colforsin has been researched along with pd 98059 in 86 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 16 (18.60) | 18.2507 |
2000's | 61 (70.93) | 29.6817 |
2010's | 9 (10.47) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Anderson, NG; Kilgour, E; Yarwood, SJ | 1 |
Gould, GW; Plevin, R; Robinson, CJ; Scott, PH | 1 |
Glembotski, CC; Hanford, DS | 1 |
Cobb, MH; Khoo, S | 1 |
Fertel, R; Rampersaud, AA; Van Brocklyn, JR; Vandenheede, JR; Yates, AJ | 1 |
Barad, M; Casadio, A; Kandel, ER; Martin, KC; Michael, D; Rose, JC; Zhu, H | 1 |
Häussinger, D; Kurz, AK; Schliess, F; vom Dahl, S | 1 |
Ballotti, R; Bertolotto, C; Brunet, A; Buscà, R; Englaro, W; Ortonne, JP; Pagès, G | 1 |
Du, X; Guo, Z; Iacovitti, L | 1 |
Funder, JW; Kawashima, S; Li, H; Liu, JP; Robinson, PJ | 1 |
Hinoue, T; Kidd, M; Läuffer, JM; Modlin, IM; Schmid, SW; Tang, LH; Zhang, T | 1 |
Arita, J; Suzuki, S; Yamamoto, I | 1 |
Johansen, B; Moens, U; Seternes, OM | 1 |
Ai, W; Gong, J; Yu, L | 1 |
Cheng, HL; Delaney, CL; Feldman, EL | 1 |
De Petrocellis, L; Di Marzo, V; Galve-Roperh, I; Guzmán, M; Melck, D; Rueda, D | 1 |
Chen, X; Tang, S; Tashjian, AH | 1 |
Bonner, JC; Wang, YZ | 1 |
Boushey, RP; Drucker, DJ; Yusta, B | 1 |
Enjalbert, A; Gérard, C; Le Péchon-Vallée, C; Magalon, K; Rasolonjanahary, R | 1 |
Kubo, Y; Miyashita, T | 1 |
Abraham, JA; Chen, MM; Joly, AH; Lam, A; Schreiner, GF | 1 |
Grewal, SS; McCleskey, EW; Molliver, DC; Stenberg, PE; Stork, PJ; York, RD | 1 |
Birnbaum, MJ; Heidenreich, KA; Laessig, T; Li, M; Meintzer, MK; Wang, X | 1 |
Kuemmerle, JF; Murthy, KS | 1 |
Choi, SL; Choi, YK; Ha, J; Kang, I; Kim, J; Kim, SS; Kim, YS; Yoon, MY | 1 |
Kievit, P; Lauten, JD; Maurer, RA | 1 |
Amsterdam, A; Dantes, A; Hanoch, T; Merz, WE; Rosenberg, R; Seger, R; Strauss, JF | 1 |
Bauer, CK; Schledermann, W; Schwarz, JR; Wulfsen, I | 1 |
Lee, JK; Suh, HW; Won, JS | 1 |
Byrnes, HD; Fine, JS; Hipkin, RW; Zavodny, PJ | 1 |
Kitahara, M; Naitoh, T; Tsuruzoe, N | 1 |
Combes, P; Crumiere, M; Dickenson, JM; Graham, S; Klotz, KN | 1 |
Esselman, WJ; Lee, K | 1 |
Bayatti, N; Engele, J | 1 |
Låg, M; Refsnes, M; Schwarze, PE; Thoresen, GH; Thrane, EV | 1 |
Haycock, JW; Salvatore, MF; Waymire, JC | 1 |
Frey, BM; Frey, FJ; Heiniger, CD; Rochat, MK | 1 |
Kandolf, R; Küpper, JH; Meyer, RG; Rodemann, HP | 1 |
Elliott-Hunt, CR; Grammatopoulos, DK; Hillhouse, EW; Kazlauskaite, J; Wilde, GJ | 1 |
Hashiba, Y; Hashimoto, K; Kohga, H; Monden, T; Mori, M; Ozawa, A; Sasaki, T; Satoh, T; Yamada, M | 1 |
Brentani, RR; Chiarini, LB; Freitas, AR; Linden, R; Martins, VR; Zanata, SM | 1 |
Mann, GE; Morgan, AJ; Pearson, JD; Sobrevia, L; Steinert, JR; Sugden, D; Wheeler-Jones, CP; Wyatt, AW | 1 |
Ding, WQ; Dong, M; Holicky, EL; Miller, LJ; Ninova, D; Stegall, MD | 1 |
Hughes, TR; Irvine, SA; Mead, JR; Ramji, DP; Singh, NN | 1 |
Coulonval, K; Dumont, JE; Lamy, F; Perpete, S; Vandeput, F | 1 |
Amsterdam, A; Dantes, A; Kotsuji, F; Seger, R; Sorokina, K; Tajima, K; Yao, Z | 1 |
Kinane, J; Oliver, RP | 1 |
Andersson, TP; Karlsson, AM; Svensson, SP | 1 |
Dhein, S; Hagendorff, A; Pfeiffer, D; Polontchouk, L; Salameh, A | 1 |
Hansen, Tv; Nielsen, FC; Rehfeld, JF | 1 |
Agarwal, SK; Bierden, RM; Geller, DH; Magoffin, DA; Munir, I; Torbati, D; Weitsman, SR; Yen, HW | 1 |
Guerrero, J; Martínez, J; Olivares, D; Santibáñez, JF | 1 |
Lisinicchia, JG; Watts, VJ | 1 |
Ishikawa, K; Tokumoto, T; Watanabe, K | 1 |
Damiano, N; Galdiero, E; Galdiero, M; Longanella, A; Tortora, A; Vitiello, M | 1 |
Slomiany, A; Slomiany, BL | 2 |
Gosmanov, AR; Thomason, DB; Thompson, DB | 1 |
Asher, O; Constantinescu, A; Diamond, I; Wu, M | 1 |
Chen, DY; Peng, A; Sun, QY; Tan, X; Tang, YZ; Wang, YC | 1 |
Creaven, BS; Egan, DA; Finn, GJ | 1 |
Chen, SD; Fan, GH; Qi, C; Wang, G; Zhou, HY | 1 |
Ahn, SC; Choi, JM; Ghil, SH; Ham, DS; Hong, SY; Kim, JW; Kim, MK; Kim, SS; Kim, SU; Kim-Kwon, Y; Lee, YD; Suh-Kim, H | 1 |
Allagnat, F; Condorelli, DF; Haefliger, JA; Martin, D; Waeber, G | 1 |
Anand-Srivastava, MB; Daou, GB; Lappas, G | 1 |
Antunes, TT; Bell, A; Gagnon, A; Sorisky, A | 1 |
Blume, N; Friedrichsen, BN; Gram, VK; Lee, YC; Møldrup, A; Neubauer, N; Nielsen, JH; Petersen, JS | 1 |
Croxatto, HB; Orihuela, PA; Parada-Bustamante, A; Zuñiga, LM | 1 |
Hahn, SJ; Jeong, IK; Jo, YH; Kang, JH; Kim, MJ; Kim, MS; Ko, SH; Koh, KH; Park, YG; Rhie, DJ; Ryu, GR; Yoon, SH | 1 |
Benninghoff, AD; Thomas, P | 1 |
Eggo, MC; Susarla, R; Watkinson, JC | 1 |
Fujii, Y; Ghooray, D; Kakar, SS; Moore, JP; Nevitt, JR; Winters, SJ | 1 |
Arai, K; Chaturvedi, G; Roby, KF; Terranova, PF | 1 |
Dayma, K; Gupta, RK; Radha, V; Rajanna, A; Raman, T | 1 |
Hanada, K; Iwasaki, Y; Kageyama, K; Nigawara, T; Sakihara, S; Suda, T; Takayasu, S | 1 |
Bell, TJ; Oberholtzer, JC | 1 |
Barrett, KE; Hoda, MR; Keely, SJ; McCole, DF; Scharl, M | 1 |
Adachi, S; Kato, K; Kozawa, O; Matsushima-Nishiwaki, R; Minamitani, C; Mizutani, J; Natsume, H; Otsuka, T; Tokuda, H | 1 |
Lin, HW; Wang, PS; Wang, SW; Yu, PL | 1 |
Kintzios, S; Mayor-Lopez, L; Moschopoulou, G; Valero, T | 1 |
Abbondanza, C; Avvedimento, EV; Di Santi, A; Migliaccio, A; Ombra, MN; Perillo, B | 1 |
Abdel-Rahman, AA; Penumarti, A | 1 |
Baran, CN; Clason, TA; Girard, BM; Hardwick, JC; May, V; Merriam, LA; Parsons, RL; Tompkins, JD | 1 |
Caiafa, I; Capasso, L; Chiosi, E; Illiano, M; Naviglio, S; Salzillo, A; Sapio, L; Spina, A | 1 |
86 other study(ies) available for colforsin and pd 98059
Article | Year |
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Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Cyclic AMP stimulates the phosphorylation and activation of p42 and p44 mitogen-activated protein kinases in 3T3-F442A preadipocytes.
