Page last updated: 2024-08-23

colforsin and quinpirole

colforsin has been researched along with quinpirole in 56 studies

Research

Studies (56)

TimeframeStudies, this research(%)All Research%
pre-19908 (14.29)18.7374
1990's28 (50.00)18.2507
2000's16 (28.57)29.6817
2010's4 (7.14)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hampson, EC; Vaney, DI; Weiler, R1
Boroni, F; Castelletti, L; Dal Toso, R; Gabellini, N; Missale, C; Sigala, S; Spano, P1
Nowak, JZ; Schorderet, M; Sek, B1
Bates, MD; Bunzow, JR; Caron, MG; Civelli, O; Liggett, SB; Senogles, SE1
De Boer, P; Dolleman-Van der Weel, MJ; Drukarch, B; Schepens, E; Stoof, JC; Van Vliet, BJ1
Nowak, JZ; Schorderet, M1
Lam, DM; Pachter, JA1
Beaulieu, M; Felder, R; Kebabian, JW1
Bowyer, JF; Weiner, N1
Ashby, CR; Hitzemann, R; Rubinstein, JE; Wang, RY1
Olianas, MC; Onali, P1
Leysen, JE; Stoof, JC; Verheijden, PF1
Burnside, B; Dearry, A1
Battaglia, G; Creese, I; Hess, EJ; Norman, AB1
Chang, JP; van der Kraak, G; Wong, AO1
Di Marzo, V; Piomelli, D; Schwartz, JC; Sokoloff, P; Vial, D1
Levavi-Sivan, B; Ofir, M; Yaron, Z1
Burnside, B; Hillman, DW; Lin, D1
Duman, RS; Hartigan, DJ; Hayward, MD; Le, HN; Nestler, EJ; Vaccarino, FM1
Ball, S; Boyfield, I; Coldwell, MC; Cook, T; Gloger, IS; Herrity, N; McHale, M; Robinson, JH; Winn, FM1
Florijn, WJ; Gispen, WH; Mulder, AH; Versteeg, DH1
Allard, S; Falardeau, P; Lapointe, S1
Hoffman, BB; Thomas, JM1
Felder, RA; Jose, PA; Walk, SF; Yamaguchi, I1
Harvey, J; Lacey, MG1
Griffon, N; Pilon, C; Sautel, F; Schwartz, JC; Sokoloff, P2
Login, IS1
Caron, MG; Robinson, SW1
Greengard, P; Nishi, A; Snyder, GL1
Backlund Höök, B; Hacksell, U; Johansson, AM; Malmberg, A; Mohell, N; Nordvall, G1
Cumbay, MG; Neve, KA; Neve, RL; Vu, MN; Watts, VJ; Wiens, BL1
Batchelor, M; Schenk, JO1
Chen, JC; Hsieh, MM; Huang, LI; Su, HJ1
Coronas, V; Jourdan, F; Krantic, S; Moyse, E1
Alberts, GL; Gill, GS; Im, WB; Pregenzer, JF; Slightom, JL; Zaworski, PG1
Huang, W; Lee, D; Lim, AT1
Kumar, U; Lange, DC; Patel, RC; Patel, SC; Patel, YC; Rocheville, M1
Armogida, M; Chiacchio, S; Colzi, A; Corsini, GU; DeMontis, MG; Maggio, R; Scarselli, M1
Ashby, B; Sakolsky, DJ1
Fisone, G; Haycock, J; Herrera-Marschitz, M; Hökfelt, T; Lindgren, N; Xu, ZQ1
Cumbay, MG; Watts, VJ1
Ahnert-Hilger, G; Faiss, S; Grabowski, P; Hoegerle, S; Höpfner, M; Jockers-Scherübl, M; Lemmer, K; Riecken, EO; Scherübl, H; Zeitz, M1
Beazely, MA; Johnston, CA; Vancura, AF; Wang, JK; Watts, VJ1
Boehm, S; Freissmuth, M; Just, H; Klinger, M; Korkhov, VM; Kudlacek, O; Nanoff, C; Pankevych, H; Vartian, N; Yang, Q1
Fukunaga, K; Takeuchi, Y1
Ebadi, M; Govitrapong, P; Santanavanich, C1
Kamiya, T; Nakata, H; Saitoh, O1
Hablitz, JJ; Wu, J1
Bastepe, M; Jüppner, H; Nguyen, CH; Vortherms, TA; Watts, VJ1
Feenstra, RW; Glennon, JC; Hesselink, MB; Long, SK; McCreary, AC; Reinders, JH; Ronken, E; Van Der Neut, M; Van Scharrenburg, G1
Cummings, DF; Ericksen, SS; Schetz, JA; Weinstein, H1
Emala, CW; Masaki, E; Mizuta, K; Panettieri, RA; Xu, D; Zhang, Y1
Berson, DM; Van Hook, MJ; Wong, KY1
Cao, BB; Huang, Y; Liu, Z; Peng, YP; Qiu, YH; Zhao, W1
Dillon, GH; Griffin, SA; Huang, R; Luedtke, RR; Mach, RH; Taylor, M; Vangveravong, S1

