combretastatin has been researched along with colchicine in 20 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (10.00) | 18.7374 |
1990's | 3 (15.00) | 18.2507 |
2000's | 8 (40.00) | 29.6817 |
2010's | 6 (30.00) | 24.3611 |
2020's | 1 (5.00) | 2.80 |
Authors | Studies |
---|---|
Chu, PS; Getahun, Z; Hamel, E; Jurd, L; Lin, CM | 1 |
Chu, PS; Dempcy, RO; Hamel, E; Lin, CM; Pettit, GR; Schmidt, JM; Singh, SB | 1 |
Hamel, E; Lin, CM | 1 |
Kajiyama, S; Kobayashi, A | 1 |
Day, BW; Hamel, E; Rosenkranz, HS; ter Haar, E | 1 |
Brown, ML; Macdonald, TL; Rieger, JM | 1 |
Kovar, P; Ng, SC; Rosenberg, SH; Tahir, SK | 1 |
Chaudhuri, AR; Hausheer, FH; Ludueña, RF; Schwarz, PM; Seetharamalu, P | 1 |
Iwasaki, S; Shirai, R | 1 |
Bane, SL; Janik, ME | 1 |
Ducki, S; Lawrence, NJ; Mackenzie, G; Snyder, JP | 1 |
Alloatti, D; Baruchello, R; Bucci, F; Carminati, P; Castorina, M; Giannini, G; Guglielmi, MB; Marcellini, M; Pavani, MG; Pisano, C; Riccioni, T; Rizzi, M; Romagnoli, R; Rondanin, R; Simoni, D | 1 |
Armitage, S; Bennett, E; Chabert, JF; Ducki, S; Greedy, B; Lawrence, NJ; Mackenzie, G; Nettles, J; Snyder, JP | 1 |
Baraldi, PG; Basso, G; Bortolozzi, R; Brancale, A; Carrion, MD; Chen, L; Cruz-Lopez, O; Hamel, E; Lopez Cara, C; Romagnoli, R; Viola, G | 1 |
Chaplin, DJ; Garner, CM; Ghatak, A; Hadimani, MB; Hall, JJ; Hamel, E; Kessler, RJ; Liu, L; Lopez, R; Macdonough, MT; Mason, RP; Nguyen, BL; Pettit, GR; Pinney, KG; Shirali, AR; Sriram, M; Strecker, TE; Trawick, ML | 1 |
Lemelle, E; McFerrin, H; Mottamal, M; Wang, G; Zhang, C; Zhang, Q; Zheng, S; Zhong, Q | 1 |
Álvarez, R; López, V; Mateo, C; Medarde, M; Peláez, R | 1 |
Bai, Z; Bao, K; Feng, D; Guan, Q; Jiang, M; Jiang, N; Li, C; Qi, H; Wu, Y; Yang, L; Zhai, Y; Zhang, W; Zuo, D | 1 |
Bartenschlager, R; Boldescu, V; Dimoglo, A; Graf, D; Klein, CD; Richter, M; Streicher, F | 1 |
Kumar, D; Kumar, S; Sharma, P; Shri, R | 1 |
3 review(s) available for combretastatin and colchicine
Article | Year |
---|---|
[Molecular basis of probes for cytoskeletal proteins].
Topics: Animals; Bibenzyls; Colchicine; Cytoskeletal Proteins; Fertilization; Microtubules; Mitosis; Paclitaxel; Sea Urchins; Stilbenes; Zearalenone | 1993 |
[Natural organic compounds that affect to microtubule functions: syntheses and structure-activity relationships of combretastatins, curacin A and their analogs as the colchicine-site ligands on tubulin].
Topics: Bibenzyls; Binding Sites; Cell Cycle; Colchicine; Cyclopropanes; Ligands; Microtubules; Protein Binding; Stilbenes; Structure-Activity Relationship; Thiazoles; Tubulin | 2000 |
Mechanistic Insights and Docking Studies of Phytomolecules as Potential Candidates in the Management of Cancer.
