colforsin has been researched along with phentolamine in 33 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 10 (30.30) | 18.7374 |
1990's | 19 (57.58) | 18.2507 |
2000's | 3 (9.09) | 29.6817 |
2010's | 1 (3.03) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET | 1 |
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM | 1 |
Atkinson, BN; Minneman, KP | 1 |
Fukumitsu, T; Hayashi, H; Tokuno, H; Tomita, T | 1 |
Langeler, EG; van Hinsbergh, VW | 1 |
Hadcock, JR; Malbon, CC; Morris, GM | 1 |
Carpéné, C; Galitzky, J; Lafontan, M; Langin, D; Larrouy, D | 1 |
Abrahamsen, J; Nedergaard, OA | 1 |
Romani, A; Scarpa, A | 1 |
Nezu, E; Yoneyama, T; Yoshimura, K | 1 |
Mulder, AH; Schoffelmeer, AN; Wierenga, EA | 1 |
Giudicelli, Y; Leneveu, MC; Pecquery, R | 1 |
Hermansen, K | 1 |
Ernst, SA; Lowy, RJ | 1 |
Andersson, RG; Elwing, H; Grundström, N; Karlsson, JO | 1 |
Mulder, AH; Putters, J; Schoffelmeer, AN | 1 |
Hwang, KS; Van Breemen, C | 1 |
Chiba, S; Horiuchi, A; Iwatsuki, K; Yamagishi, F | 1 |
Ade, T; Hanke, W; Segner, H | 1 |
Hara, M; Inoue, M; Irie, T; Mikami, T; Mikami, Y; Minato, A; Omori, K; Uyama, M; Yasukura, T; Zeng, XT | 1 |
Cooke, HJ; Wood, JD; Zafirov, DH | 1 |
Bramuglia, GF; Enero, MA; Kazanietz, MG; Pezman, E | 1 |
Izawa, T; Komabayashi, T; Noguchi, M; Suda, K; Tsuboi, M | 1 |
Celuch, SM | 1 |
Daller, M; Goldstein, I; Gupta, S; Krane, RJ; Mulhall, JP; Park, K; Payton, TR; Salimpour, P; Traish, AM | 1 |
Edwards, RH; Grodsky, GM; Ma, YH | 1 |
Soares-da-Silva, P; Vieira-Coelho, MA | 1 |
Kamagata, S; Nakata, E; Ohta, M; Oshima, N | 1 |
Gerhardt, CC; Gros, J; Issad, T; Strosberg, AD | 1 |
Jun, IO; Kim, SC; Lee, MY; Oh, MM; Seo, KK | 1 |
Delgado, M; Fernández-Alfonso, MS; Fuentes, A | 1 |
Amour, J; Birenbaum, A; Heymes, C; Loyer, X; Michelet, P; Riou, B | 1 |
Bloomquist, JR; Gross, AD | 1 |
1 review(s) available for colforsin and phentolamine
Article | Year |
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The role of receptor binding in drug discovery.
Topics: Animals; Drug Design; Humans; Receptors, Drug | 1993 |
1 trial(s) available for colforsin and phentolamine
Article | Year |
---|---|
Intracavernosal forskolin: role in management of vasculogenic impotence resistant to standard 3-agent pharmacotherapy.
Topics: Alprostadil; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Resistance; Drug Therapy, Combination; Humans; Impotence, Vasculogenic; Injections; Male; Papaverine; Penis; Phentolamine; Rabbits; Vasodilator Agents | 1997 |
31 other study(ies) available for colforsin and phentolamine
Article | Year |
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[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium | 1985 |
Multiple adrenergic receptor subtypes controlling cyclic AMP formation: comparison of brain slices and primary neuronal and glial cultures.
Topics: Adrenergic alpha-Agonists; Aging; Animals; Animals, Newborn; Cells, Cultured; Cerebral Cortex; Colforsin; Cyclic AMP; Drug Synergism; Isoproterenol; Kinetics; Neuroglia; Neurons; Norepinephrine; Phentolamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine | 1991 |
Increase in calcium channel current by beta-adrenoceptor agonists in single smooth muscle cells isolated from porcine coronary artery.