Reviews

1 review(s) available for colforsin and quinpirole

ArticleYear
Retinal dopamine D1 and D2 receptors: characterization by binding or pharmacological studies and physiological functions.
    Cellular and molecular neurobiology, 1990, Volume: 10, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Arylamine N-Acetyltransferase; Benzazepines; Colforsin; Cyclic AMP; Dopamine; Ergolines; Light; Quinpirole; Receptors, Dopamine; Retina; Second Messenger Systems; Species Specificity; Spiperone; Sulpiride; Vertebrates

1990

Other Studies

55 other study(ies) available for colforsin and quinpirole

ArticleYear
Dopaminergic modulation of gap junction permeability between amacrine cells in mammalian retina.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1992, Volume: 12, Issue:12

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Amphetamine; Animals; Benzazepines; Bicuculline; Cadmium; Cadmium Chloride; Cell Membrane Permeability; Chlorides; Colforsin; Dopamine; Ergolines; Female; Hydrogen-Ion Concentration; In Vitro Techniques; Intercellular Junctions; Male; Quinpirole; Rabbits; Retina; Synapses; Veratridine

1992
Lack of coupling of D-2 receptors to adenylate cyclase in GH-3 cells exposed to epidermal growth factor. Possible role of a differential expression of Gi protein subtypes.
    The Journal of biological chemistry, 1991, Dec-05, Volume: 266, Issue:34

    Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Base Sequence; Cell Membrane; Colforsin; Cyclic AMP; DNA; Dopamine; Dopamine Agents; Dopamine Antagonists; Epidermal Growth Factor; Ergolines; GTP-Binding Proteins; Molecular Sequence Data; Neurotensin; Potassium Channels; Prolactin; Quinpirole; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Rubidium; Tumor Cells, Cultured; Vasoactive Intestinal Peptide

1991
Bidirectional regulation of cAMP generating system by dopamine-D1 and D2-receptors in the rat retina.
    Journal of neural transmission. General section, 1990, Volume: 81, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Benzazepines; Colforsin; Cyclic AMP; Ergolines; In Vitro Techniques; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Retina

1990
Regulation of responsiveness at D2 dopamine receptors by receptor desensitization and adenylyl cyclase sensitization.
    Molecular pharmacology, 1991, Volume: 39, Issue:1

    Topics: Adenylyl Cyclases; Animals; Cell Line; Colforsin; Cyclic AMP; Dopamine; Ergolines; Gene Expression Regulation; Quinpirole; Radioimmunoassay; Rats; Receptors, Dopamine; Receptors, Dopamine D2; Recombinant Proteins

1991
Lack of a dopamine autoreceptor selective profile of B-HT 920 in functional in vitro model systems of D2 receptors in rat striatum.
    European journal of pharmacology, 1990, Oct-09, Volume: 187, Issue:2

    Topics: Adenylyl Cyclases; Animals; Azepines; Colforsin; Corpus Striatum; Dopamine Agents; Ergolines; Hydroxydopamines; In Vitro Techniques; Male; Neurotransmitter Agents; Oxidopamine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stereoisomerism; Sympathectomy, Chemical

1990
Interactions between vasoactive intestinal peptide and dopamine in the rabbit retina: stimulation of a common adenylate cyclase.
    Journal of neurochemistry, 1986, Volume: 46, Issue:1

    Topics: Adenylyl Cyclases; Animals; Butaclamol; Chickens; Colforsin; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Metoclopramide; Quinpirole; Rabbits; Receptors, Cell Surface; Receptors, Dopamine; Receptors, Vasoactive Intestinal Peptide; Retina; Sodium Fluoride; Vasoactive Intestinal Peptide

1986
D-2 dopaminergic agonists and adenosine 3',5'-monophosphate directly regulate the synthesis of alpha-melanocyte-stimulating hormone-like peptides by cultured rat melanotrophs.
    Endocrinology, 1986, Volume: 118, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Benzamides; Benzazepines; Bromocriptine; Cells, Cultured; Chemical Precipitation; Cholera Toxin; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Dopamine; Ergolines; Immunologic Techniques; Melanocyte-Stimulating Hormones; Pituitary Gland; Pro-Opiomelanocortin; Quinpirole; Rats; Receptors, Dopamine; Spiperone

