Page last updated: 2024-09-05

cp 100356 and quinidine

cp 100356 has been researched along with quinidine in 2 studies

Compound Research Comparison

Studies
(cp 100356)
Trials
(cp 100356)
Recent Studies (post-2010)
(cp 100356)
Studies
(quinidine)
Trials
(quinidine)
Recent Studies (post-2010) (quinidine)
8036,608387594

Protein Interaction Comparison

ProteinTaxonomycp 100356 (IC50)quinidine (IC50)
Voltage-dependent L-type calcium channel subunit alpha-1FHomo sapiens (human)6.4
CholinesteraseHomo sapiens (human)1.23
ATP-dependent translocase ABCB1Mus musculus (house mouse)10
ATP-dependent translocase ABCB1Homo sapiens (human)3.32
Cytochrome P450 2D26Rattus norvegicus (Norway rat)2.8
Cytochrome P450 2D6Homo sapiens (human)0.3532
Potassium voltage-gated channel subfamily A member 5Homo sapiens (human)7.3
CholinesteraseEquus caballus (horse)7.37
Voltage-dependent L-type calcium channel subunit alpha-1D Homo sapiens (human)6.4
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)0.7882
Voltage-dependent L-type calcium channel subunit alpha-1SHomo sapiens (human)6.4
Voltage-dependent L-type calcium channel subunit alpha-1CHomo sapiens (human)6.4
Sodium channel protein type 5 subunit alphaHomo sapiens (human)6.9
Potassium voltage-gated channel subfamily D member 2Rattus norvegicus (Norway rat)2.2

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
de Graaf, IA; de Jager, MH; Groothuis, GM; Li, M1
de Graaf, IA; de Jager, MH; Groothuis, GM; Li, M; van de Steeg, E1

Other Studies

2 other study(ies) available for cp 100356 and quinidine

ArticleYear
Rat precision-cut intestinal slices to study P-gp activity and the potency of its inhibitors ex vivo.
    Toxicology in vitro : an international journal published in association with BIBRA, 2015, Volume: 29, Issue:5

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cyclosporine; Cyclosporins; In Vitro Techniques; Intestinal Mucosa; Isoquinolines; Ketoconazole; Male; Quinazolines; Quinidine; Rats, Wistar; Rhodamine 123; Verapamil

2015
The consequence of regional gradients of P-gp and CYP3A4 for drug-drug interactions by P-gp inhibitors and the P-gp/CYP3A4 interplay in the human intestine ex vivo.
    Toxicology in vitro : an international journal published in association with BIBRA, 2017, Volume: 40

    Topics: Adult; Aged; Aged, 80 and over; ATP Binding Cassette Transporter, Subfamily B, Member 1; Colon; Cyclosporins; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Female; Humans; Ileum; In Vitro Techniques; Isoquinolines; Jejunum; Ketoconazole; Male; Middle Aged; Quinazolines; Quinidine; Verapamil

2017