Page last updated: 2024-08-23

colforsin and kainic acid

colforsin has been researched along with kainic acid in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-19903 (10.34)18.7374
1990's14 (48.28)18.2507
2000's9 (31.03)29.6817
2010's3 (10.34)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Batista-Gonzalez, A; Brunhofer, G; Fallarero, A; Gopi Mohan, C; Karlsson, D; Shinde, P; Vuorela, P1
Castrén, E; Hartikka, J; Lindholm, D; Thoenen, H; Zafra, F1
D'Mello, SR; Heinrich, G; Jiang, C; Lamberti, C; Martin, SC1
Adler, R; Avendano, G; Butler, BJ; Iuvone, PM1
Greengard, P; Jen, J; Nairn, AC; Stevens, CF1
Deckert, J; Jorgensen, MB1
Cramer, H; Jenner, P; Marsden, CD; Moser, A; Reavill, C1
Baraban, JM; De Souza, EB; Snyder, SH; Worley, PF1
Dawson, TM; Filloux, FM; Gehlert, DR; Hanbauer, I; Sanna, E; Wamsley, JK1
Baudry, M; Ferguson, G; Herschman, HR; Lim, IK; Tocco, G; Vician, L1
Fernández, MT; Gascón, S; Novelli, A; Torreblanca, A; Zitko, V1
Suter-Crazzolara, C; Unsicker, K1
Durkin, JP; Mealing, GA; Morley, P; Murray, CL; Poulter, MO; Small, DL; Stanimirovic, DB1
Hirose, G; Kitasato, H; Pleasure, D; Shimizu, Y; Yoshioka, A1
Benes, C; Creuzet, C; Fagard, R; Miyazaki, J; Roisin, MP; Van Tan, H1
Baudry, M; Crispino, M; Feldman, JD; Herschman, HR; Tocco, G; Vician, L1
Akinshola, BE; Ogunseitan, AB; Onaivi, ES; Taylor, RE1
Egebjerg, J; Hughes, K; Poulsen, F; Price-Jones, M; Shank, RP; Smith, L; Wiberg, FC1
Baudry, M; Crispino, M; Feldman, JD; Herschman, HR; Hoe, W; Vician, L1
Farias-Eisner, R; Feldman, JD; Ferguson, GD; Herschman, HR; Vician, L1
Caman-Krzan, M; Carman-Krzan, M; Juric, DM; Miklic, S1
Feldman, JD; Herschman, HR; Liu, W; Machado, HB; Vician, LJ; Xu, G1
Delgado-García, JM; Negrete-Díaz, JV; Rodríguez-Moreno, A; Sihra, TS1
Gaestel, M; Hitti, E; Kotlyarov, A; Potschka, H; Thomas, T1
Behrens, CJ; Chakrabarty, A; Haq, RU; Heinemann, U; Maggio, N; van den Boom, L; Wójtowicz, AM1
Colbert, CM; Eskin, A; Pita-Almenar, JD; Zou, S1

Reviews

1 review(s) available for colforsin and kainic acid

ArticleYear
The role of receptor binding in drug discovery.
    Journal of natural products, 1993, Volume: 56, Issue:4

    Topics: Animals; Drug Design; Humans; Receptors, Drug

1993

Other Studies

28 other study(ies) available for colforsin and kainic acid

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
Exploration of natural compounds as sources of new bifunctional scaffolds targeting cholinesterases and beta amyloid aggregation: the case of chelerythrine.
    Bioorganic & medicinal chemistry, 2012, Nov-15, Volume: 20, Issue:22

    Topics: Acetylcholinesterase; Amyloid beta-Peptides; Benzophenanthridines; Binding Sites; Butyrylcholinesterase; Catalytic Domain; Cholinesterase Inhibitors; Humans; Isoquinolines; Kinetics; Molecular Docking Simulation; Structure-Activity Relationship

2012
Regulation of brain-derived neurotrophic factor and nerve growth factor mRNA in primary cultures of hippocampal neurons and astrocytes.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1992, Volume: 12, Issue:12

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Astrocytes; Brain-Derived Neurotrophic Factor; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Cytokines; Glutamates; Glutamic Acid; Growth Substances; Hippocampus; Ionomycin; Isoquinolines; Kainic Acid; Kinetics; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Nifedipine; Norepinephrine; Piperazines; Potassium; Protein Kinase Inhibitors; Quisqualic Acid; Rats; RNA, Messenger; Tetradecanoylphorbol Acetate

1992
Differential regulation of the nerve growth factor and brain-derived neurotrophic factor genes in L929 mouse fibroblasts.
    Journal of neuroscience research, 1992, Volume: 33, Issue:4