1986
K+ channel and adenylate cyclase involvement in regulation of Ca2+-evoked release of [3H]dopamine from synaptosomes.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; Adenylate Cyclase Toxin; Adenylyl Cyclases; Aminopyridines; Animals; Calcium; Colforsin; Dopamine; Ergolines; Ethylmaleimide; In Vitro Techniques; Pertussis Toxin; Potassium Channels; Quinpirole; Rats; Synaptosomes; Tetraethylammonium Compounds; Virulence Factors, Bordetella

1989
One year treatment with haloperidol or clozapine fails to alter neostriatal D1- and D2-dopamine receptor sensitivity in the rat.
    Brain research, 1989, Jul-24, Volume: 493, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Antipsychotic Agents; Benzazepines; Clozapine; Colforsin; Corpus Striatum; Cyclic AMP; Dibenzazepines; Drug Synergism; Ergolines; Haloperidol; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2

1989
Involvement of adenylate cyclase inhibition in dopamine autoreceptor regulation of tyrosine hydroxylase in rat nucleus accumbens.
    Neuroscience letters, 1989, Jul-17, Volume: 102, Issue:1

    Topics: Adenylyl Cyclases; Animals; Bucladesine; Colforsin; Ergolines; Male; Nucleus Accumbens; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Septal Nuclei; Sulpiride; Tyrosine 3-Monooxygenase

1989
Stimulation of D2-receptors in rat nucleus accumbens slices inhibits dopamine and acetylcholine release but not cyclic AMP formation.
    Brain research, 1987, Oct-13, Volume: 423, Issue:1-2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Benzazepines; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine; Dopamine Antagonists; Ergolines; In Vitro Techniques; Male; Nucleus Accumbens; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Septal Nuclei; Sulpiride

1987
Stimulation of distinct D2 dopaminergic and alpha 2-adrenergic receptors induces light-adaptive pigment dispersion in teleost retinal pigment epithelium.
    Journal of neurochemistry, 1988, Volume: 51, Issue:5

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Clonidine; Colforsin; Dopamine; Ergolines; Fishes; Light; Pigment Epithelium of Eye; Quinpirole; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Dopamine D2; Retinal Pigments

1988
D2 dopamine receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in rat striatum.
    Neuroscience letters, 1985, Aug-30, Volume: 59, Issue:2

    Topics: Adenylyl Cyclases; Animals; Benzazepines; Bromocriptine; Butyrophenones; Colforsin; Corpus Striatum; Ergolines; In Vitro Techniques; Male; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Dopamine D2; Spiperone

1985
Cyclic 3',5'-adenosine monophosphate mediates dopamine D1-stimulated growth hormone release from goldfish pituitary cells.
    Neuroendocrinology, 1994, Volume: 60, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dopamine Agonists; Ergolines; Goldfish; Growth Hormone; In Vitro Techniques; Indicators and Reagents; Isoquinolines; Pituitary Gland; Quinpirole; Receptors, Dopamine D1; Sulfonamides

1994
Selection of alternative G-mediated signaling pathways at the dopamine D2 receptor by protein kinase C.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1993, Volume: 13, Issue:11

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Alkaloids; Animals; Arachidonic Acid; Calcimycin; Calcium; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Diglycerides; Diterpenes; Dopamine D2 Receptor Antagonists; Ergolines; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Kinetics; Protein Kinase C; Quinpirole; Raclopride; Receptors, Dopamine D2; Recombinant Proteins; Salicylamides; Signal Transduction; Staurosporine; Tetradecanoylphorbol Acetate; Transfection

1993
Possible sites of dopaminergic inhibition of gonadotropin release from the pituitary of a teleost fish, tilapia.
    Molecular and cellular endocrinology, 1995, Volume: 109, Issue:1

    Topics: Animals; Apomorphine; Arachidonic Acid; Bromocriptine; Calcimycin; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Diglycerides; Dopamine; Dopamine Agonists; Ergolines; Gonadotropin-Releasing Hormone; Gonadotropins, Pituitary; Ionomycin; Pituitary Gland; Quinpirole; Signal Transduction; Tilapia

1995
Evidence for D4 receptor regulation of retinomotor movement in isolated teleost cone inner-outer segments.
    Journal of neurochemistry, 1995, Volume: 64, Issue:3