Topics: 3T3 Cells; Adipocytes; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cell Differentiation; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; Flavonoids; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Phosphorylation; Protein-Tyrosine Kinases | 1996 |
Efficacy of agonist-stimulated MEK activation determines the susceptibility of mitogen-activated protein (MAP) kinase to inhibition in rat aortic smooth muscle cells.
Topics: Angiotensin II; Animals; Aorta; Bradykinin; Calcium-Calmodulin-Dependent Protein Kinases; Cattle; Cell Line; Cells, Cultured; Colforsin; DNA; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Mitogen-Activated Protein Kinase Kinases; Muscle, Smooth; Muscle, Smooth, Vascular; Platelet-Derived Growth Factor; Protein Kinases; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-raf; Rats; Trachea | 1996 |
Stabilization of the B-type natriuretic peptide mRNA in cardiac myocytes by alpha-adrenergic receptor activation: potential roles for protein kinase C and mitogen-activated protein kinase.
Topics: Adrenergic alpha-Agonists; Animals; Atrial Natriuretic Factor; Calcium-Calmodulin-Dependent Protein Kinases; Cell Division; Cells, Cultured; Colforsin; Dose-Response Relationship, Drug; Endothelin-1; Enzyme Inhibitors; Flavonoids; Half-Life; Heart; Indoles; Maleimides; Myocardium; Natriuretic Peptide, Brain; Phenylephrine; Protein Kinase C; Rats; Receptors, Adrenergic, alpha; Signal Transduction | 1996 |
Activation of mitogen-activating protein kinase by glucose is not required for insulin secretion.
Topics: Animals; Calcium-Calmodulin-Dependent Protein Kinases; Colforsin; Deoxyglucose; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Glucose; Insulin; Insulin Secretion; Insulinoma; JNK Mitogen-Activated Protein Kinases; Kinetics; Mannoheptulose; MAP Kinase Kinase 1; MAP Kinase Kinase 2; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Pancreatic Neoplasms; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Rats; Tolbutamide; Tumor Cells, Cultured | 1997 |
Ganglioside GM1 activates the mitogen-activated protein kinase Erk2 and p70 S6 kinase in U-1242 MG human glioma cells.
Topics: Calcium-Calmodulin-Dependent Protein Kinases; Colforsin; Cyclic AMP; DNA; Enzyme Activation; Enzyme Inhibitors; Flavonoids; G(M1) Ganglioside; Glioma; Humans; Immunosuppressive Agents; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase Kinases; Mitogens; Platelet-Derived Growth Factor; Polyenes; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Ribosomal Protein S6 Kinases; Signal Transduction; Sirolimus; Tumor Cells, Cultured | 1997 |
MAP kinase translocates into the nucleus of the presynaptic cell and is required for long-term facilitation in Aplysia.
Topics: Amino Acid Sequence; Animals; Aplysia; Calcium-Calmodulin-Dependent Protein Kinases; Cell Compartmentation; Cell Nucleus; Cells, Cultured; Colforsin; Cyclic AMP; Enzyme Inhibitors; Flavonoids; Hippocampus; Long-Term Potentiation; MAP Kinase Kinase 1; Mitogen-Activated Protein Kinase Kinases; Molecular Sequence Data; Neuronal Plasticity; Neurons, Afferent; Peptides; Presynaptic Terminals; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Serotonin; Synapses; Synaptic Transmission | 1997 |
Mitogen-activated protein kinases mediate the stimulation of bile acid secretion by tauroursodeoxycholate in rat liver.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Bucladesine; Calcium-Calmodulin-Dependent Protein Kinases; Cells, Cultured; Colforsin; Enzyme Activation; Enzyme Inhibitors; Flavonoids; GTP-Binding Proteins; Indoles; Isomerism; Isoproterenol; Kinetics; Liver; Male; Maleimides; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Models, Biological; Protein Kinase C; Protein-Tyrosine Kinases; Rats; Rats, Wistar; Signal Transduction; Taurochenodeoxycholic Acid; Taurocholic Acid; Tetradecanoylphorbol Acetate | 1997 |
Inhibition of the mitogen-activated protein kinase pathway triggers B16 melanoma cell differentiation.
Topics: Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cell Differentiation; Colforsin; Cyclic AMP; Enzyme Inhibitors; Flavonoids; Luciferases; Melanoma, Experimental; Mice; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Monophenol Monooxygenase; Protein Kinase Inhibitors; Protein Kinases; Recombinant Fusion Proteins; Tetradecanoylphorbol Acetate; Transfection; Tumor Cells, Cultured | 1998 |
Regulation of tyrosine hydroxylase gene expression during transdifferentiation of striatal neurons: changes in transcription factors binding the AP-1 site.
Topics: 1-Methyl-3-isobutylxanthine; Activating Transcription Factor 2; Animals; Base Sequence; Calcium-Calmodulin-Dependent Protein Kinases; Carcinogens; Cell Differentiation; Chamomile; Colforsin; Corpus Striatum; Cyclic AMP Response Element Modulator; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; DNA-Binding Proteins; Dopamine; Enzyme Inhibitors; Female; Fibroblast Growth Factor 1; Flavonoids; Gene Expression Regulation, Developmental; Gene Expression Regulation, Enzymologic; Molecular Sequence Data; Neurons; Oils, Volatile; Phosphodiesterase Inhibitors; Plants, Medicinal; Pregnancy; Protein Binding; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-jun; Rats; Rats, Sprague-Dawley; Repressor Proteins; Signal Transduction; Tetradecanoylphorbol Acetate; Transcription Factor AP-1; Transcription Factors; Tyrosine 3-Monooxygenase | 1998 |
Differential regulation of MAP kinase activity by corticotropin-releasing hormone in normal and neoplastic corticotropes.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Atrial Natriuretic Factor; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Colforsin; Corticotropin-Releasing Hormone; Cyclic AMP; DNA Replication; Enzyme Inhibitors; Flavonoids; Isoquinolines; Mice; Pituitary Gland, Anterior; Pituitary Neoplasms; Sheep; Sulfonamides; Thymidine | 1998 |
Pituitary adenylate cyclase-activating polypeptide modulates gastric enterochromaffin-like cell proliferation in rats.
