Page last updated: 2024-08-23

colforsin and phentolamine

colforsin has been researched along with phentolamine in 33 studies

Research

Studies (33)

TimeframeStudies, this research(%)All Research%
pre-199010 (30.30)18.7374
1990's19 (57.58)18.2507
2000's3 (9.09)29.6817
2010's1 (3.03)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM1
Atkinson, BN; Minneman, KP1
Fukumitsu, T; Hayashi, H; Tokuno, H; Tomita, T1
Langeler, EG; van Hinsbergh, VW1
Hadcock, JR; Malbon, CC; Morris, GM1
Carpéné, C; Galitzky, J; Lafontan, M; Langin, D; Larrouy, D1
Abrahamsen, J; Nedergaard, OA1
Romani, A; Scarpa, A1
Nezu, E; Yoneyama, T; Yoshimura, K1
Mulder, AH; Schoffelmeer, AN; Wierenga, EA1
Giudicelli, Y; Leneveu, MC; Pecquery, R1
Hermansen, K1
Ernst, SA; Lowy, RJ1
Andersson, RG; Elwing, H; Grundström, N; Karlsson, JO1
Mulder, AH; Putters, J; Schoffelmeer, AN1
Hwang, KS; Van Breemen, C1
Chiba, S; Horiuchi, A; Iwatsuki, K; Yamagishi, F1
Ade, T; Hanke, W; Segner, H1
Hara, M; Inoue, M; Irie, T; Mikami, T; Mikami, Y; Minato, A; Omori, K; Uyama, M; Yasukura, T; Zeng, XT1
Cooke, HJ; Wood, JD; Zafirov, DH1
Bramuglia, GF; Enero, MA; Kazanietz, MG; Pezman, E1
Izawa, T; Komabayashi, T; Noguchi, M; Suda, K; Tsuboi, M1
Celuch, SM1
Daller, M; Goldstein, I; Gupta, S; Krane, RJ; Mulhall, JP; Park, K; Payton, TR; Salimpour, P; Traish, AM1
Edwards, RH; Grodsky, GM; Ma, YH1
Soares-da-Silva, P; Vieira-Coelho, MA1
Kamagata, S; Nakata, E; Ohta, M; Oshima, N1
Gerhardt, CC; Gros, J; Issad, T; Strosberg, AD1
Jun, IO; Kim, SC; Lee, MY; Oh, MM; Seo, KK1
Delgado, M; Fernández-Alfonso, MS; Fuentes, A1
Amour, J; Birenbaum, A; Heymes, C; Loyer, X; Michelet, P; Riou, B1
Bloomquist, JR; Gross, AD1

Reviews

1 review(s) available for colforsin and phentolamine

ArticleYear
The role of receptor binding in drug discovery.
    Journal of natural products, 1993, Volume: 56, Issue:4

    Topics: Animals; Drug Design; Humans; Receptors, Drug

1993

Trials

1 trial(s) available for colforsin and phentolamine

ArticleYear
Intracavernosal forskolin: role in management of vasculogenic impotence resistant to standard 3-agent pharmacotherapy.
    The Journal of urology, 1997, Volume: 158, Issue:5

    Topics: Alprostadil; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Resistance; Drug Therapy, Combination; Humans; Impotence, Vasculogenic; Injections; Male; Papaverine; Penis; Phentolamine; Rabbits; Vasodilator Agents

1997

Other Studies

31 other study(ies) available for colforsin and phentolamine

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Multiple adrenergic receptor subtypes controlling cyclic AMP formation: comparison of brain slices and primary neuronal and glial cultures.
    Journal of neurochemistry, 1991, Volume: 56, Issue:2

    Topics: Adrenergic alpha-Agonists; Aging; Animals; Animals, Newborn; Cells, Cultured; Cerebral Cortex; Colforsin; Cyclic AMP; Drug Synergism; Isoproterenol; Kinetics; Neuroglia; Neurons; Norepinephrine; Phentolamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Yohimbine

1991
Increase in calcium channel current by beta-adrenoceptor agonists in single smooth muscle cells isolated from porcine coronary artery.
    British journal of pharmacology, 1990, Volume: 100, Issue:3

    Topics: 4-Aminopyridine; Adrenergic beta-Agonists; Animals; Cadmium; Calcium Channels; Colforsin; Coronary Vessels; In Vitro Techniques; Ion Channels; Isoproterenol; Muscle, Smooth, Vascular; Nicardipine; Norepinephrine; Phentolamine; Swine; Tetraethylammonium Compounds

1990
Norepinephrine and iloprost improve barrier function of human endothelial cell monolayers: role of cAMP.
    The American journal of physiology, 1991, Volume: 260, Issue:5 Pt 1

