colforsin has been researched along with quinpirole in 56 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 8 (14.29) | 18.7374 |
1990's | 28 (50.00) | 18.2507 |
2000's | 16 (28.57) | 29.6817 |
2010's | 4 (7.14) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Hampson, EC; Vaney, DI; Weiler, R | 1 |
Boroni, F; Castelletti, L; Dal Toso, R; Gabellini, N; Missale, C; Sigala, S; Spano, P | 1 |
Nowak, JZ; Schorderet, M; Sek, B | 1 |
Bates, MD; Bunzow, JR; Caron, MG; Civelli, O; Liggett, SB; Senogles, SE | 1 |
De Boer, P; Dolleman-Van der Weel, MJ; Drukarch, B; Schepens, E; Stoof, JC; Van Vliet, BJ | 1 |
Nowak, JZ; Schorderet, M | 1 |
Lam, DM; Pachter, JA | 1 |
Beaulieu, M; Felder, R; Kebabian, JW | 1 |
Bowyer, JF; Weiner, N | 1 |
Ashby, CR; Hitzemann, R; Rubinstein, JE; Wang, RY | 1 |
Olianas, MC; Onali, P | 1 |
Leysen, JE; Stoof, JC; Verheijden, PF | 1 |
Burnside, B; Dearry, A | 1 |
Battaglia, G; Creese, I; Hess, EJ; Norman, AB | 1 |
Chang, JP; van der Kraak, G; Wong, AO | 1 |
Di Marzo, V; Piomelli, D; Schwartz, JC; Sokoloff, P; Vial, D | 1 |
Levavi-Sivan, B; Ofir, M; Yaron, Z | 1 |
Burnside, B; Hillman, DW; Lin, D | 1 |
Duman, RS; Hartigan, DJ; Hayward, MD; Le, HN; Nestler, EJ; Vaccarino, FM | 1 |
Ball, S; Boyfield, I; Coldwell, MC; Cook, T; Gloger, IS; Herrity, N; McHale, M; Robinson, JH; Winn, FM | 1 |
Florijn, WJ; Gispen, WH; Mulder, AH; Versteeg, DH | 1 |
Allard, S; Falardeau, P; Lapointe, S | 1 |
Hoffman, BB; Thomas, JM | 1 |
Felder, RA; Jose, PA; Walk, SF; Yamaguchi, I | 1 |
Harvey, J; Lacey, MG | 1 |
Griffon, N; Pilon, C; Sautel, F; Schwartz, JC; Sokoloff, P | 2 |
Login, IS | 1 |
Caron, MG; Robinson, SW | 1 |
Greengard, P; Nishi, A; Snyder, GL | 1 |
Backlund Höök, B; Hacksell, U; Johansson, AM; Malmberg, A; Mohell, N; Nordvall, G | 1 |
Cumbay, MG; Neve, KA; Neve, RL; Vu, MN; Watts, VJ; Wiens, BL | 1 |
Batchelor, M; Schenk, JO | 1 |
Chen, JC; Hsieh, MM; Huang, LI; Su, HJ | 1 |
Coronas, V; Jourdan, F; Krantic, S; Moyse, E | 1 |
Alberts, GL; Gill, GS; Im, WB; Pregenzer, JF; Slightom, JL; Zaworski, PG | 1 |
Huang, W; Lee, D; Lim, AT | 1 |
Kumar, U; Lange, DC; Patel, RC; Patel, SC; Patel, YC; Rocheville, M | 1 |
Armogida, M; Chiacchio, S; Colzi, A; Corsini, GU; DeMontis, MG; Maggio, R; Scarselli, M | 1 |
Ashby, B; Sakolsky, DJ | 1 |
Fisone, G; Haycock, J; Herrera-Marschitz, M; Hökfelt, T; Lindgren, N; Xu, ZQ | 1 |
Cumbay, MG; Watts, VJ | 1 |
Ahnert-Hilger, G; Faiss, S; Grabowski, P; Hoegerle, S; Höpfner, M; Jockers-Scherübl, M; Lemmer, K; Riecken, EO; Scherübl, H; Zeitz, M | 1 |
Beazely, MA; Johnston, CA; Vancura, AF; Wang, JK; Watts, VJ | 1 |
Boehm, S; Freissmuth, M; Just, H; Klinger, M; Korkhov, VM; Kudlacek, O; Nanoff, C; Pankevych, H; Vartian, N; Yang, Q | 1 |
Fukunaga, K; Takeuchi, Y | 1 |
Ebadi, M; Govitrapong, P; Santanavanich, C | 1 |
Kamiya, T; Nakata, H; Saitoh, O | 1 |
Hablitz, JJ; Wu, J | 1 |
Bastepe, M; Jüppner, H; Nguyen, CH; Vortherms, TA; Watts, VJ | 1 |
