conessine has been researched along with pitolisant in 2 studies
Studies (conessine) | Trials (conessine) | Recent Studies (post-2010) (conessine) | Studies (pitolisant) | Trials (pitolisant) | Recent Studies (post-2010) (pitolisant) |
---|---|---|---|---|---|
80 | 0 | 28 | 97 | 14 | 77 |
Protein | Taxonomy | conessine (IC50) | pitolisant (IC50) |
---|---|---|---|
Cholinesterase | Equus caballus (horse) | 8.41 | |
Potassium voltage-gated channel subfamily H member 2 | Homo sapiens (human) | 1.7 | |
Histamine H3 receptor | Homo sapiens (human) | 0.012 |
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (50.00) | 29.6817 |
2010's | 1 (50.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Kieć-Kononowicz, K; Kuder, K; Ligneau, X; Schunack, W; Schwartz, JC; Stark, H; Łazewska, D | 1 |
Chazot, PL; Cowart, M; Gutzmer, R; Haas, HL; Leurs, R; Liu, WL; Panula, P; Stark, H; Thurmond, RL | 1 |
1 review(s) available for conessine and pitolisant
Article | Year |
---|---|
International Union of Basic and Clinical Pharmacology. XCVIII. Histamine Receptors.
Topics: Animals; Drug Design; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Ligands; Receptors, Histamine | 2015 |
1 other study(ies) available for conessine and pitolisant
Article | Year |
---|---|
Piperidine variations in search for non-imidazole histamine H(3) receptor ligands.
Topics: Animals; Binding Sites; CHO Cells; Cricetinae; Cricetulus; Humans; Imidazoles; Ligands; Piperidines; Radioligand Assay; Receptors, Histamine H3; Structure-Activity Relationship | 2008 |