Topics: 4-Aminopyridine; Adrenergic beta-Agonists; Animals; Cadmium; Calcium Channels; Colforsin; Coronary Vessels; In Vitro Techniques; Ion Channels; Isoproterenol; Muscle, Smooth, Vascular; Nicardipine; Norepinephrine; Phentolamine; Swine; Tetraethylammonium Compounds | 1990 |
Norepinephrine and iloprost improve barrier function of human endothelial cell monolayers: role of cAMP.
Topics: 1-Methyl-3-isobutylxanthine; Aorta; Cells, Cultured; Colforsin; Cyclic AMP; Electric Conductivity; Endothelium, Vascular; Fluorescent Antibody Technique; Horseradish Peroxidase; Humans; Iloprost; Isoproterenol; Kinetics; Norepinephrine; Phentolamine; Propranolol; Umbilical Arteries; Venae Cavae | 1991 |
Cross-regulation between G-protein-coupled receptors. Activation of beta 2-adrenergic receptors increases alpha 1-adrenergic receptor mRNA levels.
Topics: Animals; Blotting, Northern; Cell Line; Cholera Toxin; Colforsin; Cricetinae; Cyclic AMP; Epinephrine; GTP-Binding Proteins; Male; Phentolamine; Propranolol; Receptors, Adrenergic, alpha; RNA, Messenger; Thionucleotides; Vas Deferens | 1991 |
Non-adrenergic sites for imidazolines are not directly involved in the alpha 2-adrenergic antilipolytic effect of UK 14304 in rat adipocytes.
Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Brimonidine Tartrate; Bucladesine; Cell Membrane; Colforsin; Dioxanes; Idazoxan; Kinetics; Lipolysis; Phentolamine; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine | 1990 |
Lack of presynaptic modulation by isoprenaline of 3H-noradrenaline release from rabbit isolated ear artery.
Topics: Animals; Arteries; Autonomic Fibers, Postganglionic; Colforsin; Ear, External; Electric Stimulation; Female; In Vitro Techniques; Isoproterenol; Male; Norepinephrine; Phentolamine; Phosphodiesterase Inhibitors; Propranolol; Pyrimidines; Rabbits; Tritium; Yohimbine | 1991 |
Norepinephrine evokes a marked Mg2+ efflux from liver cells.
Topics: Animals; Carbachol; Cell Membrane; Colforsin; Cyclic AMP; In Vitro Techniques; Liver; Magnesium; Male; Norepinephrine; Phentolamine; Propranolol; Rats; Rats, Inbred Strains; Vasopressins | 1990 |
Augmentation of isoproterenol-stimulated tissue cyclic AMP level by cholinergic agonists in rat parotid gland.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Calcimycin; Calcium; Carbachol; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Isoproterenol; Male; Methacholine Chloride; Methacholine Compounds; Norepinephrine; Oxotremorine; Parotid Gland; Phentolamine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains | 1985 |
Role of adenylate cyclase in presynaptic alpha 2-adrenoceptor- and mu-opioid receptor-mediated inhibition of [3H]noradrenaline release from rat brain cortex slices.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Bucladesine; Cadmium; Calcimycin; Cerebral Cortex; Clonidine; Colforsin; Cyclic AMP; Electric Stimulation; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Morphine; Norepinephrine; Phentolamine; Pyrrolidinones; Rats; Receptors, Adrenergic, alpha; Receptors, Opioid; Receptors, Opioid, mu; Rolipram | 1986 |
Influence of androgenic status on the alpha 2/beta-adrenergic control of lipolysis in white fat cells: predominant alpha 2-antilipolytic response in testosterone-treated-castrated hamsters.
