Page last updated: 2024-08-23

colforsin and sirolimus

colforsin has been researched along with sirolimus in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's10 (43.48)18.2507
2000's5 (21.74)29.6817
2010's8 (34.78)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cuddon, P; Fleming, A; Floto, RA; Goldsmith, P; Jahreiss, L; O'Kane, CJ; Pask, D; Rubinsztein, DC; Saiki, S; Sarkar, S; Siddiqi, FH; Ttofi, EK; Williams, A1
Auld, DS; Austin, CP; Huang, R; Moeller, TA; Sakamuru, S; Shinn, P; Shukla, SJ; Vanleer, D; Xia, M1
Batista-Gonzalez, A; Brunhofer, G; Fallarero, A; Gopi Mohan, C; Karlsson, D; Shinde, P; Vuorela, P1
Argast, GM; Bornfeldt, KE; Graves, LM; Kong, X; Krebs, EG; Lawrence, JC; Lin, TA1
Bloom, SR; Rozengurt, E; Withers, DJ1
al-Hafidh, J; Belham, CM; Chilvers, ER; Gould, GW; Peacock, AJ; Plevin, R; Scott, PH1
Blenis, J; Monfar, M1
Ballotti, R; Bertolotto, C; Buscà, R; Ortonne, JP1
Earp, HS; Graves, LM; Li, X; Yu, H1
Fertel, R; Rampersaud, AA; Van Brocklyn, JR; Vandenheede, JR; Yates, AJ1
Lawrence, JC; Scott, PH1
DePinho, RA; Eisen, AM; Gallo, V; Ghiani, CA; Knutson, PL; McBain, CJ; Yuan, X1
Coulonval, K; Dumont, JE; Kozma, SC; Lamy, F; Stein, RC; Vandeput, F1
Bach, LA; Leeding, KS; Leng, SL1
Comellas, A; Guerrero, C; Pesce, L; Ridge, KM; Sznajder, JI1
Arita, J; Kawashima, K; Yamakawa, K1
Alier, KA; Morris, BJ1
Anderson, AA; Child, ES; Elphick, LM; Mann, DJ; Prasad, A1
Choi, BS; Ghee, JY; Han, DH; Hwang, HS; Kim, J; Piao, SG; Song, JH; Yang, CW1
Béliveau, È; Guillemette, G; Lapointe, F1
Menon, KM; Palaniappan, M1
Denning, G; Doering, CB; Johnston, JM; Le Doux, JM; Moot, R; Shields, J; Spencer, HT; Whitehead, D1
Baek, D; Ha, Y; Kim, Y; Oh, J1

Other Studies

23 other study(ies) available for colforsin and sirolimus

ArticleYear
Novel targets for Huntington's disease in an mTOR-independent autophagy pathway.
    Nature chemical biology, 2008, Volume: 4, Issue:5

    Topics: Animals; Autophagy; Calcium Channels, L-Type; Clonidine; Cyclic AMP; Humans; Huntington Disease; Imidazoline Receptors; Minoxidil; Protein Kinases; Signal Transduction; TOR Serine-Threonine Kinases; Type C Phospholipases; Verapamil

2008
Identification of clinically used drugs that activate pregnane X receptors.
    Drug metabolism and disposition: the biological fate of chemicals, 2011, Volume: 39, Issue:1

    Topics: Animals; Cell Line, Tumor; Cytochrome P-450 CYP3A; Drug Interactions; Hep G2 Cells; Hepatocytes; Humans; Pharmaceutical Preparations; Pregnane X Receptor; Rats; Receptors, Steroid; Small Molecule Libraries; Species Specificity; Structure-Activity Relationship; Xenobiotics

2011
Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.
    Bioorganic & medicinal chemistry, 2012, Nov-15, Volume: 20, Issue:22

    Topics: Acetylcholinesterase; Amyloid beta-Peptides; Benzophenanthridines; Binding Sites; Butyrylcholinesterase; Catalytic Domain; Cholinesterase Inhibitors; Humans; Isoquinolines; Kinetics; Molecular Docking Simulation; Structure-Activity Relationship

2012
cAMP- and rapamycin-sensitive regulation of the association of eukaryotic initiation factor 4E and the translational regulator PHAS-I in aortic smooth muscle cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1995, Aug-01, Volume: 92, Issue:16

    Topics: 3T3 Cells; Adaptor Proteins, Signal Transducing; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Carrier Proteins; Cell Cycle Proteins; Cells, Cultured; Colforsin; Cyclic AMP; Eukaryotic Initiation Factor-4E; Eukaryotic Initiation Factors; Insulin-Like Growth Factor I; Intracellular Signaling Peptides and Proteins; Mice; Muscle, Smooth, Vascular; Peptide Initiation Factors; Phosphoproteins; Phosphorylation; Platelet-Derived Growth Factor; Polyenes; Protein Serine-Threonine Kinases; Rats; Ribosomal Protein S6 Kinases; Sirolimus