Feenstra, RW; Glennon, JC; Hesselink, MB; Long, SK; McCreary, AC; Reinders, JH; Ronken, E; Van Der Neut, M; Van Scharrenburg, G | 1 |
Cummings, DF; Ericksen, SS; Schetz, JA; Weinstein, H | 1 |
Emala, CW; Masaki, E; Mizuta, K; Panettieri, RA; Xu, D; Zhang, Y | 1 |
Berson, DM; Van Hook, MJ; Wong, KY | 1 |
Cao, BB; Huang, Y; Liu, Z; Peng, YP; Qiu, YH; Zhao, W | 1 |
Dillon, GH; Griffin, SA; Huang, R; Luedtke, RR; Mach, RH; Taylor, M; Vangveravong, S | 1 |
1 review(s) available for colforsin and quinpirole
Article | Year |
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Retinal dopamine D1 and D2 receptors: characterization by binding or pharmacological studies and physiological functions.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Arylamine N-Acetyltransferase; Benzazepines; Colforsin; Cyclic AMP; Dopamine; Ergolines; Light; Quinpirole; Receptors, Dopamine; Retina; Second Messenger Systems; Species Specificity; Spiperone; Sulpiride; Vertebrates | 1990 |
55 other study(ies) available for colforsin and quinpirole
Article | Year |
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Dopaminergic modulation of gap junction permeability between amacrine cells in mammalian retina.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Benzazepines; Bicuculline; Cadmium; Cadmium Chloride; Cell Membrane Permeability; Chlorides; Colforsin; Dopamine; Ergolines; Female; Hydrogen-Ion Concentration; In Vitro Techniques; Intercellular Junctions; Male; Quinpirole; Rabbits; Retina; Synapses; Veratridine | 1992 |
Lack of coupling of D-2 receptors to adenylate cyclase in GH-3 cells exposed to epidermal growth factor. Possible role of a differential expression of Gi protein subtypes.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Cell Membrane; Colforsin; Cyclic AMP; DNA; Dopamine; Dopamine Agents; Dopamine Antagonists; Epidermal Growth Factor; Ergolines; GTP-Binding Proteins; Molecular Sequence Data; Neurotensin; Potassium Channels; Prolactin; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Rubidium; Tumor Cells, Cultured; Vasoactive Intestinal Peptide | 1991 |
Bidirectional regulation of cAMP generating system by dopamine-D1 and D2-receptors in the rat retina.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Benzazepines; Colforsin; Cyclic AMP; Ergolines; In Vitro Techniques; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Retina | 1990 |
Regulation of responsiveness at D2 dopamine receptors by receptor desensitization and adenylyl cyclase sensitization.
Topics: Adenylyl Cyclases; Animals; Cell Line; Colforsin; Cyclic AMP; Dopamine; Ergolines; Gene Expression Regulation; Quinpirole; Radioimmunoassay; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Recombinant Proteins | 1991 |
Lack of a dopamine autoreceptor selective profile of B-HT 920 in functional in vitro model systems of D2 receptors in rat striatum.