    Topics: 1-Methyl-3-isobutylxanthine; Aorta; Cells, Cultured; Colforsin; Cyclic AMP; Electric Conductivity; Endothelium, Vascular; Fluorescent Antibody Technique; Horseradish Peroxidase; Humans; Iloprost; Isoproterenol; Kinetics; Norepinephrine; Phentolamine; Propranolol; Umbilical Arteries; Venae Cavae

1991
Cross-regulation between G-protein-coupled receptors. Activation of beta 2-adrenergic receptors increases alpha 1-adrenergic receptor mRNA levels.
    The Journal of biological chemistry, 1991, Feb-05, Volume: 266, Issue:4

    Topics: Animals; Blotting, Northern; Cell Line; Cholera Toxin; Colforsin; Cricetinae; Cyclic AMP; Epinephrine; GTP-Binding Proteins; Male; Phentolamine; Propranolol; Receptors, Adrenergic, alpha; RNA, Messenger; Thionucleotides; Vas Deferens

1991
Non-adrenergic sites for imidazolines are not directly involved in the alpha 2-adrenergic antilipolytic effect of UK 14304 in rat adipocytes.
    Biochemical pharmacology, 1990, Aug-01, Volume: 40, Issue:3

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Brimonidine Tartrate; Bucladesine; Cell Membrane; Colforsin; Dioxanes; Idazoxan; Kinetics; Lipolysis; Phentolamine; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1990
Lack of presynaptic modulation by isoprenaline of 3H-noradrenaline release from rabbit isolated ear artery.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 343, Issue:2

    Topics: Animals; Arteries; Autonomic Fibers, Postganglionic; Colforsin; Ear, External; Electric Stimulation; Female; In Vitro Techniques; Isoproterenol; Male; Norepinephrine; Phentolamine; Phosphodiesterase Inhibitors; Propranolol; Pyrimidines; Rabbits; Tritium; Yohimbine

1991
Norepinephrine evokes a marked Mg2+ efflux from liver cells.
    FEBS letters, 1990, Aug-20, Volume: 269, Issue:1

    Topics: Animals; Carbachol; Cell Membrane; Colforsin; Cyclic AMP; In Vitro Techniques; Liver; Magnesium; Male; Norepinephrine; Phentolamine; Propranolol; Rats; Rats, Inbred Strains; Vasopressins

1990
Augmentation of isoproterenol-stimulated tissue cyclic AMP level by cholinergic agonists in rat parotid gland.
    The Japanese journal of physiology, 1985, Volume: 35, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Calcimycin; Calcium; Carbachol; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Isoproterenol; Male; Methacholine Chloride; Methacholine Compounds; Norepinephrine; Oxotremorine; Parotid Gland; Phentolamine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains

1985
Role of adenylate cyclase in presynaptic alpha 2-adrenoceptor- and mu-opioid receptor-mediated inhibition of [3H]noradrenaline release from rat brain cortex slices.
    Journal of neurochemistry, 1986, Volume: 46, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Bucladesine; Cadmium; Calcimycin; Cerebral Cortex; Clonidine; Colforsin; Cyclic AMP; Electric Stimulation; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Morphine; Norepinephrine; Phentolamine; Pyrrolidinones; Rats; Receptors, Adrenergic, alpha; Receptors, Opioid; Receptors, Opioid, mu; Rolipram

1986
Influence of androgenic status on the alpha 2/beta-adrenergic control of lipolysis in white fat cells: predominant alpha 2-antilipolytic response in testosterone-treated-castrated hamsters.
    Endocrinology, 1988, Volume: 122, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Adipose Tissue; Animals; Brimonidine Tartrate; Clonidine; Colforsin; Cricetinae; Cyclic AMP; Epinephrine; Isoproterenol; Lipolysis; Male; Mesocricetus; Niacin; Orchiectomy; Phentolamine; Propranolol; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Testosterone

1988
Forskolin, an activator of adenylate cyclase, stimulates pancreatic insulin, glucagon, and somatostatin release in the dog: studies in vitro.
    Endocrinology, 1985, Volume: 116, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Calcium; Colforsin; Diterpenes; Dogs; Dose-Response Relationship, Drug; Enzyme Activation; Glucagon; Glucose; In Vitro Techniques; Insulin; Insulin Secretion; Pancreas; Phentolamine; Propranolol; Somatostatin

1985
Beta-adrenergic stimulation of ion transport in primary cultures of avian salt glands.
    The American journal of physiology, 1987, Volume: 252, Issue:6 Pt 1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Animals; Atropine; Biological Transport, Active; Carbachol; Cells, Cultured; Colforsin; Cyclic GMP; Ducks; Epinephrine; Furosemide; Ions; Kinetics; Ouabain; Phentolamine; Propranolol; Salt Gland