1995
Dissociation of cAMP-stimulated mitogenesis from activation of the mitogen-activated protein kinase cascade in Swiss 3T3 cells.
    The Journal of biological chemistry, 1995, Sep-08, Volume: 270, Issue:36

    Topics: 3T3 Cells; Alprostadil; Amino Acid Sequence; Animals; Colforsin; Cyclic AMP; Enzyme Activation; GTP-Binding Proteins; Immunosuppressive Agents; Mice; Mitogens; Molecular Sequence Data; Polyenes; Protein Kinases; Signal Transduction; Sirolimus; Transfection

1995
A regulatory role for cAMP in phosphatidylinositol 3-kinase/p70 ribosomal S6 kinase-mediated DNA synthesis in platelet-derived-growth-factor-stimulated bovine airway smooth-muscle cells.
    The Biochemical journal, 1996, Sep-15, Volume: 318 ( Pt 3)

    Topics: Androstadienes; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cattle; Cell Division; Cells, Cultured; Colforsin; Cyclic AMP; DNA; Endothelin-1; Enzyme Inhibitors; Muscle, Smooth; Phosphatidylinositol 3-Kinases; Phosphotransferases (Alcohol Group Acceptor); Platelet-Derived Growth Factor; Polyenes; Protein Kinase C; Protein Serine-Threonine Kinases; Ribosomal Protein S6 Kinases; Sirolimus; Trachea; Wortmannin

1996
Inhibition of p70/p85 S6 kinase activities in T cells by dexamethasone.
    Molecular endocrinology (Baltimore, Md.), 1996, Volume: 10, Issue:9

    Topics: 1-Methyl-3-isobutylxanthine; Administration, Topical; Animals; Anti-Inflammatory Agents; Colforsin; Dexamethasone; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glucocorticoids; Interleukin-2; Marine Toxins; Mice; Oxazoles; Phorbol Esters; Phosphatidylinositol 3-Kinases; Phosphorylation; Phosphotransferases (Alcohol Group Acceptor); Polyenes; Protein Kinase C; Protein Serine-Threonine Kinases; Ribosomal Protein S6 Kinases; RNA, Messenger; Sirolimus; T-Lymphocytes; Tacrolimus; Tetradecanoylphorbol Acetate; Transcription, Genetic

1996
Inhibition of the phosphatidylinositol 3-kinase/p70(S6)-kinase pathway induces B16 melanoma cell differentiation.
    The Journal of biological chemistry, 1996, Dec-13, Volume: 271, Issue:50

    Topics: Animals; Cell Differentiation; Chromones; Colforsin; Cyclic AMP; Enzyme Inhibitors; Melanoma, Experimental; Mice; Microscopy, Fluorescence; Monophenol Monooxygenase; Morpholines; Phosphatidylinositol 3-Kinases; Phosphotransferases (Alcohol Group Acceptor); Polyenes; Protein Serine-Threonine Kinases; Ribosomal Protein S6 Kinases; Sirolimus

1996
Protein kinase C and protein kinase A inhibit calcium-dependent but not stress-dependent c-Jun N-terminal kinase activation in rat liver epithelial cells.
    The Journal of biological chemistry, 1997, Jun-06, Volume: 272, Issue:23

    Topics: 1-Methyl-3-isobutylxanthine; Androstadienes; Angiotensin II; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; Epithelial Cells; Epithelium; Humans; JNK Mitogen-Activated Protein Kinases; Kinetics; Liver; Mitogen-Activated Protein Kinases; Models, Biological; Polyenes; Protein Kinases; Rats; Recombinant Proteins; Signal Transduction; Sirolimus; Tetradecanoylphorbol Acetate; Thapsigargin; Wortmannin

1997
Ganglioside GM1 activates the mitogen-activated protein kinase Erk2 and p70 S6 kinase in U-1242 MG human glioma cells.
    Journal of neurochemistry, 1997, Volume: 69, Issue:1

    Topics: Calcium-Calmodulin-Dependent Protein Kinases; Colforsin; Cyclic AMP; DNA; Enzyme Activation; Enzyme Inhibitors; Flavonoids; G(M1) Ganglioside; Glioma; Humans; Immunosuppressive Agents; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase Kinases; Mitogens; Platelet-Derived Growth Factor; Polyenes; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Ribosomal Protein S6 Kinases; Signal Transduction; Sirolimus; Tumor Cells, Cultured

