and dihydroergotamine

ArticleYear
Neurogenic inflammation in the context of migraine.
    Microscopy research and technique, 2001, May-01, Volume: 53, Issue:3

    Topics: Animals; Blood Proteins; Bosentan; Calcitonin Gene-Related Peptide; Capillary Permeability; Dihydroergotamine; Dura Mater; Humans; Migraine Disorders; Narcotics; Neurogenic Inflammation; Neurokinin-1 Receptor Antagonists; Pyrrolidines; Receptor, Serotonin, 5-HT1D; Receptor, Serotonin, 5-HT1F; Receptors, Neurokinin-1; Receptors, Serotonin; Serotonin Receptor Agonists; Skull; Sulfonamides; Sumatriptan; Trigeminal Nerve; Vasoconstrictor Agents; Vasodilation

2001

Other Studies

1 other study(ies) available for cp 122288 and dihydroergotamine

ArticleYear
5-Carboxamido-tryptamine, CP-122,288 and dihydroergotamine but not sumatriptan, CP-93,129, and serotonin-5-O-carboxymethyl-glycyl -tyrosinamide block dural plasma protein extravasation in knockout mice that lack 5-hydroxytryptamine1B receptors.
    Molecular pharmacology, 1996, Volume: 49, Issue:5

    Topics: Animals; Capillary Permeability; Dihydroergotamine; Dipeptides; Mice; Mice, Knockout; Pyridines; Pyrroles; Pyrrolidines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Sumatriptan; Trigeminal Ganglion

1996