coumarin and thiazoles

coumarin has been researched along with thiazoles in 22 studies

Research

Studies (22)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (9.09)18.2507
2000's3 (13.64)29.6817
2010's12 (54.55)24.3611
2020's5 (22.73)2.80

Authors

AuthorsStudies
Beamand, JA; Lake, BG; Mistry, H; Price, RJ; Renwick, AB; Wield, PT1
Funae, Y; Funayama, M; Green, C; Inoue, K; Kamataki, T; Kimura, K; Kinoshita, M; Kodama, T; Nagashima, K; Nunoya, K; Yokoi, T1
Deligeorgiev, TG; Katerinopoulos, HE; Liepouri, F; Savakis, C; Veneti, Z1
Hadjipavlou-Litina, D; Kontogiorgis, CA; Luo, Y; Xu, Y1
Baudoin, C; Féron, C; Koyama, S; Novotny, MV; Soini, HA; Wiesler, D1
Fleita, DH; Mohareb, RM; Sakka, OK1
Arshad, A; Bagley, MC; Lam, CK; Mohamad, S; Osman, H; Zahariluddin, AS1
Ballazhi, L; Dräger, G; Huwiler, A; Imeri, F; Jashari, A; Mikhova, B; Popovski, E; Shabani, A1
Duan, YW; En, D; Guo, Y; Li, CW; Li, J; Peng, MJ; Suzenet, F; Yang, XF; Yin, B1
Das, S; Dhar, SK; Govindaraju, T; Kumar, M; Kundu, TK; Narayanaswamy, N; Pati, SK; Samanta, PK; Sharma, R1
MegallyAbdo, NY; Mohareb, RM1
He, D; Li, J; Li, X; Peng, Z; Wang, G1
Gul, S; Imran, S; Ismail, NH; Khan, KM; Perveen, S; Salar, U; Taha, M; Wadood, A1
Bajorath, J; Furtmann, N; Hameed, A; Ibrar, A; Iqbal, J; Khan, I; Saeed, A; Tehseen, Y1
Abbas, Q; Channar, PA; Hassan, M; Larik, FA; Mahesar, PA; Raza, H; Saeed, A; Seo, SY1
Abd El-Karim, SS; Abdelghany, TM; El Kerdawy, AM; Syam, YM1
Alvala, M; Alvala, R; Ghouse, MS; Goud, NS; Pranay, J; Qureshi, IA; Talla, V; Vishnu, J1
Ahsan Halim, S; Al-Harrasi, A; Csuk, R; Ibrar, A; Khan, A; Khan, I; Mehsud, S; Saeed, A1
Ahmad, Z; Al-Qawasmeh, RA; Al-Tel, TH; Hersi, F; Jaber, AM; Omar, HA; Zaher, DM1
Ansari, MF; Cheng, Y; Hu, C; Hu, Y; Pan, G; Yadav Bheemanaboina, RR; Yu, C; Zhang, J; Zhou, C1
Ciszkowicz, E; Creaven, B; Jenkins, H; Kamiński, D; Karcz, D; Lecka-Szlachta, K; Matwijczuk, A; Miłoś, A; Radomski, P; Ślusarczyk, L; Starzak, K1
Abdel-Aziem, A; Elsharabasy, SA; Sayed, MT1

Other Studies

22 other study(ies) available for coumarin and thiazoles

ArticleYear
Comparison of the toxicity of allyl alcohol, coumarin and menadione in precision-cut rat, guinea-pig, cynomolgus monkey and human liver slices.
    Archives of toxicology, 1996, Volume: 71, Issue:1-2

    Topics: 1-Propanol; Animals; Coloring Agents; Coumarins; Guinea Pigs; Humans; Liver; Macaca fascicularis; Male; Potassium; Propanols; Protein Biosynthesis; Rats; Tetrazolium Salts; Thiazoles; Toxicity Tests; Vitamin K

1996
A new deleted allele in the human cytochrome P450 2A6 (CYP2A6) gene found in individuals showing poor metabolic capacity to coumarin and (+)-cis-3,5-dimethyl-2-(3-pyridyl)thiazolidin-4-one hydrochloride (SM-12502).
    Pharmacogenetics, 1998, Volume: 8, Issue:3

    Topics: Aryl Hydrocarbon Hydroxylases; Base Sequence; Cloning, Molecular; Coumarins; Cytochrome P-450 CYP2A6; Cytochrome P-450 Enzyme System; Gene Deletion; Genomic Library; Humans; Hydroxylation; Microsomes, Liver; Mixed Function Oxygenases; Molecular Sequence Data; Polymerase Chain Reaction; Polymorphism, Genetic; Polymorphism, Restriction Fragment Length; Sequence Analysis, DNA; Substrate Specificity; Thiazoles; Thiazolidines

1998
Near-membrane iminocoumarin-based low affinity fluorescent Ca(2+) indicators.
    Cell calcium, 2002, Volume: 31, Issue:5

