Page last updated: 2024-08-23

colforsin and thapsigargin

colforsin has been researched along with thapsigargin in 101 studies

Research

Studies (101)

TimeframeStudies, this research(%)All Research%
pre-19901 (0.99)18.7374
1990's60 (59.41)18.2507
2000's33 (32.67)29.6817
2010's7 (6.93)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Cuddon, P; Fleming, A; Floto, RA; Goldsmith, P; Jahreiss, L; O'Kane, CJ; Pask, D; Rubinsztein, DC; Saiki, S; Sarkar, S; Siddiqi, FH; Ttofi, EK; Williams, A1
Batista-Gonzalez, A; Brunhofer, G; Fallarero, A; Gopi Mohan, C; Karlsson, D; Shinde, P; Vuorela, P1
Brayden, DJ; Cuthbert, AW; Pickles, RJ1
Bismuth, G; Cefai, D; Christensen, SB; Debre, P; Gouy, H1
Nahorski, SR; Wojcikiewicz, RJ1
Chew, CS; Petropoulos, AC1
Aakerlund, L; Fuhlendorff, J; Gether, U; Schwartz, TW; Thastrup, O1
Brayden, DJ; Cuthbert, AW; Hanley, MR; Thastrup, O1
De Pont, JJ; Van Emst-de Vries, SE; Willems, PH1
Boddeke, HG; Seuwen, K1
Reich, H; Sei, Y1
Akaike, N; Uneyama, C; Uneyama, H1
Komatsu, M; McDermott, AM; Sharp, GW1
Gérard, C; Mauchamp, J; Penel, C; Verrier, B1
Eaton, DC; Kokko, KE; Ling, BN1
Doubell, AF; Thibault, G1
Gillison, SL; Komatsu, M; McDermott, AM; Sharp, GW1
Ahlström, M; Törnquist, K1
Brooker, G; Debernardi, MA; Munshi, R1
Anwer, MS; Engelking, LR; Grüne, S1
Brayden, DJ; Krouse, ME; Law, T; Wine, JJ1
Baird, AW; Taylor, CT1
Böhmer, FD; Böhmer, SA1
Kao, LS; Lin, YJ; Liu, PS1
Akaike, N; Takahashi, M; Uneyama, C; Uneyama, H1
Brabant, G; Mader, T; Rossig, L; Schöfl, C; von zur Mühlen, A1
Komatsu, M; Schermerhorn, T; Sharp, GW; Straub, SG1
Ahrén, B; Karlsson, S1
An, S; Goetzl, EJ; Zeng, L1
Dowd, DR; Kamradt, MC; MacDonald, PN; Miesfeld, RL; Ryerse, JS1
Earp, HS; Graves, LM; Li, X; Yu, H1
Naderali, EK; Poyser, NL1
Amano, K; Hori, M; Karaki, H; Ozaki, H; Sato, K1
Laychock, SG; Lee, B1
Akbarali, HI; Hrnjez, BJ; Matthews, JB; Mayol, JM; Smith, JA; Song, JC1
Dukhanin, AS; Gubaeva, FR; Sergeev, PV1
al Hussaini, M; Gath, J; Himmel, H; Ravens, U1
Kocić, I1
Jung, JS; Kang, DS; Kim, MG; Lee, SH; Oh, SO1
Krouse, ME; Moon, S; Singh, M; Wine, JJ1
Barritt, GJ; Fernando, KC; Gregory, RB1
Gibson, WJ; Pinnock, RD; Young, JM; Young, KW1
Cooper, DM; Fagan, KA; Mons, N1
Hiramatsu, Y; Murakami, M; Yoshimura, K1
Alper, SL; Jiang, L; Lencer, WI; Madara, JL; Merlin, D; Nusrat, A; Strohmeier, GR1
Braiman, A; Priel, Z; Zagoory, O1
Christensen, G; Holt, E; Lunde, PK; Sejersted, OM; Semb, SO; Tønnessen, T; Wasserstrom, JA1
O'Farrell, AM; O'Reilly, CM; Ryan, MP1
Chan, HC; Chew, SB; Ko, WH; Wong, PY1
Choi, SY; Kim, KT; Song, SK1
Balasubramaniam, A; Chance, W; Dayal, R; Fischer, J; Kasckow, J; Regmi, A; Sheriff, S1
Davia, K; Harding, SE1
Carraway, RE; Mitra, SP1
Glushakov, AV; Glushakova, HY; Skok, VI1
Arrese, EL; Flowers, MT; Gazard, JL; Wells, MA1
Doms, RW; Edinger, AL; Funk, CD; Hoffman, TL; Martin, V; Ronde, P; Unett, D; Wong, A1
Bobryshev, AIu; Skok, VI; Voĭtenko, SV1
Kozawa, O; Shinoda, J; Tokuda, H; Uematsu, T1
Hayashi, M; Ichihara, A; Miyashita, Y; Naitoh, M; Saruta, T; Suzuki, H1
Dun, NJ; Dun, SL; Leung, GP; Wong, PY1
Martinez, JR; Zhang, GH1
Shuttleworth, TJ; Thompson, JL1
Eade, J; Hill, CE; Sandow, SL1
Buxbaum, JD; Corfas, G; Peschon, JJ; Rio, C1
Belinsky, GS; Tashjian, AH1
Conner, TD; Dickson, JL; Ecay, TW1
Berggren, PO; Islam, MS; Larsson, O; Lemmens, R1
Botana, LM; de la Rosa, LA; Vieytes, MR; Vilariño, N1
Jacobson, KL; Ott, SM; Singh, JC; Watson, EL1
Cooper, DM; Fagan, KA; Gu, C; Hu, B; Smith, KE1
Chandrasekhar, S; Halladay, DL; Martin, TJ; Miles, RR; Onyia, JE; Thirunavukkarasu, K1
Balasubramaniam, A; F Qureshy, A; Kasckow, JW; Sheriff, S; T Chance, W1
Chen, ZY; Huang, Y; Ko, WH; Lau, CW; Law, VW; Yip, WC; Yue, GG1
Duszyk, M1
Joo, NS; Krouse, ME; Saenz, Y; Wine, JJ1
Greger, R; Herbst, M; Hescheler, J; Sasse, P; Ullrich, S; Yu, H1
Delbecque, JP; Gautron, F; Manière, G; Vanhems, E1
Andrade, R; Cooley, D; Ge, Q; Legakis, JE; Mattingly, RR; Yang, H1
Hughes, TR; Irvine, SA; Mead, JR; Ramji, DP; Singh, NN1
Hanafusa, T; Hosoi, K; Min, KY; Mori, H; Nakahari, T; Shiima, C1
Fabbro, M; Nair, SV; Raftos, DA1
Haggie, PM; Song, Y; Thiagarajah, JR; Verkman, AS1
Bendhack, LM; Callera, GE; Caperuto, LC; Carvalho, CR; Tostes, RC; Yeh, E1
Belmadani, S; Fischmeister, R; Méry, PF; Poüs, C1
Irokawa, T; Joo, NS; Krouse, ME; Wine, JJ; Wu, JV1
Joo, NS; Krouse, ME; Lee, MM; Talbott, JF; Wine, JJ1
Jan, CR; Liu, CP1
Grünberger, C; Klar, J; Kurtz, A; Obermayer, B; Schweda, F1
Caron, AZ; Chaloux, B; Guillemette, G1
Cristino, L; De Petrocellis, L; Di Marzo, V; Marini, P; Matias, I; Moriello, AS; Nigam, S; Starowicz, K1
Ciruela, A; Cooper, DM; Macdougall, DA; Sinz, A; Wachten, S1
Chakraborty, T; Fromm, M; Gitter, AH; Günzel, D; Mohamed, W; Richter, JF; Schulzke, JD; Weiss, S1
Fletcher, PA; Li, YX1
Xie, X; Xu, Y1
Choi, HS; Kim, HJ; Kim, HS; Kim, MK; Kim, NK; Lee, IK; Lee, KM; Lee, KU; Min, AK; Park, KG; Ryu, SY; Seo, HY1
Bertelsen, LS; Frankson, M; Keely, SJ; Kelly, OB; Mroz, MS; Toumi, F; Ward, JB1
Aoyagi, H; Higa, T; Horinouchi, T; Miwa, S; Nishiya, T; Terada, K1
Dalal, S; Das, BC; Foster, CR; Singh, K; Singh, M1
Ayala, JE; Burmeister, MA; Younce, CW1
Aygün, O; Bittker, JA; Carr, S; Clark, A; Greka, A; Gutierrez, J; Jehle, AW; Mandinova, A; Matan, S; Mundel, P; Reitberger, M; Schoenfelder, J; Sieber, J; Udeshi, N; Wieder, N; Zhang, J1

