Page last updated: 2024-09-05

cp 100356 and tacrolimus

cp 100356 has been researched along with tacrolimus in 1 studies

Compound Research Comparison

Studies
(cp 100356)
Trials
(cp 100356)
Recent Studies (post-2010)
(cp 100356)
Studies
(tacrolimus)
Trials
(tacrolimus)
Recent Studies (post-2010) (tacrolimus)
80317,7572,3196,661

Protein Interaction Comparison

ProteinTaxonomycp 100356 (IC50)tacrolimus (IC50)
Bile salt export pumpHomo sapiens (human)7.18
Cytochrome P450 3A4Homo sapiens (human)0.58
Cytochrome P450 3A5Homo sapiens (human)0.385
Serine/threonine-protein kinase mTORHomo sapiens (human)0.0021
Peptidyl-prolyl cis-trans isomerase FKBP1AHomo sapiens (human)0.2547
Serine/threonine-protein phosphatase 2B catalytic subunit alpha isoformHomo sapiens (human)0.0148
Splicing factor 3B subunit 3Homo sapiens (human)0.0123
Broad substrate specificity ATP-binding cassette transporter ABCG2Homo sapiens (human)3.3
Solute carrier organic anion transporter family member 1B1Homo sapiens (human)3.7

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Guengerich, P; Kajiji, S; Kim, RB; Wandel, C; Wilkinson, GR; Wood, AJ1

Other Studies

1 other study(ies) available for cp 100356 and tacrolimus

ArticleYear
P-glycoprotein and cytochrome P-450 3A inhibition: dissociation of inhibitory potencies.
    Cancer research, 1999, Aug-15, Volume: 59, Issue:16

    Topics: Aryl Hydrocarbon Hydroxylases; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Caco-2 Cells; Cytochrome P-450 CYP3A; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Digoxin; Down-Regulation; Enzyme Inhibitors; Humans; Oxidoreductases, N-Demethylating; Substrate Specificity

1999