Topics: Androstadienes; Animals; Cell Division; Cells, Cultured; Colforsin; DNA; Enterochromaffin Cells; Female; Flavonoids; Gastric Mucosa; Gastrins; Genistein; Humans; Neuropeptides; Neurotransmitter Agents; Octreotide; Peptide Fragments; Pituitary Adenylate Cyclase-Activating Polypeptide; Polymerase Chain Reaction; Rats; Rats, Sprague-Dawley; Receptors, Pituitary Adenylate Cyclase-Activating Polypeptide; Receptors, Pituitary Hormone; Receptors, Vasoactive Intestinal Peptide; Signal Transduction; Terfenadine; Vasoactive Intestinal Peptide; Wortmannin | 1999 |
Mitogen-activated protein kinase-dependent stimulation of proliferation of rat lactotrophs in culture by 3',5'-cyclic adenosine monophosphate.
Topics: Animals; Bromocriptine; Bucladesine; Calcium-Calmodulin-Dependent Protein Kinases; Cell Division; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Female; Flavonoids; Insulin; Pituitary Gland, Anterior; Rats; Rats, Wistar | 1999 |
A dominant role for the Raf-MEK pathway in forskolin, 12-O-tetradecanoyl-phorbol acetate, and platelet-derived growth factor-induced CREB (cAMP-responsive element-binding protein) activation, uncoupled from serine 133 phosphorylation in NIH 3T3 cells.
Topics: 3T3 Cells; Amino Acid Sequence; Animals; Calcium-Calmodulin-Dependent Protein Kinases; Cell Cycle Proteins; Colforsin; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; DNA-Binding Proteins; Dual Specificity Phosphatase 1; Dual Specificity Phosphatase 6; Enzyme Activation; Enzyme Inhibitors; ets-Domain Protein Elk-1; Flavonoids; Immediate-Early Proteins; MAP Kinase Kinase Kinase 1; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Molecular Sequence Data; Phosphoprotein Phosphatases; Phosphorylation; Platelet-Derived Growth Factor; Protein Kinase C; Protein Phosphatase 1; Protein Serine-Threonine Kinases; Protein Tyrosine Phosphatases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-raf; Serine; Tetradecanoylphorbol Acetate; Transcription Factors; Transcriptional Activation | 1999 |
MAP kinase activation by mu opioid receptor involves phosphatidylinositol 3-kinase but not the cAMP/PKA pathway.
Topics: Androstadienes; Animals; Calcium-Calmodulin-Dependent Protein Kinases; CHO Cells; Chromones; Colforsin; Cricetinae; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Genistein; Indoles; Maleimides; Morphine; Morpholines; Naloxone; Narcotic Antagonists; Narcotics; Phosphatidylinositol 3-Kinases; Protein Kinase C; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Rats; Receptors, Opioid, mu; Recombinant Proteins; Thionucleotides; Transfection; Wortmannin | 1999 |
Insulin-like growth factor-I prevents caspase-mediated apoptosis in Schwann cells.
Topics: Animals; Animals, Newborn; Apoptosis; Caspase 3; Caspase Inhibitors; Caspases; Cells, Cultured; Chromones; Colforsin; Enzyme Inhibitors; Flavonoids; Flow Cytometry; Insulin; Insulin-Like Growth Factor I; Mitogen-Activated Protein Kinases; Morpholines; Phosphatidylinositol 3-Kinases; Rats; Rats, Sprague-Dawley; Schwann Cells; Sciatic Nerve | 1999 |
Involvement of the cAMP/protein kinase A pathway and of mitogen-activated protein kinase in the anti-proliferative effects of anandamide in human breast cancer cells.
Topics: Arachidonic Acids; Breast Neoplasms; Cell Division; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Down-Regulation; Endocannabinoids; Flavonoids; Humans; Mitogen-Activated Protein Kinases; Nerve Growth Factor; Piperidines; Polyunsaturated Alkamides; Prolactin; Proto-Oncogene Proteins c-raf; Pyrazoles; Receptors, Prolactin; Rimonabant; Tumor Cells, Cultured | 1999 |
Novel action of pituitary adenylate cyclase-activating polypeptide. Stimulation of extracellular acidification in rat pituitary GH4C1 cells.
Topics: Animals; Calcium; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Extracellular Space; Flavonoids; Hydrogen-Ion Concentration; Kinetics; Mitogen-Activated Protein Kinases; Naphthalenes; Neuropeptides; Pituitary Adenylate Cyclase-Activating Polypeptide; Pituitary Gland; Protein Kinase C; Rats; Signal Transduction; Tetradecanoylphorbol Acetate; Thyrotropin-Releasing Hormone | 2000 |
Mechanism of extracellular signal-regulated kinase (ERK)-1 and ERK-2 activation by vanadium pentoxide in rat pulmonary myofibroblasts.
Topics: Acetylcysteine; Animals; Asthma; Bronchitis; Carbon; Coal Ash; Colforsin; Enzyme Activation; ErbB Receptors; Fibroblasts; Flavonoids; Intracellular Signaling Peptides and Proteins; Lung; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Particulate Matter; Phosphorylation; Phosphotyrosine; Protein Tyrosine Phosphatase, Non-Receptor Type 11; Protein Tyrosine Phosphatase, Non-Receptor Type 6; Protein Tyrosine Phosphatases; Quinazolines; Rats; Titanium; Tyrphostins; Vanadium Compounds | 2000 |
The glucagon-like peptide-2 receptor mediates direct inhibition of cellular apoptosis via a cAMP-dependent protein kinase-independent pathway.
Topics: Amino Acid Chloromethyl Ketones; Animals; Apoptosis; Caspase 3; Caspase 8; Caspase 9; Caspases; Cell Division; Cell Line; Cell Survival; Chromones; Colforsin; Cricetinae; Cyclic AMP-Dependent Protein Kinases; Cycloheximide; Cysteine Proteinase Inhibitors; Cytochrome c Group; Cytosol; DNA Fragmentation; Electrophoresis, Agar Gel; Enzyme Activation; Enzyme Inhibitors; Epithelium; Fibroblasts; Flavonoids; Glucagon-Like Peptide 2; Glucagon-Like Peptide-1 Receptor; Glucagon-Like Peptides; Intestinal Mucosa; Isoquinolines; Microscopy, Fluorescence; Mitochondria; Morpholines; Peptides; Poly(ADP-ribose) Polymerases; Protein Synthesis Inhibitors; Receptors, Cell Surface; Receptors, Glucagon; Signal Transduction; Sulfonamides; Time Factors; Transfection | 2000 |
Vasoactive intestinal polypeptide and pituitary adenylate cyclase-activating polypeptides stimulate mitogen-activated protein kinase in the pituitary cell line GH4C1 by a 3',5'-cyclic adenosine monophosphate pathway.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adjuvants, Immunologic; Animals; Butadienes; Cell Line; Cholera Toxin; Colforsin; Cyclic AMP; Enzyme Inhibitors; Extracellular Space; Flavonoids; Gene Expression; Indoles; Isoquinolines; Maleimides; MAP Kinase Kinase 1; MAP Kinase Kinase 2; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Neuropeptides; Nitriles; Pituitary Adenylate Cyclase-Activating Polypeptide; Pituitary Gland; Prolactin; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Receptor Cross-Talk; RNA, Messenger; Sulfonamides; Thyrotropin-Releasing Hormone; Vasoactive Intestinal Peptide | 2000 |
Extracellular Ca2+ sensitivity of mGluR1alpha induces an increase in the basal cAMP level by direct coupling with Gs protein in transfected CHO cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actins; Animals; Calcium; Cell Size; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Flavonoids; Fluorescent Dyes; Glutamic Acid; GTP-Binding Protein alpha Subunits, Gs; Isoquinolines; MAP Kinase Signaling System; Protein Kinase C; Receptors, Metabotropic Glutamate; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Transfection; Type C Phospholipases | 2000 |
CTGF expression is induced by TGF- beta in cardiac fibroblasts and cardiac myocytes: a potential role in heart fibrosis.