Topics: Adenylyl Cyclases; Animals; Azepines; Colforsin; Corpus Striatum; Dopamine Agents; Ergolines; Hydroxydopamines; In Vitro Techniques; Male; Neurotransmitter Agents; Oxidopamine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Sympathectomy, Chemical | 1990 |
Interactions between vasoactive intestinal peptide and dopamine in the rabbit retina: stimulation of a common adenylate cyclase.
Topics: Adenylyl Cyclases; Animals; Butaclamol; Chickens; Colforsin; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Metoclopramide; Quinpirole; Rabbits; Receptors, Cell Surface; Receptors, Dopamine; Receptors, Vasoactive Intestinal Peptide; Retina; Sodium Fluoride; Vasoactive Intestinal Peptide | 1986 |
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone | 1986 |
K+ channel and adenylate cyclase involvement in regulation of Ca2+-evoked release of [3H]dopamine from synaptosomes.
Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; Adenylate Cyclase Toxin; Adenylyl Cyclases; Aminopyridines; Animals; Calcium; Colforsin; Dopamine; Ergolines; Ethylmaleimide; In Vitro Techniques; Pertussis Toxin; Potassium Channels; Quinpirole; Rats; Synaptosomes; Tetraethylammonium Compounds; Virulence Factors, Bordetella | 1989 |
One year treatment with haloperidol or clozapine fails to alter neostriatal D1- and D2-dopamine receptor sensitivity in the rat.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Clozapine; Colforsin; Corpus Striatum; Cyclic AMP; Dibenzazepines; Drug Synergism; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2 | 1989 |
Involvement of adenylate cyclase inhibition in dopamine autoreceptor regulation of tyrosine hydroxylase in rat nucleus accumbens.
Topics: Adenylyl Cyclases; Animals; Bucladesine; Colforsin; Ergolines; Male; Nucleus Accumbens; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Septal Nuclei; Sulpiride; Tyrosine 3-Monooxygenase | 1989 |
Stimulation of D2-receptors in rat nucleus accumbens slices inhibits dopamine and acetylcholine release but not cyclic AMP formation.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Benzazepines; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine; Dopamine Antagonists; Ergolines; In Vitro Techniques; Male; Nucleus Accumbens; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Sulpiride | 1987 |
Stimulation of distinct D2 dopaminergic and alpha 2-adrenergic receptors induces light-adaptive pigment dispersion in teleost retinal pigment epithelium.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Clonidine; Colforsin; Dopamine; Ergolines; Fishes; Light; Pigment Epithelium of Eye; Quinpirole; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Dopamine D2; Retinal Pigments | 1988 |
D2 dopamine receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in rat striatum.
Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Butyrophenones; Colforsin; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone | 1985 |
Cyclic 3',5'-adenosine monophosphate mediates dopamine D1-stimulated growth hormone release from goldfish pituitary cells.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dopamine Agonists; Ergolines; Goldfish; Growth Hormone; In Vitro Techniques; Indicators and Reagents; Isoquinolines; Pituitary Gland; Quinpirole; Receptors, Dopamine D1; Sulfonamides | 1994 |
Selection of alternative G-mediated signaling pathways at the dopamine D2 receptor by protein kinase C.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Alkaloids; Animals; Arachidonic Acid; Calcimycin; Calcium; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Diglycerides; Diterpenes; Dopamine D2 Receptor Antagonists; Ergolines; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Kinetics; Protein Kinase C; Quinpirole; Raclopride; Receptors, Dopamine D2; Recombinant Proteins; Salicylamides; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate; Transfection | 1993 |
Possible sites of dopaminergic inhibition of gonadotropin release from the pituitary of a teleost fish, tilapia.
