Page last updated: 2024-08-23

colforsin and prazosin

colforsin has been researched along with prazosin in 64 studies

Research

Studies (64)

TimeframeStudies, this research(%)All Research%
pre-199017 (26.56)18.7374
1990's35 (54.69)18.2507
2000's9 (14.06)29.6817
2010's3 (4.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Azuma, H; Oshima, H; Tsujii, T; Yamaguchi, T1
Schachter, JB; Wolfe, BB1
Bradley, ME; Buxton, IL; Keef, KD; Zhang, L1
Chan, CB; MacPhail, RM1
Haimo, LT; Thaler, CD1
Atkinson, BN; Minneman, KP1
Mori-Okamoto, J; Namii, Y; Tatsuno, J1
Cannon, B; Herron, D; Néchad, M; Nedergaard, J; Rehnmark, S1
Felder, CC; Kanterman, RY; McCune, SK; Voigt, MM1
Berger, HJ; Pfeifer, A; Rupp, H; Werdan, K1
Hescheler, J; Wallukat, G; Wobus, AM1
Bylund, DB; Halenda, SP; Jones, SB1
Andriantsitohaina, R; Stoclet, JC1
Medgett, IC; Rajanayagam, MA; Rand, MJ1
Alari, L; Axelsson, KL; Persson, ML; Post, C; Uhlén, S; Wikberg, JE1
Baudysová, M; Houstĕk, J; Kopecký, J; Pavelka, S1
Corda, D; Kohn, LD1
Costa, E; Eva, C; Fabrazzo, M1
Arkinstall, SJ; Jones, CT1
Etgen, AM; Petitti, N1
Filburn, CR; Guggino, S; Kumagai, H; Sacktor, B; Sakamoto, H1
Larsen, PR; Raasmaja, A1
Lim, AT; Vale, W; Widmaier, EP1
Insel, PA; Maisel, AS; Motulsky, HJ; Ziegler, MG1
Connolly, E; Nedergaard, J1
Hashimoto, K; Kato, K; Tsujimoto, A; Tsujimoto, G1
Uhlén, S; Wikberg, JE1
Andersson, RG; Elwing, H; Grundström, N; Karlsson, JO1
Larsen, PR; Lemack, G; Mills, I; Moolten, N; Raasmaja, A; Silva, JE1
Fredholm, BB; Larsson, O1
Colucci, WS1
Flaim, SF; Gleason, MM1
Kendall, DA; Wilson, VG; Wright, IK1
Arilla, E; López-Sañudo, S1
Bogoyevitch, MA; Fuller, SJ; Sugden, PH1
Harling, R; Kendall, DA; Wilson, VG; Wright, IK1
Ahlström, M; Lamberg-Allardt, C; Törnquist, K1
Bruggemann, EP; Cardarelli, C; Gottesman, MM; Greenberger, LM; Morris, DI; Pastan, I; Seamon, KB1
Ernsberger, P; Furin, J; Liedtke, CM1
Ehara, T; Hirahara, K; Iyadomi, I1
Delton-Vandenbroucke, I; Gharib, A; Lagarde, M; Molière, P; Sarda, N1
Hernández, ML; Martínez, MJ; Ochoa, B; Ruiz, JI1
Osnes, JB; Skomedal, T; Viko, H1
Aikawa, R; Hiroi, Y; Komuro, I; Kudoh, S; Mizuno, T; Shiojima, I; Takano, H; Yamazaki, T; Yazaki, Y; Zou, Y1
Andersson, RG; Moartensson, LG1
Bond, M; McConnell, BK; Morano, I; Moravec, CS1
Altschuld, R; Bogdanov, KY; Cheng, H; Hohl, C; Lakatta, EG; Xiao, RP; Zhou, YY1
Allen, LF; Fatima, S; Kan, H; Malik, KU; Parmentier, JH; Ruan, Y1
Soares-da-Silva, P; Vieira-Coelho, MA1
Gerhardt, CC; Gros, J; Issad, T; Strosberg, AD1
Bobirnac, I; Gazi, L; Loetscher, E; Parsley, S; Schoeffter, P1
Adya, HV; Faisal, M; Mallick, BN1
Kaloyianni, M; Papaefthimiou, I; Simeonidou, V1
Gutierrez, A; Kornfeld, M; Persson, AE; Salomonsson, M1
Sugimoto, M; Uchida-Oka, N1
Alarcón, P; García-Sancho, J; Núñez, L1
Greger, R; Herbst, M; Hescheler, J; Sasse, P; Ullrich, S; Yu, H1
Chakir, K; Crow, MT; Jo, SH; Lakatta, EG; Leblais, V; Maltsev, V; Wang, W; Xiao, RP; Zheng, M1
Cox, CL; Govindaiah, G1
Centurión, D; Gupta, S; Mehrotra, S; Saxena, PR; VandenBrink, AM; Villalón, CM1
Bossard, F; Gauthier, C; Lavazais-Blancou, E; Robay, A; Rozec, B; Sagan, C; Silantieff, E1
Amodeo, FS; Brummett, CM; Hong, EK; Janda, AM; Lydic, R1