Topics: Adult; Aged; Animals; Animals, Newborn; Biomarkers; Blotting, Northern; Cells, Cultured; Colforsin; Collagen; Connective Tissue Growth Factor; Disease Models, Animal; Enzyme-Linked Immunosorbent Assay; Extracellular Matrix; Female; Fibroblasts; Fibronectins; Fibrosis; Flavonoids; Genes, Reporter; Growth Substances; Heart Diseases; Heart Ventricles; Humans; Immediate-Early Proteins; Intercellular Signaling Peptides and Proteins; Luciferases; Male; MAP Kinase Signaling System; Middle Aged; Myocardial Infarction; Myocardium; Plasminogen Activator Inhibitor 1; Promoter Regions, Genetic; Rats; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors; Tissue Distribution; Transforming Growth Factor beta; Up-Regulation | 2000 |
Role of phosphoinositide 3-kinase and endocytosis in nerve growth factor-induced extracellular signal-regulated kinase activation via Ras and Rap1.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Blotting, Western; Cell Differentiation; Cell Survival; Cells, Cultured; Chromatography, Affinity; Chromones; Colforsin; Dose-Response Relationship, Drug; Endocytosis; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Ganglia, Spinal; Immunohistochemistry; Luciferases; Microscopy, Electron; Microscopy, Fluorescence; Mitogen-Activated Protein Kinases; Models, Biological; Morpholines; Nerve Growth Factor; PC12 Cells; Phosphatidylinositol 3-Kinases; Proto-Oncogene Proteins c-raf; rap1 GTP-Binding Proteins; ras Proteins; Rats; Receptor, trkA; Signal Transduction; Time Factors; Transfection | 2000 |
Cyclic AMP promotes neuronal survival by phosphorylation of glycogen synthase kinase 3beta.
Topics: Animals; Apoptosis; Brain Chemistry; Calcium-Calmodulin-Dependent Protein Kinases; Cell Fractionation; Cell Survival; Cells, Cultured; Cerebellum; Colforsin; Culture Media, Serum-Free; Cyclic AMP; Enzyme Inhibitors; Flavonoids; Glycogen Synthase Kinase 3; Glycogen Synthase Kinases; Immunoblotting; Isoquinolines; Neurons; Phosphorylation; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Rats; Recombinant Fusion Proteins; Sulfonamides; Transfection | 2000 |
Coupling of the insulin-like growth factor-I receptor tyrosine kinase to Gi2 in human intestinal smooth muscle: Gbetagamma -dependent mitogen-activated protein kinase activation and growth.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Cell Division; Cells, Cultured; Chromones; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flavonoids; GTP-Binding Protein alpha Subunit, Gi2; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein beta Subunits; GTP-Binding Protein gamma Subunits; Heterotrimeric GTP-Binding Proteins; Humans; Insulin-Like Growth Factor II; Intestinal Mucosa; MAP Kinase Signaling System; Morpholines; Muscle, Smooth; Pertussis Toxin; Phosphatidylinositol 3-Kinases; Phosphorylation; Protein Binding; Protein-Tyrosine Kinases; Proto-Oncogene Proteins; Receptor, IGF Type 1; Recombinant Proteins; Time Factors; Virulence Factors, Bordetella | 2001 |
Effects of stimulation of AMP-activated protein kinase on insulin-like growth factor 1- and epidermal growth factor-dependent extracellular signal-regulated kinase pathway.
Topics: 3T3 Cells; Aminoimidazole Carboxamide; AMP-Activated Protein Kinases; Animals; Catalysis; Cell Line; Colforsin; COS Cells; DNA; DNA, Complementary; Enzyme Activation; Enzyme Inhibitors; Epidermal Growth Factor; Flavonoids; Insulin-Like Growth Factor I; Mice; Mitogen-Activated Protein Kinases; Multienzyme Complexes; Phosphorylation; Protein Binding; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins c-raf; Ribonucleotides; RNA; RNA, Antisense; Serine; Signal Transduction; Time Factors; Transfection | 2001 |
Analysis of the role of the mitogen-activated protein kinase in mediating cyclic-adenosine 3',5'-monophosphate effects on prolactin promoter activity.
Topics: Animals; Binding Sites; Colforsin; CREB-Binding Protein; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; DNA-Binding Proteins; E1A-Associated p300 Protein; Enzyme Inhibitors; Epidermal Growth Factor; ets-Domain Protein Elk-1; Flavonoids; Isoquinolines; Mitogen-Activated Protein Kinases; Nuclear Proteins; Pituitary Neoplasms; Potassium Channels; Prolactin; Promoter Regions, Genetic; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-ets; rap1 GTP-Binding Proteins; Rats; Sulfonamides; Thyrotropin-Releasing Hormone; Trans-Activators; Transcription Factors; Transcription, Genetic; Tumor Cells, Cultured | 2001 |
The ERK signaling cascade inhibits gonadotropin-stimulated steroidogenesis.
Topics: Animals; Cell Line; Chorionic Gonadotropin; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Down-Regulation; Enzyme Activation; Enzyme Inhibitors; Female; Flavonoids; Follicle Stimulating Hormone; Gonadotropins; Granulosa Cells; Humans; Luteinizing Hormone; MAP Kinase Signaling System; Microscopy, Fluorescence; Mitogen-Activated Protein Kinases; Models, Biological; Phosphoproteins; Phosphorylation; Plasmids; Progesterone; Protein Binding; Rats; Signal Transduction; Steroids; Time Factors; Transfection | 2001 |
Modulation of rat erg1, erg2, erg3 and HERG K+ currents by thyrotropin-releasing hormone in anterior pituitary cells via the native signal cascade.
Topics: Animals; Arachidonic Acid; Cation Transport Proteins; Cells, Cultured; Cholecystokinin; Colforsin; DNA-Binding Proteins; Enzyme Inhibitors; ERG1 Potassium Channel; Ether-A-Go-Go Potassium Channels; Flavonoids; Humans; Indoles; Isoquinolines; Kinetics; Maleimides; Membrane Potentials; Membrane Transport Proteins; Patch-Clamp Techniques; Pituitary Gland, Anterior; Potassium Channels; Potassium Channels, Voltage-Gated; Protein Kinase Inhibitors; Protein Kinases; Rats; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Thyrotropin-Releasing Hormone; Trans-Activators; Transcriptional Regulator ERG; Tyrphostins; Vasoactive Intestinal Peptide | 2001 |
Forskolin inhibits expression of inducible nitric oxide synthase mRNA via inhibiting the mitogen activated protein kinase in C6 cells.
Topics: Animals; Colforsin; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation, Enzymologic; Glioma; Imidazoles; Isoquinolines; Lipopolysaccharides; Mitogen-Activated Protein Kinases; NF-kappa B; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; p38 Mitogen-Activated Protein Kinases; Pyridines; Rats; RNA, Messenger; Sulfonamides; Transcription, Genetic; Tumor Cells, Cultured | 2001 |
Evaluation of signal transduction pathways in chemoattractant-induced human monocyte chemotaxis.
Topics: 1-Methyl-3-isobutylxanthine; Androstadienes; Chemokine CCL2; Chemokine CCL3; Chemokine CCL4; Chemokine CCL5; Chemotactic Factors; Chemotaxis, Leukocyte; Chromones; Colforsin; Flavonoids; Humans; In Vitro Techniques; Macrophage Inflammatory Proteins; Mitogen-Activated Protein Kinases; Monocytes; Morpholines; N-Formylmethionine Leucyl-Phenylalanine; Phosphatidylinositol 3-Kinases; Signal Transduction; Wortmannin | 2001 |
Tumor necrosis factor-alpha is induced through phorbol ester--and glycated human albumin-dependent pathway in THP-1 cells.