1987
Pigment migration in fish erythrophores is controlled by alpha 2-adrenoceptors.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1988, Volume: 91, Issue:2

    Topics: Animals; Chromatophores; Colforsin; Electric Stimulation; Fishes; Norepinephrine; Phentolamine; Prazosin; Receptors, Adrenergic, alpha; Yohimbine

1988
Activation of presynaptic alpha 2-adrenoceptors attenuates the inhibitory effect of mu-opioid receptor agonists on noradrenaline release from brain slices.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 333, Issue:4

    Topics: Animals; Brain Chemistry; Cadmium; Clonidine; Colforsin; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; In Vitro Techniques; Male; Morphine; Norepinephrine; Phentolamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Opioid; Receptors, Opioid, mu

1986
Effect of dB-c-AMP and forskolin on the 45Ca influx, net Ca uptake and tension in rabbit aortic smooth muscle.
    European journal of pharmacology, 1987, Feb-10, Volume: 134, Issue:2

    Topics: Animals; Aorta, Thoracic; Bucladesine; Calcium; Calcium Radioisotopes; Colforsin; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Phentolamine; Propranolol; Rats

1987
Effects of forskolin on pancreatic exocrine secretion and cyclic nucleotide concentrations of the dog pancreas.
    Archives internationales de pharmacodynamie et de therapie, 1987, Volume: 286, Issue:2

    Topics: Animals; Atropine; Cimetidine; Colforsin; Cyclic AMP; Cyclic GMP; Dogs; Female; Male; Nucleotides, Cyclic; Pancreatic Juice; Phentolamine; Propranolol; Sulpiride; Verapamil

1987
Hormonal response of primary hepatocytes of the clawed toad, Xenopus laevis.
    Experimental and clinical endocrinology & diabetes : official journal, German Society of Endocrinology [and] German Diabetes Association, 1995, Volume: 103, Issue:1

    Topics: Animals; Cell Survival; Cells, Cultured; Colforsin; Deamino Arginine Vasopressin; Epinephrine; Female; Glucose; Hormones; Kinetics; Liver; Liver Glycogen; Male; Phentolamine; Propranolol; Vasotocin; Xenopus laevis

1995
Adrenergic receptor-mediated Cl- transport in rabbit corneal endothelial cells.
    Japanese journal of pharmacology, 1995, Volume: 67, Issue:4

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acetates; Acetazolamide; Adrenergic Agonists; Adrenergic Antagonists; Affinity Labels; Animals; Brimonidine Tartrate; Cells, Cultured; Chlorides; Colforsin; Dose-Response Relationship, Drug; Endothelium, Corneal; Fluorescent Dyes; Ion Transport; Isoproterenol; Microscopy, Fluorescence; Norepinephrine; Phentolamine; Phenylephrine; Photometry; Quinolines; Quinoxalines; Rabbits; Receptors, Adrenergic; Yohimbine

1995
Elevation of cAMP facilitates noradrenergic transmission in submucous neurons of guinea pig ileum.
    The American journal of physiology, 1993, Volume: 264, Issue:3 Pt 1

    Topics: 1-Methyl-3-isobutylxanthine; Adrenergic alpha-Antagonists; Animals; Colforsin; Cyclic AMP; Dioxanes; Electric Stimulation; Ganglia; Guinea Pigs; Idazoxan; Ileum; Membrane Potentials; Microelectrodes; Neurons; Norepinephrine; Phentolamine; Receptors, Purinergic; Synaptic Transmission; Yohimbine

1993
Beta-adrenoceptor desensitization by/clenbuterol in rat uterus.
    General pharmacology, 1993, Volume: 24, Issue:3

    Topics: Adrenergic beta-Antagonists; Animals; Clenbuterol; Colforsin; Cyclic AMP; Estradiol; Female; In Vitro Techniques; Isoproterenol; Kinetics; Muscle Relaxation; Phentolamine; Potassium Chloride; Rats; Rats, Wistar; Uterus

1993
Mechanism of isoprenaline-stimulated diacylglycerol formation in rat parotid acinar cells.
    Japanese journal of pharmacology, 1993, Volume: 62, Issue:4

    Topics: Alkaloids; Animals; Bucladesine; Cells, Cultured; Colforsin; Diglycerides; In Vitro Techniques; Isoproterenol; Kinetics; Male; Parotid Gland; Phentolamine; Phosphatidylcholines; Phosphatidylethanolamines; Phosphatidylinositol 4,5-Diphosphate; Phosphatidylinositol Phosphates; Propranolol; Protein Kinase C; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta; Staurosporine; Stimulation, Chemical; Vasoactive Intestinal Peptide

1993
Possible participation of histamine H3 receptors in the modulation of noradrenaline release from rat spinal cord slices.
    European journal of pharmacology, 1995, Dec-12, Volume: 287, Issue:2