Topics: Antineoplastic Agents; Bibenzyls; Colchicine; Curcumin; Humans; Molecular Docking Simulation; Neoplasms; Paclitaxel | 2022 |
17 other study(ies) available for combretastatin and colchicine
Article | Year |
---|---|
Synthesis of alkoxy-substituted diaryl compounds and correlation of ring separation with inhibition of tubulin polymerization: differential enhancement of inhibitory effects under suboptimal polymerization reaction conditions.
Topics: Animals; Antineoplastic Agents; Bibenzyls; Binding Sites; Bridged-Ring Compounds; Colchicine; Leukemia L1210; Mice; Stilbenes; Structure-Activity Relationship; Tubulin | 1992 |
Interactions of tubulin with potent natural and synthetic analogs of the antimitotic agent combretastatin: a structure-activity study.
Topics: Animals; Anisoles; Antineoplastic Agents; Bibenzyls; Binding Sites; Binding, Competitive; Colchicine; Leukemia L1210; Mice; Mitosis; Podophyllotoxin; Protein Binding; Stilbenes; Structure-Activity Relationship; Tubulin | 1988 |
Interactions of combretastatin, a new plant-derived antimitotic agent, with tubulin.
Topics: Animals; Anisoles; Bibenzyls; Binding Sites; Brain Chemistry; Cattle; Cells, Cultured; Colchicine; Leukemia L1210; Mice; Mitosis; Protein Binding; Stilbenes; Tubulin | 1983 |
Computational and molecular modeling evaluation of the structural basis for tubulin polymerization inhibition by colchicine site agents.
Topics: Antineoplastic Agents, Phytogenic; Bibenzyls; Binding Sites; Colchicine; Models, Molecular; Paclitaxel; Podophyllotoxin; Protein Conformation; Software; Stilbenes; Tubulin; Tubulin Modulators | 1996 |
Comparative molecular field analysis of colchicine inhibition and tubulin polymerization for combretastatins binding to the colchicine binding site on beta-tubulin.
Topics: Bibenzyls; Binding Sites; Biopolymers; Colchicine; Molecular Conformation; Stilbenes; Tubulin | 2000 |
Rapid colchicine competition-binding scintillation proximity assay using biotin-labeled tubulin.
Topics: Aminophenols; Bibenzyls; Binding Sites; Binding, Competitive; Biotinylation; Colchicine; Demecolcine; Mebendazole; Microspheres; Podophyllotoxin; Scintillation Counting; Solvents; Stilbenes; Streptavidin; Sulfonamides; Tritium; Tubulin; Yttrium | 2000 |
The interaction of the B-ring of colchicine with alpha-tubulin: a novel footprinting approach.
Topics: Amino Acid Sequence; Animals; Bibenzyls; Binding Sites; Cattle; Chromatography, High Pressure Liquid; Colchicine; Fluorescence; Models, Molecular; Molecular Sequence Data; Peptide Fragments; Podophyllotoxin; Protein Conformation; Protein Footprinting; Stilbenes; Tropolone; Tryptophan; Tubulin; Urea | 2000 |
Synthesis and antimicrotubule activity of combretatropone derivatives.
Topics: Antineoplastic Agents; Bibenzyls; Colchicine; Magnetic Resonance Spectroscopy; Microtubules; Molecular Structure; Stilbenes; Structure-Activity Relationship; Tubulin; Tubulin Modulators | 2002 |
Quantitative structure-activity relationship (5D-QSAR) study of combretastatin-like analogues as inhibitors of tubulin assembly.
Topics: Antineoplastic Agents; Bibenzyls; Binding Sites; Colchicine; Ligands; Models, Molecular; Molecular Conformation; Monte Carlo Method; Quantitative Structure-Activity Relationship; Stilbenes; Tubulin; Tubulin Modulators | 2005 |
Novel combretastatin analogues endowed with antitumor activity.
