colforsin has been researched along with oxotremorine in 29 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 8 (27.59) | 18.7374 |
1990's | 14 (48.28) | 18.2507 |
2000's | 6 (20.69) | 29.6817 |
2010's | 1 (3.45) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Ehlert, FJ; Griffin, MT | 1 |
Bleasdale, JE; Denlinger, LC; Fisher, SK; Mostafapour, SP; Thompson, AK | 1 |
Lovenberg, TW; Mailman, RB; Nichols, DE; Roth, RH | 1 |
Nezu, E; Yoneyama, T; Yoshimura, K | 1 |
Baumgold, J; Fishman, PH | 1 |
Fertel, R; Hadjiconstantinou, M; Neff, NH; Qu, ZX | 1 |
Henis, YI; Moscona-Amir, E; Sokolovsky, M | 1 |
Brown, BL; Dobson, PR; Quilliam, LA | 1 |
Costa, E; Eva, C | 1 |
Desjardins, D; Heisler, S; Nguyen, MH | 1 |
Evans, T; Harden, TK; Hepler, JR; Hughes, AR; Martin, MW; Meeker, RB; Smith, MM; Tanner, LI | 1 |
Ehlert, FJ; Thomas, EA | 2 |
Ehlert, FJ; Gerstin, EH | 1 |
Ehlert, FJ; Esqueda, EE; Gerstin, EH; Griffin, MT | 1 |
Anand-Srivastava, MB; Marcil, J; Thibault, C | 1 |
Ehlert, FJ; Sawyer, GW | 1 |
Ehlert, FJ; Ostrom, RS | 2 |
Islam, MA; Kimura, I; Nojima, H | 1 |
Berger, JG; Brown, J; Clader, J; Duffy, RA; Guzik, H; Kozlowski, J; Lachowicz, JE; Lowe, D; McQuade, R; Murgolo, N; Ruperto, V; Strader, CD; Taylor, LA; Tice, M | 1 |
Ehlert, F; Sawyer, G | 1 |
Anand-Srivastava, MB; Boumati, M; Li, Y | 1 |
Anand-Srivastava, MB; Di Fusco, F | 1 |
Abe, DM; Ehlert, FJ; Griffin, MT; Manabe, T; Matsui, M; Taketo, MM; Vo, TH | 1 |
Barak, D; Pittel, Z; Segall, Y | 1 |
Ehlert, FJ; Figueroa, KW; Griffin, MT; Liller, S | 1 |
Aguirre, A; Cerveñansky, C; Colettis, N; Jerusalinsky, D; Kornisiuk, E; Quillfeldt, JA; Sánchez, G; Vázquez, P | 1 |
Ehlert, FJ; Matsui, M; Ostrom, RS; Pak, KJ | 1 |
1 review(s) available for colforsin and oxotremorine
Article | Year |
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Functional role of M2 muscarinic receptors in the guinea pig ileum.
Topics: Animals; Colforsin; Cyclic AMP; Guinea Pigs; Heart; Histamine; Ileum; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pertussis Toxin; Piperidines; Rats; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Signal Transduction; Submandibular Gland; Virulence Factors, Bordetella | 1995 |
28 other study(ies) available for colforsin and oxotremorine
Article | Year |
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Specific inhibition of isoproterenol-stimulated cyclic AMP accumulation by M2 muscarinic receptors in rat intestinal smooth muscle.
Topics: Adenylyl Cyclases; Animals; Binding Sites; Colforsin; Cyclic AMP; Enzyme Activation; Ileum; Isoproterenol; Male; Muscle, Smooth; Oxotremorine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic | 1992 |
The aminosteroid U-73122 inhibits muscarinic receptor sequestration and phosphoinositide hydrolysis in SK-N-SH neuroblastoma cells. A role for Gp in receptor compartmentation.