    Topics: Animals; Cell Movement; Colforsin; Darkness; Dopamine; Dopamine Agonists; Dopamine Antagonists; Ergolines; In Vitro Techniques; Light; Perciformes; Quinpirole; Receptors, Dopamine; Retinal Cone Photoreceptor Cells

1995
Induction of immediate early genes by cyclic AMP in primary cultures of neurons from rat cerebral cortex.
    Brain research. Molecular brain research, 1993, Volume: 19, Issue:1-2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Animals, Newborn; Bucladesine; Cells, Cultured; Cerebral Cortex; Colforsin; Cyclic AMP; DNA-Binding Proteins; Dopamine Agents; Early Growth Response Protein 1; Ergolines; Gene Expression Regulation; Genes, fos; Genes, jun; Glutamates; Glutamic Acid; Immediate-Early Proteins; Immunohistochemistry; Kinetics; Neuroglia; Neurons; Quinpirole; Rats; RNA, Messenger; Second Messenger Systems; Transcription Factors; Vasoactive Intestinal Peptide

1993
Expression and functional characterisation of a synthetic version of the human D4 dopamine receptor in a stable human cell line.
    FEBS letters, 1994, May-30, Volume: 345, Issue:2-3

    Topics: Adenylyl Cyclases; Animals; Base Sequence; Binding, Competitive; Cell Line; Chlorocebus aethiops; Colforsin; DNA; Ergolines; Genes, Synthetic; Humans; Kidney; Kinetics; Molecular Sequence Data; Plasmids; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D2; Receptors, Dopamine D4; Restriction Mapping; Spiperone; Transfection

1994
Adrenocorticotropin/alpha-melanocyte-stimulating hormone (ACTH/MSH)-like peptides modulate adenylate cyclase activity in rat brain slices: evidence for an ACTH/MSH receptor-coupled mechanism.
    Journal of neurochemistry, 1993, Volume: 60, Issue:6

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 3,4-Dihydroxyphenylacetic Acid; Adenylyl Cyclases; Adrenocorticotropic Hormone; alpha-MSH; Animals; Brain; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Desipramine; Dopamine; Dose-Response Relationship, Drug; Ergolines; In Vitro Techniques; Kinetics; Male; Organ Specificity; Oxidopamine; Quinpirole; Rats; Rats, Wistar; Receptors, Corticotropin; Receptors, Pituitary Hormone; Sulpiride

1993
Specific induction of a functional endogenous D2 short dopamine receptor in GH4C1 cells.
    Biochemical and biophysical research communications, 1993, Jun-15, Volume: 193, Issue:2

    Topics: Animals; Apomorphine; Base Sequence; Colforsin; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Ergolines; Gene Expression; Kanamycin Kinase; Kinetics; Molecular Sequence Data; Oligodeoxyribonucleotides; Phosphotransferases; Pituitary Neoplasms; Polymerase Chain Reaction; Potassium Chloride; Prolactin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Sulpiride; Transfection; Tumor Cells, Cultured; Vasoactive Intestinal Peptide

1993
Isoform-specific sensitization of adenylyl cyclase activity by prior activation of inhibitory receptors: role of beta gamma subunits in transducing enhanced activity of the type VI isoform.
    Molecular pharmacology, 1996, Volume: 49, Issue:5

    Topics: Adenylyl Cyclases; Alprostadil; Carbachol; Cells, Cultured; Chorionic Gonadotropin; Colforsin; Cyclic AMP; Dopamine Agonists; Enzyme Activation; Ergolines; Humans; Isoenzymes; Muscarinic Agonists; Quinpirole; Receptors, Muscarinic; Recombinant Proteins; Signal Transduction; Transducin

1996
Dopamine D2L receptors stimulate Na+/K(+)-ATPase activity in murine LTK- cells.
    Molecular pharmacology, 1996, Volume: 49, Issue:2

    Topics: Adenylyl Cyclases; Animals; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; Dideoxyadenosine; Dopamine Agonists; Ergolines; Kinetics; L Cells; Mice; Ouabain; Pertussis Toxin; Quinpirole; Rats; Receptors, Dopamine D2; Recombinant Proteins; Rubidium; Sodium-Potassium-Exchanging ATPase; Spiperone; Transfection; Virulence Factors, Bordetella

1996
Endogenous and exogenous dopamine depress EPSCs in rat nucleus accumbens in vitro via D1 receptors activation.
    The Journal of physiology, 1996, Apr-01, Volume: 492 ( Pt 1)

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Amphetamine; Animals; Benzazepines; Cocaine; Colforsin; Dopamine; Dopamine Agonists; Evoked Potentials; In Vitro Techniques; Male; Nucleus Accumbens; Patch-Clamp Techniques; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Synaptic Transmission