1997
Attenuation of mammalian target of rapamycin activity by increased cAMP in 3T3-L1 adipocytes.
    The Journal of biological chemistry, 1998, Dec-18, Volume: 273, Issue:51

    Topics: 3T3 Cells; Adaptor Proteins, Signal Transducing; Adipocytes; Amino Acid Sequence; Animals; Carrier Proteins; Cell Cycle Proteins; Colforsin; Cyclic AMP; Eukaryotic Initiation Factors; Immunoassay; Insulin; Intracellular Signaling Peptides and Proteins; Mice; Molecular Sequence Data; Peptide Fragments; Peptide Mapping; Phosphoproteins; Phosphorylation; Phosphotransferases (Alcohol Group Acceptor); Protein Kinases; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Rats; Recombinant Proteins; Repressor Proteins; Sequence Alignment; Sequence Homology, Amino Acid; Sirolimus; Theophylline; Thionucleotides; TOR Serine-Threonine Kinases

1998
Voltage-activated K+ channels and membrane depolarization regulate accumulation of the cyclin-dependent kinase inhibitors p27(Kip1) and p21(CIP1) in glial progenitor cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Jul-01, Volume: 19, Issue:13

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cell Cycle Proteins; Cell Division; Cell Lineage; Cerebellum; Colforsin; Cyclin D; Cyclin-Dependent Kinase Inhibitor p21; Cyclin-Dependent Kinase Inhibitor p27; Cyclins; Deferoxamine; Ion Channel Gating; Isoproterenol; Membrane Potentials; Mice; Microtubule-Associated Proteins; Oligodendroglia; Potassium; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Sirolimus; Stem Cells; Tetraethylammonium; Tumor Suppressor Proteins; Veratridine

1999
Phosphatidylinositol 3-kinase, protein kinase B and ribosomal S6 kinases in the stimulation of thyroid epithelial cell proliferation by cAMP and growth factors in the presence of insulin.
    The Biochemical journal, 2000, Jun-01, Volume: 348 Pt 2

    Topics: Androstadienes; Animals; Cell Division; Cells, Cultured; Colforsin; Cyclic AMP; Dogs; Enzyme Inhibitors; Epidermal Growth Factor; Epithelial Cells; Growth Substances; Hepatocyte Growth Factor; Insulin; Kinetics; Phosphatidylinositol 3-Kinases; Phosphatidylinositols; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Ribosomal Protein S6 Kinases; Sirolimus; Tetradecanoylphorbol Acetate; Thyroid Gland; Thyrotropin; Wortmannin

2000
Cyclic AMP agonists increase levels of insulin-like growth factor (IGF) binding protein-6 in PC12 rat phaeochromocytoma cells.
    Growth hormone & IGF research : official journal of the Growth Hormone Research Society and the International IGF Research Society, 1998, Volume: 8, Issue:3

    Topics: Animals; Cell Division; Colforsin; Cyclic AMP; Dexamethasone; Dose-Response Relationship, Drug; Extracellular Matrix; Insulin-Like Growth Factor Binding Protein 6; Insulin-Like Growth Factor II; Neurites; PC12 Cells; Rats; Sirolimus; Thionucleotides

1998
beta-agonists regulate Na,K-ATPase via novel MAPK/ERK and rapamycin-sensitive pathways.
    FEBS letters, 2000, Dec-15, Volume: 486, Issue:3

    Topics: Adrenergic beta-Agonists; Animals; Cell Membrane; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Epithelial Cells; Isoproterenol; Male; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Propranolol; Pulmonary Alveoli; Rats; Rats, Sprague-Dawley; RNA, Messenger; Signal Transduction; Sirolimus; Sodium-Potassium-Exchanging ATPase

2000
Involvement of phosphoinositide-3-kinase and p70 S6 kinase in regulation of proliferation of rat lactotrophs in culture.
    Endocrine, 2000, Volume: 13, Issue:3

    Topics: Adenylyl Cyclases; Androstadienes; Animals; Bromocriptine; Bromodeoxyuridine; Bucladesine; Cell Division; Cells, Cultured; Chromones; Colforsin; Cyclic AMP; Enzyme Activation; Enzyme Inhibitors; Estradiol; Female; Homeostasis; Insulin; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Wistar; Ribosomal Protein S6 Kinases; Sirolimus; Wortmannin

2000
Differential regulation of MAP2 and alphaCamKII expression in hippocampal neurones by forskolin and calcium ionophore treatment.
    Brain research. Molecular brain research, 2004, Mar-17, Volume: 122, Issue:1