Other Studies

101 other study(ies) available for colforsin and thapsigargin

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Novel targets for Huntington's disease in an mTOR-independent autophagy pathway.
    Nature chemical biology, 2008, Volume: 4, Issue:5

    Topics: Animals; Autophagy; Calcium Channels, L-Type; Clonidine; Cyclic AMP; Humans; Huntington Disease; Imidazoline Receptors; Minoxidil; Protein Kinases; Signal Transduction; TOR Serine-Threonine Kinases; Type C Phospholipases; Verapamil

2008
Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.
    Bioorganic & medicinal chemistry, 2012, Nov-15, Volume: 20, Issue:22

    Topics: Acetylcholinesterase; Amyloid beta-Peptides; Benzophenanthridines; Binding Sites; Butyrylcholinesterase; Catalytic Domain; Cholinesterase Inhibitors; Humans; Isoquinolines; Kinetics; Molecular Docking Simulation; Structure-Activity Relationship

2012
Ion transport in cultured epithelia from human sweat glands: comparison of normal and cystic fibrosis tissues.
    British journal of pharmacology, 1991, Volume: 102, Issue:1

    Topics: Adenylyl Cyclases; Amiloride; Barium; Calcium; Carbachol; Cells, Cultured; Colforsin; Cyclic AMP; Cystic Fibrosis; Epithelium; Humans; Kallidin; Lanthanum; Sodium Channels; Sweat Glands; Terpenes; Thapsigargin

1991
Cyclic AMP- and inositol phosphate-independent inhibition of Ca2+ influx by cholera toxin in CD3-stimulated Jurkat T cells. A study with a cholera toxin-resistant cell variant and the Ca2+ endoplasmic reticulum-ATPase inhibitor thapsigargin.
    Journal of immunology (Baltimore, Md. : 1950), 1991, Aug-01, Volume: 147, Issue:3

    Topics: Antigens, Differentiation, T-Lymphocyte; Calcium; Calcium-Transporting ATPases; CD3 Complex; Cell Division; Cell Line; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dinoprostone; Drug Antagonism; Gene Expression Regulation; Humans; In Vitro Techniques; Inositol Phosphates; Receptors, Antigen, T-Cell; T-Lymphocytes; Terpenes; Thapsigargin

1991
Chronic muscarinic stimulation of SH-SY5Y neuroblastoma cells suppresses inositol 1,4,5-trisphosphate action. Parallel inhibition of inositol 1,4,5-trisphosphate-induced Ca2+ mobilization and inositol 1,4,5-trisphosphate binding.
    The Journal of biological chemistry, 1991, Nov-25, Volume: 266, Issue:33

    Topics: Calcium; Calcium Channels; Carbachol; Cell Line; Cell Membrane; Cell Membrane Permeability; Colforsin; Humans; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Inositol Phosphates; Kinetics; Neuroblastoma; Phorbol 12,13-Dibutyrate; Plant Extracts; Receptors, Cell Surface; Receptors, Cytoplasmic and Nuclear; Terpenes; Thapsigargin; Tretinoin

1991
Thapsigargin potentiates histamine-stimulated HCl secretion in gastric parietal cells but does not mimic cholinergic responses.
    Cell regulation, 1991, Volume: 2, Issue:1

    Topics: Aminopyrine; Animals; Calcium; Carbachol; Colforsin; Cyclic AMP; Drug Synergism; Gastric Acid; Gastric Mucosa; Histamine; In Vitro Techniques; Rabbits; Receptors, Cholinergic; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin

1991
Y1 receptors for neuropeptide Y are coupled to mobilization of intracellular calcium and inhibition of adenylate cyclase.
    FEBS letters, 1990, Jan-15, Volume: 260, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Animals; Binding Sites; Calcium; Colforsin; Cytosol; Fluorescent Dyes; Intracellular Membranes; Neuroblastoma; Neuropeptide Y; Plant Extracts; Receptors, Neuropeptide Y; Receptors, Neurotransmitter; Swine; Thapsigargin; Tumor Cells, Cultured

1990
Thapsigargin, a new calcium-dependent epithelial anion secretagogue.
    British journal of pharmacology, 1989, Volume: 98, Issue:3

    Topics: Adenocarcinoma; Anions; Calcimycin; Calcium; Colforsin; Colonic Neoplasms; Electrophysiology; Epithelium; Humans; Plant Extracts; Thapsigargin; Tumor Cells, Cultured

1989
Cholecystokinin-stimulated enzyme secretion from dispersed rabbit pancreatic acinar cells: phosphorylation-dependent changes in potency and efficacy.
    Pflugers Archiv : European journal of physiology, 1995, Volume: 430, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Alkaloids; Amylases; Animals; Calcium-Transporting ATPases; Cells, Cultured; Cholecystokinin; Colforsin; Cyclic AMP; Enzyme Activation; Enzyme Inhibitors; Pancreas; Phosphodiesterase Inhibitors; Phosphorylation; Protein Kinase Inhibitors; Protein Kinases; Rabbits; Sincalide; Staurosporine; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Time Factors

1995
Heparin-insensitive calcium release from intracellular stores triggered by the recombinant human parathyroid hormone receptor.
    British journal of pharmacology, 1995, Volume: 114, Issue:8

    Topics: Calcium; Calcium-Transporting ATPases; Carbachol; Cells, Cultured; Colforsin; Cyclic AMP; Egtazic Acid; Heparin; Humans; Parathyroid Hormone; Receptors, Parathyroid Hormone; Ryanodine; Terpenes; Thapsigargin

1995
Thapsigargin induces IL-2 receptor alpha-chain in human peripheral and Jurkat T cells via a protein kinase C-independent mechanism.
    Immunology letters, 1995, Volume: 45, Issue:1-2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Base Sequence; Calcimycin; Calcium; Calcium-Transporting ATPases; Cholera Toxin; Colforsin; Drug Synergism; Gene Expression Regulation; Gene Expression Regulation, Leukemic; Humans; Hydroquinones; Isoquinolines; Leukemia-Lymphoma, Adult T-Cell; Molecular Sequence Data; Neoplasm Proteins; NF-kappa B; Piperazines; Protein Kinase C; Receptors, Interleukin-2; RNA, Messenger; RNA, Neoplasm; Signal Transduction; Staurosporine; T-Lymphocytes; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin

1995
Intracellular mechanisms of cytoplasmic Ca2+ oscillation in rat megakaryocyte.
    The Journal of biological chemistry, 1993, Jan-05, Volume: 268, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine Triphosphate; Alkaloids; Animals; Calcimycin; Calcium; Calcium-Transporting ATPases; Calmodulin; Colforsin; Cyclic AMP; Cytoplasm; Egtazic Acid; Female; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Kinetics; Male; Megakaryocytes; Models, Biological; Oscillometry; Protein Kinase C; Rats; Staurosporine; Sulfonamides; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Trifluoperazine

1993
Sodium fluoride stimulates exocytosis at a late site of calcium interaction in stimulus-secretion coupling: studies with the RINm5F beta cell line.
    Molecular pharmacology, 1995, Volume: 47, Issue:3

    Topics: Aluminum; Animals; Arachidonic Acid; Calcium; Calcium-Binding Proteins; Cell Line; Colforsin; Cyclic AMP; Deferoxamine; Exocytosis; Extracellular Space; Insulin; Insulin Secretion; Ionomycin; Islets of Langerhans; Kinetics; Melitten; Nitrendipine; Potassium Chloride; Protein Kinase C; Secretory Rate; Sodium Fluoride; Stimulation, Chemical; Sulfonamides; Temperature; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Trifluoperazine