Other Studies

64 other study(ies) available for colforsin and prazosin

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
A possible role of decreased relaxation mediated by beta-adrenoceptors in bladder outlet obstruction by benign prostatic hyperplasia.
    British journal of pharmacology, 1992, Volume: 107, Issue:3

    Topics: Adult; Aged; Aged, 80 and over; Colforsin; Dihydroalprenolol; Humans; In Vitro Techniques; Isometric Contraction; Isoproterenol; Kinetics; Male; Membranes; Middle Aged; Muscle Relaxation; Potassium Chloride; Prazosin; Propranolol; Prostatic Hyperplasia; Radioligand Assay; Receptors, Adrenergic, beta; Urinary Bladder Neck Obstruction

1992
Cyclic AMP differentiates two separate but interacting pathways of phosphoinositide hydrolysis in the DDT1-MF2 smooth muscle cell line.
    Molecular pharmacology, 1992, Volume: 41, Issue:3

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Alkylating Agents; Cell Line; Colforsin; Cyclic AMP; Hydrolysis; Muscle, Smooth; Norepinephrine; Pertussis Toxin; Phosphatidylinositols; Prazosin; Propranolol; Protein Kinase Inhibitors; Receptors, Adrenergic, alpha; Receptors, Purinergic; Virulence Factors, Bordetella

1992
Action of alpha 2A-adrenergic receptors in circular smooth muscle of canine proximal colon.
    The American journal of physiology, 1992, Volume: 262, Issue:3 Pt 1

    Topics: Adenylate Cyclase Toxin; Animals; Binding, Competitive; Cell Membrane; Clonidine; Colforsin; Colon; Dogs; Epinephrine; Female; In Vitro Techniques; Isoproterenol; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Oxymetazoline; Pertussis Toxin; Prazosin; Receptors, Adrenergic, alpha; Tetrodotoxin; Virulence Factors, Bordetella; Yohimbine

1992
Functional characterization of alpha-adrenoceptors on pancreatic islets of fa/fa Zucker rats.
    Molecular and cellular endocrinology, 1992, Volume: 84, Issue:1-2

    Topics: Animals; Cells, Cultured; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Epinephrine; Female; Glucose; Insulin; Islets of Langerhans; Obesity; Prazosin; Rats; Rats, Zucker; Receptors, Adrenergic, alpha; Yohimbine

1992
Control of organelle transport in melanophores: regulation of Ca2+ and cAMP levels.
    Cell motility and the cytoskeleton, 1992, Volume: 22, Issue:3

    Topics: Animals; Biological Transport; Calcium; Cell Movement; Colforsin; Cyclic AMP; Egtazic Acid; Epinephrine; Fishes; Melanophores; Models, Biological; Organelles; Prazosin; Second Messenger Systems

1992
Multiple adrenergic receptor subtypes controlling cyclic AMP formation: comparison of brain slices and primary neuronal and glial cultures.
    Journal of neurochemistry, 1991, Volume: 56, Issue:2

    Topics: Adrenergic alpha-Agonists; Aging; Animals; Animals, Newborn; Cells, Cultured; Cerebral Cortex; Colforsin; Cyclic AMP; Drug Synergism; Isoproterenol; Kinetics; Neuroglia; Neurons; Norepinephrine; Phentolamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine

1991
Subtypes of adrenergic receptors and intracellular mechanisms involved in modulatory effects of noradrenaline on glutamate.
    Brain research, 1991, Jan-18, Volume: 539, Issue:1

    Topics: Acebutolol; Albuterol; Animals; Cells, Cultured; Cerebellum; Chick Embryo; Clonidine; Colforsin; Electric Conductivity; Ethanolamines; Glutamates; Glutamic Acid; Isoproterenol; Membrane Potentials; Neurons; Norepinephrine; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tolazoline; Yohimbine

1991
Alpha- and beta-adrenergic induction of the expression of the uncoupling protein thermogenin in brown adipocytes differentiated in culture.
    The Journal of biological chemistry, 1990, Sep-25, Volume: 265, Issue:27

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adipose Tissue, Brown; Adrenergic beta-Antagonists; Animals; Blotting, Northern; Carrier Proteins; Cells, Cultured; Colforsin; Gene Expression; Insulin; Ion Channels; Male; Membrane Proteins; Mice; Mitochondrial Proteins; Norepinephrine; Nucleic Acid Hybridization; Oxymetazoline; Phenylephrine; Prazosin; Propanolamines; Propranolol; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; RNA; RNA, Messenger; Thyroxine; Triiodothyronine; Uncoupling Protein 1