1996
Two intracellular signaling pathways for the dopamine D3 receptor: opposite and synergistic interactions with cyclic AMP.
    Journal of neurochemistry, 1997, Volume: 68, Issue:1

    Topics: Cell Line; Colforsin; Cyclic AMP; Dopamine Agonists; Enzyme Inhibitors; Genistein; Humans; Intracellular Membranes; Isoflavones; Mitosis; Protein-Tyrosine Kinases; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Signal Transduction; Time Factors

1997
Antipsychotics with inverse agonist activity at the dopamine D3 receptor.
    Journal of neural transmission (Vienna, Austria : 1996), 1996, Volume: 103, Issue:10

    Topics: Animals; Antipsychotic Agents; Calcium; CHO Cells; Clozapine; Colforsin; Cricetinae; Cyclic AMP; DNA Replication; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Flupenthixol; Glioma; Haloperidol; Humans; Hybrid Cells; Naphthalenes; Neuroblastoma; Pertussis Toxin; Phenothiazines; Pimozide; Pyrrolidines; Quinpirole; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Proteins; Risperidone; Salicylamides; Second Messenger Systems; Sulpiride; Tetrahydronaphthalenes; Tumor Cells, Cultured; Virulence Factors, Bordetella

1996
D2 dopamine receptor activation inhibits basal and forskolin-evoked acetylcholine release from dissociated striatal cholinergic interneurons.
    Brain research, 1997, Feb-21, Volume: 749, Issue:1

    Topics: Acetylcholine; Adenylyl Cyclases; Animals; Colforsin; Dopamine Agonists; Dopamine Antagonists; In Vitro Techniques; Interneurons; Male; Neostriatum; Neuromuscular Depolarizing Agents; Parasympathetic Nervous System; Piperidines; Quinpirole; Rats; Receptors, Dopamine D2; Salicylamides

1997
Selective inhibition of adenylyl cyclase type V by the dopamine D3 receptor.
    Molecular pharmacology, 1997, Volume: 52, Issue:3

    Topics: Adenylyl Cyclase Inhibitors; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Dogs; Dopamine Agonists; Drug Interactions; Embryo, Mammalian; Humans; Isoenzymes; Kidney; Quinpirole; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3; Transfection

1997
Bidirectional regulation of DARPP-32 phosphorylation by dopamine.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Nov-01, Volume: 17, Issue:21

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Antipsychotic Agents; Calcineurin; Calcineurin Inhibitors; Calcium; Chelating Agents; Colforsin; Corpus Striatum; Cyclosporine; Dopamine; Dopamine Agonists; Dopamine and cAMP-Regulated Phosphoprotein 32; Egtazic Acid; Fenoldopam; Male; Mice; Mice, Inbred C57BL; Nerve Tissue Proteins; Neurotoxins; Nucleus Accumbens; Phosphoproteins; Phosphorylation; Protein Processing, Post-Translational; Quinpirole; Raclopride; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, N-Methyl-D-Aspartate; Salicylamides; Signal Transduction; Tetrodotoxin

1997
Interactions of ligands with active and inactive conformations of the dopamine D2 receptor.
    European journal of pharmacology, 1998, Apr-10, Volume: 346, Issue:2-3

    Topics: Cells, Cultured; Cloning, Molecular; Colforsin; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Humans; Ligands; Protein Conformation; Quinpirole; Raclopride; Receptors, Dopamine D2; Salicylamides; Structure-Activity Relationship

1998
Selective activation of Galphao by D2L dopamine receptors in NS20Y neuroblastoma cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Nov-01, Volume: 18, Issue:21

    Topics: Adenylate Cyclase Toxin; Animals; Colforsin; Cyclic AMP; Enzyme Activation; Genetic Vectors; GTP-Binding Proteins; Mice; Neuroblastoma; Neurons; Pertussis Toxin; Quinpirole; Receptors, Dopamine D2; Simplexvirus; Transfection; Tumor Cells, Cultured; Virulence Factors, Bordetella

1998
Protein kinase A activity may kinetically upregulate the striatal transporter for dopamine.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1998, Dec-15, Volume: 18, Issue:24

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Biological Transport; Carrier Proteins; Colforsin; Corpus Striatum; Cyclic AMP-Dependent Protein Kinases; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Enzyme Activation; Enzyme Inhibitors; Isoquinolines; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Quinpirole; Rats; Rats, Sprague-Dawley; Sulfonamides; Sulpiride; Up-Regulation

1998
Reductions in binding and functions of D2 dopamine receptors in the rat ventral striatum during amphetamine sensitization.
    Life sciences, 1999, Volume: 64, Issue:5