1995
Thyrotropin regulation of basolateral Cl- and I- effluxes in thyroid follicles in culture.
    Molecular and cellular endocrinology, 1994, Volume: 106, Issue:1-2

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Animals; Antiporters; Calcimycin; Calcium; Cell Membrane; Cells, Cultured; Chloride Channels; Chlorides; Colforsin; Cyclic AMP; Iodides; Kinetics; Nitrobenzoates; Probenecid; Swine; Terpenes; Thapsigargin; Thyroid Gland; Thyrotropin

1994
Prostaglandin E2 activates clusters of apical Cl- channels in principal cells via a cyclic adenosine monophosphate-dependent pathway.
    The Journal of clinical investigation, 1994, Volume: 93, Issue:2

    Topics: Animals; Arginine Vasopressin; Bucladesine; Calcium-Transporting ATPases; Cell Membrane; Cells, Cultured; Chloride Channels; Colforsin; Cyclic AMP; Dinoprostone; Electric Conductivity; Kidney Cortex; Kidney Tubules, Collecting; Membrane Potentials; Rabbits; Terpenes; Thapsigargin

1994
Calcium is involved in both positive and negative modulation of the secretory system for ANP.
    The American journal of physiology, 1994, Volume: 266, Issue:5 Pt 2

    Topics: Animals; Animals, Newborn; Atrial Natriuretic Factor; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Cells, Cultured; Chromatography, High Pressure Liquid; Colforsin; Egtazic Acid; Endothelins; Fibroblast Growth Factors; Gallic Acid; Heart; Heart Atria; Kinetics; Models, Cardiovascular; Myocardium; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Ryanodine; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Time Factors

1994
Mastoparan stimulates exocytosis at a Ca(2+)-independent late site in stimulus-secretion coupling. Studies with the RINm5F beta-cell line.
    The Journal of biological chemistry, 1993, Nov-05, Volume: 268, Issue:31

    Topics: Animals; Calcium; Cell Line; Colforsin; Exocytosis; Hydroquinones; In Vitro Techniques; Insulin; Insulin Secretion; Intercellular Signaling Peptides and Proteins; Islets of Langerhans; Nitrendipine; Peptides; Pertussis Toxin; Rats; Secretory Rate; Terpenes; Thapsigargin; Virulence Factors, Bordetella; Wasp Venoms

1993
Modulatory effect of cyclic AMP on calcium fluxes in FRTL-5 cells.
    Journal of cellular physiology, 1993, Volume: 157, Issue:3

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenosine Triphosphate; Animals; Calcium; Calcium-Transporting ATPases; Cell Line; Colforsin; Cyclic AMP; Fura-2; Rats; Terpenes; Thapsigargin; Thyroid Gland

1993
Ca2+ inhibition of beta-adrenergic receptor- and forskolin-stimulated cAMP accumulation in C6-2B rat glioma cells is independent of protein kinase C.
    Molecular pharmacology, 1993, Volume: 43, Issue:3

    Topics: Animals; Calcium; Colforsin; Cyclic AMP; Enzyme Activation; Glioma; Hydrolysis; Isoproterenol; Phosphatidylinositols; Protein Kinase C; Rats; Receptors, Adrenergic, beta; Signal Transduction; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Tumor Cells, Cultured

1993
Role of intracellular calcium and protein kinases in the activation of hepatic Na+/taurocholate cotransport by cyclic AMP.
    The Journal of biological chemistry, 1993, Aug-25, Volume: 268, Issue:24

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Bucladesine; Calcium; Calcium-Transporting ATPases; Cells, Cultured; Colforsin; Cyclic AMP; Ionomycin; Kinetics; Liver; Phenylephrine; Protein Kinase Inhibitors; Protein Kinases; Rats; Sodium; Taurocholic Acid; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin; Vasopressins

1993
Stilbenes stimulate T84 Cl- secretion by elevating Ca2+.
    The American journal of physiology, 1993, Volume: 264, Issue:2 Pt 1

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Calcium; Cell Line; Chlorides; Colforsin; Colon; Drug Synergism; Electrophysiology; Stilbenes; Terpenes; Thapsigargin

1993
Berberine inhibition of electrogenic ion transport in rat colon.
    British journal of pharmacology, 1995, Volume: 116, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Bacterial Toxins; Berberine; Biological Transport; Chlorides; Colforsin; Colon; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Cytochalasin D; Enterotoxins; Epithelium; Escherichia coli Proteins; In Vitro Techniques; Ions; Male; Membrane Potentials; Rats; Rats, Wistar; Secretory Rate; Sensitivity and Specificity; Signal Transduction; Terpenes; Thapsigargin

1995
Activation of platelet-derived growth factor (PDGF) receptor dephosphorylation in intact Swiss 3T3 cells by elevators of intracellular Ca2+ and cAMP.
    FEBS letters, 1996, Aug-05, Volume: 391, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; 3T3 Cells; Animals; Calcimycin; Calcium; Calcium-Transporting ATPases; Cell Division; Colforsin; Cyclic AMP; Enzyme Inhibitors; Kinetics; Mice; Platelet-Derived Growth Factor; Protein Tyrosine Phosphatases; Receptors, Platelet-Derived Growth Factor; Terpenes; Thapsigargin

1996
Effects of caffeine on Ca2+ fluxes and secretion in bovine chromaffin cells.
    European journal of pharmacology, 1995, Nov-30, Volume: 291, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Adrenal Medulla; Animals; Bucladesine; Caffeine; Calcium; Calcium-Transporting ATPases; Carbachol; Catecholamines; Cattle; Colforsin; Dimethylphenylpiperazinium Iodide; Inositol Phosphates; Nicotinic Agonists; Phosphodiesterase Inhibitors; Terpenes; Thapsigargin; Veratridine

1995
Pharmacological studies on mechanisms involved in Ca2+ oscillations in rat megakaryocytes.
    European journal of pharmacology, 1995, Nov-30, Volume: 291, Issue:3

    Topics: Adenosine Triphosphate; Alkaloids; Animals; Calcium; Calcium-Transporting ATPases; Calmodulin; Colforsin; Female; Indoles; Male; Megakaryocytes; Protein Kinase C; Rats; Rats, Wistar; Staurosporine; Sulfonamides; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin

1995
CYCLIC adenosine 3',5'-monophosphate potentiates Ca2+ signaling and insulin secretion by phospholipase C-linked hormones in HIT cells.
    Endocrinology, 1996, Volume: 137, Issue:7

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Arginine Vasopressin; Bombesin; Calcium; Calcium-Transporting ATPases; Cell Line; Colforsin; Cricetinae; Cyclic AMP; Egtazic Acid; Enzyme Inhibitors; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Mesocricetus; Nifedipine; Signal Transduction; Terpenes; Thapsigargin; Time Factors

1996
Pituitary adenylate cyclase-activating peptide, carbachol, and glucose stimulate insulin release in the absence of an increase in intracellular Ca2+.
    Molecular pharmacology, 1996, Volume: 50, Issue:4

    Topics: Animals; Calcium; Calcium Channel Blockers; Carbachol; Cells, Cultured; Colforsin; Glucose; Insulin; Insulin Secretion; Intracellular Fluid; Islets of Langerhans; Neuropeptides; Nitrendipine; Pituitary Adenylate Cyclase-Activating Polypeptide; Rats; Stimulation, Chemical; Tetradecanoylphorbol Acetate; Thapsigargin

1996
Gastrin-releasing peptide mobilizes calcium from intracellular stores in HIT-T15 cells.
    Peptides, 1996, Volume: 17, Issue:6

    Topics: Animals; Calcium; Cell Line; Colforsin; Cricetinae; Cyclic AMP; Egtazic Acid; Enzyme Inhibitors; Estrenes; Gastrin-Releasing Peptide; Gastrointestinal Hormones; Glucose; Islets of Langerhans; Peptides; Protein Kinase C; Pyrrolidinones; Ryanodine; Signal Transduction; Thapsigargin; Type C Phospholipases

1996
Regulation of expression of matrix metalloproteinase-9 in early human T cells of the HSB.2 cultured line by the EP3 subtype of prostaglandin E2 receptor.
    The Journal of biological chemistry, 1996, Nov-01, Volume: 271, Issue:44

