Page last updated: 2024-08-23

colforsin and methacholine chloride

colforsin has been researched along with methacholine chloride in 31 studies

Research

Studies (31)

TimeframeStudies, this research(%)All Research%
pre-19907 (22.58)18.7374
1990's13 (41.94)18.2507
2000's9 (29.03)29.6817
2010's2 (6.45)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Diamond, J; Giembycz, MA1
Nezu, E; Yoneyama, T; Yoshimura, K1
Linden, J1
Sato, F; Sato, K1
Brown, JK; Madison, JM1
Fiscus, RR; Mayer, SE; Peterson, SM; Rinard, GA; Torphy, TJ; Zheng, C1
Shuttleworth, TJ; Thompson, JL1
Armour, CL; Hogg, JC; Paré, PD; Schellenberg, RR; Taylor, SM1
Finkbeiner, WE; Mrsny, RJ; Shen, BQ; Widdicombe, JH; Wine, JJ1
Pyne, NJ; Stevens, PA1
Cavallin, S; Sato, F; Sato, K; Sato, KT1
Jackson, WF1
Black, C; Curry, C; Emala, C; Hirshman, CA; Levine, MA1
Ohtsuyama, M; Sato, F; Sato, K1
Adem, A; Karlsson, E; Olianas, MC; Onali, P1
Elzinga, CR; Hoiting, BH; Kuipers, R; Meurs, H; Schuiling, M; Zaagsma, J1
Knutsen, D; Sato, K; Soos, G; Toyomoto, T1
Kume, H; Takagi, K1
Bast, A; Kramer, K; Smink, CG1
Tabrizchi, R1
Heijenbrok, FJ; Mathy, MJ; Pfaffendorf, M; van Zwieten, PA1
Ito, S; Ito, Y; Kume, H; Yamaki, K1
Ishikawa, T; Ito, S; Kotlikoff, MI; Kume, H; Oguma, T; Shimokata, K1
Ishikawa, T; Ito, Y; Kondo, M; Kume, H; Shimokata, K; Yamaki, K1
Boterman, M; Elzinga, CR; Eppens, PB; Meurs, H; Wagemakers, D; Zaagsma, J1
Honjo, H; Ito, S; Kamiya, K; Kodama, I; Kume, H; Oguma, T; Shimokata, K; Takeda, N1
Bai, Y; Sanderson, MJ1
de la Cal, C; Elverdin, JC; Fernández-Solari, J; Iribarne, M; McCann, SM; Prestifilippo, JP; Rettori, V; Suburo, AM1
Elverdin, JC; Fernandez-Solari, J; Ossola, CA; Prestifilippo, JP; Rettori, V1
Danielsson, J; Emala, CW; Funayama, H; Gallos, G; Kim, B; Worgall, TS; Xu, D; Yim, PD; Zaidi, S1

Other Studies

31 other study(ies) available for colforsin and methacholine chloride

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Partial characterization of cyclic AMP-dependent protein kinases in guinea-pig lung employing the synthetic heptapeptide substrate, kemptide. In vitro sensitivity of the soluble enzyme to isoprenaline, forskolin, methacholine and leukotriene D4.
    Biochemical pharmacology, 1990, Apr-15, Volume: 39, Issue:8

    Topics: Adenosine Triphosphate; Animals; Carrier Proteins; Chromatography, DEAE-Cellulose; Colforsin; Cyclic AMP; Cyclic GMP; Enzyme Activation; Guinea Pigs; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Isoenzymes; Isoproterenol; Lung; Magnesium; Male; Methacholine Chloride; Methacholine Compounds; Oligopeptides; Protein Kinase Inhibitors; Protein Kinases; Solubility; SRS-A

1990
Augmentation of isoproterenol-stimulated tissue cyclic AMP level by cholinergic agonists in rat parotid gland.
    The Japanese journal of physiology, 1985, Volume: 35, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Calcimycin; Calcium; Carbachol; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Isoproterenol; Male; Methacholine Chloride; Methacholine Compounds; Norepinephrine; Oxotremorine; Parotid Gland; Phentolamine; Pilocarpine; Quinuclidinyl Benzilate; Rats; Rats, Inbred Strains