    Topics: Animals; Benzimidazoles; Benzopyrans; Binding Sites; Calcium; Cell Membrane; Coumarins; Drosophila melanogaster; Embryo, Nonmammalian; Fluorescent Dyes; Indicators and Reagents; Magnetic Resonance Spectroscopy; Mass Spectrometry; Membrane Lipids; Microscopy, Fluorescence; Spectrum Analysis; Thiazoles

2002
Coumarin derivatives protection against ROS production in cellular models of Abeta toxicities.
    Free radical research, 2007, Volume: 41, Issue:10

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Animals; Cell Line, Tumor; Coumarins; Free Radicals; Humans; Hydrogen Peroxide; Mice; Mice, Transgenic; Models, Chemical; Mutation; Oxidative Stress; Reactive Oxygen Species; Tetrazolium Salts; Thiazoles

2007
Comparison of urinary scents of two related mouse species, Mus spicilegus and Mus domesticus.
    Journal of chemical ecology, 2009, Volume: 35, Issue:5

    Topics: Animals; Coumarins; Gas Chromatography-Mass Spectrometry; Lactones; Male; Mice; Pheromones; Smell; Species Specificity; Thiazoles

2009
Novel synthesis of hydrazide-hydrazone derivatives and their utilization in the synthesis of coumarin, pyridine, thiazole and thiophene derivatives with antitumor activity.
    Molecules (Basel, Switzerland), 2010, Dec-23, Volume: 16, Issue:1

    Topics: Antineoplastic Agents; Azides; Cell Division; Cell Line, Tumor; Coumarins; Drug Screening Assays, Antitumor; Humans; Hydrazones; Magnetic Resonance Spectroscopy; Pyridines; Thiazoles; Thiophenes

2010
Synthesis and antimicrobial properties of some new thiazolyl coumarin derivatives.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:9

    Topics: Anti-Infective Agents; Candida albicans; Coumarins; Crystallography, X-Ray; Gram-Negative Bacteria; Gram-Positive Bacteria; Magnetic Resonance Spectroscopy; Microbial Sensitivity Tests; Models, Molecular; Mycobacterium tuberculosis; Spectrophotometry, Infrared; Thiazoles

2011
Synthesis and cellular characterization of novel isoxazolo- and thiazolohydrazinylidene-chroman-2,4-diones on cancer and non-cancer cell growth and death.
    Bioorganic & medicinal chemistry, 2014, May-01, Volume: 22, Issue:9

    Topics: 4-Hydroxycoumarins; Antineoplastic Agents; Apoptosis; Cell Line; Cell Proliferation; Coumarins; Humans; Isoxazoles; MCF-7 Cells; Poly(ADP-ribose) Polymerases; Thiazoles; U937 Cells

2014
A hybrid coumarin-thiazole fluorescent sensor for selective detection of bisulfite anions in vivo and in real samples.
    Chemistry, an Asian journal, 2014, Volume: 9, Issue:7

    Topics: Anions; Biosensing Techniques; Color; Coumarins; Female; Fluorescent Dyes; Humans; MCF-7 Cells; Molecular Structure; Sensitivity and Specificity; Sulfites; Thiazoles

2014
A thiazole coumarin (TC) turn-on fluorescence probe for AT-base pair detection and multipurpose applications in different biological systems.
    Scientific reports, 2014, Sep-25, Volume: 4

    Topics: Base Pairing; Carbocyanines; Cell Cycle; Coumarins; DNA; Flow Cytometry; Fluorescence; Fluorescent Dyes; HEK293 Cells; HeLa Cells; Humans; Molecular Imaging; Thiazoles

2014
Uses of 3-(2-Bromoacetyl)-2H-chromen-2-one in the Synthesis of Heterocyclic Compounds Incorporating Coumarin: Synthesis, Characterization and Cytotoxicity.
    Molecules (Basel, Switzerland), 2015, Jun-23, Volume: 20, Issue:6

    Topics: Antineoplastic Agents; Cell Line, Tumor; Cell Proliferation; Coumarins; Drug Screening Assays, Antitumor; Humans; Neoplasms; Pyrans; Structure-Activity Relationship; Thiazoles

2015
Design, synthesis and biological evaluation of novel coumarin thiazole derivatives as α-glucosidase inhibitors.
    Bioorganic chemistry, 2016, Volume: 65

    Topics: alpha-Glucosidases; Coumarins; Dose-Response Relationship, Drug; Drug Design; Glycoside Hydrolase Inhibitors; Molecular Docking Simulation; Molecular Structure; Saccharomyces cerevisiae; Structure-Activity Relationship; Thiazoles

2016
Syntheses of new 3-thiazolyl coumarin derivatives, in vitro α-glucosidase inhibitory activity, and molecular modeling studies.
    European journal of medicinal chemistry, 2016, Oct-21, Volume: 122

    Topics: alpha-Glucosidases; Chemistry Techniques, Synthetic; Coumarins; Glycoside Hydrolase Inhibitors; Molecular Docking Simulation; Protein Conformation; Thiazoles