    Topics: Animals; Base Sequence; Blotting, Northern; Brain-Derived Neurotrophic Factor; Colforsin; Corticosterone; Cyclic AMP; Fibroblasts; Gene Expression Regulation; Hippocampus; Kainic Acid; L Cells; Male; Mice; Molecular Sequence Data; Nerve Growth Factors; Nerve Tissue Proteins; Oligodeoxyribonucleotides; Polymerase Chain Reaction; Rats; Rats, Sprague-Dawley; RNA, Messenger; Seizures; Tetradecanoylphorbol Acetate

1992
Cyclic AMP-dependent induction of serotonin N-acetyltransferase activity in photoreceptor-enriched chick retinal cell cultures: characterization and inhibition by dopamine.
    Journal of neurochemistry, 1990, Volume: 55, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Acetyltransferases; Animals; Arylamine N-Acetyltransferase; Cells, Cultured; Chick Embryo; Colforsin; Cyclic AMP; Cycloheximide; Dactinomycin; Dopamine; Dopamine Antagonists; Enzyme Induction; Kainic Acid; Photoreceptor Cells; Receptors, Dopamine; Receptors, Dopamine D2; Retina; Time Factors

1990
Enhancement of the glutamate response by cAMP-dependent protein kinase in hippocampal neurons.
    Science (New York, N.Y.), 1991, Sep-06, Volume: 253, Issue:5024

    Topics: Adenosine Triphosphate; Animals; Animals, Newborn; Cells, Cultured; Colforsin; Electric Conductivity; Glutamates; Hippocampus; Ion Channel Gating; Ion Channels; Kainic Acid; Kinetics; Membrane Potentials; N-Methylaspartate; Neurons; Protein Kinases; Rats; Receptors, Glutamate; Receptors, Neurotransmitter

1991
Post- and presynaptic lesions in the CA1 region of hippocampus: effect on [3H]forskolin and [3H]phorboldibutyrate ester binding.
    Journal of neural transmission. General section, 1991, Volume: 83, Issue:3

    Topics: Adenylyl Cyclases; Animals; Colforsin; Enzyme Activation; Hippocampus; Humans; Injections, Intraventricular; Ischemic Attack, Transient; Kainic Acid; Male; Neurons; Phorbol 12,13-Dibutyrate; Protein Kinase C; Rats; Rats, Inbred Strains; Second Messenger Systems

1991
Effects of somatostatin on dopamine sensitive adenylate cyclase activity in the caudate-putamen of the rat.
    Experimental brain research, 1986, Volume: 62, Issue:3

    Topics: Adenylyl Cyclases; Animals; Caudate Nucleus; Colforsin; Dopamine; Enzyme Activation; Female; Guanylyl Imidodiphosphate; Hydroxydopamines; Kainic Acid; Oxidopamine; Putamen; Rats; Rats, Inbred Strains; Sodium Fluoride; Somatostatin

1986
Mapping second messenger systems in the brain: differential localizations of adenylate cyclase and protein kinase C.
    Proceedings of the National Academy of Sciences of the United States of America, 1986, Volume: 83, Issue:11

    Topics: Adenylyl Cyclases; Animals; Autoradiography; Binding Sites; Brain; Brain Mapping; Cerebellum; Colforsin; Hippocampus; Kainic Acid; Phorbol Esters; Protein Kinase C; Quinolinic Acid; Quinolinic Acids; Rats; Synaptic Transmission

1986
Evidence that [3H]forskolin binding in the substantia nigra is intrinsic to a striatal-nigral projection: an autoradiographic study of rat brain.
    Neuroscience letters, 1987, Jan-14, Volume: 73, Issue:2

    Topics: Adenylyl Cyclases; Animals; Autoradiography; Caudate Nucleus; Colforsin; Corpus Striatum; Ibotenic Acid; Kainic Acid; Neural Pathways; Putamen; Rats; Substantia Nigra

1987
Synaptotagmin IV is an immediate early gene induced by depolarization in PC12 cells and in brain.
    Proceedings of the National Academy of Sciences of the United States of America, 1995, Mar-14, Volume: 92, Issue:6

    Topics: Adrenal Gland Neoplasms; Amino Acid Sequence; Animals; Base Sequence; Brain; Calcium-Binding Proteins; Cell Line; Colforsin; DNA Primers; Gene Expression; Gene Library; Genes, Immediate-Early; Hippocampus; Kainic Acid; Male; Membrane Glycoproteins; Membrane Potentials; Mice; Molecular Sequence Data; Nerve Tissue Proteins; Oligonucleotide Probes; Organ Specificity; PC12 Cells; Pheochromocytoma; Polymerase Chain Reaction; Potassium; Rats; Rats, Sprague-Dawley; RNA, Messenger; Seizures; Sequence Homology, Amino Acid; Synaptotagmins; Tetradecanoylphorbol Acetate

