Page last updated: 2024-09-04

conivaptan and sitagliptin

conivaptan has been researched along with sitagliptin in 3 studies

Compound Research Comparison

Studies
(conivaptan)
Trials
(conivaptan)
Recent Studies (post-2010)
(conivaptan)
Studies
(sitagliptin)
Trials
(sitagliptin)
Recent Studies (post-2010) (sitagliptin)
188176497070

Protein Interaction Comparison

ProteinTaxonomyconivaptan (IC50)sitagliptin (IC50)
Chain A, Dipeptidyl peptidase IVHomo sapiens (human)0.018
Dipeptidyl peptidase 4Rattus norvegicus (Norway rat)0.0255
Thromboxane-A synthase Homo sapiens (human)0.0194
Dipeptidyl peptidase 4Homo sapiens (human)0.0236
Dipeptidyl peptidase 4Mus musculus (house mouse)0.046
Prolyl endopeptidase FAPHomo sapiens (human)2.93
Dipeptidyl peptidase 8Homo sapiens (human)0.4715
Dipeptidyl peptidase 9Homo sapiens (human)1.539
Dipeptidyl peptidase 2Homo sapiens (human)0.022

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Lombardo, F; Obach, RS; Waters, NJ1
Chang, G; El-Kattan, A; Miller, HR; Obach, RS; Rotter, C; Steyn, SJ; Troutman, MD; Varma, MV1
Chen, M; Hu, C; Suzuki, A; Thakkar, S; Tong, W; Yu, K1

Reviews

1 review(s) available for conivaptan and sitagliptin

ArticleYear
DILIrank: the largest reference drug list ranked by the risk for developing drug-induced liver injury in humans.
    Drug discovery today, 2016, Volume: 21, Issue:4

    Topics: Chemical and Drug Induced Liver Injury; Databases, Factual; Drug Labeling; Humans; Pharmaceutical Preparations; Risk

2016

Other Studies

2 other study(ies) available for conivaptan and sitagliptin

ArticleYear
Trend analysis of a database of intravenous pharmacokinetic parameters in humans for 670 drug compounds.
    Drug metabolism and disposition: the biological fate of chemicals, 2008, Volume: 36, Issue:7

    Topics: Blood Proteins; Half-Life; Humans; Hydrogen Bonding; Infusions, Intravenous; Pharmacokinetics; Protein Binding

2008
Physicochemical space for optimum oral bioavailability: contribution of human intestinal absorption and first-pass elimination.
    Journal of medicinal chemistry, 2010, Feb-11, Volume: 53, Issue:3

    Topics: Administration, Oral; Biological Availability; Humans; Intestinal Absorption; Pharmaceutical Preparations

2010