Topics: Carcinogens; Catalase; Cell Differentiation; Cell Line; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Glycated Serum Albumin; Glycation End Products, Advanced; Humans; Insulin Resistance; Mitogen-Activated Protein Kinases; Monocytes; Protein Kinase C; Serum Albumin; Signal Transduction; Staurosporine; Superoxide Dismutase; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 2001 |
Regulation of p42/p44 mitogen-activated protein kinase by the human adenosine A3 receptor in transfected CHO cells.
Topics: Adenosine; Androstadienes; Animals; CHO Cells; Chromones; Colforsin; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Humans; Luciferases; Mitogen-Activated Protein Kinase 1; Morpholines; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Receptor, Adenosine A3; Receptors, Purinergic P1; Recombinant Fusion Proteins; Wortmannin | 2001 |
cAMP potentiates H(2)O(2)-induced ERK1/2 phosphorylation without the requirement for MEK1/2 phosphorylation.
Topics: Colforsin; Cyclic AMP; Drug Synergism; Enzyme Inhibitors; Estrenes; Flavonoids; Humans; Hydrogen Peroxide; Jurkat Cells; Lymphocyte Specific Protein Tyrosine Kinase p56(lck); MAP Kinase Kinase 1; MAP Kinase Kinase 2; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Pyrrolidinones; Receptors, Antigen, T-Cell; T-Lymphocytes | 2001 |
Cyclic AMP modulates the response of central nervous system glia to fibroblast growth factor-2 by redirecting signalling pathways.
Topics: Animals; Astrocytes; Bucladesine; Cell Division; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Enzyme Inhibitors; Fibroblast Growth Factor 2; Flavonoids; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Phosphorylation; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley | 2001 |
Mechanisms in fluoride-induced interleukin-8 synthesis in human lung epithelial cells.
Topics: Androstadienes; Benzylamines; Cell Line; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Egtazic Acid; Epithelial Cells; Flavonoids; Genistein; Humans; Indoles; Interleukin-8; Isoquinolines; Lung; Maleimides; Okadaic Acid; Pertussis Toxin; Protein Kinase C; Signal Transduction; Sodium Fluoride; Sulfonamides; Tetradecanoylphorbol Acetate; Vanadates; Virulence Factors, Bordetella; Wortmannin | 2001 |
Depolarization-stimulated catecholamine biosynthesis: involvement of protein kinases and tyrosine hydroxylase phosphorylation sites in situ.
Topics: Animals; Catecholamines; Cell Line; Chemical Phenomena; Chemistry; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Electrophysiology; Enzyme Inhibitors; Flavonoids; Mathematics; Mitogen-Activated Protein Kinases; Nerve Growth Factor; PC12 Cells; Phosphorylation; Potassium; Protein Kinases; Rats; Tyrosine 3-Monooxygenase | 2001 |
TNF-alpha enhances intracellular glucocorticoid availability.
Topics: 11-beta-Hydroxysteroid Dehydrogenase Type 2; Animals; Cells, Cultured; Colforsin; Corticosterone; Cyclic AMP-Dependent Protein Kinases; Down-Regulation; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Glucocorticoids; Glucose; Hydroxysteroid Dehydrogenases; Imidazoles; Indoles; Maleimides; Mitogen-Activated Protein Kinases; Pyridines; Tetradecanoylphorbol Acetate; Tumor Necrosis Factor-alpha | 2001 |
Early growth response-1 gene (Egr-1) promoter induction by ionizing radiation in U87 malignant glioma cells in vitro.
Topics: Androstadienes; Anisomycin; Blotting, Western; Colforsin; DNA-Binding Proteins; Early Growth Response Protein 1; Epidermal Growth Factor; Flavonoids; Glioma; Humans; Imidazoles; Immediate-Early Proteins; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Promoter Regions, Genetic; Pyridines; Suramin; Transcription Factors; Wortmannin | 2002 |
Potential signalling pathways underlying corticotrophin-releasing hormone-mediated neuroprotection from excitotoxicity in rat hippocampus.
Topics: Animals; Cell Death; Colforsin; Corticotropin-Releasing Hormone; Cyclic AMP; Enzyme Inhibitors; Flavonoids; Glutamic Acid; Hippocampus; In Situ Hybridization, Fluorescence; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Neurons; Neurotoxins; Organ Culture Techniques; Proto-Oncogene Proteins c-jun; Rats | 2002 |
Transcriptional regulation of the human PRL-releasing peptide (PrRP) receptor gene by a dopamine 2 Receptor agonist: cloning and characterization of the human PrRP receptor gene and its promoter region.
Topics: Amino Acid Sequence; Base Sequence; Blotting, Northern; Bromocriptine; Cell Line; Cloning, Molecular; Colforsin; Cyclic AMP Response Element-Binding Protein; Dopamine Agonists; Flavonoids; Humans; Molecular Sequence Data; Nimodipine; Promoter Regions, Genetic; Receptors, Dopamine D2; Receptors, Neuropeptide; Serine; Transcription, Genetic | 2002 |
Cellular prion protein transduces neuroprotective signals.
Topics: Animals; Animals, Newborn; Anisomycin; Antibodies, Monoclonal; Apoptosis; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Eye Proteins; Flavonoids; Gene Expression Regulation, Developmental; Immune Sera; MAP Kinase Signaling System; Mice; Mice, Inbred C57BL; Mice, Knockout; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Neurons; Organ Culture Techniques; Peptide Fragments; Phosphatidylinositol Diacylglycerol-Lyase; Phosphoinositide Phospholipase C; Phosphorylation; Protein Processing, Post-Translational; PrPC Proteins; Rats; Rats, Inbred Strains; Retina; Signal Transduction; Thionucleotides; Type C Phospholipases | 2002 |
Early activation of the p42/p44MAPK pathway mediates adenosine-induced nitric oxide production in human endothelial cells: a novel calcium-insensitive mechanism.
Topics: Adenosine; Androstadienes; Arginine; Biological Transport; Butadienes; Calcium; Cells, Cultured; Chromones; Colforsin; Cyclic AMP; Cyclic GMP; Endothelium, Vascular; Enzyme Inhibitors; Fetus; Flavonoids; Gene Expression; Genistein; Humans; Hydrogen-Ion Concentration; MAP Kinase Signaling System; Membrane Potentials; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Morpholines; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Nitriles; Phenethylamines; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Potassium; Protein Isoforms; Purinergic P1 Receptor Agonists; Receptors, Purinergic P1; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Wortmannin | 2002 |
Forskolin suppresses insulin gene transcription in islet beta-cells through a protein kinase A-independent pathway.
Topics: Base Sequence; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Down-Regulation; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation; Humans; Insulin; Islets of Langerhans; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; Promoter Regions, Genetic; Transcription, Genetic | 2003 |
Interferon-gamma stimulates the expression of the inducible cAMP early repressor in macrophages through the activation of casein kinase 2. A potentially novel pathway for interferon-gamma-mediated inhibition of gene transcription.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Apigenin; Blotting, Western; Calcimycin; Calcium; Casein Kinase II; Cell Line; Cloning, Molecular; Colforsin; Cyclic AMP; Cyclic AMP Response Element Modulator; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; DNA; DNA-Binding Proteins; Electrophoresis, Polyacrylamide Gel; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation, Enzymologic; Genetic Vectors; Imidazoles; Indoles; Interferon-gamma; Macrophages; Maleimides; Mice; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Protein Binding; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; Repressor Proteins; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Thapsigargin; Time Factors; Transcription, Genetic; Transcriptional Activation; Tyrphostins | 2003 |
Role of the different mitogen-activated protein kinase subfamilies in the stimulation of dog and human thyroid epithelial cell proliferation by cyclic adenosine 5'-monophosphate and growth factors.