1995
Neurotoxic effect of okadaic acid, a seafood-related toxin, on cultured cerebellar neurons.
    Annals of the New York Academy of Sciences, 1993, May-28, Volume: 679

    Topics: Animals; Cell Death; Cells, Cultured; Cerebellum; Colforsin; Ethers, Cyclic; Glutamates; Glutamic Acid; Kainic Acid; Marine Toxins; Models, Neurological; Neurons; Neurotoxins; Okadaic Acid; Phosphoprotein Phosphatases; Rats; Shellfish; Tetradecanoylphorbol Acetate

1993
GDNF mRNA levels are induced by FGF-2 in rat C6 glioblastoma cells.
    Brain research. Molecular brain research, 1996, Sep-05, Volume: 41, Issue:1-2

    Topics: Animals; Astrocytes; Brain Neoplasms; Cell Division; Colforsin; Dexamethasone; Fibroblast Growth Factor 1; Fibroblast Growth Factor 2; Gene Expression Regulation, Neoplastic; Glial Cell Line-Derived Neurotrophic Factor; Glioma; Humans; Interleukin-6; Kainic Acid; Neoplasm Proteins; Nerve Growth Factors; Nerve Tissue Proteins; Neuroblastoma; Neurons; Organ Specificity; Pheochromocytoma; Platelet-Derived Growth Factor; Polymerase Chain Reaction; Rats; Recombinant Proteins; RNA, Messenger; RNA, Neoplasm; Triiodothyronine; Tumor Cells, Cultured; Vasoactive Intestinal Peptide

1996
Evidence that functional glutamate receptors are not expressed on rat or human cerebromicrovascular endothelial cells.
    Journal of cerebral blood flow and metabolism : official journal of the International Society of Cerebral Blood Flow and Metabolism, 1998, Volume: 18, Issue:4

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Brain Ischemia; Calcium; Capillaries; Cattle; Cells, Cultured; Cerebrovascular Circulation; Colforsin; Cyclic AMP; Cycloleucine; Endothelin-1; Endothelium, Vascular; Gene Expression; Humans; Inositol 1,4,5-Trisphosphate; Kainic Acid; Mice; N-Methylaspartate; Neurons; Polymerase Chain Reaction; Rats; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; RNA, Messenger; Second Messenger Systems

1998
Cyclic AMP-elevating agents prevent oligodendroglial excitotoxicity.
    Journal of neurochemistry, 1998, Volume: 70, Issue:6

    Topics: Animals; Bucladesine; Calcium; Cell Death; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cycloheximide; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Kainic Acid; L-Lactate Dehydrogenase; Oligodendroglia; Phosphoprotein Phosphatases; Protein Synthesis Inhibitors; Pyridines; Rats; Xanthines

1998
Rapid activation and nuclear translocation of mitogen-activated protein kinases in response to physiological concentration of glucose in the MIN6 pancreatic beta cell line.
    The Journal of biological chemistry, 1998, Jun-19, Volume: 273, Issue:25

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Cell Nucleus; Colforsin; Egtazic Acid; Enzyme Activation; Glucose; Glyburide; Hypoglycemic Agents; Islets of Langerhans; Kainic Acid; Mice; Mice, Transgenic; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nifedipine; Potassium; Receptors, Glutamate

1998
Seizure activity induces PIM-1 expression in brain.
    Journal of neuroscience research, 1998, Aug-15, Volume: 53, Issue:4

    Topics: Animals; Brain; Colforsin; Cycloheximide; Female; Gene Expression Regulation; Kainic Acid; Male; Nerve Growth Factors; Organ Specificity; PC12 Cells; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-pim-1; Proto-Oncogenes; Rats; Rats, Sprague-Dawley; RNA, Messenger; Seizures; Sequence Homology, Amino Acid; Transcription, Genetic

1998
Anandamide inhibition of recombinant AMPA receptor subunits in Xenopus oocytes is increased by forskolin and 8-bromo-cyclic AMP.
    Naunyn-Schmiedeberg's archives of pharmacology, 1999, Volume: 360, Issue:3

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Arachidonic Acid; Arachidonic Acids; Benzoxazines; Colforsin; Dose-Response Relationship, Drug; Electric Stimulation; Endocannabinoids; Female; Imines; Kainic Acid; Membrane Potentials; Morpholines; Naphthalenes; Oocytes; Patch-Clamp Techniques; Polyunsaturated Alkamides; Receptors, AMPA; Recombinant Fusion Proteins; Sensitivity and Specificity; Time Factors; Xenopus laevis