1985
Enhanced cAMP accumulation after termination of cholinergic action in the heart.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 1987, Volume: 1, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Atropine; Cells, Cultured; Chick Embryo; Colforsin; Cyclic AMP; Heart; Isoproterenol; Methacholine Chloride; Methacholine Compounds; Myocardial Contraction; Myocardium; Parasympathomimetics; Pindolol; Receptors, Muscarinic

1987
Effect of VIP on sweat secretion and cAMP accumulation in isolated simian eccrine glands.
    The American journal of physiology, 1987, Volume: 253, Issue:6 Pt 2

    Topics: Animals; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Eccrine Glands; Macaca mulatta; Methacholine Chloride; Methacholine Compounds; Sweat Glands; Sweating; Vasoactive Intestinal Peptide

1987
Differential inhibitory effects of forskolin, isoproterenol, and dibutyryl cyclic adenosine monophosphate on phosphoinositide hydrolysis in canine tracheal smooth muscle.
    The Journal of clinical investigation, 1988, Volume: 82, Issue:4

    Topics: Animals; Bucladesine; Colforsin; Dogs; Histamine; Hydrolysis; Isoproterenol; Methacholine Chloride; Methacholine Compounds; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Trachea

1988
Inhibitory effect of methacholine on drug-induced relaxation, cyclic AMP accumulation, and cyclic AMP-dependent protein kinase activation in canine tracheal smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 1985, Volume: 233, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Colforsin; Cyclic AMP; Dinoprostone; Diterpenes; Dogs; Enzyme Activation; In Vitro Techniques; Isoproterenol; Methacholine Chloride; Methacholine Compounds; Muscle Relaxation; Muscle, Smooth; Prostaglandins E; Protein Kinases; Trachea

1985
Secretory activity in salt glands of birds and turtles: stimulation via cyclic AMP.
    The American journal of physiology, 1987, Volume: 252, Issue:2 Pt 2

    Topics: Animals; Calcimycin; Colforsin; Cyclic AMP; Ducks; Methacholine Chloride; Methacholine Compounds; Salt Gland; Stimulation, Chemical; Turtles

1987
Airway reactivity in chronic obstructive pulmonary disease. Failure of in vivo methacholine responsiveness to correlate with cholinergic, adrenergic, or nonadrenergic responses in vitro.
    The American review of respiratory disease, 1985, Volume: 132, Issue:1

    Topics: Aged; Albuterol; Bronchi; Bronchial Provocation Tests; Colforsin; Diterpenes; Female; Forced Expiratory Volume; Humans; In Vitro Techniques; Lung Diseases, Obstructive; Male; Methacholine Chloride; Methacholine Compounds; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Pneumonectomy

1985
Calu-3: a human airway epithelial cell line that shows cAMP-dependent Cl- secretion.
    The American journal of physiology, 1994, Volume: 266, Issue:5 Pt 1

    Topics: Bradykinin; Bumetanide; Calcimycin; Cell Line; Cell Membrane; Cell Membrane Permeability; Chloride Channels; Chlorides; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Cytoplasmic Granules; Desmosomes; Epithelium; Histamine; Humans; Intercellular Junctions; Isoproterenol; Kinetics; Lung Neoplasms; Membrane Proteins; Methacholine Chloride; Microscopy, Electron; Nystatin; Ouabain; Sodium; Trypsin; Tumor Cells, Cultured

1994
The inhibition of adenylyl cyclase activity in isolated lung membranes by muscarinic and alpha-adrenoceptor agonists: role of G-protein alpha and beta gamma sub-units.
    Cellular signalling, 1995, Volume: 7, Issue:2

    Topics: Adenosine Diphosphate Ribose; Adenylyl Cyclase Inhibitors; Adrenergic alpha-Agonists; Animals; Cholera Toxin; Clonidine; Colforsin; GTP-Binding Proteins; Guanine Nucleotides; Guanylyl Imidodiphosphate; Guinea Pigs; In Vitro Techniques; Lung; Male; Membranes; Methacholine Chloride; Muscarinic Agonists; Norepinephrine; Protein Conformation