    Topics: Animals; Colforsin; Desipramine; Dose-Response Relationship, Drug; Female; Histamine; Male; Norepinephrine; Phentolamine; Radioligand Assay; Rats; Rats, Wistar; Receptors, Histamine H3; Spinal Cord

1995
Chronic sympathetic innervation of islets in transgenic mice results in differential desensitization of alpha-adrenergic inhibition of insulin secretion.
    Advances in experimental medicine and biology, 1997, Volume: 426

    Topics: Adrenergic alpha-Antagonists; Animals; Blood Glucose; Colforsin; Female; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Mice, Inbred C57BL; Mice, Transgenic; Nerve Growth Factors; Phentolamine; Promoter Regions, Genetic; Rats; Receptors, Adrenergic, alpha; Recombinant Fusion Proteins; Reference Values; Sympathetic Nervous System; Time Factors

1997
Alpha2-adrenoceptors mediate the effect of dopamine on adult rat jejunal electrolyte transport.
    European journal of pharmacology, 1998, Aug-28, Volume: 356, Issue:1

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Amiloride; Animals; Brimonidine Tartrate; Bucladesine; Cardiotonic Agents; Colforsin; Diuretics; Dopamine; Dose-Response Relationship, Drug; Electric Impedance; Electrolytes; Furosemide; Ion Transport; Jejunum; Male; Ouabain; Phentolamine; Prazosin; Propranolol; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2

1998
Light-induced pigment aggregation in xanthophores of the medaka, Oryzias latipes.
    Pigment cell research, 1998, Volume: 11, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic alpha-Antagonists; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Chromatophores; Colforsin; Cyclic AMP; Cyclic GMP; Light; Melanosomes; Oryzias; Phentolamine; Phosphoric Diester Hydrolases; Skin Pigmentation; Sulfonamides

1998
Stimulation of the extracellular signal-regulated kinase 1/2 pathway by human beta-3 adrenergic receptor: new pharmacological profile and mechanism of activation.
    Molecular pharmacology, 1999, Volume: 55, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bupranolol; Calcium-Calmodulin-Dependent Protein Kinases; CHO Cells; Colforsin; Cricetinae; Dioxoles; Enzyme Activation; Epinephrine; Ethanolamines; Humans; Insulin; Isoproterenol; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Norepinephrine; Phentolamine; Prazosin; Propanolamines; Receptors, Adrenergic, beta; Receptors, Adrenergic, beta-3; Signal Transduction; Yohimbine

1999
Synergistic effects of sildenafil on relaxation of rabbit and rat cavernosal smooth muscles when combined with various vasoactive agents.
    BJU international, 2001, Volume: 88, Issue:6

    Topics: Animals; Antihypertensive Agents; Cardiovascular Agents; Colforsin; Drug Synergism; Drug Therapy, Combination; Erectile Dysfunction; Male; Muscle Relaxation; Muscle, Smooth; Phentolamine; Phosphodiesterase Inhibitors; Piperazines; Prostaglandins E, Synthetic; Purines; Rabbits; Rats; Sildenafil Citrate; Sulfones

2001
Effect of adrenaline and glucocorticoids on monocyte cAMP-specific phosphodiesterase (PDE4) in a monocytic cell line.
    Archives of dermatological research, 2002, Volume: 294, Issue:4

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 8-Bromo Cyclic Adenosine Monophosphate; Atenolol; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Cycloheximide; Dermatitis, Atopic; Dexamethasone; Enzyme Activation; Epinephrine; Humans; Kinetics; Monocytes; Phentolamine; Propranolol; Receptors, Adrenergic, beta-2; Stress, Physiological; U937 Cells

2002
Preservation of the positive lusitropic effect of beta-adrenoceptors stimulation in diabetic cardiomyopathy.
    Anesthesia and analgesia, 2008, Volume: 107, Issue:4

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Cardiomyopathies; Colforsin; Diabetes Complications; Diabetes Mellitus, Experimental; Echocardiography; In Vitro Techniques; Isoproterenol; Male; Myocardial Contraction; NG-Nitroarginine Methyl Ester; Nitric Oxide; Papillary Muscles; Phentolamine; Pindolol; Rats; Rats, Wistar; Receptors, Adrenergic, beta

2008
Pharmacology of central octopaminergic and muscarinic pathways in Drosophila melanogaster larvae: Assessing the target potential of GPCRs.
    Pesticide biochemistry and physiology, 2018, Volume: 151

    Topics: Animals; Atropine; Central Nervous System; Colforsin; Cyclic CMP; Drosophila melanogaster; Electrophysiology; Larva; Octopamine; Phentolamine; Pilocarpine; Receptors, G-Protein-Coupled

2018