1990
The rat alpha 2-C4 adrenergic receptor gene encodes a novel pharmacological subtype.
    FEBS letters, 1991, Jan-14, Volume: 278, Issue:1

    Topics: Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Blotting, Northern; Colforsin; Cyclic AMP; Dioxanes; DNA; Gene Expression; Humans; Molecular Sequence Data; Prazosin; Radioligand Assay; Rats; Receptors, Adrenergic, alpha; RNA; Sequence Homology, Nucleic Acid; Transfection; Yohimbine

1991
Effect of positive inotropic agents on myosin isozyme population and mechanical activity of cultured rat heart myocytes.
    Circulation research, 1991, Volume: 68, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Animals, Newborn; Bucladesine; Cardiotonic Agents; Cells, Cultured; Colforsin; Heart; Isoenzymes; Isoproterenol; Myocardial Contraction; Myocardium; Myosins; Ouabain; Phenylephrine; Prazosin; Propranolol; Rats

1991
Pluripotent mouse embryonic stem cells are able to differentiate into cardiomyocytes expressing chronotropic responses to adrenergic and cholinergic agents and Ca2+ channel blockers.
    Differentiation; research in biological diversity, 1991, Volume: 48, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Animals, Newborn; Atropine; Calcium Channel Blockers; Carbachol; Cell Differentiation; Cell Line; Colforsin; Dose-Response Relationship, Drug; Embryo, Mammalian; Embryo, Nonmammalian; Heart; Heart Rate; Isoproterenol; Membrane Potentials; Myocardium; Parasympathomimetics; Phenylephrine; Prazosin; Stem Cells; Sympathomimetics

1991
Alpha 2-adrenergic receptor stimulation of phospholipase A2 and of adenylate cyclase in transfected Chinese hamster ovary cells is mediated by different mechanisms.
    Molecular pharmacology, 1991, Volume: 39, Issue:2

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Enzyme Activation; Female; Kinetics; Membranes; Ovary; Pertussis Toxin; Phospholipases A; Phospholipases A2; Prazosin; Quinacrine; Receptors, Adrenergic, alpha; Signal Transduction; Stimulation, Chemical; Time Factors; Transfection; Tritium; Virulence Factors, Bordetella; Yohimbine

1991
Enhancement by neuropeptide Y (NPY) of the dihydropyridine-sensitive component of the response to alpha 1-adrenoceptor stimulation in rat isolated mesenteric arterioles.
    British journal of pharmacology, 1990, Volume: 99, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Arterioles; Calcium Channel Blockers; Colforsin; Dihydropyridines; Diltiazem; Female; In Vitro Techniques; Mesenteric Arteries; Muscle, Smooth, Vascular; Neuropeptide Y; Nitroprusside; Norepinephrine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains

1990
Vasoconstrictor responses of rat tail artery to sympathetic nerve stimulation contain a component due to activation of postjunctional beta- or alpha 2-adrenoceptors.
    European journal of pharmacology, 1990, Feb-20, Volume: 177, Issue:1-2

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Calcium; Colforsin; Dioxanes; Electric Stimulation; Idazoxan; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Neurotransmitter Agents; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Regional Blood Flow; Sympathetic Nervous System; Tail; Vasoconstriction

1990
Antinociceptive actions of alpha 2-adrenoceptor agonists in the rat spinal cord: evidence for antinociceptive alpha 2-adrenoceptor subtypes and dissociation of antinociceptive alpha 2-adrenoceptors from cyclic AMP.
    Journal of neurochemistry, 1990, Volume: 55, Issue:6

    Topics: Adrenergic alpha-Agonists; Animals; Benzylamines; Brimonidine Tartrate; Colforsin; Cyclic AMP; Guanfacine; Male; Neurotoxins; Nociceptors; Pain Measurement; Prazosin; Quinoxalines; Rats; Rats, Inbred Strains; Spinal Cord; Yohimbine

1990
Induction of type II iodothyronine 5'-deiodinase and mitochondrial uncoupling protein in brown adipocytes differentiated in cell culture.
    FEBS letters, 1990, Nov-12, Volume: 274, Issue:1-2

    Topics: Adipose Tissue, Brown; Animals; Bucladesine; Carrier Proteins; Cells, Cultured; Colforsin; Cycloheximide; Dactinomycin; Enzyme Induction; Iodide Peroxidase; Ion Channels; Isoproterenol; Kinetics; Membrane Proteins; Mice; Mice, Inbred BALB C; Mitochondria; Mitochondrial Proteins; Norepinephrine; Phenylephrine; Prazosin; Propranolol; Uncoupling Protein 1

1990
Thyrotropin upregulates alpha 1-adrenergic receptors in rat FRTL-5 thyroid cells.
    Proceedings of the National Academy of Sciences of the United States of America, 1985, Volume: 82, Issue:24

    Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cell Line; Cholera Toxin; Colforsin; Cyclic AMP; Cycloheximide; Dactinomycin; Norepinephrine; Prazosin; Rats; Receptors, Adrenergic, alpha; Thyroid Gland; Thyrotropin

1985
Changes of cholinergic, noradrenergic and serotonergic synaptic transmission indices elicited by ethylcholine aziridinium ion (AF64A) infused intraventricularly.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 241, Issue:1

    Topics: Acetylcholine; Animals; Aziridines; Azirines; Binding Sites; Choline; Colforsin; Cyclic AMP; Hippocampus; Hydroxyindoleacetic Acid; Injections, Intraventricular; Norepinephrine; Prazosin; Rats; Rats, Inbred Strains; Serotonin; Synaptic Transmission

1987
Myometrial alpha 1-adrenoceptors in pregnant guinea pig: their distribution and increased number.
    The American journal of physiology, 1989, Volume: 256, Issue:2 Pt 1

    Topics: Animals; Colforsin; Female; Guinea Pigs; Kinetics; Myometrium; Organ Specificity; Prazosin; Pregnancy; Pregnancy, Animal; Receptors, Adrenergic, alpha; Reference Values; Uterus

1989
Progesterone depression of norepinephrine-stimulated cAMP accumulation in hypothalamic slices.
    Brain research. Molecular brain research, 1989, Volume: 5, Issue:2

    Topics: Animals; Colforsin; Cyclic AMP; Estradiol; Female; Hypothalamus; In Vitro Techniques; Norepinephrine; Phosphoric Diester Hydrolases; Prazosin; Preoptic Area; Progesterone; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vasoactive Intestinal Peptide; Yohimbine

1989
Neurotransmitter regulation of cytosolic calcium in osteoblast-like bone cells.
    Calcified tissue international, 1989, Volume: 45, Issue:4

    Topics: Adenosine Triphosphate; Animals; Calcium; Colforsin; Cyclic AMP; Cytosol; Inositol Phosphates; Norepinephrine; Osteoblasts; Parathyroid Hormone; Prazosin; Propranolol; Rats; Tumor Cells, Cultured; Vasoactive Intestinal Peptide

1989
Alpha 1- and beta-adrenergic agents cause synergistic stimulation of the iodothyronine deiodinase in rat brown adipocytes.
    Endocrinology, 1989, Volume: 125, Issue:5

    Topics: Adipose Tissue, Brown; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Alprenolol; Animals; Bucladesine; Cells, Cultured; Colforsin; Cyclic AMP; Drug Synergism; Enzyme Activation; Imidazoles; Iodide Peroxidase; Isoproterenol; Male; Norepinephrine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Yohimbine

1989
Secretion of corticotropin-releasing factor from cultured rat hypothalamic cells: effects of catecholamines.
    Endocrinology, 1989, Volume: 124, Issue:2

    Topics: Animals; Animals, Newborn; Cells, Cultured; Colforsin; Corticotropin-Releasing Hormone; Hypothalamus; Isoproterenol; Norepinephrine; Phenylephrine; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate

1989
Ischemia- and agonist-induced changes in alpha- and beta-adrenergic receptor traffic in guinea pig hearts.
    The American journal of physiology, 1987, Volume: 253, Issue:5 Pt 2

    Topics: Animals; Colforsin; Epinephrine; Guanylyl Imidodiphosphate; Guinea Pigs; Iodocyanopindolol; Male; Microscopy, Electron; Myocardium; Pindolol; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1987
Beta-adrenergic modulation of Ca2+ uptake by isolated brown adipocytes. Possible involvement of mitochondria.
    The Journal of biological chemistry, 1988, Aug-05, Volume: 263, Issue:22

    Topics: Adipose Tissue, Brown; Animals; Biological Transport, Active; Calcium; Colforsin; Cricetinae; Cyclic AMP; Egtazic Acid; In Vitro Techniques; Kinetics; Male; Membrane Potentials; Mesocricetus; Mitochondria; Norepinephrine; Palmitic Acids; Prazosin; Receptors, Adrenergic, beta; Theophylline

1988
In vivo desensitization of glycogenolysis to Ca2+-mobilizing hormones in rat liver cells.
    The Journal of clinical investigation, 1988, Volume: 82, Issue:6

    Topics: Adrenal Gland Neoplasms; Angiotensin II; Animals; Arginine Vasopressin; Bucladesine; Calcimycin; Calcium; Colforsin; Glucagon; Hormones; Liver Glycogen; Male; Norepinephrine; Phenoxybenzamine; Phenylephrine; Pheochromocytoma; Phosphorylases; Prazosin; Rats; Receptors, Adrenergic, alpha; Second Messenger Systems

