conivaptan has been researched along with suramin in 2 studies
Studies (conivaptan) | Trials (conivaptan) | Recent Studies (post-2010) (conivaptan) | Studies (suramin) | Trials (suramin) | Recent Studies (post-2010) (suramin) |
---|---|---|---|---|---|
188 | 17 | 64 | 3,023 | 92 | 431 |
Protein | Taxonomy | conivaptan (IC50) | suramin (IC50) |
---|---|---|---|
ATP-dependent 6-phosphofructokinase | Trypanosoma brucei brucei | 3 | |
Tyrosine-protein phosphatase non-receptor type 1 | Homo sapiens (human) | 9.76 | |
P2X purinoceptor 2 | Rattus norvegicus (Norway rat) | 4 | |
DNA-dependent protein kinase catalytic subunit | Homo sapiens (human) | 1.7 | |
DNA primase | Mycobacterium tuberculosis CDC1551 | 8.2 | |
RmtA | Aspergillus nidulans | 5.9 | |
Reverse transcriptase/RNaseH | Human immunodeficiency virus 1 | 9.4 | |
NAD-dependent protein deacetylase sirtuin-2 | Homo sapiens (human) | 1.15 | |
NAD-dependent protein deacetylase sirtuin-1 | Homo sapiens (human) | 1.5667 | |
Protein arginine N-methyltransferase 1 | Homo sapiens (human) | 5.33 | |
NAD-dependent protein deacylase sirtuin-5, mitochondrial | Homo sapiens (human) | 2.5 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 1 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Lombardo, F; Obach, RS; Waters, NJ | 1 |
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV | 1 |
2 other study(ies) available for conivaptan and suramin
Article | Year |
---|---|
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding | 2008 |
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations | 2010 |