    Topics: Adenine; Alprostadil; Blotting, Northern; Bucladesine; Calcium; Cell Line; Colforsin; Collagenases; Cyclic AMP; Cycloheximide; Dactinomycin; Dinoprostone; Enzyme Inhibitors; Gene Expression Regulation, Enzymologic; Gene Expression Regulation, Neoplastic; Humans; Kinetics; Leukemia, T-Cell; Matrix Metalloproteinase 9; Misoprostol; Prostaglandins E, Synthetic; Receptors, Prostaglandin E; RNA, Messenger; T-Lymphocytes; Thapsigargin; Transcription, Genetic; Tumor Cells, Cultured

1996
Crosstalk during Ca2+-, cAMP-, and glucocorticoid-induced gene expression in lymphocytes.
    Molecular and cellular endocrinology, 1997, Apr-04, Volume: 128, Issue:1-2

    Topics: Animals; Apoptosis; Calcimycin; Calcium; Cell Division; Chloramphenicol O-Acetyltransferase; Colforsin; Cyclic AMP; Dexamethasone; Gene Expression Regulation, Neoplastic; Genes, Reporter; Glucocorticoids; Lymphocytes; Mice; Signal Transduction; Thapsigargin; Thymoma; Thymus Neoplasms; Transfection; Tumor Cells, Cultured

1997
Protein kinase C and protein kinase A inhibit calcium-dependent but not stress-dependent c-Jun N-terminal kinase activation in rat liver epithelial cells.
    The Journal of biological chemistry, 1997, Jun-06, Volume: 272, Issue:23

    Topics: 1-Methyl-3-isobutylxanthine; Androstadienes; Angiotensin II; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; Epithelial Cells; Epithelium; Humans; JNK Mitogen-Activated Protein Kinases; Kinetics; Liver; Mitogen-Activated Protein Kinases; Models, Biological; Polyenes; Protein Kinases; Rats; Recombinant Proteins; Signal Transduction; Sirolimus; Tetradecanoylphorbol Acetate; Thapsigargin; Wortmannin

1997
Prostaglandin production by guinea-pig endometrial cells: effects of caffeine and other modulators of intracellular calcium.
    Prostaglandins, leukotrienes, and essential fatty acids, 1997, Volume: 56, Issue:5

    Topics: Animals; Berberine; Caffeine; Calcium; Cell Separation; Cells, Cultured; Colforsin; Dinoprost; Drug Interactions; Endometrium; Female; Gallic Acid; Guinea Pigs; Ryanodine; Sulfonamides; Thapsigargin; Theophylline; Trifluoperazine

1997
Palytoxin-induced increase in endothelial Ca2+ concentration in the rabbit aortic valve.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 355, Issue:6

    Topics: Acrylamides; Adenosine Triphosphate; Animals; Aortic Valve; Calcium; Cnidarian Venoms; Colforsin; Endothelium, Vascular; In Vitro Techniques; Lanthanum; Marine Toxins; Microscopy, Confocal; Ouabain; Oxazoles; Potassium; Rabbits; Sodium; Thapsigargin; Vasoconstrictor Agents

1997
Atrial natriuretic peptide and cyclic nucleotides affect glucose-induced Ca2+ responses in single pancreatic islet beta-cells: correlation with (Ca[2+] + Mg2+)-ATPase activity.
    Diabetes, 1997, Volume: 46, Issue:8

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Atrial Natriuretic Factor; Ca(2+) Mg(2+)-ATPase; Calcium; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Colforsin; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Gallopamil; Glucose; Islets of Langerhans; Male; Nucleotides, Cyclic; Rats; Rats, Sprague-Dawley; Thapsigargin

1997
Ammonia effect on calcium-activated chloride secretion in T84 intestinal epithelial monolayers.
    The American journal of physiology, 1997, Volume: 273, Issue:2 Pt 1

    Topics: Ammonia; Barium; Calcimycin; Calcium; Carbachol; Cell Line; Chlorides; Colforsin; Cyclic AMP; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Humans; Intestinal Mucosa; Intracellular Membranes; Ionomycin; Ionophores; Tetradecanoylphorbol Acetate; Thapsigargin

1997
[Early stages in mechanisms of glucocorticoids action on human thrombocytes: effect of hydrocortisone on intracellular cAMP and Ca2+].
    Biulleten' eksperimental'noi biologii i meditsiny, 1997, Volume: 123, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine; Blood Platelets; Calcium; Colforsin; Collagen; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Epinephrine; Glucocorticoids; Humans; Hydrocortisone; Intracellular Fluid; Phosphodiesterase Inhibitors; Radioligand Assay; Thapsigargin

1997
Mechanical restitution in atrial muscle from human and rat hearts: effects of agents that modify sarcoplasmic reticulum function.
    Pharmacology & toxicology, 1997, Volume: 81, Issue:2

    Topics: Animals; Binding, Competitive; Caffeine; Calcium; Calcium Channels; Colforsin; Enzyme Inhibitors; Humans; Hydroquinones; Myocardial Contraction; Phosphodiesterase Inhibitors; Rats; Ryanodine; Sarcoplasmic Reticulum; Thapsigargin

1997
Pretreatment with rimalkalim changes the adrenergic responsiveness of isolated guinea pig papillary muscle.
    European journal of pharmacology, 1997, Jul-30, Volume: 332, Issue:1

    Topics: Animals; Bucladesine; Cardiotonic Agents; Chromans; Colforsin; Enzyme Inhibitors; Female; Glyburide; Guinea Pigs; Male; Metoprolol; Muscle Relaxants, Central; Papillary Muscles; Phenylephrine; Potassium Channels; Pyrrolidines; Sympathetic Nervous System; Thapsigargin

1997
Cl- secretion induced by 5-hydroxytryptamine and calcitonin gene-related peptide in rat tracheal epithelia.
    Pflugers Archiv : European journal of physiology, 1997, Volume: 435, Issue:1

    Topics: Animals; Bumetanide; Calcitonin Gene-Related Peptide; Cells, Cultured; Chlorides; Colforsin; Cyclic AMP; Egtazic Acid; Electric Conductivity; Epithelium; Indomethacin; Kinetics; Rats; Rats, Sprague-Dawley; Serotonin; Thapsigargin; Trachea

1997
Calcium-stimulated Cl- secretion in Calu-3 human airway cells requires CFTR.
    The American journal of physiology, 1997, Volume: 273, Issue:6

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Bumetanide; Calcium; Carbachol; Cell Line; Cell Membrane; Chlorides; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Electric Conductivity; Epithelial Cells; Humans; Isoproterenol; Kinetics; Lung; Models, Biological; Thapsigargin

1997
Protein kinase A regulates the disposition of Ca2+ which enters the cytoplasmic space through store-activated Ca2+ channels in rat hepatocytes by diverting inflowing Ca2+ to mitochondria.
    The Biochemical journal, 1998, Mar-15, Volume: 330 ( Pt 3)

    Topics: Adenosine Triphosphate; Aluminum Compounds; Animals; Bucladesine; Calcium; Calcium Channels; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cytoplasm; Enzyme Inhibitors; Fluorides; Genistein; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Kinetics; Liver; Mitochondria, Liver; Rats; Thapsigargin; Vasopressins

1998
Dual effects of histamine and substance P on intracellular calcium levels in human U373 MG astrocytoma cells: role of protein kinase C.
    British journal of pharmacology, 1998, Volume: 123, Issue:3

    Topics: Animals; Astrocytoma; Brain Neoplasms; Calcium; Cerebellum; Colforsin; Cyclic AMP; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Guinea Pigs; HeLa Cells; Histamine; Humans; Inositol Phosphates; Protein Kinase C; Pyrilamine; Substance P; Thapsigargin; Tritium; Tumor Cells, Cultured

1998
Dependence of the Ca2+-inhibitable adenylyl cyclase of C6-2B glioma cells on capacitative Ca2+ entry.
    The Journal of biological chemistry, 1998, Apr-10, Volume: 273, Issue:15

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Biological Transport; Brain; Calcium; Cell Membrane; Colforsin; Cyclic AMP; Egtazic Acid; Glioma; Ionomycin; Ionophores; Kinetics; Rats; Thapsigargin; Tumor Cells, Cultured