Topics: Alprostadil; Cell Line; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Down-Regulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Estrenes; GTP-Binding Proteins; Humans; Inositol; Kinetics; Neuroblastoma; Oxotremorine; Phosphatidylinositols; Pyrrolidinones; Receptors, Muscarinic; Scopolamine; Type C Phospholipases | 1991 |
D1 dopamine receptors of NS20Y neuroblastoma cells are functionally similar to rat striatal D1 receptors.
Topics: Benzazepines; Butaclamol; Carbachol; Cell Line; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine; Dopamine Agents; Flupenthixol; Kinetics; Neuroblastoma; Oxotremorine; Phenanthridines; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D1; Sulpiride; Tubocurarine | 1991 |
Augmentation of isoproterenol-stimulated tissue cyclic AMP level by cholinergic agonists in rat parotid gland.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Calcimycin; Calcium; Carbachol; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Isoproterenol; Male; Methacholine Chloride; Methacholine Compounds; Norepinephrine; Oxotremorine; Parotid Gland; Phentolamine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains | 1985 |
Muscarinic receptor-mediated increase in cAMP levels in SK-N-SH human neuroblastoma cells.
Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Carbachol; Cell Line; Colforsin; Cyclic AMP; Humans; Kinetics; Neuroblastoma; Oxotremorine; Pertussis Toxin; Receptors, Muscarinic; Virulence Factors, Bordetella | 1988 |
Pharmacological characterization of muscarinic receptors mediating inhibition of adenylate cyclase activity in the rat retina.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Adenylyl Cyclase Inhibitors; Animals; Arecoline; Aziridines; Carbachol; Choline; Colforsin; Cyclic AMP; Male; Oxotremorine; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Retina | 1988 |
Aging of rat heart myocytes disrupts muscarinic receptor coupling that leads to inhibition of cAMP accumulation and alters the pathway of muscarinic-stimulated phosphoinositide hydrolysis.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Binding, Competitive; Carbachol; Cells, Cultured; Cholera Toxin; Colforsin; Cyclic AMP; Heart; Isoproterenol; Kinetics; Myocardium; Norepinephrine; Oxotremorine; Phosphatidylinositols; Rats; Receptors, Muscarinic; Time Factors | 1989 |
Regulation of GH3 pituitary tumour-cell adenylate cyclase activity by activators of protein kinase C.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Bombesin; Cholera Toxin; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activation; Humans; Oxotremorine; Phorbol 12,13-Dibutyrate; Pituitary Neoplasms; Protein Kinase C; Tumor Cells, Cultured; Type C Phospholipases; Vasoactive Intestinal Peptide | 1989 |
In rat hippocampus, somatostatin 14 and muscarinic receptor ligands modulate an adenylate cyclase belonging to a common domain of the receptor.
Topics: Acetylcholine; Adenylyl Cyclase Inhibitors; Animals; Carbachol; Colforsin; GTP Phosphohydrolases; Hippocampus; Hydrolysis; Oxotremorine; Phosphatidylinositols; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Somatostatin | 1987 |
Muscarinic cholinergic receptors in mouse pituitary tumor cells: prolonged agonist pretreatment decreases receptor content and increases forskolin- and hormone-stimulated cyclic AMP synthesis and adrenocorticotropin secretion.
Topics: Adrenocorticotropic Hormone; Animals; Cell Line; Colforsin; Cyclic AMP; Cycloheximide; Diterpenes; Hormones; Mice; Oxotremorine; Pituitary Gland; Pituitary Neoplasms; Quinuclidinyl Benzilate; Receptors, Muscarinic; Scopolamine; Time Factors | 1985 |
Regulation of cyclic AMP metabolism by muscarinic cholinergic receptors.
Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Adenylyl Cyclases; Alprostadil; Animals; Bacterial Toxins; Calcium; Cell Line; Colforsin; Cyclic AMP; Diterpenes; Humans; Isoproterenol; Kinetics; Mice; Molecular Weight; Oxotremorine; Phosphodiesterase Inhibitors; Prostaglandins E; Receptors, Adrenergic, beta; Receptors, Muscarinic; Virulence Factors, Bordetella | 1985 |
Involvement of the M2 muscarinic receptor in contractions of the guinea pig trachea, guinea pig esophagus, and rat fundus.