    Topics: Adenylyl Cyclases; Amphetamine; Analysis of Variance; Animals; Bromocriptine; Colforsin; Corpus Striatum; Cyclic AMP; Drug Administration Schedule; GTP-Binding Proteins; Guanylyl Imidodiphosphate; Injections, Intraperitoneal; Male; Motor Activity; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Stereotyped Behavior; Substance Withdrawal Syndrome; Time Factors

1999
Dopamine receptor coupling to adenylyl cyclase in rat olfactory pathway: a combined pharmacological-radioautographic approach.
    Neuroscience, 1999, Volume: 90, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Autoradiography; Benzazepines; Bromocriptine; Carbachol; Colforsin; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Antagonists; Enzyme Activation; GTP-Binding Proteins; Guanosine Triphosphate; Male; Muscarinic Agonists; Nitriles; Odorants; Olfactory Bulb; Olfactory Mucosa; Olfactory Pathways; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Signal Transduction

1999
Efficient functional coupling of the human D3 dopamine receptor to G(o) subtype of G proteins in SH-SY5Y cells.
    British journal of pharmacology, 1999, Volume: 128, Issue:6

    Topics: Adenylyl Cyclases; Binding, Competitive; Calcium Channels; Cell Line; Colforsin; Cyclic AMP; Dopamine Agonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Membrane Potentials; Quinpirole; Radioligand Assay; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Fusion Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA; Sulfur Radioisotopes; Tritium; Tumor Cells, Cultured

1999
Dopamine induces a biphasic modulation of hypothalamic ANF neurons: a ligand concentration-dependent effect involving D5 and D2 receptor interaction.
    Molecular psychiatry, 2000, Volume: 5, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Antibodies; Atrial Natriuretic Factor; Benzazepines; Biological Transport; Blotting, Northern; Bucladesine; Cells, Cultured; CHO Cells; Colforsin; Cricetinae; Dopamine; Dopamine Agonists; Dopamine Antagonists; Gene Expression; GTP-Binding Proteins; Hypothalamus; In Situ Hybridization; Intercellular Signaling Peptides and Proteins; Ligands; Neurons; Peptides; Phosphodiesterase Inhibitors; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Dopamine D5; RNA, Messenger; Staining and Labeling; Wasp Venoms

2000
Receptors for dopamine and somatostatin: formation of hetero-oligomers with enhanced functional activity.
    Science (New York, N.Y.), 2000, Apr-07, Volume: 288, Issue:5463

    Topics: Animals; Cell Membrane; Cerebral Cortex; CHO Cells; Colforsin; Corpus Striatum; Cricetinae; Cyclic AMP; Dimerization; Dopamine D2 Receptor Antagonists; Guanosine 5'-O-(3-Thiotriphosphate); Heterotrimeric GTP-Binding Proteins; Humans; Ligands; Male; Neurons; Pyramidal Cells; Quinpirole; Rats; Receptor Cross-Talk; Receptors, Dopamine D2; Receptors, Somatostatin; Somatostatin; Spiperone; Sulpiride; Transfection

2000
Reconstitution of functional dopamine D(2s) receptor by co-expression of amino- and carboxyl-terminal receptor fragments.
    European journal of pharmacology, 2000, Jun-02, Volume: 397, Issue:2-3

    Topics: Animals; Apomorphine; Binding, Competitive; Clozapine; Colforsin; COS Cells; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Gene Expression; Haloperidol; Membranes; Peptide Fragments; Pergolide; Quinpirole; Radioligand Assay; Rats; Receptors, Dopamine D2; Recombinant Fusion Proteins; Spiperone; Transfection; Tritium

2000
Determination of D1 and D2 dopamine receptor expression by Ntera-2 cells.
    Brain research. Molecular brain research, 2000, Dec-08, Volume: 84, Issue:1-2

    Topics: Benzazepines; Colforsin; Cyclic AMP; Dopamine; Dopamine Agonists; Humans; Quinpirole; Receptors, Dopamine D1; Receptors, Dopamine D2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Teratocarcinoma; Tumor Cells, Cultured

2000
Dopamine D(2) receptors regulate tyrosine hydroxylase activity and phosphorylation at Ser40 in rat striatum.
    The European journal of neuroscience, 2001, Volume: 13, Issue:4

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Colforsin; Corpus Striatum; Dihydroxyphenylalanine; Dopamine; Dopamine Agonists; Male; N-Methylaspartate; Nerve Tissue Proteins; Okadaic Acid; Phosphodiesterase Inhibitors; Phosphoprotein Phosphatases; Phosphorylation; Phosphoserine; Protein Phosphatase 1; Protein Processing, Post-Translational; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D2; Tyrosine 3-Monooxygenase