Topics: Animals; Arsenites; Carcinogens; Cell Division; Cells, Cultured; Colforsin; Cyclic AMP; Dogs; Enzyme Inhibitors; Epidermal Growth Factor; Epithelial Cells; Flavonoids; Hepatocyte Growth Factor; Humans; Hypoglycemic Agents; Imidazoles; Insulin; MAP Kinase Signaling System; Mitogen-Activated Protein Kinases; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pyridines; Sodium Compounds; Tetradecanoylphorbol Acetate; Thyroid Gland; Thyrotropin | 2003 |
Down-regulation of steroidogenic response to gonadotropins in human and rat preovulatory granulosa cells involves mitogen-activated protein kinase activation and modulation of DAX-1 and steroidogenic factor-1.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cell Nucleus; Cells, Cultured; Chorionic Gonadotropin; Colforsin; DAX-1 Orphan Nuclear Receptor; DNA-Binding Proteins; Enzyme Activation; Enzyme Inhibitors; Female; Flavonoids; Follicle Stimulating Hormone; Fushi Tarazu Transcription Factors; Gene Expression; Gonadotropins; Granulosa Cells; Homeodomain Proteins; Humans; Luteinizing Hormone; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Ovulation; Phosphoproteins; Phosphorylation; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Repressor Proteins; Steroidogenic Factor 1; Steroids; Transcription Factors | 2003 |
Evidence that the appressorial development in barley powdery mildew is controlled by MAP kinase activity in conjunction with the cAMP pathway.
Topics: Ascomycota; Cholera Toxin; Colforsin; Cyclic AMP; Enzyme Activators; Enzyme Inhibitors; Flavonoids; Hordeum; Hyphae; Isoquinolines; Mitogen-Activated Protein Kinases; Pertussis Toxin; Signal Transduction; Sphingosine; Sulfonamides; Time Factors | 2003 |
Regulation of melanosome movement by MAP kinase.
Topics: Animals; Blotting, Western; Cell Movement; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Fibroblasts; Flavonoids; Kinetics; MAP Kinase Signaling System; Melanophores; Melanosomes; Microscopy, Phase-Contrast; Mitogen-Activated Protein Kinase 1; Models, Biological; Phosphorylation; Protein Serine-Threonine Kinases; Signal Transduction; Time Factors; Tyrosine; Xenopus laevis | 2003 |
Chronic regulation of the expression of the gap junction protein connexin 43 in transfected HeLa cells.
Topics: Adenylyl Cyclases; Blotting, Western; Colforsin; Connexin 43; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Flavonoids; Fluorescent Antibody Technique; Gap Junctions; Gene Expression Regulation; HeLa Cells; Humans; Imidazoles; Protein Kinase C; Protein-Tyrosine Kinases; Pyridines; Receptors, Tumor Necrosis Factor; Reverse Transcriptase Polymerase Chain Reaction; Signal Transduction; Transfection; Tumor Necrosis Factor-alpha | 2003 |
KCl potentiates forskolin-induced PC12 cell neurite outgrowth via protein kinase A and extracellular signal-regulated kinase signaling pathways.
Topics: Active Transport, Cell Nucleus; Animals; Calcium; Cell Differentiation; Colforsin; Cyclic AMP-Dependent Protein Kinases; Flavonoids; Isoquinolines; MAP Kinase Kinase 1; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Neurites; PC12 Cells; Phosphorylation; Potassium Chloride; Protein Serine-Threonine Kinases; Rats; Signal Transduction; Sulfonamides | 2003 |
Insulin augmentation of 17alpha-hydroxylase activity is mediated by phosphatidyl inositol 3-kinase but not extracellular signal-regulated kinase-1/2 in human ovarian theca cells.
Topics: Androgens; Cells, Cultured; Colforsin; Enzyme Inhibitors; Female; Flavonoids; Gene Expression Regulation, Enzymologic; Humans; Hypoglycemic Agents; Insulin; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Phosphatidylinositol 3-Kinases; Polycystic Ovary Syndrome; RNA, Messenger; Steroid 17-alpha-Hydroxylase; Theca Cells | 2004 |
Cyclic AMP inhibits TGFbeta1-induced cell-scattering and invasiveness in murine-transformed keratinocytes.
Topics: Animals; Cell Line, Transformed; Cell Movement; Cell Transformation, Neoplastic; Colforsin; Cyclic AMP; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation, Enzymologic; Humans; Keratinocytes; Matrix Metalloproteinase 9; Mice; Neoplasm Invasiveness; Recombinant Proteins; Transforming Growth Factor beta; Transforming Growth Factor beta1; Urokinase-Type Plasminogen Activator | 2003 |
Sensitization of adenylate cyclase by short-term activation of 5-HT1A receptors.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Arachidonic Acid; Buspirone; Calcimycin; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Cycloheximide; Dose-Response Relationship, Drug; Flavonoids; Humans; Indoles; Indomethacin; Maleimides; Pertussis Toxin; Phorbol Esters; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1A; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Time Factors; Tryptamines | 2003 |
1,10-Phenanthroline phosphorylates (activates) MAP kinase in Xenopus oocytes.
Topics: Animals; Blotting, Western; Butadienes; Cell-Free System; Chromones; Colforsin; Cycloheximide; Enzyme Inhibitors; Female; Flavonoids; Indoles; Kinetics; Maleimides; Mitogen-Activated Protein Kinase Kinases; Mitogen-Activated Protein Kinases; Morpholines; Nitriles; Oocytes; Pentetic Acid; Phenanthrolines; Phosphorylation; Progesterone; Threonine; Tyrosine; Xenopus laevis; Zinc Sulfate | 2003 |
Induction of cytokine mRNA expression in U937 cells by Salmonella typhimurium porins is regulated by different phosphorylation pathways.
Topics: Colforsin; Cytokines; Enzyme Inhibitors; Flavonoids; Gene Expression Regulation; Humans; Imidazoles; Lipopolysaccharides; Monocytes; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Porins; Proto-Oncogene Proteins c-raf; Pyridines; RNA, Messenger; Salmonella typhimurium; U937 Cells | 2005 |
Salivary phospholipid secretion in response to beta-adrenergic stimulation is mediated by Src kinase-dependent epidermal growth factor receptor transactivation.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Alprenolol; Androstadienes; Animals; Bucladesine; Choline; Colforsin; Enzyme Inhibitors; ErbB Receptors; Flavonoids; Isoproterenol; Phosphoinositide-3 Kinase Inhibitors; Phospholipids; Pyrimidines; Quinazolines; Rats; Receptors, Adrenergic, beta; Saliva; src-Family Kinases; Sublingual Gland; Transcriptional Activation; Wortmannin | 2004 |
Regulation of Na(+)-K(+)-2Cl- cotransporter activity in rat skeletal muscle and intestinal epithelial cells.
Topics: Animals; Bumetanide; Butadienes; Cell Line; Chromones; Colforsin; Cyclic AMP; Enzyme Inhibitors; Epithelial Cells; Flavonoids; Gastrointestinal Tract; Indoles; Isoproterenol; Isoquinolines; Maleimides; Mitogen-Activated Protein Kinases; Morpholines; Muscle, Skeletal; Nitriles; Potassium; Rats; Rubidium Radioisotopes; Sodium-Potassium-Chloride Symporters; Sulfonamides | 2003 |
cAMP-dependent protein kinase type I regulates ethanol-induced cAMP response element-mediated gene expression via activation of CREB-binding protein and inhibition of MAPK.