1988
Inhibition of cyclic AMP production by alpha 2-adrenoceptor stimulation in the guinea-pig spinal cord slices.
    Pharmacology & toxicology, 1988, Volume: 63, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Brimonidine Tartrate; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Male; Prazosin; Quinoxalines; Spinal Cord; Yohimbine

1988
Pigment migration in fish erythrophores is controlled by alpha 2-adrenoceptors.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1988, Volume: 91, Issue:2

    Topics: Animals; Chromatophores; Colforsin; Electric Stimulation; Fishes; Norepinephrine; Phentolamine; Prazosin; Receptors, Adrenergic, alpha; Yohimbine

1988
Effect of thyroid status on catecholamine stimulation of thyroxine 5'-deiodinase in brown adipocytes.
    The American journal of physiology, 1989, Volume: 256, Issue:1 Pt 1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adipose Tissue, Brown; Alprenolol; Animals; Catecholamines; Colforsin; Cycloheximide; Dactinomycin; Drug Synergism; Enzyme Activation; Hypothyroidism; Iodide Peroxidase; Isoproterenol; Kinetics; Male; Norepinephrine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains

1989
Carbachol stimulation of inositol phosphate accumulation in rat submandibular gland fragments is not modified by VIP.
    Acta physiologica Scandinavica, 1989, Volume: 135, Issue:3

    Topics: Animals; Atropine; Carbachol; Colforsin; Inositol Phosphates; Male; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Submandibular Gland; Sugar Phosphates; Vasoactive Intestinal Peptide

1989
Adenosine 3',5'-cyclic-monophosphate-dependent regulation of alpha 1-adrenergic receptor number in rabbit aortic smooth muscle cells.
    Circulation research, 1986, Volume: 58, Issue:2

    Topics: Adenylyl Cyclases; Alprostadil; Animals; Aorta; Calcium; Colforsin; Cyclic AMP; Muscle, Smooth, Vascular; Norepinephrine; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Tritium

1986
Phorbol ester contracts rabbit thoracic aorta by increasing intracellular calcium and by activating calcium influx.
    Biochemical and biophysical research communications, 1986, Aug-14, Volume: 138, Issue:3

    Topics: Animals; Biological Transport; Calcium; Colforsin; Cytoplasm; Extracellular Space; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Phorbol 12,13-Dibutyrate; Phorbol Esters; Prazosin; Protein Kinase C; Rabbits; Time Factors

1986
Alpha 2-adrenoceptor mediated inhibition of forskolin-stimulated cyclic AMP accumulation in isolated porcine palmar lateral veins.
    Naunyn-Schmiedeberg's archives of pharmacology, 1995, Volume: 352, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Colforsin; Cyclic AMP; Enzyme Inhibitors; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Pyrrolidinones; Receptors, Adrenergic, alpha-2; Rolipram; Swine; Veins; Yohimbine

1995
Changes in alpha 1-adrenergic neurotransmission alter the number of somatostatin receptors in the rat hippocampus.
    Neuroscience letters, 1994, Aug-15, Volume: 177, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Colforsin; Cyclic AMP; Down-Regulation; Enzyme Activation; Hippocampus; Learning; Phenylephrine; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Receptors, Somatostatin; Signal Transduction; Somatostatin

1994
cAMP and protein synthesis in isolated adult rat heart preparations.
    The American journal of physiology, 1993, Volume: 265, Issue:5 Pt 1

    Topics: 1-Methyl-3-isobutylxanthine; Adenine Nucleotides; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Energy Metabolism; Epinephrine; Glucagon; Heart; Hypertension; In Vitro Techniques; Isoproterenol; Kinetics; Male; Myocardium; Perfusion; Phenylephrine; Phosphocreatine; Prazosin; Propranolol; Protein Biosynthesis; Rats; Rats, Sprague-Dawley; Yohimbine

1993
Examination of the role of inhibition of cyclic AMP in alpha 2-adrenoceptor mediated contractions of the porcine isolated palmar lateral vein.
    British journal of pharmacology, 1995, Volume: 114, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Forelimb; Norepinephrine; Prazosin; Veins; Yohimbine

1995
1,25-Dihydroxyvitamin D3 reduces the number of alpha 1-adrenergic receptors in FRTL-5 rat thyroid cells.
    Molecular and cellular endocrinology, 1995, Feb-27, Volume: 108, Issue:1-2

    Topics: 24,25-Dihydroxyvitamin D 3; Adenosine Triphosphate; Animals; Calcitriol; Calcium; Cell Line; Colforsin; Cyclic AMP; Cycloheximide; Dose-Response Relationship, Drug; Norepinephrine; Prazosin; Rats; Receptors, Adrenergic, alpha; Thyroid Gland; Thyrotropin; Time Factors

