Page last updated: 2024-09-03

cp 122288 and 5-carboxamidotryptamine

cp 122288 has been researched along with 5-carboxamidotryptamine in 2 studies

Compound Research Comparison

Studies
(cp 122288)
Trials
(cp 122288)
Recent Studies (post-2010)
(cp 122288)
Studies
(5-carboxamidotryptamine)
Trials
(5-carboxamidotryptamine)
Recent Studies (post-2010) (5-carboxamidotryptamine)
1710392136

Protein Interaction Comparison

ProteinTaxonomycp 122288 (IC50)5-carboxamidotryptamine (IC50)
5-hydroxytryptamine receptor 1DSus scrofa (pig)0.004

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Castanon, N; Chauveau, J; Chaveau, J; Hen, R; Macor, JE; Moskowitz, MA; Scearce, K; Waeber, C; Yu, XJ1
Cutrer, FM; Moskowitz, MA; Waeber, C; Yu, XJ1

Other Studies

2 other study(ies) available for cp 122288 and 5-carboxamidotryptamine

ArticleYear
5-Carboxamido-tryptamine, CP-122,288 and dihydroergotamine but not sumatriptan, CP-93,129, and serotonin-5-O-carboxymethyl-glycyl -tyrosinamide block dural plasma protein extravasation in knockout mice that lack 5-hydroxytryptamine1B receptors.
    Molecular pharmacology, 1996, Volume: 49, Issue:5

    Topics: Animals; Capillary Permeability; Dihydroergotamine; Dipeptides; Mice; Mice, Knockout; Pyridines; Pyrroles; Pyrrolidines; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Sumatriptan; Trigeminal Ganglion

1996
The 5-HT1D receptor antagonist GR-127,935 prevents inhibitory effects of sumatriptan but not CP-122,288 and 5-CT on neurogenic plasma extravasation within guinea pig dura mater.
    Neuropharmacology, 1997, Volume: 36, Issue:1

    Topics: Animals; Dose-Response Relationship, Drug; Dura Mater; Electric Stimulation; Female; Guinea Pigs; Male; Oxadiazoles; Pertussis Toxin; Piperazines; Prosencephalon; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1D; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Sumatriptan; Trigeminal Nerve; Virulence Factors, Bordetella

1997