Topics: Animals; Apomorphine; Arachidonic Acid; Bromocriptine; Calcimycin; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Diglycerides; Dopamine; Dopamine Agonists; Ergolines; Gonadotropin-Releasing Hormone; Gonadotropins, Pituitary; Ionomycin; Pituitary Gland; Quinpirole; Signal Transduction; Tilapia | 1995 |
Evidence for D4 receptor regulation of retinomotor movement in isolated teleost cone inner-outer segments.
Topics: Animals; Cell Movement; Colforsin; Darkness; Dopamine; Dopamine Agonists; Dopamine Antagonists; Ergolines; In Vitro Techniques; Light; Perciformes; Quinpirole; Receptors, Dopamine; Retinal Cone Photoreceptor Cells | 1995 |
Induction of immediate early genes by cyclic AMP in primary cultures of neurons from rat cerebral cortex.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Bucladesine; Cells, Cultured; Cerebral Cortex; Colforsin; Cyclic AMP; DNA-Binding Proteins; Dopamine Agents; Early Growth Response Protein 1; Ergolines; Gene Expression Regulation; Genes, fos; Genes, jun; Glutamates; Glutamic Acid; Immediate-Early Proteins; Immunohistochemistry; Kinetics; Neuroglia; Neurons; Quinpirole; Rats; RNA, Messenger; Second Messenger Systems; Transcription Factors; Vasoactive Intestinal Peptide | 1993 |
Expression and functional characterisation of a synthetic version of the human D4 dopamine receptor in a stable human cell line.
Topics: Adenylyl Cyclases; Animals; Base Sequence; Binding, Competitive; Cell Line; Chlorocebus aethiops; Colforsin; DNA; Ergolines; Genes, Synthetic; Humans; Kidney; Kinetics; Molecular Sequence Data; Plasmids; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Restriction Mapping; Spiperone; Transfection | 1994 |
Adrenocorticotropin/alpha-melanocyte-stimulating hormone (ACTH/MSH)-like peptides modulate adenylate cyclase activity in rat brain slices: evidence for an ACTH/MSH receptor-coupled mechanism.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Adrenocorticotropic Hormone; alpha-MSH; Animals; Brain; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Desipramine; Dopamine; Dose-Response Relationship, Drug; Ergolines; In Vitro Techniques; Kinetics; Male; Organ Specificity; Oxidopamine; Quinpirole; Rats; Rats, Wistar; Receptors, Corticotropin; Receptors, Pituitary Hormone; Sulpiride | 1993 |
Specific induction of a functional endogenous D2 short dopamine receptor in GH4C1 cells.
Topics: Animals; Apomorphine; Base Sequence; Colforsin; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Ergolines; Gene Expression; Kanamycin Kinase; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Phosphotransferases; Pituitary Neoplasms; Polymerase Chain Reaction; Potassium Chloride; Prolactin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Sulpiride; Transfection; Tumor Cells, Cultured; Vasoactive Intestinal Peptide | 1993 |
Isoform-specific sensitization of adenylyl cyclase activity by prior activation of inhibitory receptors: role of beta gamma subunits in transducing enhanced activity of the type VI isoform.
Topics: Adenylyl Cyclases; Alprostadil; Carbachol; Cells, Cultured; Chorionic Gonadotropin; Colforsin; Cyclic AMP; Dopamine Agonists; Enzyme Activation; Ergolines; Humans; Isoenzymes; Muscarinic Agonists; Quinpirole; Receptors, Muscarinic; Recombinant Proteins; Signal Transduction; Transducin | 1996 |
Dopamine D2L receptors stimulate Na+/K(+)-ATPase activity in murine LTK- cells.