1998
Cyclic AMP potentiates substance P-induced amylase secretion by augmenting the effect of calcium in the rat parotid acinar cells.
    Biochimica et biophysica acta, 1998, Mar-27, Volume: 1402, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 2,4-Dinitrophenol; Amylases; Animals; Bucladesine; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Isoproterenol; Male; Parotid Gland; Perfusion; Phorbol 12,13-Dibutyrate; Rats; Rats, Wistar; Substance P; Thapsigargin

1998
Distinct Ca2+- and cAMP-dependent anion conductances in the apical membrane of polarized T84 cells.
    The American journal of physiology, 1998, Volume: 275, Issue:2

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Anions; Bumetanide; Calcium; Cell Membrane; Cell Polarity; Charybdotoxin; Chloride Channels; Colforsin; Colonic Neoplasms; Cyclic AMP; Cytosol; Humans; Kinetics; Membrane Potentials; Models, Biological; Thapsigargin; Tumor Cells, Cultured

1998
PKA induces Ca2+ release and enhances ciliary beat frequency in a Ca2+-dependent and -independent manner.
    The American journal of physiology, 1998, Volume: 275, Issue:3

    Topics: Animals; Bucladesine; Calcium; Cells, Cultured; Cilia; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Egtazic Acid; Enzyme Inhibitors; Esophagus; Estrenes; Homeostasis; Isoquinolines; Kinetics; Mucous Membrane; Pyrrolidinones; Rana ridibunda; Sulfonamides; Thapsigargin; Type C Phospholipases

1998
Mechanisms of cardiomyocyte dysfunction in heart failure following myocardial infarction in rats.
    Journal of molecular and cellular cardiology, 1998, Volume: 30, Issue:8

    Topics: Actin Cytoskeleton; Animals; Calcium; Calcium Channels; Calcium-Transporting ATPases; Colforsin; Fura-2; Heart Failure; Heart Ventricles; Hemodynamics; Male; Muscle Contraction; Myocardial Infarction; Myocardium; Patch-Clamp Techniques; Rats; Rats, Wistar; Sarcoplasmic Reticulum; Sodium; Thapsigargin

1998
Purinoceptor activation of chloride transport in cystic fibrosis and CFTR-transfected pancreatic cell lines.
    British journal of pharmacology, 1998, Volume: 124, Issue:8

    Topics: Adenosine Triphosphate; Cell Line; Chloride Channels; Colforsin; Cyclic AMP; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Enzyme Inhibitors; Humans; Pancreas; Purinergic Agonists; Receptors, Purinergic; Thapsigargin; Transfection; Uridine Triphosphate

1998
Regulated anion secretion in cultured epithelia from Sertoli cells of immature rats.
    The Journal of physiology, 1998, Oct-15, Volume: 512 ( Pt 2)

    Topics: Adenosine Triphosphate; Animals; Anions; Bicarbonates; Cells, Cultured; Chlorides; Colforsin; Cyclic AMP; Electric Stimulation; Enzyme Inhibitors; Epithelial Cells; Male; Membrane Potentials; Patch-Clamp Techniques; Rats; Rats, Sprague-Dawley; Seminiferous Tubules; Sertoli Cells; Thapsigargin; Thionucleotides

1998
Opposing effects of protein kinase A and C on capacitative calcium entry into HL-60 promyelocytes.
    Biochemical pharmacology, 1998, Sep-01, Volume: 56, Issue:5

    Topics: Calcium; Calcium-Transporting ATPases; Cell Differentiation; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Granulocytes; HL-60 Cells; Humans; Protein Kinase C; Tetradecanoylphorbol Acetate; Thapsigargin

1998
NPY upregulates genes containing cyclic AMP response element in human neuroblastoma cell lines bearing Y1 and Y2 receptors: involvement of CREB.
    Regulatory peptides, 1998, Sep-25, Volume: 75-76

    Topics: Animals; Artificial Gene Fusion; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Humans; Neuroblastoma; Neuropeptide Y; Phosphorylation; Rats; Receptors, Neuropeptide Y; RNA, Messenger; Thapsigargin; Transfection; Tumor Cells, Cultured; Up-Regulation

1998
Post-rest contraction amplitude in myocytes from failing human ventricle.
    Basic research in cardiology, 1998, Volume: 93 Suppl 1

    Topics: Analysis of Variance; Calcium; Cardiac Output, Low; Cardiotonic Agents; Colforsin; Digoxigenin; Drug Evaluation, Preclinical; Heart Ventricles; Humans; In Vitro Techniques; Isoproterenol; Linear Models; Myocardial Contraction; Rest; Thapsigargin

1998
Neurotensin enhances agonist-induced cAMP accumulation in PC3 cells via Ca2+ -dependent adenylyl cyclase(s).
    Molecular and cellular endocrinology, 1998, Sep-25, Volume: 144, Issue:1-2

    Topics: Adenylyl Cyclases; Calcium; Cholera Toxin; Colforsin; Cyclic AMP; Dinoprostone; Drug Synergism; Egtazic Acid; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Humans; Ionomycin; Isoproterenol; Male; Neurotensin; Prostatic Neoplasms; Thapsigargin; Tumor Cells, Cultured; Uridine Triphosphate

1998
Modulation of nicotinic acetylcholine receptor activity in submucous neurons by intracellular messengers.
    Journal of the autonomic nervous system, 1999, Jan-15, Volume: 75, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine Triphosphate; Animals; Colforsin; Enzyme Inhibitors; Genistein; Guinea Pigs; In Vitro Techniques; Intestinal Mucosa; Neurons; Parasympatholytics; Phorbol Esters; Receptors, Nicotinic; Second Messenger Systems; Thapsigargin

1999
Calcium and cAMP are second messengers in the adipokinetic hormone-induced lipolysis of triacylglycerols in Manduca sexta fat body.
    Journal of lipid research, 1999, Volume: 40, Issue:3

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Calcium; Chelating Agents; Cholera Toxin; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Fat Body; Insect Hormones; Ionomycin; Lipolysis; Male; Manduca; Oligopeptides; Pyrrolidonecarboxylic Acid; Second Messenger Systems; Signal Transduction; Thapsigargin; Triglycerides

1999
Leukotriene binding, signaling, and analysis of HIV coreceptor function in mouse and human leukotriene B4 receptor-transfected cells.
    The Journal of biological chemistry, 1999, Mar-26, Volume: 274, Issue:13

    Topics: Animals; Arachidonate 5-Lipoxygenase; Calcium; Cell Line; Cloning, Molecular; Colforsin; Cyclic AMP; GTP-Binding Proteins; Humans; Leukotriene B4; Melanophores; Mice; Protein Binding; Receptors, Chemokine; Receptors, HIV; Receptors, Leukotriene B4; Signal Transduction; Thapsigargin; Transfection

1999
[Intracellular regulation of neuronal nicotinic cholinergic receptors].
    Rossiiskii fiziologicheskii zhurnal imeni I.M. Sechenova, 1998, Volume: 84, Issue:10

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Calcium; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP-Dependent Protein Kinases; Enzyme Activation; In Vitro Techniques; Membrane Potentials; Neurons; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Protein Kinase C; Rats; Receptors, Nicotinic; Superior Cervical Ganglion; Tetradecanoylphorbol Acetate; Thapsigargin

1998
Effect of ceramide on interleukin-6 synthesis in osteoblast-like cells.
    Cellular signalling, 1999, Volume: 11, Issue:6

    Topics: Alprostadil; Animals; Bucladesine; Calcimycin; Cell Line; Cholera Toxin; Colforsin; Dinoprost; Interleukin-1; Interleukin-6; Mice; Osteoblasts; Sphingosine; Tetradecanoylphorbol Acetate; Thapsigargin; Thrombin; Tumor Necrosis Factor-alpha

1999
Transmural pressure inhibits prorenin processing in juxtaglomerular cell.
    The American journal of physiology, 1999, Volume: 277, Issue:1

    Topics: Animals; Caffeine; Calcium Channel Blockers; Cells, Cultured; Colforsin; Enzyme Inhibitors; Enzyme Precursors; Juxtaglomerular Apparatus; Male; Pressure; Rats; Rats, Sprague-Dawley; Renin; Thapsigargin; Verapamil