2016
Coumarin-thiazole and -oxadiazole derivatives: Synthesis, bioactivity and docking studies for aldose/aldehyde reductase inhibitors.
    Bioorganic chemistry, 2016, Volume: 68

    Topics: Aldehyde Reductase; Animals; Cattle; Coumarins; Dose-Response Relationship, Drug; Enzyme Inhibitors; Molecular Docking Simulation; Molecular Structure; Oxadiazoles; Structure-Activity Relationship; Thiazoles

2016
Synthesis, molecular docking studies of coumarinyl-pyrazolinyl substituted thiazoles as non-competitive inhibitors of mushroom tyrosinase.
    Bioorganic chemistry, 2017, Volume: 74

    Topics: Agaricales; Coumarins; Dose-Response Relationship, Drug; Enzyme Inhibitors; Molecular Docking Simulation; Molecular Structure; Monophenol Monooxygenase; Pyrazoles; Structure-Activity Relationship; Thiazoles

2017
New thiazol-hydrazono-coumarin hybrids targeting human cervical cancer cells: Synthesis, CDK2 inhibition, QSAR and molecular docking studies.
    Bioorganic chemistry, 2019, Volume: 86

    Topics: Antineoplastic Agents; Apoptosis; Cell Cycle; Cell Proliferation; Coumarins; Cyclin-Dependent Kinase 2; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; HeLa Cells; Humans; Hydrazones; Molecular Docking Simulation; Molecular Structure; Protein Kinase Inhibitors; Quantitative Structure-Activity Relationship; Thiazoles; Tumor Cells, Cultured

2019
Synthesis and Biological Evaluation of Novel Heterocyclic Imines Linked Coumarin- Thiazole Hybrids as Anticancer Agents.
    Anti-cancer agents in medicinal chemistry, 2019, Volume: 19, Issue:4

    Topics: Antineoplastic Agents; Cell Line, Tumor; Coumarins; Drug Screening Assays, Antitumor; Heterocyclic Compounds; Humans; Imines; Membrane Potential, Mitochondrial; Molecular Docking Simulation; Thiazoles

2019
Exploring biological efficacy of coumarin clubbed thiazolo[3,2-b][1,2,4]triazoles as efficient inhibitors of urease: A biochemical and in silico approach.
    International journal of biological macromolecules, 2020, Jan-01, Volume: 142

    Topics: Binding Sites; Catalytic Domain; Coumarins; Enzyme Inhibitors; Models, Molecular; Molecular Structure; Protein Binding; Structure-Activity Relationship; Thiazoles; Triazoles; Urease

2020
Design and synthesis of new energy restriction mimetic agents: Potent anti-tumor activities of hybrid motifs of aminothiazoles and coumarins.
    Scientific reports, 2020, 02-19, Volume: 10, Issue:1

    Topics: Antineoplastic Agents; Cell Cycle Checkpoints; Cell Proliferation; Cisplatin; Colorectal Neoplasms; Coumarins; Drug Design; Drug Screening Assays, Antitumor; Energy Metabolism; G1 Phase; Glucose; HCT116 Cells; HT29 Cells; Humans; Inhibitory Concentration 50; Reactive Oxygen Species; Thiazoles

2020
Novel chalcone-conjugated, multi-flexible end-group coumarin thiazole hybrids as potential antibacterial repressors against methicillin-resistant Staphylococcus aureus.
    European journal of medicinal chemistry, 2021, Oct-15, Volume: 222

    Topics: Animals; Anti-Bacterial Agents; Cell Line; Chalcones; Coumarins; Dose-Response Relationship, Drug; Humans; Methicillin-Resistant Staphylococcus aureus; Mice; Microbial Sensitivity Tests; Molecular Docking Simulation; Molecular Structure; Structure-Activity Relationship; Thiazoles

2021
Novel Coumarin-Thiadiazole Hybrids and Their Cu(II) and Zn(II) Complexes as Potential Antimicrobial Agents and Acetylcholinesterase Inhibitors.
    International journal of molecular sciences, 2021, Sep-08, Volume: 22, Issue:18

    Topics: Acetylcholinesterase; Anti-Bacterial Agents; Anti-Infective Agents; Cholinesterase Inhibitors; Copper; Coumarins; Crystallography, X-Ray; Escherichia coli; Ligands; Magnetic Resonance Spectroscopy; Metals; Microbial Sensitivity Tests; Neurodegenerative Diseases; Pseudomonas aeruginosa; Schiff Bases; Spectrometry, Fluorescence; Spectrophotometry, Atomic; Staphylococcus aureus; Staphylococcus epidermidis; Thiadiazoles; Thiazoles; Zinc

2021
Synthesis and antimicrobial activity of new series of thiazoles, pyridines and pyrazoles based on coumarin moiety.
    Scientific reports, 2023, 06-19, Volume: 13, Issue:1

    Topics: Anti-Bacterial Agents; Anti-Infective Agents; Coumarins; Microbial Sensitivity Tests; Molecular Structure; Pyrazoles; Pyridines; Thiazoles

2023