Topics: Adenylyl Cyclases; Animals; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; Dideoxyadenosine; Dopamine Agonists; Ergolines; Kinetics; L Cells; Mice; Ouabain; Pertussis Toxin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Proteins; Rubidium; Sodium-Potassium-Exchanging ATPase; Spiperone; Transfection; Virulence Factors, Bordetella | 1996 |
Endogenous and exogenous dopamine depress EPSCs in rat nucleus accumbens in vitro via D1 receptors activation.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Amphetamine; Animals; Benzazepines; Cocaine; Colforsin; Dopamine; Dopamine Agonists; Evoked Potentials; In Vitro Techniques; Male; Nucleus Accumbens; Patch-Clamp Techniques; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Synaptic Transmission | 1996 |
Two intracellular signaling pathways for the dopamine D3 receptor: opposite and synergistic interactions with cyclic AMP.
Topics: Cell Line; Colforsin; Cyclic AMP; Dopamine Agonists; Enzyme Inhibitors; Genistein; Humans; Intracellular Membranes; Isoflavones; Mitosis; Protein-Tyrosine Kinases; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Signal Transduction; Time Factors | 1997 |
Antipsychotics with inverse agonist activity at the dopamine D3 receptor.
Topics: Animals; Antipsychotic Agents; Calcium; CHO Cells; Clozapine; Colforsin; Cricetinae; Cyclic AMP; DNA Replication; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Flupenthixol; Glioma; Haloperidol; Humans; Hybrid Cells; Naphthalenes; Neuroblastoma; Pertussis Toxin; Phenothiazines; Pimozide; Pyrrolidines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Proteins; Risperidone; Salicylamides; Second Messenger Systems; Sulpiride; Tetrahydronaphthalenes; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1996 |
D2 dopamine receptor activation inhibits basal and forskolin-evoked acetylcholine release from dissociated striatal cholinergic interneurons.
Topics: Acetylcholine; Adenylyl Cyclases; Animals; Colforsin; Dopamine Agonists; Dopamine Antagonists; In Vitro Techniques; Interneurons; Male; Neostriatum; Neuromuscular Depolarizing Agents; Parasympathetic Nervous System; Piperidines; Quinpirole; Rats; Receptors, Dopamine D2; Salicylamides | 1997 |
Selective inhibition of adenylyl cyclase type V by the dopamine D3 receptor.
Topics: Adenylyl Cyclase Inhibitors; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Dogs; Dopamine Agonists; Drug Interactions; Embryo, Mammalian; Humans; Isoenzymes; Kidney; Quinpirole; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3; Transfection | 1997 |
Bidirectional regulation of DARPP-32 phosphorylation by dopamine.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Antipsychotic Agents; Calcineurin; Calcineurin Inhibitors; Calcium; Chelating Agents; Colforsin; Corpus Striatum; Cyclosporine; Dopamine; Dopamine Agonists; Dopamine and cAMP-Regulated Phosphoprotein 32; Egtazic Acid; Fenoldopam; Male; Mice; Mice, Inbred C57BL; Nerve Tissue Proteins; Neurotoxins; Nucleus Accumbens; Phosphoproteins; Phosphorylation; Protein Processing, Post-Translational; Quinpirole; Raclopride; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate; Salicylamides; Signal Transduction; Tetrodotoxin | 1997 |
Interactions of ligands with active and inactive conformations of the dopamine D2 receptor.
Topics: Cells, Cultured; Cloning, Molecular; Colforsin; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Humans; Ligands; Protein Conformation; Quinpirole; Raclopride; Receptors, Dopamine D2; Salicylamides; Structure-Activity Relationship | 1998 |
Selective activation of Galphao by D2L dopamine receptors in NS20Y neuroblastoma cells.
Topics: Adenylate Cyclase Toxin; Animals; Colforsin; Cyclic AMP; Enzyme Activation; Genetic Vectors; GTP-Binding Proteins; Mice; Neuroblastoma; Neurons; Pertussis Toxin; Quinpirole; Receptors, Dopamine D2; Simplexvirus; Transfection; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1998 |
Protein kinase A activity may kinetically upregulate the striatal transporter for dopamine.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Biological Transport; Carrier Proteins; Colforsin; Corpus Striatum; Cyclic AMP-Dependent Protein Kinases; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Enzyme Activation; Enzyme Inhibitors; Isoquinolines; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Quinpirole; Rats; Rats, Sprague-Dawley; Sulfonamides; Sulpiride; Up-Regulation | 1998 |
Reductions in binding and functions of D2 dopamine receptors in the rat ventral striatum during amphetamine sensitization.