2001
Heterologous sensitization of recombinant adenylate cyclases by activation of D(2) dopamine receptors.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 297, Issue:3

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Cell Line; Colforsin; Cyclic AMP; Dopamine Agonists; Enzyme Activation; GTP-Binding Protein alpha Subunits, Gs; Humans; Ionophores; Isoenzymes; Isoproterenol; Kidney; Quinpirole; Receptors, Dopamine D2; Recombinant Proteins; Tetradecanoylphorbol Acetate

2001
Expression of dopamine receptors and transporter in neuroendocrine gastrointestinal tumor cells.
    Life sciences, 2002, Jun-28, Volume: 71, Issue:6

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Base Sequence; Biological Transport; Colforsin; Cyclic AMP; DNA Primers; Dopamine; Dopamine Plasma Membrane Transport Proteins; Gastrointestinal Neoplasms; Gene Expression Regulation, Neoplastic; Humans; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Nerve Tissue Proteins; Neuroendocrine Tumors; Pancreatic Neoplasms; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Transcription, Genetic; Tumor Cells, Cultured

2002
Heterologous sensitization of adenylate cyclase is protein kinase A-dependent in Cath.a differentiated (CAD)-D2L cells.
    Journal of neurochemistry, 2002, Volume: 82, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cell Differentiation; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dopamine Agonists; Enzyme Activation; Enzyme Activators; Enzyme Inhibitors; Isoenzymes; Mice; Neurons; Phosphodiesterase Inhibitors; Quinpirole; Receptors, Dopamine D2; RNA, Messenger

2002
The human D2 dopamine receptor synergizes with the A2A adenosine receptor to stimulate adenylyl cyclase in PC12 cells.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2003, Volume: 28, Issue:7

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenine; Adenosine; Adenosine Deaminase; Adenosine Diphosphate; Adenylyl Cyclases; Animals; Benzamides; Binding, Competitive; Cell Cycle; Cell Membrane; Cofilin 1; Colforsin; Cyclic AMP; Cytoskeletal Proteins; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Enzyme Activation; Gene Expression; Glutamic Acid; Humans; Membrane Potentials; Patch-Clamp Techniques; PC12 Cells; Pertussis Toxin; Phenethylamines; Phosphodiesterase Inhibitors; Phosphoproteins; Propionates; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Pyrrolidines; Quinpirole; Radioligand Assay; Rats; Receptors, Dopamine D2; Receptors, Purinergic P1; Thionucleotides; Transfection; Triazines; Triazoles; Xenopus Proteins

2003
Dopamine D2 receptor activates extracellular signal-regulated kinase through the specific region in the third cytoplasmic loop.
    Journal of neurochemistry, 2004, Volume: 89, Issue:6

    Topics: Animals; Cell Line; Colforsin; Enzyme Activation; Genes, Reporter; Intracellular Space; Mice; Mitogen-Activated Protein Kinases; Neuroblastoma; NF-kappa B; Protein Structure, Tertiary; Quinpirole; Rats; Receptors, Dopamine D2; Response Elements; Sequence Deletion; Structure-Activity Relationship; Transfection

2004
Dopamine receptor activation in bovine pinealocyte via a cAMP-dependent transcription pathway.
    Journal of pineal research, 2005, Volume: 38, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acyltransferases; Animals; Benzazepines; Cattle; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Melatonin; Phosphorylation; Pineal Gland; Quinpirole; Receptors, Dopamine; Receptors, Dopamine D1; Receptors, Dopamine D2; RNA, Messenger; Spiperone; Transcription, Genetic

2005
Functional expression of single-chain heterodimeric G-protein-coupled receptors for adenosine and dopamine.
    Cell structure and function, 2005, Volume: 29, Issue:5-6

    Topics: Adenosine; Cell Line; Cell Membrane; Colforsin; Cyclic AMP; Dimerization; Dopamine Agonists; Drug Interactions; Fluorescent Antibody Technique, Indirect; Humans; Ligands; Models, Biological; Phenethylamines; Protein Binding; Purinergic P1 Receptor Agonists; Purinergic P2 Receptor Agonists; Quinpirole; Radioligand Assay; Receptor, Adenosine A2A; Receptors, Dopamine D2; Receptors, Purinergic P1; Receptors, Purinergic P2; Transfection

2005
Cooperative activation of D1 and D2 dopamine receptors enhances a hyperpolarization-activated inward current in layer I interneurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Jul-06, Volume: 25, Issue:27