1995
Localization of the forskolin labeling sites to both halves of P-glycoprotein: similarity of the sites labeled by forskolin and prazosin.
    Molecular pharmacology, 1994, Volume: 46, Issue:2

    Topics: Amino Acid Sequence; ATP Binding Cassette Transporter, Subfamily B, Member 1; Binding Sites; Carrier Proteins; Cell Line; Colforsin; Humans; Immune Sera; Iodine Radioisotopes; Membrane Glycoproteins; Molecular Sequence Data; Peptide Fragments; Prazosin; Precipitin Tests; Protein Conformation; Trypsin; Tumor Cells, Cultured

1994
Alpha 2-adrenergic, but not imidazole, agonists activate NaCl cotransport in rabbit tracheal epithelial cells.
    The American journal of physiology, 1993, Volume: 264, Issue:3 Pt 1

    Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Carrier Proteins; Cells, Cultured; Chloride-Bicarbonate Antiporters; Clonidine; Colforsin; Cyclic AMP; Drug Interactions; Epithelial Cells; Epithelium; Guanabenz; Imidazoles; Imidazoline Receptors; Iodine Radioisotopes; Isoproterenol; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Receptors, Drug; Second Messenger Systems; Sodium Chloride Symporters; Symporters; Thromboxane-A Synthase; Trachea

1993
alpha-Adrenergic inhibition of the beta-adrenoceptor-dependent chloride current in guinea-pig ventricular myocytes.
    The Journal of physiology, 1995, Nov-15, Volume: 489 ( Pt 1)

    Topics: Animals; Chloride Channels; Colforsin; Epinephrine; Guinea Pigs; Heart Ventricles; Patch-Clamp Techniques; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Ventricular Function

1995
Modulation of norepinephrine-stimulated cyclic AMP accumulation in rat pinealocytes by n-3 fatty acids.
    European journal of pharmacology, 1996, Oct-03, Volume: 312, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Animals; Colforsin; Cyclic AMP; Drug Synergism; Fatty Acids; Male; Norepinephrine; Phospholipids; Pineal Gland; Prazosin; Rats; Rats, Sprague-Dawley; Triglycerides

1996
Stimulation of microsomal cholesterol ester hydrolase by glucagon, cyclic AMP analogues, and vasopressin in isolated rat hepatocytes.
    Lipids, 1996, Volume: 31, Issue:3

    Topics: Animals; Bucladesine; Cholesterol Esters; Colforsin; Cyclic AMP; Diglycerides; Glucagon; Microsomes, Liver; Particle Size; Prazosin; Rats; Sterol Esterase; Thionucleotides; Vasopressins

1996
Alpha(1)- and beta-adrenoceptor-mediated increase in 86Rb(+)-uptake in isolated cardiomyocytes from adult rat heart: evidence for interaction between the two receptor systems.
    Pharmacology & toxicology, 1996, Volume: 79, Issue:6

    Topics: Adrenergic alpha-Agonists; Adrenergic Antagonists; Animals; Cells, Cultured; Colforsin; Dose-Response Relationship, Drug; Heart; Myocardium; Norepinephrine; Prazosin; Rats; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Rubidium Radioisotopes; Timolol

1996
Norepinephrine induces the raf-1 kinase/mitogen-activated protein kinase cascade through both alpha 1- and beta-adrenoceptors.
    Circulation, 1997, Mar-04, Volume: 95, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Adrenergic alpha-1 Receptor Antagonists; Amino Acids; Animals; Animals, Newborn; Biological Transport; Bucladesine; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Cardiomegaly; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Heart; Kinetics; Myocardium; Norepinephrine; Phenylephrine; Prazosin; Propranolol; Protein Kinase C; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-raf; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Sarcolemma

1997
Denervation of pigment cells lead to a receptor that is ultrasensitive to melatonin and noradrenaline.
    Life sciences, 1997, Volume: 60, Issue:18

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Colforsin; Denervation; Fishes; Melanins; Melanophores; Melatonin; Norepinephrine; Peripheral Nervous System; Prazosin; Yohimbine

1997
Troponin I phosphorylation in spontaneously hypertensive rat heart: effect of beta-adrenergic stimulation.
    The American journal of physiology, 1997, Volume: 273, Issue:3 Pt 2

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Animals; Calcium; Calcium-Binding Proteins; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Electric Stimulation; Enzyme Inhibitors; Heart; Heart Ventricles; Hypertension; Isoproterenol; Marine Toxins; Myocardial Contraction; Myocardium; Myosin Light Chains; Norepinephrine; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Troponin I

1997
Localized cAMP-dependent signaling mediates beta 2-adrenergic modulation of cardiac excitation-contraction coupling.
    The American journal of physiology, 1997, Volume: 273, Issue:3 Pt 2