1999
Serotonin via 5-HT1B and 5-HT2B receptors stimulates anion secretion in the rat epididymal epithelium.
    The Journal of physiology, 1999, Sep-15, Volume: 519 Pt 3

    Topics: Animals; Anions; Chelating Agents; Colforsin; Culture Techniques; Cyclic AMP; Egtazic Acid; Enzyme Inhibitors; Epididymis; Epithelium; Imines; Isoquinolines; Male; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1B; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin; Serotonin; Sulfonamides; Thapsigargin

1999
Effects of forksolin, dibutyryl cAMP and H89 on Ca2+ mobilization in submandibular salivary cells of newborn rats.
    Archives of oral biology, 1999, Volume: 44, Issue:9

    Topics: Acetylcholine; Age Factors; Animals; Animals, Newborn; Bucladesine; Calcium; Calcium Signaling; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Female; Inositol 1,4,5-Trisphosphate; Isoquinolines; Male; Rats; Rats, Sprague-Dawley; Submandibular Gland; Sulfonamides; Thapsigargin

1999
Discriminating between capacitative and arachidonate-activated Ca(2+) entry pathways in HEK293 cells.
    The Journal of biological chemistry, 1999, Oct-29, Volume: 274, Issue:44

    Topics: Adenylyl Cyclases; Arachidonic Acid; Biological Transport; Calcium; Cell Membrane; Colforsin; Models, Biological; Recombinant Proteins; Thapsigargin

1999
Mechanisms underlying spontaneous rhythmical contractions in irideal arterioles of the rat.
    The Journal of physiology, 1999, Dec-01, Volume: 521 Pt 2

    Topics: Adenosine Triphosphate; Age Factors; Animals; Arterioles; Cadmium Chloride; Caffeine; Calcium; Capsaicin; Central Nervous System Stimulants; Colforsin; Cyclic AMP; Dinucleoside Phosphates; Enzyme Inhibitors; Felodipine; Female; Gap Junctions; Iris; Male; Membrane Potentials; Muscle, Smooth, Vascular; Neuropeptide Y; NG-Nitroarginine Methyl Ester; Peptides, Cyclic; Periodicity; Platelet Aggregation Inhibitors; Pyridoxal Phosphate; Rats; Rats, Wistar; Ryanodine; Thapsigargin; Vasoconstriction; Vasodilator Agents

1999
Tumor necrosis factor-alpha-converting enzyme is required for cleavage of erbB4/HER4.
    The Journal of biological chemistry, 2000, Apr-07, Volume: 275, Issue:14

    Topics: 3T3 Cells; ADAM Proteins; ADAM17 Protein; Animals; Clone Cells; Cloning, Molecular; Colforsin; Disintegrins; Drosophila Proteins; ErbB Receptors; Kinetics; Marine Toxins; Metalloendopeptidases; Mice; Mice, Inbred C57BL; Mice, Knockout; Okadaic Acid; Oxazoles; Protein Isoforms; Receptor, ErbB-4; Recombinant Proteins; Substrate Specificity; Tetradecanoylphorbol Acetate; Thapsigargin; Transfection; Tumor Necrosis Factor-alpha; Vanadates

2000
Direct measurement of hormone-induced acidification in intact bone.
    Journal of bone and mineral research : the official journal of the American Society for Bone and Mineral Research, 2000, Volume: 15, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Animals, Newborn; Bone and Bones; Bone Neoplasms; Bucladesine; Calcium Signaling; Carbonic Anhydrases; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Extracellular Space; Humans; Hydrogen-Ion Concentration; Mice; Organ Culture Techniques; Organ Specificity; Osteoblasts; Osteosarcoma; Parathyroid Hormone; Protein Kinase C; Second Messenger Systems; Skull; Tetradecanoylphorbol Acetate; Thapsigargin; Tumor Cells, Cultured

2000
Inhibition of phosphatidylinositol 3-kinase does not alter forskolin-stimulated Cl(-) secretion by T84 cells.
    American journal of physiology. Cell physiology, 2000, Volume: 278, Issue:5

    Topics: Androstadienes; Cell Compartmentation; Cell Line; Cell Membrane; Chlorides; Chromones; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Endocytosis; Enzyme Inhibitors; Epidermal Growth Factor; Humans; Ion Transport; Morpholines; Phosphoinositide-3 Kinase Inhibitors; Thapsigargin; Wortmannin

2000
Ca2+-induced Ca2+ release from the endoplasmic reticulum amplifies the Ca2+ signal mediated by activation of voltage-gated L-type Ca2+ channels in pancreatic beta-cells.
    The Journal of biological chemistry, 2001, Mar-30, Volume: 276, Issue:13

    Topics: Animals; Caffeine; Calcium; Calcium Channels; Colforsin; Cytoplasm; Electrophysiology; Endoplasmic Reticulum; Estrenes; Fura-2; Glucose; Islets of Langerhans; Mice; Mice, Obese; Phosphodiesterase Inhibitors; Potassium Chloride; Pyrrolidinones; Ryanodine Receptor Calcium Release Channel; Signal Transduction; Spectrometry, Fluorescence; Strontium; Thapsigargin; Time Factors; Type C Phospholipases

2001
Modulation of thapsigargin-induced calcium mobilisation by cyclic AMP-elevating agents in human lymphocytes is insensitive to the action of the protein kinase A inhibitor H-89.
    Cellular signalling, 2001, Volume: 13, Issue:6

    Topics: Adenosine Triphosphatases; Bucladesine; Calcium; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cytosol; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Humans; Isoquinolines; Lymphocytes; Microscopy, Fluorescence; Milrinone; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Rolipram; Sulfonamides; Thapsigargin; Time Factors

2001
Nitric oxide inhibition of cAMP synthesis in parotid acini: regulation of type 5/6 adenylyl cyclase.
    Cellular signalling, 2001, Volume: 13, Issue:10

    Topics: Adenylyl Cyclases; Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Isoenzymes; Isoproterenol; Mice; Nitric Oxide; Nitric Oxide Donors; Oxadiazoles; Parotid Gland; Phosphoric Diester Hydrolases; Quinoxalines; Thapsigargin; Triazoles

2001
Residence of adenylyl cyclase type 8 in caveolae is necessary but not sufficient for regulation by capacitative Ca(2+) entry.
    The Journal of biological chemistry, 2002, Feb-22, Volume: 277, Issue:8

    Topics: Adenylyl Cyclases; Calcium; Calcium Channel Blockers; Caveolae; Cell Line; Cholesterol; Colforsin; Cyclic AMP; Humans; Imidazoles; Ionomycin; Kinetics; Mutagenesis; Recombinant Proteins; Sequence Deletion; Thapsigargin; Transfection

2002
Identification of signal transduction pathways and promoter sequences that mediate parathyroid hormone 1-38 inhibition of osteoprotegerin gene expression.
    Journal of cellular biochemistry, 2001, Volume: 84, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Bucladesine; Calcimycin; Colforsin; Gene Expression; Glycoproteins; Osteoblasts; Osteoprotegerin; Parathyroid Hormone; Parathyroid Hormone-Related Protein; Peptide Fragments; Promoter Regions, Genetic; Proteins; Rats; Receptors, Cytoplasmic and Nuclear; Receptors, Tumor Necrosis Factor; Signal Transduction; Tetradecanoylphorbol Acetate; Thapsigargin

2001
Predominant role by CaM kinase in NPY Y(1) receptor signaling: involvement of CREB [corrected].
    Peptides, 2002, Volume: 23, Issue:1

    Topics: Benzylamines; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Dose-Response Relationship, Drug; Enzyme Inhibitors; Genes, Reporter; Humans; Leucine; Luciferases; Peptides; Phosphorylation; Proline; Protein Binding; Proto-Oncogene Proteins c-fos; Receptors, Neuropeptide Y; Signal Transduction; Sulfonamides; Thapsigargin; Time Factors; Transfection; Tumor Cells, Cultured

2002
Stimulation of chloride secretion by baicalein in isolated rat distal colon.
    American journal of physiology. Gastrointestinal and liver physiology, 2002, Volume: 282, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Amiloride; Animals; Atropine; Calcium; Carbachol; Chlorides; Colforsin; Colon; Cyclic AMP; Dinoprostone; Electric Conductivity; Female; Flavanones; Flavonoids; Indomethacin; Intestinal Mucosa; Male; Muscarinic Antagonists; Potassium Channel Blockers; Rats; Rats, Sprague-Dawley; Tetrodotoxin; Thapsigargin