1995
Secretion of ions and pharmacological responsiveness in the mouse paw sweat gland.
    Clinical science (London, England : 1979), 1994, Volume: 86, Issue:2

    Topics: Aging; Animals; Colforsin; Culture Techniques; Cyclic AMP; Eccrine Glands; Forelimb; Isoproterenol; Male; Methacholine Chloride; Mice; Mice, Inbred BALB C; Potassium; Sodium

1994
Arteriolar tone is determined by activity of ATP-sensitive potassium channels.
    The American journal of physiology, 1993, Volume: 265, Issue:5 Pt 2

    Topics: Adenosine Triphosphate; Animals; Arterioles; Benzopyrans; Bucladesine; Colforsin; Cricetinae; Cromakalim; Epoprostenol; Glyburide; Guanidines; Isoproterenol; Male; Mesocricetus; Methacholine Chloride; Muscle Tonus; Muscle, Smooth, Vascular; Muscles; Nitroprusside; Pinacidil; Potassium Channels; Pyrroles; Quaternary Ammonium Compounds; Vasoconstriction; Vasodilation; Vasodilator Agents

1993
Impaired beta-adrenergic receptor activation of adenylyl cyclase in airway smooth muscle in the basenji-greyhound dog model of airway hyperresponsiveness.
    American journal of respiratory cell and molecular biology, 1993, Volume: 8, Issue:6

    Topics: Adenylyl Cyclases; Analysis of Variance; Animals; Bronchial Hyperreactivity; Bucladesine; Cholera Toxin; Colforsin; Dinoprostone; Disease Models, Animal; Dogs; Enzyme Activation; Immunoblotting; Isoproterenol; Lung; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Radioimmunoassay; Receptors, Adrenergic, beta; Trachea

1993
Whole cell K and Cl currents in dissociated eccrine secretory coil cells during stimulation.
    The Journal of membrane biology, 1993, Volume: 134, Issue:2

    Topics: Animals; Barium; Cells, Cultured; Chloride Channels; Colforsin; Cyclic AMP; Eccrine Glands; Electric Stimulation; Ionomycin; Isoproterenol; Macaca mulatta; Membrane Potentials; Methacholine Chloride; Models, Biological; Potassium Channels; Quinidine; Sodium; Time Factors

1993
Rat striatal muscarinic receptors coupled to the inhibition of adenylyl cyclase activity: potent block by the selective m4 ligand muscarinic toxin 3 (MT3).
    British journal of pharmacology, 1996, Volume: 118, Issue:2

    Topics: Acetylcholine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Cerebral Cortex; Colforsin; Corpus Striatum; Enzyme Activation; In Vitro Techniques; Inositol Phosphates; Intercellular Signaling Peptides and Proteins; Ligands; Male; Methacholine Chloride; Muscarinic Antagonists; Peptides; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M4; Receptors, Dopamine D1; Receptors, Muscarinic; Tritium

1996
Modulation of agonist-induced phosphoinositide metabolism, Ca2+ signalling and contraction of airway smooth muscle by cyclic AMP-dependent mechanisms.
    British journal of pharmacology, 1996, Volume: 117, Issue:3

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic beta-Agonists; Animals; Calcium; Cattle; Cells, Cultured; Cholinergic Agents; Colforsin; Cyclic AMP; Histamine; Isoproterenol; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Signal Transduction; Trachea

1996
Na-K-2Cl cotransporters are present and regulated in simian eccrine clear cells.
    The American journal of physiology, 1997, Volume: 273, Issue:1 Pt 2

    Topics: Amiloride; Animals; Bumetanide; Carrier Proteins; Cells, Cultured; Colforsin; Cyclic AMP; Eccrine Glands; Hand; Homeostasis; Humans; Hypertonic Solutions; Hypotonic Solutions; Isoproterenol; Macaca mulatta; Methacholine Chloride; Ouabain; Polymerase Chain Reaction; RNA, Messenger; Sodium; Sodium-Potassium-Chloride Symporters; Tetradecanoylphorbol Acetate; Transcription, Genetic

