Page last updated: 2024-09-02

conessine and pitolisant

conessine has been researched along with pitolisant in 2 studies

Compound Research Comparison

Studies
(conessine)
Trials
(conessine)
Recent Studies (post-2010)
(conessine)
Studies
(pitolisant)
Trials
(pitolisant)
Recent Studies (post-2010) (pitolisant)
80028971477

Protein Interaction Comparison

ProteinTaxonomyconessine (IC50)pitolisant (IC50)
CholinesteraseEquus caballus (horse)8.41
Potassium voltage-gated channel subfamily H member 2Homo sapiens (human)1.7
Histamine H3 receptorHomo sapiens (human)0.012

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kieć-Kononowicz, K; Kuder, K; Ligneau, X; Schunack, W; Schwartz, JC; Stark, H; Łazewska, D1
Chazot, PL; Cowart, M; Gutzmer, R; Haas, HL; Leurs, R; Liu, WL; Panula, P; Stark, H; Thurmond, RL1

Reviews

1 review(s) available for conessine and pitolisant

ArticleYear
International Union of Basic and Clinical Pharmacology. XCVIII. Histamine Receptors.
    Pharmacological reviews, 2015, Volume: 67, Issue:3

    Topics: Animals; Drug Design; Histamine; Histamine Agonists; Histamine Antagonists; Humans; Ligands; Receptors, Histamine

2015

Other Studies

1 other study(ies) available for conessine and pitolisant

ArticleYear
Piperidine variations in search for non-imidazole histamine H(3) receptor ligands.
    Bioorganic & medicinal chemistry, 2008, Sep-15, Volume: 16, Issue:18

    Topics: Animals; Binding Sites; CHO Cells; Cricetinae; Cricetulus; Humans; Imidazoles; Ligands; Piperidines; Radioligand Assay; Receptors, Histamine H3; Structure-Activity Relationship

2008