2002
CFTR and lysozyme secretion in human airway epithelial cells.
    Pflugers Archiv : European journal of physiology, 2001, Volume: 443 Suppl 1

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Biological Transport; Cell Line; Chlorides; Colforsin; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Enzyme Inhibitors; Humans; Muramidase; Nitric Oxide Donors; Oligonucleotides, Antisense; Respiratory Mucosa; S-Nitrosoglutathione; Thapsigargin

2001
Mucus secretion from single submucosal glands of pig. Stimulation by carbachol and vasoactive intestinal peptide.
    The Journal of biological chemistry, 2002, Aug-02, Volume: 277, Issue:31

    Topics: Animals; Bumetanide; Carbachol; Cell Membrane; Colforsin; Exocrine Glands; Female; Hydrogen-Ion Concentration; Kinetics; Mucus; Muscle, Smooth; Swine; Thapsigargin; Trachea; Vasoactive Intestinal Peptide

2002
Membrane potential dependent modulations of calcium oscillations in insulin-secreting INS-1 cells.
    Cell calcium, 2002, Volume: 31, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Calcium Signaling; Cell Line; Clonidine; Colforsin; Diazoxide; Enzyme Inhibitors; Epinephrine; Fluorescent Dyes; Fura-2; Glucose; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Membrane Potentials; Mice; Patch-Clamp Techniques; Potassium Channels; Prazosin; Receptors, Adrenergic, alpha-2; Thapsigargin; Tolbutamide

2002
Calcium inhibits ovarian steroidogenesis in the blowfly Phormia regina.
    The Journal of endocrinology, 2002, Volume: 173, Issue:3

    Topics: Animals; Calcimycin; Calcium; Colforsin; Cyclic AMP; Depression, Chemical; Diptera; Ecdysteroids; Enzyme Inhibitors; Female; Ionophores; Organ Culture Techniques; Ovary; Thapsigargin; Vitellogenesis

2002
Phosphorylation of the Ras-GRF1 exchange factor at Ser916/898 reveals activation of Ras signaling in the cerebral cortex.
    The Journal of biological chemistry, 2003, Apr-11, Volume: 278, Issue:15

    Topics: Animals; Binding Sites; Cerebral Cortex; Chlorocebus aethiops; Colforsin; COS Cells; In Vitro Techniques; Peptide Fragments; Phosphopeptides; Phosphorylation; Phosphoserine; Prosencephalon; ras Guanine Nucleotide Exchange Factors; ras-GRF1; Rats; Recombinant Proteins; Serine; Thapsigargin; Transfection

2003
Interferon-gamma stimulates the expression of the inducible cAMP early repressor in macrophages through the activation of casein kinase 2. A potentially novel pathway for interferon-gamma-mediated inhibition of gene transcription.
    The Journal of biological chemistry, 2003, May-16, Volume: 278, Issue:20

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Apigenin; Blotting, Western; Calcimycin; Calcium; Casein Kinase II; Cell Line; Cloning, Molecular; Colforsin; Cyclic AMP; Cyclic AMP Response Element Modulator; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; DNA; DNA-Binding Proteins; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation, Enzymologic; Genetic Vectors; Imidazoles; Indoles; Interferon-gamma; Macrophages; Maleimides; Mice; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Binding; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; Repressor Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Thapsigargin; Time Factors; Transcription, Genetic; Transcriptional Activation; Tyrphostins

2003
Terbutaline-induced triphasic changes in volume of rat alveolar type II cells: the role of cAMP.
    The Japanese journal of physiology, 2002, Volume: 52, Issue:6

    Topics: Adrenergic beta-Agonists; Amiloride; Animals; Calcium; Cell Size; Cells, Cultured; Colforsin; Cyclic AMP; Ionomycin; Male; Microscopy, Video; Potassium Channels; Pulmonary Alveoli; Quinine; Rats; Rats, Wistar; Sodium Channels; Terbutaline; Thapsigargin

2002
Exocytosis of a complement component C3-like protein by tunicate hemocytes.
    Developmental and comparative immunology, 2004, Volume: 28, Issue:3

    Topics: Alkaloids; Animals; Benzophenanthridines; Blotting, Western; Calcimycin; Carrageenan; Cell Survival; Cholera Toxin; Colchicine; Colforsin; Complement C3; Cytochalasin D; Cytoplasmic Vesicles; Enzyme-Linked Immunosorbent Assay; Exocytosis; Hemocytes; Immunohistochemistry; Kinetics; Lipopolysaccharides; Mannans; Microscopy, Electron; Phenanthridines; Staurosporine; Tetradecanoylphorbol Acetate; Thapsigargin; Urochordata

2004
A small molecule CFTR inhibitor produces cystic fibrosis-like submucosal gland fluid secretions in normal airways.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2004, Volume: 18, Issue:7

    Topics: Animals; Benzoates; Body Fluids; Bronchi; Cells, Cultured; Chlorides; Cholinergic Agents; Colforsin; Cyclic AMP; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Exocrine Glands; Humans; Hydrogen-Ion Concentration; Pilocarpine; Second Messenger Systems; Sodium; Swine; Thapsigargin; Thiazoles; Thiazolidines; Viscosity

2004
Changes in the vascular beta-adrenoceptor-activated signalling pathway in 2Kidney-1Clip hypertensive rats.
    British journal of pharmacology, 2004, Volume: 141, Issue:7

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Aorta, Thoracic; Caffeine; Calcium-Transporting ATPases; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Gene Expression; Glyburide; Hypertension, Renovascular; Isoproterenol; Kidney; Male; Membrane Proteins; Muscle, Smooth, Vascular; Phenylephrine; Potassium Channels; Rats; Rats, Wistar; Receptors, Adrenergic, beta; RNA, Messenger; Sarcolemma; Signal Transduction; Thapsigargin; Vasoconstriction; Vasodilation

2004
Post-translational modifications of tubulin and microtubule stability in adult rat ventricular myocytes and immortalized HL-1 cardiomyocytes.
    Molecular and cellular biochemistry, 2004, Volume: 258, Issue:1-2

    Topics: Adrenergic beta-Agonists; Animals; Antineoplastic Agents; Caffeine; Calcium Signaling; Cell Line, Transformed; Cholera Toxin; Colforsin; Cyclic AMP; Enzyme Inhibitors; Heart Ventricles; Isoproterenol; Male; Microtubules; Myocytes, Cardiac; Nocodazole; Phosphodiesterase Inhibitors; Protein Processing, Post-Translational; Rats; Rats, Wistar; Thapsigargin; Tubulin

2004
A "virtual gland" method for quantifying epithelial fluid secretion.
    American journal of physiology. Lung cellular and molecular physiology, 2004, Volume: 287, Issue:4

    Topics: Cell Line; Colforsin; Humans; Kinetics; Models, Biological; Respiratory Mucosa; Thapsigargin; User-Computer Interface

2004
Acid and base secretion in the Calu-3 model of human serous cells.
    American journal of physiology. Lung cellular and molecular physiology, 2004, Volume: 287, Issue:6

    Topics: Acetazolamide; Bicarbonates; Cell Line; Chlorides; Colforsin; Humans; Hydrogen-Ion Concentration; Models, Biological; Potassium Channels; Respiratory Mucosa; Thapsigargin

2004
Effect of carvedilol on Ca2+ movement and cytotoxicity in human MG63 osteosarcoma cells.
    Basic & clinical pharmacology & toxicology, 2004, Volume: 95, Issue:2

    Topics: Adenylyl Cyclases; Calcium; Calcium Channels; Calcium Signaling; Carbazoles; Carvedilol; Cell Compartmentation; Cell Line, Tumor; Cell Proliferation; Cell Survival; Colforsin; Dose-Response Relationship, Drug; Endoplasmic Reticulum; Estrenes; Fluorescence; Fura-2; Histamine; Histamine Antagonists; Humans; Inositol 1,4,5-Trisphosphate; Manganese; Osteosarcoma; Phorbol Esters; Propanolamines; Protein Kinase C; Pyrrolidinones; Tetrazolium Salts; Thapsigargin; Time Factors; Type C Phospholipases