Topics: Adenylyl Cyclases; Amphetamine; Analysis of Variance; Animals; Bromocriptine; Colforsin; Corpus Striatum; Cyclic AMP; Drug Administration Schedule; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Injections, Intraperitoneal; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Stereotyped Behavior; Substance Withdrawal Syndrome; Time Factors | 1999 |
Dopamine receptor coupling to adenylyl cyclase in rat olfactory pathway: a combined pharmacological-radioautographic approach.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Autoradiography; Benzazepines; Bromocriptine; Carbachol; Colforsin; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Enzyme Activation; GTP-Binding Proteins; Guanosine Triphosphate; Male; Muscarinic Agonists; Nitriles; Odorants; Olfactory Bulb; Olfactory Mucosa; Olfactory Pathways; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Signal Transduction | 1999 |
Efficient functional coupling of the human D3 dopamine receptor to G(o) subtype of G proteins in SH-SY5Y cells.
Topics: Adenylyl Cyclases; Binding, Competitive; Calcium Channels; Cell Line; Colforsin; Cyclic AMP; Dopamine Agonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Membrane Potentials; Quinpirole; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Fusion Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA; Sulfur Radioisotopes; Tritium; Tumor Cells, Cultured | 1999 |
Dopamine induces a biphasic modulation of hypothalamic ANF neurons: a ligand concentration-dependent effect involving D5 and D2 receptor interaction.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Antibodies; Atrial Natriuretic Factor; Benzazepines; Biological Transport; Blotting, Northern; Bucladesine; Cells, Cultured; CHO Cells; Colforsin; Cricetinae; Dopamine; Dopamine Agonists; Dopamine Antagonists; Gene Expression; GTP-Binding Proteins; Hypothalamus; In Situ Hybridization; Intercellular Signaling Peptides and Proteins; Ligands; Neurons; Peptides; Phosphodiesterase Inhibitors; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D5; RNA, Messenger; Staining and Labeling; Wasp Venoms | 2000 |
Receptors for dopamine and somatostatin: formation of hetero-oligomers with enhanced functional activity.
Topics: Animals; Cell Membrane; Cerebral Cortex; CHO Cells; Colforsin; Corpus Striatum; Cricetinae; Cyclic AMP; Dimerization; Dopamine D2 Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Heterotrimeric GTP-Binding Proteins; Humans; Ligands; Male; Neurons; Pyramidal Cells; Quinpirole; Rats; Receptor Cross-Talk; Receptors, Dopamine D2; Receptors, Somatostatin; Somatostatin; Spiperone; Sulpiride; Transfection | 2000 |
Reconstitution of functional dopamine D(2s) receptor by co-expression of amino- and carboxyl-terminal receptor fragments.
Topics: Animals; Apomorphine; Binding, Competitive; Clozapine; Colforsin; COS Cells; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Gene Expression; Haloperidol; Membranes; Peptide Fragments; Pergolide; Quinpirole; Radioligand Assay; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Transfection; Tritium | 2000 |
Determination of D1 and D2 dopamine receptor expression by Ntera-2 cells.
Topics: Benzazepines; Colforsin; Cyclic AMP; Dopamine; Dopamine Agonists; Humans; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Teratocarcinoma; Tumor Cells, Cultured | 2000 |
Dopamine D(2) receptors regulate tyrosine hydroxylase activity and phosphorylation at Ser40 in rat striatum.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Colforsin; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Agonists; Male; N-Methylaspartate; Nerve Tissue Proteins; Okadaic Acid; Phosphodiesterase Inhibitors; Phosphoprotein Phosphatases; Phosphorylation; Phosphoserine; Protein Phosphatase 1; Protein Processing, Post-Translational; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Tyrosine 3-Monooxygenase | 2001 |
Heterologous sensitization of recombinant adenylate cyclases by activation of D(2) dopamine receptors.
Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Cell Line; Colforsin; Cyclic AMP; Dopamine Agonists; Enzyme Activation; GTP-Binding Protein alpha Subunits, Gs; Humans; Ionophores; Isoenzymes; Isoproterenol; Kidney; Quinpirole; Receptors, Dopamine D2; Recombinant Proteins; Tetradecanoylphorbol Acetate | 2001 |
Expression of dopamine receptors and transporter in neuroendocrine gastrointestinal tumor cells.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Base Sequence; Biological Transport; Colforsin; Cyclic AMP; DNA Primers; Dopamine; Dopamine Plasma Membrane Transport Proteins; Gastrointestinal Neoplasms; Gene Expression Regulation, Neoplastic; Humans; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Nerve Tissue Proteins; Neuroendocrine Tumors; Pancreatic Neoplasms; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Transcription, Genetic; Tumor Cells, Cultured | 2002 |
Heterologous sensitization of adenylate cyclase is protein kinase A-dependent in Cath.a differentiated (CAD)-D2L cells.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cell Differentiation; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dopamine Agonists; Enzyme Activation; Enzyme Activators; Enzyme Inhibitors; Isoenzymes; Mice; Neurons; Phosphodiesterase Inhibitors; Quinpirole; Receptors, Dopamine D2; RNA, Messenger | 2002 |
The human D2 dopamine receptor synergizes with the A2A adenosine receptor to stimulate adenylyl cyclase in PC12 cells.
Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenine; Adenosine; Adenosine Deaminase; Adenosine Diphosphate; Adenylyl Cyclases; Animals; Benzamides; Binding, Competitive; Cell Cycle; Cell Membrane; Cofilin 1; Colforsin; Cyclic AMP; Cytoskeletal Proteins; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Enzyme Activation; Gene Expression; Glutamic Acid; Humans; Membrane Potentials; Patch-Clamp Techniques; PC12 Cells; Pertussis Toxin; Phenethylamines; Phosphodiesterase Inhibitors; Phosphoproteins; Propionates; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyrrolidines; Quinpirole; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Purinergic P1; Thionucleotides; Transfection; Triazines; Triazoles; Xenopus Proteins | 2003 |
Dopamine D2 receptor activates extracellular signal-regulated kinase through the specific region in the third cytoplasmic loop.
Topics: Animals; Cell Line; Colforsin; Enzyme Activation; Genes, Reporter; Intracellular Space; Mice; Mitogen-Activated Protein Kinases; Neuroblastoma; NF-kappa B; Protein Structure, Tertiary; Quinpirole; Rats; Receptors, Dopamine D2; Response Elements; Sequence Deletion; Structure-Activity Relationship; Transfection | 2004 |
Dopamine receptor activation in bovine pinealocyte via a cAMP-dependent transcription pathway.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acyltransferases; Animals; Benzazepines; Cattle; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Melatonin; Phosphorylation; Pineal Gland; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Spiperone; Transcription, Genetic | 2005 |
Functional expression of single-chain heterodimeric G-protein-coupled receptors for adenosine and dopamine.
Topics: Adenosine; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; Dimerization; Dopamine Agonists; Drug Interactions; Fluorescent Antibody Technique, Indirect; Humans; Ligands; Models, Biological; Phenethylamines; Protein Binding; Purinergic P1 Receptor Agonists; Purinergic P2 Receptor Agonists; Quinpirole; Radioligand Assay; Receptor, Adenosine A2A; Receptors, Dopamine D2; Receptors, Purinergic P1; Receptors, Purinergic P2; Transfection | 2005 |
Cooperative activation of D1 and D2 dopamine receptors enhances a hyperpolarization-activated inward current in layer I interneurons.