Topics: 1-Methyl-3-isobutylxanthine; Adipose Tissue; Animals; Brimonidine Tartrate; Clonidine; Colforsin; Cricetinae; Cyclic AMP; Epinephrine; Isoproterenol; Lipolysis; Male; Mesocricetus; Niacin; Orchiectomy; Phentolamine; Propranolol; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Testosterone | 1988 |
Forskolin, an activator of adenylate cyclase, stimulates pancreatic insulin, glucagon, and somatostatin release in the dog: studies in vitro.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Calcium; Colforsin; Diterpenes; Dogs; Dose-Response Relationship, Drug; Enzyme Activation; Glucagon; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Pancreas; Phentolamine; Propranolol; Somatostatin | 1985 |
Beta-adrenergic stimulation of ion transport in primary cultures of avian salt glands.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Animals; Atropine; Biological Transport, Active; Carbachol; Cells, Cultured; Colforsin; Cyclic GMP; Ducks; Epinephrine; Furosemide; Ions; Kinetics; Ouabain; Phentolamine; Propranolol; Salt Gland | 1987 |
Pigment migration in fish erythrophores is controlled by alpha 2-adrenoceptors.
Topics: Animals; Chromatophores; Colforsin; Electric Stimulation; Fishes; Norepinephrine; Phentolamine; Prazosin; Receptors, Adrenergic, alpha; Yohimbine | 1988 |
Activation of presynaptic alpha 2-adrenoceptors attenuates the inhibitory effect of mu-opioid receptor agonists on noradrenaline release from brain slices.
Topics: Animals; Brain Chemistry; Cadmium; Clonidine; Colforsin; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; In Vitro Techniques; Male; Morphine; Norepinephrine; Phentolamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Opioid; Receptors, Opioid, mu | 1986 |
Effect of dB-c-AMP and forskolin on the 45Ca influx, net Ca uptake and tension in rabbit aortic smooth muscle.
Topics: Animals; Aorta, Thoracic; Bucladesine; Calcium; Calcium Radioisotopes; Colforsin; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Phentolamine; Propranolol; Rats | 1987 |
Effects of forskolin on pancreatic exocrine secretion and cyclic nucleotide concentrations of the dog pancreas.
Topics: Animals; Atropine; Cimetidine; Colforsin; Cyclic AMP; Cyclic GMP; Dogs; Female; Male; Nucleotides, Cyclic; Pancreatic Juice; Phentolamine; Propranolol; Sulpiride; Verapamil | 1987 |
Hormonal response of primary hepatocytes of the clawed toad, Xenopus laevis.
Topics: Animals; Cell Survival; Cells, Cultured; Colforsin; Deamino Arginine Vasopressin; Epinephrine; Female; Glucose; Hormones; Kinetics; Liver; Liver Glycogen; Male; Phentolamine; Propranolol; Vasotocin; Xenopus laevis | 1995 |
Adrenergic receptor-mediated Cl- transport in rabbit corneal endothelial cells.
Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acetates; Acetazolamide; Adrenergic Agonists; Adrenergic Antagonists; Affinity Labels; Animals; Brimonidine Tartrate; Cells, Cultured; Chlorides; Colforsin; Dose-Response Relationship, Drug; Endothelium, Corneal; Fluorescent Dyes; Ion Transport; Isoproterenol; Microscopy, Fluorescence; Norepinephrine; Phentolamine; Phenylephrine; Photometry; Quinolines; Quinoxalines; Rabbits; Receptors, Adrenergic; Yohimbine | 1995 |
Elevation of cAMP facilitates noradrenergic transmission in submucous neurons of guinea pig ileum.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic alpha-Antagonists; Animals; Colforsin; Cyclic AMP; Dioxanes; Electric Stimulation; Ganglia; Guinea Pigs; Idazoxan; Ileum; Membrane Potentials; Microelectrodes; Neurons; Norepinephrine; Phentolamine; Receptors, Purinergic; Synaptic Transmission; Yohimbine | 1993 |
Beta-adrenoceptor desensitization by/clenbuterol in rat uterus.
Topics: Adrenergic beta-Antagonists; Animals; Clenbuterol; Colforsin; Cyclic AMP; Estradiol; Female; In Vitro Techniques; Isoproterenol; Kinetics; Muscle Relaxation; Phentolamine; Potassium Chloride; Rats; Rats, Wistar; Uterus | 1993 |
Mechanism of isoprenaline-stimulated diacylglycerol formation in rat parotid acinar cells.