2004
The calcium paradoxon of renin release: calcium suppresses renin exocytosis by inhibition of calcium-dependent adenylate cyclases AC5 and AC6.
    Circulation research, 2006, Nov-24, Volume: 99, Issue:11

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Angiotensin II; Animals; Calcium; Cell Line; Colforsin; Cyclic AMP; Endothelin-1; Enzyme Inhibitors; Exocytosis; In Vitro Techniques; Intracellular Membranes; Isoproterenol; Kidney; Mice; Mice, Inbred C57BL; Renin; RNA, Small Interfering; Thapsigargin

2006
Protein kinase A increases the binding affinity and the Ca2+ release activity of the inositol 1,4,5-trisphosphate receptor type 3 in RINm5F cells.
    Biology of the cell, 2007, Volume: 99, Issue:7

    Topics: Animals; Calcium; Carbachol; Cell Line; Cholinergic Agonists; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Phosphorylation; Rats; RNA, Small Interfering; Thapsigargin

2007
Mechanisms for the coupling of cannabinoid receptors to intracellular calcium mobilization in rat insulinoma beta-cells.
    Experimental cell research, 2007, Aug-15, Volume: 313, Issue:14

    Topics: Animals; Arachidonic Acids; Bombesin; Calcium; Cannabinoids; Capsaicin; Cell Line, Tumor; Colforsin; Dose-Response Relationship, Drug; Dronabinol; Enzyme Inhibitors; Estrenes; Insulinoma; Neuroprotective Agents; Neurotransmitter Agents; Pertussis Toxin; Phosphoinositide Phospholipase C; Pyrrolidinones; Rats; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Sensory System Agents; Signal Transduction; Thapsigargin; TRPV Cation Channels

2007
Separate elements within a single IQ-like motif in adenylyl cyclase type 8 impart ca2+/calmodulin binding and autoinhibition.
    The Journal of biological chemistry, 2009, Jun-05, Volume: 284, Issue:23

    Topics: Adenylyl Cyclases; Amino Acid Substitution; Animals; Cloning, Molecular; Colforsin; Cyclic AMP; DNA Primers; DNA, Complementary; Glutathione Transferase; Kinetics; Models, Molecular; Mutagenesis, Site-Directed; Plasmids; Polymerase Chain Reaction; Protein Conformation; Rats; Recombinant Fusion Proteins; Sequence Deletion; Thapsigargin

2009
Listeriolysin O affects barrier function and induces chloride secretion in HT-29/B6 colon epithelial cells.
    American journal of physiology. Gastrointestinal and liver physiology, 2009, Volume: 296, Issue:6

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Bacterial Toxins; Biological Transport; Calcium Signaling; Cell Survival; Chelating Agents; Chlorides; Colforsin; Egtazic Acid; Electric Impedance; Electrophysiological Phenomena; Epithelial Cells; Heat-Shock Proteins; Hemolysin Proteins; HT29 Cells; Humans; Intestinal Mucosa; L-Lactate Dehydrogenase; Mannitol; Permeability; Protein Kinase Inhibitors; Recombinant Proteins; Sodium; Thapsigargin; Theophylline

2009
An integrated model of electrical spiking, bursting, and calcium oscillations in GnRH neurons.
    Biophysical journal, 2009, Jun-03, Volume: 96, Issue:11

    Topics: Action Potentials; Algorithms; Apamin; Calcium; Colforsin; Cyclic AMP; Enzyme Inhibitors; Gonadotropin-Releasing Hormone; Membrane Potentials; Models, Neurological; Neurons; Neurotoxins; Sodium; Thapsigargin

2009
Glucagon receptor mediates calcium signaling by coupling to G alpha q/11 and G alpha i/o in HEK293 cells.
    Journal of receptor and signal transduction research, 2009, Volume: 29, Issue:6

    Topics: Calcium; Calcium Signaling; Cell Line; Colforsin; Cyclic AMP; Enzyme Inhibitors; Glucagon; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gq-G11; Humans; Pertussis Toxin; Receptors, Glucagon; RNA Interference; Signal Transduction; Thapsigargin

2009
Endoplasmic reticulum stress-induced activation of activating transcription factor 6 decreases cAMP-stimulated hepatic gluconeogenesis via inhibition of CREB.
    Endocrinology, 2010, Volume: 151, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Activating Transcription Factor 6; Animals; Carcinoma, Hepatocellular; Cell Line, Tumor; Colforsin; CREB-Binding Protein; Cyclic AMP; Endoplasmic Reticulum; Gluconeogenesis; Hep G2 Cells; Humans; Liver; Liver Neoplasms; Mice; Rats; RNA Splicing; RNA, Messenger; RNA, Small Interfering; Thapsigargin; Tunicamycin

2010
Chronic regulation of colonic epithelial secretory function by activation of G protein-coupled receptors.
    Neurogastroenterology and motility, 2011, Volume: 23, Issue:2

    Topics: Adenocarcinoma; Calcium; Carbachol; Cell Line, Tumor; Chlorides; Colforsin; Colonic Neoplasms; Epithelial Cells; Histamine; Humans; Patch-Clamp Techniques; Protein Kinase C; Receptor, Muscarinic M3; Receptors, G-Protein-Coupled; Thapsigargin

2011
Adenylate cyclase/cAMP/protein kinase A signaling pathway inhibits endothelin type A receptor-operated Ca²⁺ entry mediated via transient receptor potential canonical 6 channels.
    The Journal of pharmacology and experimental therapeutics, 2012, Volume: 340, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Blotting, Western; Calcium; Calcium Signaling; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; HEK293 Cells; Humans; Microscopy, Confocal; Mutation; Papaverine; Phosphorylation; Protein Kinase Inhibitors; Receptor, Endothelin A; Retroviridae; Signal Transduction; Subcellular Fractions; Thapsigargin; TRPC Cation Channels; TRPC6 Cation Channel

2012
Β-adrenergic receptor stimulation induces endoplasmic reticulum stress in adult cardiac myocytes: role in apoptosis.
    Molecular and cellular biochemistry, 2012, Volume: 364, Issue:1-2

    Topics: Adenylyl Cyclases; Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Animals; Antigens, Differentiation; Apoptosis; Brefeldin A; Caspase 12; Caspase Inhibitors; Cells, Cultured; Cinnamates; Colforsin; eIF-2 Kinase; Endoplasmic Reticulum Stress; Eukaryotic Initiation Factor-2; Gene Expression Regulation; Heat-Shock Proteins; Isoproterenol; Male; Mice; Myocytes, Cardiac; Phosphorylation; Proto-Oncogene Proteins; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Signal Transduction; Thapsigargin; Thiourea; Transcription Factor CHOP

2012
Exendin-4 attenuates high glucose-induced cardiomyocyte apoptosis via inhibition of endoplasmic reticulum stress and activation of SERCA2a.
    American journal of physiology. Cell physiology, 2013, Volume: 304, Issue:6

    Topics: Animals; Apoptosis; Calcium-Binding Proteins; Cells, Cultured; Colforsin; Diabetic Cardiomyopathies; Endoplasmic Reticulum Stress; Enzyme Activation; Exenatide; Glucagon-Like Peptide-1 Receptor; Glucose; Heat-Shock Proteins; HSP70 Heat-Shock Proteins; Hydrogen Peroxide; Hyperglycemia; Hypoglycemic Agents; Isoquinolines; Membrane Proteins; Myocytes, Cardiac; Oxidative Stress; Peptide Fragments; Peptides; Phosphorylation; Protein Kinase Inhibitors; Rats; Receptors, Glucagon; RNA, Messenger; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Sulfonamides; Thapsigargin; Transcription Factor CHOP; Tunicamycin; Unfolded Protein Response; Venoms

2013
GDC-0879, a BRAF
    Cell chemical biology, 2018, 02-15, Volume: 25, Issue:2

    Topics: Cell Death; Colforsin; Humans; Indenes; Kidney Diseases; MAP Kinase Signaling System; Podocytes; Pyrazoles; Signal Transduction; Thapsigargin

2018