Topics: Action Potentials; Animals; Benzazepines; Cations; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dopamine; Dopamine Agonists; Dopamine Antagonists; gamma-Aminobutyric Acid; Interneurons; Ion Transport; Membrane Potentials; Neocortex; Patch-Clamp Techniques; Peptide Fragments; Prefrontal Cortex; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2 | 2005 |
D2 dopamine receptor-induced sensitization of adenylyl cyclase type 1 is G alpha(s) independent.
Topics: Adenylyl Cyclases; Animals; Calcimycin; Calcium; Colforsin; Cyclic AMP; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Activation; GTP-Binding Protein alpha Subunits; Hybrid Cells; Ionophores; Isoproterenol; Mice; Quinpirole; Rabbits; Receptors, Dopamine D2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Transfection; Tritium | 2006 |
In vitro characterization of SLV308 (7-[4-methyl-1-piperazinyl]-2(3H)-benzoxazolone, monohydrochloride): a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist.
Topics: Animals; Benzoxazoles; Binding, Competitive; Brain; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Lisuride; Male; Molecular Structure; Parkinson Disease; Piperazines; Quinpirole; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Fusion Proteins; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists | 2006 |
Ligand selectivity of D2 dopamine receptors is modulated by changes in local dynamics produced by sodium binding.
Topics: Amebicides; Colforsin; Cyclic AMP; Gentamicins; Humans; Kidney; Kinetics; Ligands; Models, Molecular; Mutagenesis, Site-Directed; Protein Conformation; Quinpirole; Radioligand Assay; Receptors, Dopamine D2; Recombinant Proteins; Sodium; Transfection | 2009 |
The dopamine D(2) receptor is expressed and sensitizes adenylyl cyclase activity in airway smooth muscle.
Topics: Adenylyl Cyclases; Animals; Cells, Cultured; Colforsin; Estrenes; Gene Expression; Guinea Pigs; Humans; Inositol Phosphates; Male; Muscle Relaxation; Muscle, Smooth; Myocytes, Smooth Muscle; Primary Cell Culture; Pyrrolidinones; Quinpirole; Receptors, Dopamine D2; Reverse Transcriptase Polymerase Chain Reaction; Trachea; Type C Phospholipases | 2012 |
Dopaminergic modulation of ganglion-cell photoreceptors in rat.
Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Actins; Animals; Carbazoles; Cells, Cultured; Colforsin; Cyclic AMP; Dopamine; Dopamine Agonists; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Gene Expression Regulation; In Vitro Techniques; Light; Light Signal Transduction; Male; Membrane Potentials; Patch-Clamp Techniques; Photic Stimulation; Photoreceptor Cells; Pyrroles; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Retina; Retinal Ganglion Cells; Rod Opsins; Sodium Channel Blockers; Tetrodotoxin; Visual Pathways | 2012 |
Dopamine receptors modulate cytotoxicity of natural killer cells via cAMP-PKA-CREB signaling pathway.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzazepines; Cell Line, Tumor; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Cytotoxicity, Immunologic; Dopamine Agonists; Dopamine Antagonists; Enzyme Activators; Gene Expression; Isoquinolines; Killer Cells, Natural; Mice, Inbred ICR; Phosphorylation; Protein Processing, Post-Translational; Quinpirole; Receptors, Dopamine D3; Receptors, Dopamine D4; Receptors, Dopamine D5; Second Messenger Systems; Sulfonamides | 2013 |
The effect of SV 293, a D2 dopamine receptor-selective antagonist, on D2 receptor-mediated GIRK channel activation and adenylyl cyclase inhibition.
Topics: Adenylyl Cyclase Inhibitors; Animals; Cell Line, Tumor; Colforsin; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Humans; Indoles; Mice; Piperidines; Quinpirole; Receptors, Dopamine D2 | 2013 |