Topics: Alkaloids; Animals; Bucladesine; Cells, Cultured; Colforsin; Diglycerides; In Vitro Techniques; Isoproterenol; Kinetics; Male; Parotid Gland; Phentolamine; Phosphatidylcholines; Phosphatidylethanolamines; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Phosphates; Propranolol; Protein Kinase C; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Staurosporine; Stimulation, Chemical; Vasoactive Intestinal Peptide | 1993 |
Possible participation of histamine H3 receptors in the modulation of noradrenaline release from rat spinal cord slices.
Topics: Animals; Colforsin; Desipramine; Dose-Response Relationship, Drug; Female; Histamine; Male; Norepinephrine; Phentolamine; Radioligand Assay; Rats; Rats, Wistar; Receptors, Histamine H3; Spinal Cord | 1995 |
Chronic sympathetic innervation of islets in transgenic mice results in differential desensitization of alpha-adrenergic inhibition of insulin secretion.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Glucose; Colforsin; Female; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Mice, Inbred C57BL; Mice, Transgenic; Nerve Growth Factors; Phentolamine; Promoter Regions, Genetic; Rats; Receptors, Adrenergic, alpha; Recombinant Fusion Proteins; Reference Values; Sympathetic Nervous System; Time Factors | 1997 |
Alpha2-adrenoceptors mediate the effect of dopamine on adult rat jejunal electrolyte transport.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Amiloride; Animals; Brimonidine Tartrate; Bucladesine; Cardiotonic Agents; Colforsin; Diuretics; Dopamine; Dose-Response Relationship, Drug; Electric Impedance; Electrolytes; Furosemide; Ion Transport; Jejunum; Male; Ouabain; Phentolamine; Prazosin; Propranolol; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2 | 1998 |
Light-induced pigment aggregation in xanthophores of the medaka, Oryzias latipes.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic alpha-Antagonists; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Chromatophores; Colforsin; Cyclic AMP; Cyclic GMP; Light; Melanosomes; Oryzias; Phentolamine; Phosphoric Diester Hydrolases; Skin Pigmentation; Sulfonamides | 1998 |
Stimulation of the extracellular signal-regulated kinase 1/2 pathway by human beta-3 adrenergic receptor: new pharmacological profile and mechanism of activation.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Calcium-Calmodulin-Dependent Protein Kinases; CHO Cells; Colforsin; Cricetinae; Dioxoles; Enzyme Activation; Epinephrine; Ethanolamines; Humans; Insulin; Isoproterenol; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Norepinephrine; Phentolamine; Prazosin; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Signal Transduction; Yohimbine | 1999 |
Synergistic effects of sildenafil on relaxation of rabbit and rat cavernosal smooth muscles when combined with various vasoactive agents.
Topics: Animals; Antihypertensive Agents; Cardiovascular Agents; Colforsin; Drug Synergism; Drug Therapy, Combination; Erectile Dysfunction; Male; Muscle Relaxation; Muscle, Smooth; Phentolamine; Phosphodiesterase Inhibitors; Piperazines; Prostaglandins E, Synthetic; Purines; Rabbits; Rats; Sildenafil Citrate; Sulfones | 2001 |
Effect of adrenaline and glucocorticoids on monocyte cAMP-specific phosphodiesterase (PDE4) in a monocytic cell line.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 8-Bromo Cyclic Adenosine Monophosphate; Atenolol; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Cycloheximide; Dermatitis, Atopic; Dexamethasone; Enzyme Activation; Epinephrine; Humans; Kinetics; Monocytes; Phentolamine; Propranolol; Receptors, Adrenergic, beta-2; Stress, Physiological; U937 Cells | 2002 |
Preservation of the positive lusitropic effect of beta-adrenoceptors stimulation in diabetic cardiomyopathy.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiomyopathies; Colforsin; Diabetes Complications; Diabetes Mellitus, Experimental; Echocardiography; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Papillary Muscles; Phentolamine; Pindolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta | 2008 |
Pharmacology of central octopaminergic and muscarinic pathways in Drosophila melanogaster larvae: Assessing the target potential of GPCRs.
Topics: Animals; Atropine; Central Nervous System; Colforsin; Cyclic CMP; Drosophila melanogaster; Electrophysiology; Larva; Octopamine; Phentolamine; Pilocarpine; Receptors, G-Protein-Coupled | 2018 |