1997
Inhibitory effects of Gs on desensitization of beta-adrenergic receptors in tracheal smooth muscle.
    The American journal of physiology, 1997, Volume: 273, Issue:3 Pt 1

    Topics: Adrenergic beta-Agonists; Animals; Cholera Toxin; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; GTP-Binding Proteins; Guinea Pigs; In Vitro Techniques; Isometric Contraction; Isoproterenol; Kinetics; Male; Methacholine Chloride; Muscle Relaxation; Muscle, Smooth; Receptors, Adrenergic, beta; Thionucleotides; Time Factors; Trachea

1997
Effect of phospholipase A2 activation on the receptor function in the rat left atrium: unmasking of a positive inotropic effect of methacholine.
    General pharmacology, 1997, Volume: 29, Issue:3

    Topics: Adrenergic beta-Agonists; Animals; Cardiotonic Agents; Colforsin; Enzyme Activation; Enzyme Inhibitors; Heart; Heart Atria; In Vitro Techniques; Isoproterenol; Melitten; Methacholine Chloride; Muscarinic Agonists; Myocardial Contraction; Phospholipases A; Phospholipases A2; Quinacrine; Rats; Rats, Wistar; Receptors, Neurotransmitter

1997
Influence of increase in osmotic pressure with sucrose on relaxation and cyclonucleotides levels in isolated rat aorta.
    European journal of pharmacology, 1999, Oct-15, Volume: 382, Issue:3

    Topics: Adrenergic beta-Agonists; Animals; Aorta, Thoracic; Colforsin; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Hypertonic Solutions; In Vitro Techniques; Isoproterenol; Male; Methacholine Chloride; Muscarinic Agonists; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Osmotic Pressure; Pinacidil; Rats; Rats, Sprague-Dawley; Sucrose; Vasodilator Agents

1999
The influence of chronic inhibition of nitric oxide synthesis on contractile and relaxant properties of rat carotid and mesenteric arteries.
    Naunyn-Schmiedeberg's archives of pharmacology, 2000, Volume: 362, Issue:6

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Carotid Artery, Common; Colforsin; Endothelium, Vascular; Enzyme Inhibitors; Isometric Contraction; Isoproterenol; Male; Mesenteric Arteries; Methacholine Chloride; Muscarinic Agonists; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Phenylephrine; Potassium Chloride; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Adrenergic, beta; Receptors, Muscarinic; Vasoconstrictor Agents; Vasodilation

2000
Role of lysophosphatidylcholine in the desensitization of beta-adrenergic receptors by Ca(2+) sensitization in tracheal smooth muscle.
    American journal of respiratory cell and molecular biology, 2001, Volume: 25, Issue:3

    Topics: Adenylate Cyclase Toxin; Adrenergic beta-Agonists; Amides; Animals; Bucladesine; Calcium; Cholera Toxin; Colforsin; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Inhibitors; Guinea Pigs; In Vitro Techniques; Indoles; Isoproterenol; Lysophosphatidylcholines; Male; Maleimides; Methacholine Chloride; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Pyridines; Receptors, Adrenergic, beta; rho GTP-Binding Proteins; Spectrometry, Fluorescence; Theophylline; Trachea; Virulence Factors, Bordetella

2001
Involvement of Ca2+ mobilization in tachyphylaxis to beta-adrenergic receptors in trachealis.
    American journal of respiratory cell and molecular biology, 2003, Volume: 29, Issue:3 Pt 1

    Topics: Adenylyl Cyclases; Analysis of Variance; Animals; Calcium; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Fluorescent Dyes; Fura-2; Guinea Pigs; Male; Methacholine Chloride; Muscle, Smooth; Potassium; Potassium Channels; Protein Binding; Receptors, Adrenergic, beta; Swine; Tachyphylaxis; Temperature; Time Factors; Trachea; Verapamil