Topics: Blotting, Western; Cell Line, Tumor; Cell Nucleus; Colforsin; CREB-Binding Protein; Cyclic AMP; Cyclic AMP-Dependent Protein Kinase Type II; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Ethanol; Flavonoids; Gene Expression Regulation; Humans; Immunohistochemistry; Immunoprecipitation; Luciferases; MAP Kinase Signaling System; Models, Biological; Nuclear Proteins; Phosphorylation; Proto-Oncogene Proteins B-raf; Ribosomal Protein S6 Kinases, 90-kDa; Time Factors; Trans-Activators; Transcriptional Activation | 2004 |
Secretion of gastric mucus phospholipids in response to beta-adrenergic G protein-coupled receptor activation is mediated by SRC kinase-dependent epidermal growth factor receptor transactivation.
Topics: Adrenergic beta-Agonists; Animals; Bucladesine; Cells, Cultured; Colforsin; ErbB Receptors; Flavonoids; Gastric Mucosa; Isoproterenol; Phospholipids; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; src-Family Kinases; Transcriptional Activation | 2004 |
Effects of MAP kinase pathway and other factors on meiosis of Urechis unicinctus eggs.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Annelida; Calcimycin; Chromosomes; Colforsin; Cycloheximide; Diglycerides; Extracellular Signal-Regulated MAP Kinases; Fertilization; Flavonoids; MAP Kinase Signaling System; Meiosis; Okadaic Acid; Ovum; Parthenogenesis; Phosphorylation | 2005 |
Activation of mitogen activated protein kinase pathways and melanogenesis by novel nitro-derivatives of 7-hydroxycomarin in human malignant melanoma cells.
Topics: Antineoplastic Agents; Cell Differentiation; Cell Line, Tumor; Colforsin; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Flavonoids; Humans; Imidazoles; MAP Kinase Signaling System; Melanins; Melanoma; Mitogen-Activated Protein Kinases; Monophenol Monooxygenase; Nitro Compounds; Pyridines; Umbelliferones | 2005 |
PACAP protects neuronal differentiated PC12 cells against the neurotoxicity induced by a mitochondrial complex I inhibitor, rotenone.
Topics: Animals; Bucladesine; Caspase 3; Caspases; Cell Differentiation; Cell Survival; Colforsin; Dose-Response Relationship, Drug; Enzyme Inhibitors; Flavonoids; Intracellular Membranes; Isoquinolines; MAP Kinase Signaling System; Membrane Potentials; Mitochondria; Nerve Growth Factors; Neurons; Neuropeptides; Neurosecretory Systems; Neurotransmitter Agents; p38 Mitogen-Activated Protein Kinases; Parkinson Disease; PC12 Cells; Pituitary Adenylate Cyclase-Activating Polypeptide; Protein Kinase Inhibitors; Rats; Rotenone; Signal Transduction; Sulfonamides | 2005 |
cAMP induces neuronal differentiation of mesenchymal stem cells via activation of extracellular signal-regulated kinase/MAPK.
Topics: Adolescent; Blotting, Western; Cell Differentiation; Cells, Cultured; Child; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Enzyme Activation; Enzyme Inhibitors; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Humans; Mesenchymal Stem Cells; Phosphorylation; raf Kinases; Time Factors | 2005 |
Glucose represses connexin36 in insulin-secreting cells.
Topics: Animals; Base Sequence; Cell Line, Tumor; Colforsin; Connexins; Cyclic AMP; Cyclic AMP Response Element Modulator; Cyclic AMP-Dependent Protein Kinases; DNA-Binding Proteins; Down-Regulation; Flavonoids; Gap Junction delta-2 Protein; Glucose; Humans; Insulin-Secreting Cells; Isoquinolines; Mitogen-Activated Protein Kinases; Nifedipine; Promoter Regions, Genetic; Rats; Response Elements; RNA, Messenger; Sequence Deletion; Sulfonamides; Tetradecanoylphorbol Acetate | 2005 |
Oxidative stress contributes to the enhanced expression of Gialpha proteins and adenylyl cyclase signaling in vascular smooth muscle cells from spontaneously hypertensive rats.
Topics: Acetylcysteine; Adenylyl Cyclases; Animals; Antioxidants; Cells, Cultured; Colforsin; Flavonoids; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Guanosine 5'-O-(3-Thiotriphosphate); Hypertension; Isoproterenol; MAP Kinase Signaling System; Models, Biological; Muscle, Smooth, Vascular; Onium Compounds; Oxidative Stress; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Signal Transduction; Superoxides | 2005 |
Thyroid-stimulating hormone stimulates interleukin-6 release from 3T3-L1 adipocytes through a cAMP-protein kinase A pathway.
Topics: 3T3 Cells; Adipocytes; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dactinomycin; Flavonoids; Humans; Interleukin-6; Isoquinolines; Mice; Protein Synthesis Inhibitors; Signal Transduction; Sulfonamides; Thyroid Gland; Thyrotropin | 2005 |
Stimulation of pancreatic beta-cell replication by incretins involves transcriptional induction of cyclin D1 via multiple signalling pathways.
Topics: Adenylyl Cyclases; Androstadienes; Animals; Animals, Newborn; Cell Line; Cell Proliferation; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyclin D1; Enzyme Activation; Flavonoids; Gastric Inhibitory Polypeptide; Glucagon-Like Peptide 1; Human Growth Hormone; Imidazoles; Insulin-Secreting Cells; Isoquinolines; Liraglutide; Mitogen-Activated Protein Kinase Kinases; Phosphoinositide-3 Kinase Inhibitors; Pyridines; Rats; Signal Transduction; Stimulation, Chemical; Sulfonamides; Transcription, Genetic; Transduction, Genetic; Wortmannin | 2006 |
Inositol triphosphate participates in an oestradiol nongenomic signalling pathway involved in accelerated oviductal transport in cycling rats.
Topics: Adenine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Estradiol; Estrus; Fallopian Tubes; Female; Flavonoids; Inositol Phosphates; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase Kinases; Oocytes; Ovum Transport; Phosphatidylcholines; Phospholipid Ethers; Rats; Rats, Sprague-Dawley; Signal Transduction; Type C Phospholipases | 2006 |
Exendin-4 induction of cyclin D1 expression in INS-1 beta-cells: involvement of cAMP-responsive element.
Topics: Animals; Blotting, Western; Cell Line; Cell Proliferation; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Cyclin D1; Dose-Response Relationship, Drug; Exenatide; Flavonoids; Gene Expression; Glucagon-Like Peptide-1 Receptor; Insulin-Secreting Cells; Isoquinolines; Mitogen-Activated Protein Kinase Kinases; Mutagenesis, Site-Directed; Peptides; Phosphorylation; Proto-Oncogene Proteins c-raf; Rats; Rats, Sprague-Dawley; Receptors, Glucagon; Response Elements; RNA, Messenger; Sulfonamides; Venoms | 2006 |
Gonadotropin regulation of testosterone production by primary cultured theca and granulosa cells of Atlantic croaker: II. Involvement of a mitogen-activated protein kinase pathway.
Topics: Adenylyl Cyclases; Animals; Calcium; Cell Culture Techniques; Coculture Techniques; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Extracellular Signal-Regulated MAP Kinases; Female; Flavonoids; Gonadotropins; Granulosa Cells; MAP Kinase Kinase 1; MAP Kinase Kinase 2; Mitogen-Activated Protein Kinase 3; Models, Biological; Ovarian Follicle; Perciformes; Signal Transduction; Testosterone; Theca Cells | 2006 |
Regulation of plasminogen activators in human thyroid follicular cells and their relationship to differentiated function.