    Topics: Action Potentials; Animals; Benzazepines; Cations; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dopamine; Dopamine Agonists; Dopamine Antagonists; gamma-Aminobutyric Acid; Interneurons; Ion Transport; Membrane Potentials; Neocortex; Patch-Clamp Techniques; Peptide Fragments; Prefrontal Cortex; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2

2005
D2 dopamine receptor-induced sensitization of adenylyl cyclase type 1 is G alpha(s) independent.
    Neuropharmacology, 2006, Volume: 50, Issue:5

    Topics: Adenylyl Cyclases; Animals; Calcimycin; Calcium; Colforsin; Cyclic AMP; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Activation; GTP-Binding Protein alpha Subunits; Hybrid Cells; Ionophores; Isoproterenol; Mice; Quinpirole; Rabbits; Receptors, Dopamine D2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Transfection; Tritium

2006
In vitro characterization of SLV308 (7-[4-methyl-1-piperazinyl]-2(3H)-benzoxazolone, monohydrochloride): a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist.
    Synapse (New York, N.Y.), 2006, Dec-15, Volume: 60, Issue:8

    Topics: Animals; Benzoxazoles; Binding, Competitive; Brain; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Lisuride; Male; Molecular Structure; Parkinson Disease; Piperazines; Quinpirole; Radioligand Assay; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine D2; Receptors, Dopamine D3; Recombinant Fusion Proteins; Serotonin 5-HT1 Receptor Agonists; Serotonin Receptor Agonists

2006
Ligand selectivity of D2 dopamine receptors is modulated by changes in local dynamics produced by sodium binding.
    The Journal of pharmacology and experimental therapeutics, 2009, Volume: 328, Issue:1

    Topics: Amebicides; Colforsin; Cyclic AMP; Gentamicins; Humans; Kidney; Kinetics; Ligands; Models, Molecular; Mutagenesis, Site-Directed; Protein Conformation; Quinpirole; Radioligand Assay; Receptors, Dopamine D2; Recombinant Proteins; Sodium; Transfection

2009
The dopamine D(2) receptor is expressed and sensitizes adenylyl cyclase activity in airway smooth muscle.
    American journal of physiology. Lung cellular and molecular physiology, 2012, Feb-01, Volume: 302, Issue:3

    Topics: Adenylyl Cyclases; Animals; Cells, Cultured; Colforsin; Estrenes; Gene Expression; Guinea Pigs; Humans; Inositol Phosphates; Male; Muscle Relaxation; Muscle, Smooth; Myocytes, Smooth Muscle; Primary Cell Culture; Pyrrolidinones; Quinpirole; Receptors, Dopamine D2; Reverse Transcriptase Polymerase Chain Reaction; Trachea; Type C Phospholipases

2012
Dopaminergic modulation of ganglion-cell photoreceptors in rat.
    The European journal of neuroscience, 2012, Volume: 35, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Actins; Animals; Carbazoles; Cells, Cultured; Colforsin; Cyclic AMP; Dopamine; Dopamine Agonists; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Gene Expression Regulation; In Vitro Techniques; Light; Light Signal Transduction; Male; Membrane Potentials; Patch-Clamp Techniques; Photic Stimulation; Photoreceptor Cells; Pyrroles; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Retina; Retinal Ganglion Cells; Rod Opsins; Sodium Channel Blockers; Tetrodotoxin; Visual Pathways

2012
Dopamine receptors modulate cytotoxicity of natural killer cells via cAMP-PKA-CREB signaling pathway.
    PloS one, 2013, Volume: 8, Issue:6

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adenylyl Cyclases; Animals; Benzazepines; Cell Line, Tumor; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Cytotoxicity, Immunologic; Dopamine Agonists; Dopamine Antagonists; Enzyme Activators; Gene Expression; Isoquinolines; Killer Cells, Natural; Mice, Inbred ICR; Phosphorylation; Protein Processing, Post-Translational; Quinpirole; Receptors, Dopamine D3; Receptors, Dopamine D4; Receptors, Dopamine D5; Second Messenger Systems; Sulfonamides

2013
The effect of SV 293, a D2 dopamine receptor-selective antagonist, on D2 receptor-mediated GIRK channel activation and adenylyl cyclase inhibition.
    Pharmacology, 2013, Volume: 92, Issue:1-2

    Topics: Adenylyl Cyclase Inhibitors; Animals; Cell Line, Tumor; Colforsin; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; G Protein-Coupled Inwardly-Rectifying Potassium Channels; Humans; Indoles; Mice; Piperidines; Quinpirole; Receptors, Dopamine D2

2013