2003
Inhibitory effects of interferon-gamma on the heterologous desensitization of beta-adrenoceptors by transforming growth factor-beta 1 in tracheal smooth muscle.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 2003, Volume: 33, Issue:6

    Topics: Adrenergic beta-Agonists; Animals; Colforsin; Cyclic AMP; Female; Guinea Pigs; In Vitro Techniques; Interferon-gamma; Isoproterenol; Methacholine Chloride; Muscle, Smooth; Receptors, Adrenergic, beta; Trachea; Transforming Growth Factor beta

2003
Potentiation of beta-adrenoceptor function in bovine tracheal smooth muscle by inhibition of protein kinase C.
    European journal of pharmacology, 2005, May-23, Volume: 516, Issue:1

    Topics: Adrenergic beta-Agonists; Animals; Cattle; Colforsin; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Histamine; In Vitro Techniques; Indoles; Isoproterenol; Maleimides; Methacholine Chloride; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Protein Kinase C; Receptors, Adrenergic, beta; Trachea

2005
Involvement of reduced sensitivity to Ca in beta-adrenergic action on airway smooth muscle.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 2006, Volume: 36, Issue:2

    Topics: Adrenergic beta-Agonists; Amides; Animals; Asthma; Bucladesine; Calcium; Calcium Channel Blockers; Colforsin; Cyclic AMP Receptor Protein; Cyclic AMP-Dependent Protein Kinases; Depression, Chemical; Fura-2; Guinea Pigs; Imidazoles; In Vitro Techniques; Indoles; Intracellular Signaling Peptides and Proteins; Isoproterenol; Male; Maleimides; Marine Toxins; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Myosin-Light-Chain Phosphatase; Oxazoles; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Trachea

2006
Modulation of the Ca2+ sensitivity of airway smooth muscle cells in murine lung slices.
    American journal of physiology. Lung cellular and molecular physiology, 2006, Volume: 291, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Arterioles; Bronchoconstrictor Agents; Caffeine; Calcium; Central Nervous System Stimulants; Colforsin; Cyclic AMP; Enzyme Inhibitors; In Vitro Techniques; Male; Methacholine Chloride; Mice; Mice, Inbred BALB C; Muscle Contraction; Myocytes, Smooth Muscle; Protein Kinase C; Respiratory System; Ryanodine

2006
Inhibition of salivary secretion by activation of cannabinoid receptors.
    Experimental biology and medicine (Maywood, N.J.), 2006, Volume: 231, Issue:8

    Topics: Animals; Arachidonic Acids; Cannabinoid Receptor Modulators; Colforsin; Cyclic AMP; Endocannabinoids; Immunohistochemistry; Indoles; Male; Methacholine Chloride; Norepinephrine; Parasympathomimetics; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Saliva; Submandibular Gland; Sympathomimetics

2006
Participation of the endocannabinoid system in lipopolysaccharide-induced inhibition of salivary secretion.
    Archives of oral biology, 2010, Volume: 55, Issue:8

    Topics: Amidohydrolases; Animals; Arachidonic Acid; Arachidonic Acids; Cannabinoid Receptor Modulators; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Endocannabinoids; Etanercept; Immunoglobulin G; Immunologic Factors; In Vitro Techniques; Indoles; Lipopolysaccharides; Male; Methacholine Chloride; Muscarinic Agonists; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Receptors, Tumor Necrosis Factor; Recombinant Fusion Proteins; Saliva; Salivation; Secretory Rate; Submandibular Gland; Tumor Necrosis Factor-alpha

2010
Airway Epithelial Cell Release of GABA is Regulated by Protein Kinase A.
    Lung, 2016, Volume: 194, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bronchoalveolar Lavage Fluid; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activators; Epithelial Cells; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Guanine Nucleotide Exchange Factors; Humans; Male; Methacholine Chloride; Mice; Mice, Inbred C57BL; Myocytes, Smooth Muscle; Platelet-Derived Growth Factor; Propranolol; Receptor Protein-Tyrosine Kinases; Respiratory Mucosa; Rifabutin; RNA, Messenger; Signal Transduction; Terbutaline

2016