Topics: Adrenergic beta-Agonists; Animals; Colforsin; Cyclic AMP; Esophagus; Gastric Fundus; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Pertussis Toxin; Pirenzepine; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Serotonin; Trachea; Virulence Factors, Bordetella | 1996 |
Inhibition of muscarinic stimulated phosphoinositide hydrolysis in the rat parotid gland by cAMP.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic beta-Antagonists; Animals; Calcium; Colforsin; Cyclic AMP; Dinoprostone; Drug Interactions; Hydrolysis; Isoproterenol; Male; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Parotid Gland; Phosphatidylinositols; Phosphodiesterase Inhibitors; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Sodium Fluoride; Stimulation, Chemical | 1996 |
Stimulation of cyclic AMP accumulation and phosphoinositide hydrolysis by M3 muscarinic receptors in the rat peripheral lung.
Topics: Animals; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Hydrolysis; Lung; Male; Oxotremorine; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic | 1996 |
Enhanced expression of Gi-protein precedes the development of blood pressure in spontaneously hypertensive rats.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Age Factors; Animals; Animals, Newborn; Aorta; Atrial Natriuretic Factor; Blood Pressure; Colforsin; Enzyme Inhibitors; Gene Expression Regulation, Developmental; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Hormones; Hypertension; Muscarinic Agonists; Myocardium; Oxotremorine; Rats; Rats, Inbred SHR; RNA, Messenger | 1997 |
Contractile roles of the M2 and M3 muscarinic receptors in the guinea pig colon.
Topics: Animals; Colforsin; Colon; Cyclic AMP; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Oxotremorine; Pertussis Toxin; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Receptors, Muscarinic; Virulence Factors, Bordetella | 1998 |
M2 muscarinic receptors inhibit forskolin- but not isoproterenol-mediated relaxation in bovine tracheal smooth muscle.
Topics: Animals; Cattle; Colforsin; Cyclic AMP; Diphenylacetic Acids; Histamine; In Vitro Techniques; Isoproterenol; Muscle Relaxation; Muscle, Smooth; Oxotremorine; Piperidines; Receptor, Muscarinic M2; Receptors, Muscarinic; Trachea | 1998 |
Acetylcholine-induced biphasic effect on the maximum upstroke velocity of action potential in mouse right atria: interaction with beta-adrenergic signaling cascade.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Action Potentials; Adenylate Cyclase Toxin; Adjuvants, Immunologic; Adrenergic beta-Agonists; Animals; Cholera Toxin; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; GTP-Binding Protein alpha Subunits, Gi-Go; Heart; Heart Atria; Heart Rate; In Vitro Techniques; Isoproterenol; Isoquinolines; Kinetics; Male; Mice; Muscarinic Agonists; Naphthalenes; Oxotremorine; Protein Kinase C; Receptors, Adrenergic, beta; Sulfonamides; Virulence Factors, Bordetella | 1998 |
Comparison of functional antagonism between isoproterenol and M2 muscarinic receptors in guinea pig ileum and trachea.
Topics: Animals; Colforsin; Diphenylacetic Acids; Guinea Pigs; Histamine; Ileum; Isoproterenol; Muscle Relaxation; Oxotremorine; Pertussis Toxin; Piperidines; Pirenzepine; Receptor, Muscarinic M2; Receptors, Muscarinic; Trachea; Virulence Factors, Bordetella | 1999 |
SCH 57790: a novel M2 receptor selective antagonist.
Topics: Acetylcholine; Adenylyl Cyclases; Alzheimer Disease; Animals; Binding Sites; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Humans; Muscarinic Agonists; Muscarinic Antagonists; Oxotremorine; Piperazines; Quinuclidinyl Benzilate; Receptor, Muscarinic M2; Receptors, Muscarinic; Transfection | 1999 |
Pertussis toxin increases isoproterenol induced relaxation in field-stimulated ileum.