Topics: Adenylyl Cyclases; Aprotinin; Cell Differentiation; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activators; Epidermal Growth Factor; Fibroblast Growth Factors; Flavonoids; Humans; Indoles; Insulin; Iodine; Iodine Radioisotopes; Maleimides; Mesylates; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Plasminogen Inactivators; Protein Kinase C; Protein Kinase C beta; Protein Kinase Inhibitors; Pyrroles; RNA, Messenger; Serine Proteinase Inhibitors; Signal Transduction; Tetradecanoylphorbol Acetate; Thyroid Gland; Thyrotropin; Time Factors; Tissue Plasminogen Activator; Urokinase-Type Plasminogen Activator | 2007 |
Transcriptional regulation of follistatin expression by GnRH in mouse gonadotroph cell lines: evidence for a role for cAMP signaling.
Topics: Animals; Cell Line; Colforsin; Cyclic AMP; Enzyme Inhibitors; Flavonoids; Follistatin; Gene Expression Regulation; Genes, Reporter; Gonadotrophs; Gonadotropin-Releasing Hormone; Mice; Promoter Regions, Genetic; Recombinant Fusion Proteins; Second Messenger Systems; Transcription, Genetic | 2007 |
The Src tyrosine kinase pathway regulates thecal CYP17 expression and androstenedione secretion.
Topics: Androstenedione; Animals; Cholesterol Side-Chain Cleavage Enzyme; Colforsin; Cyclic AMP; Dual Specificity Phosphatase 1; Female; Flavonoids; MAP Kinase Kinase 1; Mice; Mice, Inbred C57BL; Phosphoproteins; Promoter Regions, Genetic; Pyrimidines; src-Family Kinases; Steroid 17-alpha-Hydroxylase; Steroidogenic Factor 1; Theca Cells | 2008 |
The guanine nucleotide exchange factor, C3G regulates differentiation and survival of human neuroblastoma cells.
Topics: cdc42 GTP-Binding Protein; Cell Differentiation; Cell Line, Tumor; Cell Survival; Colforsin; Culture Media, Serum-Free; Enzyme Inhibitors; Flavonoids; Green Fluorescent Proteins; Guanine Nucleotide-Releasing Factor 2; Humans; Nerve Growth Factor; Neurites; Neuroblastoma; rap1 GTP-Binding Proteins; RNA, Small Interfering; Transfection | 2008 |
Involvement of regulatory elements on corticotropin-releasing factor gene promoter in hypothalamic 4B cells.
Topics: Anthracenes; Cell Line; Chromones; Colforsin; Corticotropin-Releasing Hormone; Dexamethasone; Flavonoids; Genes, Reporter; Humans; Hypothalamus; Imidazoles; Isoquinolines; Morpholines; Promoter Regions, Genetic; Protein Kinase Inhibitors; Pyridines; Regulatory Elements, Transcriptional; Sequence Deletion; Sulfonamides; Transfection | 2008 |
cAMP-induced auditory supporting cell proliferation is mediated by ERK MAPK signaling pathway.
Topics: Animals; Antimetabolites; Apigenin; Birds; Bromodeoxyuridine; Butadienes; Cell Division; Colforsin; Cyclic AMP; Enzyme Inhibitors; Epithelial Cells; Extracellular Signal-Regulated MAP Kinases; Flavonoids; Hair Cells, Auditory; Macrolides; MAP Kinase Signaling System; Myosin VIIa; Myosins; Nitriles; Organ Culture Techniques; Organ of Corti; Proto-Oncogene Proteins B-raf | 2010 |
Apical leptin induces chloride secretion by intestinal epithelial cells and in a rat model of acute chemotherapy-induced colitis.
Topics: Androstadienes; Animals; Carbachol; Cell Line; Chlorides; Colforsin; Enterocolitis; Epithelial Cells; Flavonoids; Humans; Leptin; Male; MAP Kinase Signaling System; Methotrexate; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Rats; Rats, Sprague-Dawley; Signal Transduction; Wortmannin | 2010 |
Synergistic effect of vasoactive intestinal peptides on TNF-alpha-induced IL-6 synthesis in osteoblasts: amplification of p44/p42 MAP kinase activation.
Topics: 3T3 Cells; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cells, Cultured; Colforsin; Enzyme Activation; Flavonoids; Interleukin-6; Isoquinolines; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Osteoblasts; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Sulfonamides; Tumor Necrosis Factor-alpha; Vasoactive Intestinal Peptide | 2010 |
Effects of nonylphenol on the production of progesterone on the rats granulosa cells.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cells, Cultured; Chorionic Gonadotropin; Colforsin; Environmental Pollutants; Estrogens; Female; Flavonoids; Granulosa Cells; Humans; Maternal Exposure; Phenols; Phosphoproteins; Pregnancy; Pregnenolone; Prenatal Exposure Delayed Effects; Progesterone; Rats; Reproductive Control Agents | 2011 |
Moderate superoxide production is an early promoter of mitochondrial biogenesis in differentiating N2a neuroblastoma cells.
Topics: Animals; Biomarkers; Bucladesine; Cell Cycle; Cell Line, Tumor; Colforsin; Culture Media, Serum-Free; Cyclic AMP; Flavonoids; Free Radical Scavengers; Hormesis; MAP Kinase Signaling System; Metalloporphyrins; Mice; Mitochondria; Neurites; Neuroblastoma; Neurogenesis; Second Messenger Systems; Superoxides | 2012 |
Retinoic acid impairs estrogen signaling in breast cancer cells by interfering with activation of LSD1 via PKA.
Topics: Breast Neoplasms; Catalytic Domain; Chromatin; Colforsin; Cyclic AMP-Dependent Protein Kinases; Estrogens; Female; Flavonoids; Histone Demethylases; Histones; Humans; Isoquinolines; MAP Kinase Signaling System; MCF-7 Cells; Methylation; Protein Processing, Post-Translational; Proto-Oncogene Proteins c-bcl-2; RNA, Small Interfering; Sulfonamides; Transcription, Genetic; Tretinoin | 2013 |
Neuronal nitric oxide synthase-dependent elevation in adiponectin in the rostral ventrolateral medulla underlies g protein-coupled receptor 18-mediated hypotension in conscious rats.
Topics: Adenylyl Cyclases; Adiponectin; Androstadienes; Animals; Anisoles; Arginine; Colforsin; Consciousness; Cyclic AMP; Cyclohexanes; Flavonoids; Hypotension; Male; Medulla Oblongata; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Nitric Oxide; Nitric Oxide Synthase Type I; Oxidative Stress; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Phosphorylation; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Wortmannin | 2014 |
Recruitment of endosomal signaling mediates the forskolin modulation of guinea pig cardiac neuron excitability.
Topics: Adenylyl Cyclases; Animals; Carbazoles; Clathrin; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Endosomes; Flavonoids; Guinea Pigs; Heart; Humans; MAP Kinase Signaling System; Myocardium; Neurons; Pituitary Adenylate Cyclase-Activating Polypeptide; Pyrroles; Receptors, G-Protein-Coupled; Receptors, Pituitary Adenylate Cyclase-Activating Polypeptide, Type I | 2017 |
Forskolin improves sensitivity to doxorubicin of triple negative breast cancer cells via Protein Kinase A-mediated ERK1/2 inhibition.
Topics: Cell Line, Tumor; Colforsin; Cyclic AMP-Dependent Protein Kinases; Doxorubicin; Extracellular Signal-Regulated MAP Kinases; Female; Flavonoids; Gene Expression Regulation, Enzymologic; Gene Expression Regulation, Neoplastic; Humans; Protein Kinase Inhibitors; Triple Negative Breast Neoplasms | 2018 |