Topics: Animals; Antineoplastic Agents; Benzofurans; Bibenzyls; Binding, Competitive; Biopolymers; Cell Line, Tumor; Cell Nucleus; Colchicine; Endothelial Cells; Endothelium, Vascular; Female; Humans; Mice; Mice, Nude; Microtubules; Organophosphates; Prodrugs; Stereoisomerism; Stilbenes; Structure-Activity Relationship; Thiophenes; Tubulin; Xenograft Model Antitumor Assays | 2006 |
Combretastatin-like chalcones as inhibitors of microtubule polymerisation. Part 2: Structure-based discovery of alpha-aryl chalcones.
Topics: Algorithms; Bibenzyls; Binding Sites; Cell Line; Chalcones; Colchicine; Drug Discovery; Humans; Hydrocarbons, Cyclic; Microtubules; Structure-Activity Relationship; Tubulin Modulators | 2009 |
Synthesis and antitumor activity of 1,5-disubstituted 1,2,4-triazoles as cis-restricted combretastatin analogues.
Topics: Angiogenesis Inhibitors; Animals; Antineoplastic Agents; Apoptosis; Bibenzyls; Caspase 3; Cell Line, Tumor; Cell Shape; Cells, Cultured; Chick Embryo; Colchicine; Drug Screening Assays, Antitumor; Endothelial Cells; Enzyme Activation; G2 Phase; Humans; Membrane Potential, Mitochondrial; Mitochondria; Models, Molecular; Poly(ADP-ribose) Polymerases; Protein Binding; Proto-Oncogene Proteins c-bcl-2; Reactive Oxygen Species; Structure-Activity Relationship; Triazoles; Tubulin; Tubulin Modulators | 2010 |
Synthesis of a 2-aryl-3-aroyl indole salt (OXi8007) resembling combretastatin A-4 with application as a vascular disrupting agent.
Topics: Animals; Antineoplastic Agents; Bibenzyls; Colchicine; Drug Screening Assays, Antitumor; Humans; Indoles; Inhibitory Concentration 50; Male; Mice; Molecular Structure; Organophosphates; Prodrugs; Prostatic Neoplasms; Stilbenes; Structure-Activity Relationship; Tubulin | 2013 |
Design, synthesis, and biological evaluation of novel pyridine-bridged analogues of combretastatin-A4 as anticancer agents.
Topics: Animals; Antineoplastic Agents; Bibenzyls; Binding Sites; Cell Cycle Checkpoints; Cell Line, Tumor; Chick Embryo; Colchicine; Drug Design; Female; Humans; Mice; Mice, Inbred C57BL; Models, Molecular; Polymerization; Pyridines; Structure-Activity Relationship; Tubulin; Tubulin Modulators | 2014 |
p,p-Dihydroxydihydrostilbenophanes related to antimitotic combretastatins. Conformational analysis and its relationship to tubulin inhibition.
Topics: Antimitotic Agents; Bibenzyls; Colchicine; Macrocyclic Compounds; Magnetic Resonance Spectroscopy; Models, Molecular; Molecular Conformation; Polymerization; Stilbenes; Tubulin Modulators | 2014 |
Microwave-assisted synthesis and biological evaluation of 3,4-diaryl maleic anhydride/N-substituted maleimide derivatives as combretastatin A-4 analogues.
Topics: Bibenzyls; Binding Sites; Cell Line, Tumor; Cell Proliferation; Colchicine; Drug Design; Humans; Maleic Anhydrides; Maleimides; Microwaves; Molecular Docking Simulation; Protein Structure, Tertiary; Structure-Activity Relationship; Tubulin; Tubulin Modulators | 2015 |
Synthesis, Biological Evaluation, and Molecular Docking of Combretastatin and Colchicine Derivatives and their hCE1-Activated Prodrugs as Antiviral Agents.
Topics: Antiviral Agents; Bibenzyls; Binding Sites; Carboxylesterase; Cell Line, Tumor; Cell Survival; Colchicine; Drug Design; Humans; Molecular Docking Simulation; Prodrugs; Protein Structure, Tertiary; Structure-Activity Relationship; Tubulin; Tubulin Modulators; Zika Virus | 2019 |