    Topics: Animals; Animals, Newborn; Blotting, Western; Calcimycin; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Colforsin; Drug Interactions; Gene Expression Regulation; Hippocampus; Immunohistochemistry; Immunosuppressive Agents; Ionophores; Microtubule-Associated Proteins; Neurons; Rats; Sirolimus

2004
Cyclin D1 and cyclin D3 show divergent responses to distinct mitogenic stimulation.
    Journal of cellular physiology, 2010, Volume: 225, Issue:3

    Topics: Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclin D1; Cyclin D3; Cyclin-Dependent Kinase 4; Enzyme Activation; Enzyme Activators; Fibroblasts; Humans; Intracellular Signaling Peptides and Proteins; Mice; Mitogen-Activated Protein Kinases; Mitogens; Mitosis; Phorbol 12,13-Dibutyrate; Protein Kinase C; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Protein Transport; Signal Transduction; Sirolimus; Swiss 3T3 Cells; Time Factors; TOR Serine-Threonine Kinases; Transfection

2010
Effect of sirolimus on calcineurin inhibitor-induced nephrotoxicity using renal expression of KLOTHO, an antiaging gene.
    Transplantation, 2010, Jul-27, Volume: 90, Issue:2

    Topics: Aging; Animals; Calcineurin Inhibitors; Colforsin; Cyclosporine; DNA Primers; Fibroblast Growth Factor-23; Gene Expression Regulation; Glucuronidase; Immunosuppressive Agents; Kidney; Klotho Proteins; Mice; Nephritis, Interstitial; Oxidative Stress; Reverse Transcriptase Polymerase Chain Reaction; RNA; RNA, Messenger; Sirolimus; Tacrolimus

2010
The activation state of the inositol 1,4,5-trisphosphate receptor regulates the velocity of intracellular Ca2+ waves in bovine aortic endothelial cells.
    Journal of cellular biochemistry, 2011, Volume: 112, Issue:12

    Topics: Adenosine Triphosphate; Animals; Aorta; Calcium; Calcium Signaling; Cattle; Cells, Cultured; Colforsin; Endothelium, Vascular; Inositol 1,4,5-Trisphosphate Receptors; Protein Kinases; Signal Transduction; Sirolimus; Tetradecanoylphorbol Acetate; TOR Serine-Threonine Kinases

2011
Luteinizing hormone/human chorionic gonadotropin-mediated activation of mTORC1 signaling is required for androgen synthesis by theca-interstitial cells.
    Molecular endocrinology (Baltimore, Md.), 2012, Volume: 26, Issue:10

    Topics: Androgens; Androstenedione; Animals; Cells, Cultured; Cholesterol Side-Chain Cleavage Enzyme; Chorionic Gonadotropin; Colforsin; Cyclic AMP Response Element-Binding Protein; Enzyme Induction; Eukaryotic Initiation Factor-4E; Female; Gene Knockdown Techniques; Luteinizing Hormone; Mechanistic Target of Rapamycin Complex 1; Multiprotein Complexes; Phosphoproteins; Phosphorylation; Protein Processing, Post-Translational; Proteins; Rats; Rats, Sprague-Dawley; Ribosomal Protein S6 Kinases; RNA Interference; Signal Transduction; Sirolimus; Steroid 17-alpha-Hydroxylase; Theca Cells; TOR Serine-Threonine Kinases

2012
High-throughput screening identifies compounds that enhance lentiviral transduction.
    Gene therapy, 2014, Volume: 21, Issue:12

    Topics: Animals; Antigens, CD34; Camptothecin; Cell Line, Tumor; Colforsin; Genetic Therapy; Genetic Vectors; Green Fluorescent Proteins; HEK293 Cells; Hematopoietic Stem Cells; High-Throughput Screening Assays; Humans; Lentivirus; Mice; NIH 3T3 Cells; Sirolimus; Tetradecanoylphorbol Acetate; Transduction, Genetic; U937 Cells

2014
Malignant gliomas can be converted to non‑proliferating glial cells by treatment with a combination of small molecules.
    Oncology reports, 2019, Volume: 41, Issue:1

    Topics: 2',3'-Cyclic Nucleotide 3'-Phosphodiesterase; Animals; Antineoplastic Combined Chemotherapy Protocols; Brain Neoplasms; Cell Differentiation; Cell Line, Tumor; Cell Proliferation; Cellular Reprogramming; Colforsin; Drug Therapy, Combination; Gene Expression Profiling; Gene Expression Regulation, Neoplastic; Glial Fibrillary Acidic Protein; Glioma; Heterocyclic Compounds, 4 or More Rings; Humans; Neuroglia; Oligonucleotide Array Sequence Analysis; Rats; Sirolimus; Small Molecule Libraries

2019