Topics: Animals; Colforsin; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Histamine; Histamine Agonists; Ileum; In Vitro Techniques; Isoproterenol; Male; Muscarinic Agonists; Muscle Contraction; Muscle Relaxation; Oxotremorine; Pertussis Toxin; Sympathomimetics; Virulence Factors, Bordetella | 1999 |
Modulation of ANP-C receptor signaling by endothelin-1 in A-10 smooth muscle cells.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Angiotensin II; Animals; Atrial Natriuretic Factor; Cell Line; Colforsin; Down-Regulation; Endothelin-1; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; GTP-Binding Proteins; Guanylate Cyclase; Kinetics; Muscle, Smooth, Vascular; Oxotremorine; Peptide Fragments; Rats; Receptors, Atrial Natriuretic Factor; Signal Transduction; Sodium Fluoride | 2002 |
Redox modulation of Gi protein expression and adenylyl cyclase signaling: role of nitric oxide.
Topics: Adenylyl Cyclases; Angiotensin II; Animals; Blood Pressure; Cholera Toxin; Colforsin; Enzyme Inhibitors; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Guanosine 5'-O-(3-Thiotriphosphate); Heart; Male; Muscarinic Agonists; Myocardium; NG-Nitroarginine Methyl Ester; Nitric Oxide; Oxidation-Reduction; Oxotremorine; Rats; Rats, Sprague-Dawley; Signal Transduction; Tissue Extracts | 2004 |
The M2 muscarinic receptor mediates contraction through indirect mechanisms in mouse urinary bladder.
Topics: Adrenergic beta-Agonists; Animals; Binding, Competitive; Colforsin; Dinoprost; Diphenylacetic Acids; In Vitro Techniques; Isoproterenol; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscarinic Agonists; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Oxotremorine; Piperidines; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Urinary Bladder | 2005 |
Function-specific blockage of M(1) and M(3) muscarinic acetylcholine receptors by VX and echothiophate.
Topics: Animals; Atropine; CHO Cells; Cholinesterase Inhibitors; Colforsin; Cricetinae; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Echothiophate Iodide; Muscarinic Agonists; Muscarinic Antagonists; N-Methylscopolamine; Organothiophosphorus Compounds; Oxotremorine; Phosphatidylinositols; Protein Binding; Receptor, Muscarinic M1; Receptor, Muscarinic M3; Transfection; Tritium | 2006 |
Estimation of agonist activity at G protein-coupled receptors: analysis of M2 muscarinic receptor signaling through Gi/o,Gs, and G15.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Algorithms; Animals; Carbachol; Cell Line; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Diphenylacetic Acids; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gq-G11; GTP-Binding Protein alpha Subunits, Gs; Heterotrimeric GTP-Binding Proteins; Humans; Isoproterenol; Oxotremorine; Pertussis Toxin; Phosphatidylinositols; Piperidines; Pirenzepine; Quinuclidines; Receptor, Muscarinic M2; Signal Transduction; Transfection | 2007 |
Muscarinic inhibition of hippocampal and striatal adenylyl cyclase is mainly due to the M(4) receptor.
Topics: Adenylyl Cyclases; Amygdala; Animals; Colforsin; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Hippocampus; Male; Muscarinic Agonists; Muscarinic Antagonists; Neostriatum; Oxotremorine; Rats; Rats, Wistar; Receptor, Muscarinic M4 | 2009 |
Impaired M3 and enhanced M2 muscarinic receptor contractile function in a streptozotocin model of mouse diabetic urinary bladder.
Topics: Animals; Colforsin; Diabetes Mellitus, Experimental; Disease Models, Animal; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscarinic Agonists; Muscle Contraction; Oxotremorine; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Streptozocin; Time Factors; Urinary Bladder | 2010 |