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Calcium; Calcium Channels; Calcium Channels, L-Type; Colforsin; Cyclic AMP; Ethanolamines; Heart; Heart Ventricles; Imidazoles; In Vitro Techniques; Isoproterenol; Myocardial Contraction; Myocardium; Norepinephrine; Prazosin; Rats; Receptors, Adrenergic, beta-2; Signal Transduction; Thionucleotides

1997
Alpha-1A adrenergic receptor stimulation with phenylephrine promotes arachidonic acid release by activation of phospholipase D in rat-1 fibroblasts: inhibition by protein kinase A.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:2

    Topics: Adenine; Adenylate Cyclase Toxin; Animals; Arachidonic Acid; Calcimycin; Carbazoles; Cell Line; Cholera Toxin; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Diglycerides; Enzyme Activation; Enzyme Inhibitors; Glycerides; GTP-Binding Proteins; Indoles; Lipase; Phenylephrine; Phospholipase D; Phospholipases A; Phospholipases A2; Prazosin; Pyrroles; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Transfection; Virulence Factors, Bordetella

1998
Alpha2-adrenoceptors mediate the effect of dopamine on adult rat jejunal electrolyte transport.
    European journal of pharmacology, 1998, Aug-28, Volume: 356, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Amiloride; Animals; Brimonidine Tartrate; Bucladesine; Cardiotonic Agents; Colforsin; Diuretics; Dopamine; Dose-Response Relationship, Drug; Electric Impedance; Electrolytes; Furosemide; Ion Transport; Jejunum; Male; Ouabain; Phentolamine; Prazosin; Propranolol; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2

1998
Stimulation of the extracellular signal-regulated kinase 1/2 pathway by human beta-3 adrenergic receptor: new pharmacological profile and mechanism of activation.
    Molecular pharmacology, 1999, Volume: 55, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Calcium-Calmodulin-Dependent Protein Kinases; CHO Cells; Colforsin; Cricetinae; Dioxoles; Enzyme Activation; Epinephrine; Ethanolamines; Humans; Insulin; Isoproterenol; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Norepinephrine; Phentolamine; Prazosin; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Signal Transduction; Yohimbine

1999
Functional alpha2C-adrenoceptors in human neuroblastoma SH-SY5Y cells.
    European journal of pharmacology, 1999, May-07, Volume: 372, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Brimonidine Tartrate; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Guanfacine; Humans; Idazoxan; Isoquinolines; Neuroblastoma; Oxymetazoline; Piperazines; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured; Yohimbine

1999
Norepinephrine-stimulated increase in Na+, K+-ATPase activity in the rat brain is mediated through alpha1A-adrenoceptor possibly by dephosphorylation of the enzyme.
    Journal of neurochemistry, 2000, Volume: 74, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Anticoagulants; Brain; Calcimycin; Calcineurin; Calcium; Calmodulin; Colforsin; Cyclosporine; Dioxanes; Enzyme Activation; Enzyme Inhibitors; Heparin; Ionophores; Male; Norepinephrine; Phosphorylation; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Signal Transduction; Sodium-Potassium-Exchanging ATPase; Sulfonamides

2000
Metabolic effects induced by epinephrine in Rana balcanica erythrocytes under normoxic and hypoxic conditions.
    Cell biochemistry and function, 2000, Volume: 18, Issue:3

    Topics: Adenosine Triphosphate; Adrenergic Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Colforsin; Cyclic AMP; Epinephrine; Erythrocytes; Glucose; Hypoxia; Lactic Acid; Ouabain; Oxygen; Perchlorates; Phosphofructokinase-1; Prazosin; Propranolol; Pyruvic Acid; Ranidae; Sodium-Potassium-Exchanging ATPase; Time Factors; Yohimbine

2000
The influence of beta-adrenergic activation on noradrenergic alpha1 activation of rabbit afferent arterioles.
    Pflugers Archiv : European journal of physiology, 2000, Volume: 441, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic alpha-Antagonists; Afferent Pathways; Animals; Arterioles; Calcium; Colforsin; Cyclic AMP; Cytosol; Enzyme Activation; Fluorescent Dyes; Fura-2; Isoproterenol; Muscle, Smooth, Vascular; Norepinephrine; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine

2000
Norepinephrine induces apoptosis in skin melanophores by attenuating cAMP-PKA signals via alpha2-adrenoceptors in the medaka, Oryzias latipes.
    Pigment cell research, 2001, Volume: 14, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Apoptosis; Clonidine; Colforsin; Culture Techniques; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cysteine Proteinase Inhibitors; Isoquinolines; Melanophores; Norepinephrine; Oligopeptides; Oryzias; Phenylephrine; Prazosin; Protein Isoforms; Receptors, Adrenergic, alpha-2; Signal Transduction; Skin; Skin Pigmentation; Sulfonamides; Yohimbine

2001
Direct actions of adrenergic agents on rat anterior pituitary cells.
    Pflugers Archiv : European journal of physiology, 2001, Volume: 442, Issue:6

    Topics: Adrenergic Agents; Adrenocorticotropic Hormone; Animals; Calcium; Cells, Cultured; Clonidine; Colforsin; Corticotropin-Releasing Hormone; Culture Media; Epinephrine; Follicle Stimulating Hormone; Growth Hormone; Growth Hormone-Releasing Hormone; Isoproterenol; Luteinizing Hormone; Male; Phenylephrine; Pituitary Gland, Anterior; Prazosin; Prolactin; Propranolol; Rats; Thyrotropin

2001
Membrane potential dependent modulations of calcium oscillations in insulin-secreting INS-1 cells.
    Cell calcium, 2002, Volume: 31, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Calcium Signaling; Cell Line; Clonidine; Colforsin; Diazoxide; Enzyme Inhibitors; Epinephrine; Fluorescent Dyes; Fura-2; Glucose; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Membrane Potentials; Mice; Patch-Clamp Techniques; Potassium Channels; Prazosin; Receptors, Adrenergic, alpha-2; Thapsigargin; Tolbutamide

2002
Phosphatidylinositol 3-kinase offsets cAMP-mediated positive inotropic effect via inhibiting Ca2+ influx in cardiomyocytes.
    Circulation research, 2004, Dec-10, Volume: 95, Issue:12

    Topics: Androstadienes; Animals; Calcium; Calcium Channels, L-Type; Calcium Signaling; Cells, Cultured; Chromones; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein beta Subunits; GTP-Binding Protein gamma Subunits; Insulin-Like Growth Factor I; Ion Transport; Isoproterenol; Morpholines; Myocardial Contraction; Myocytes, Cardiac; Norepinephrine; Patch-Clamp Techniques; Peptide Fragments; Pertussis Toxin; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Prazosin; Propanolamines; Protein Processing, Post-Translational; Rats; Receptors, Adrenergic, beta-1; Recombinant Proteins; Second Messenger Systems; Signal Transduction; Wortmannin

2004
Excitatory actions of dopamine via D1-like receptors in the rat lateral geniculate nucleus.
    Journal of neurophysiology, 2005, Volume: 94, Issue:6

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Action Potentials; Adrenergic alpha-Antagonists; Analysis of Variance; Anesthetics, Local; Animals; Animals, Newborn; Benzazepines; Bromocriptine; Carbazoles; Colforsin; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Enzyme Inhibitors; Geniculate Bodies; In Vitro Techniques; Indoles; Neurons; Patch-Clamp Techniques; Prazosin; Pyrimidines; Pyrroles; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Tetrodotoxin; Thionucleotides

2005
A61603-induced contractions of the porcine meningeal artery are mediated by alpha1- and alpha2-adrenoceptors.
    Basic & clinical pharmacology & toxicology, 2007, Volume: 100, Issue:4

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Antagonists; Alkaloids; Animals; Benzophenanthridines; Colforsin; Dose-Response Relationship, Drug; Female; Forecasting; Imidazoles; In Vitro Techniques; Meningeal Arteries; Methiothepin; Norepinephrine; Oxadiazoles; Phenylephrine; Piperazines; Potassium Chloride; Prazosin; Protein Kinase C; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Ritanserin; Serotonin 5-HT1 Receptor Antagonists; Serotonin Antagonists; Swine; Tetrahydronaphthalenes; Vasoconstriction; Yohimbine

2007
β1, β2, and β3 adrenoceptors and Na+/H+ exchanger regulatory factor 1 expression in human bronchi and their modifications in cystic fibrosis.
    American journal of respiratory cell and molecular biology, 2011, Volume: 44, Issue:1

    Topics: Adrenergic beta-Agonists; Adult; Aged; Albuterol; Benzoates; Bronchi; Case-Control Studies; Cell Line; Colforsin; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Dobutamine; Female; Gene Expression Regulation; Humans; Male; Middle Aged; Phosphoproteins; Prazosin; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; RNA, Messenger; Sodium-Hydrogen Exchangers; Thiazolidines; Young Adult

2011
Perineural dexmedetomidine added to ropivacaine for sciatic nerve block in rats prolongs the duration of analgesia by blocking the hyperpolarization-activated cation current.
    Anesthesiology, 2011, Volume: 115, Issue:4

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Amides; Analgesia; Anesthetics, Local; Animals; Behavior, Animal; Colforsin; Cyclic Nucleotide-Gated Cation Channels; Dexmedetomidine; Dose-Response Relationship, Drug; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Hypnotics and Sedatives; Idazoxan; Male; Nerve Block; Pain Measurement; Potassium Channel Blockers; Potassium Channels; Prazosin; Pyrimidines; Rats; Rats, Sprague-Dawley; Ropivacaine; Sciatic Nerve

2011