1999
Effects of topiramate on kainate- and domoate-activated [14C]guanidinium ion flux through GluR6 channels in transfected BHK cells using Cytostar-T scintillating microplates.
    Epilepsia, 2000, Volume: 41, Issue:S1

    Topics: Animals; Anticonvulsants; Carbon Radioisotopes; Cell Line; Colforsin; Cricetinae; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Fructose; Guanidine; Kainic Acid; Kidney; Phosphorylation; Receptors, AMPA; Receptors, Glutamate; Receptors, Kainic Acid; Scintillation Counting; Topiramate; Transfection

2000
The salt-inducible kinase, SIK, is induced by depolarization in brain.
    Journal of neurochemistry, 2000, Volume: 74, Issue:6

    Topics: Animals; Blotting, Northern; Cerebral Cortex; Colforsin; Cycloheximide; Epilepsy; Excitatory Amino Acid Agonists; Gene Expression Regulation, Enzymologic; Genes, Immediate-Early; Hippocampus; Kainic Acid; Membrane Potentials; Molecular Sequence Data; Neurons; PC12 Cells; Phylogeny; Protein Synthesis Inhibitors; Protein-Tyrosine Kinases; Rats; RNA, Messenger; Salts; Seizures; Sequence Homology, Amino Acid; Serine; src-Family Kinases

2000
Searching for depolarization-induced genes that modulate synaptic plasticity and neurotrophin-induced genes that mediate neuronal differentiation.
    Neurochemical research, 2000, Volume: 25, Issue:5

    Topics: Adrenal Gland Neoplasms; Animals; Cell Differentiation; Colforsin; Epidermal Growth Factor; Gene Expression Regulation; Genes, Immediate-Early; Kainic Acid; Male; Nerve Growth Factors; Neuronal Plasticity; Neurons; PC12 Cells; Pheochromocytoma; Rats; Synapses

2000
Differences in the regulation of BDNF and NGF synthesis in cultured neonatal rat astrocytes.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 2004, Volume: 22, Issue:3

    Topics: Animals; Animals, Newborn; Astrocytes; Brain-Derived Neurotrophic Factor; Cells, Cultured; Cerebellum; Cerebral Cortex; Colforsin; Cytokines; Dopamine; Dose-Response Relationship, Drug; Homeostasis; Kainic Acid; Nerve Growth Factor; Rats; Rats, Wistar; Tissue Distribution; Tissue Plasminogen Activator

2004
MAPKAP kinase-2 is a primary response gene induced by depolarization in PC12 cells and in brain.
    Journal of neuroscience research, 2004, Nov-01, Volume: 78, Issue:3

    Topics: Amino Acid Sequence; Animals; Blotting, Northern; Blotting, Southern; Brain; Calcium; Cell Differentiation; Cloning, Molecular; Colforsin; Cycloheximide; Drug Interactions; Enzyme Activation; Excitatory Amino Acid Agonists; Gene Expression Regulation, Enzymologic; In Situ Hybridization; Intracellular Signaling Peptides and Proteins; Kainic Acid; Male; Molecular Sequence Data; PC12 Cells; Potassium Chloride; Protein Serine-Threonine Kinases; Protein Synthesis Inhibitors; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Time Factors

2004
Kainate receptor-mediated inhibition of glutamate release involves protein kinase A in the mouse hippocampus.
    Journal of neurophysiology, 2006, Volume: 96, Issue:4

    Topics: Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electrophysiology; Excitatory Postsynaptic Potentials; Glutamic Acid; GTP-Binding Proteins; Hippocampus; Kainic Acid; Mice; Mice, Inbred C57BL; Mossy Fibers, Hippocampal; Pyramidal Cells; Receptors, Kainic Acid; Second Messenger Systems; Signal Transduction

2006
MAP-kinase-activated protein kinase 2 expression and activity is induced after neuronal depolarization.
    The European journal of neuroscience, 2008, Volume: 28, Issue:4

    Topics: Animals; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Stability; Excitatory Amino Acid Agonists; Hippocampus; Humans; Intracellular Signaling Peptides and Proteins; Isoquinolines; Kainic Acid; Membrane Potentials; Mice; Mice, Knockout; Neurons; p38 Mitogen-Activated Protein Kinases; PC12 Cells; Potassium Chloride; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Rats; RNA, Messenger; Seizures; Signal Transduction; Sulfonamides

2008
Monoamines block kainate- and carbachol-induced gamma-oscillations but augment stimulus-induced gamma-oscillations in rat hippocampus in vitro.
    Hippocampus, 2009, Volume: 19, Issue:3

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Biogenic Monoamines; Carbachol; Central Nervous System Agents; Colforsin; Dopamine; Electric Stimulation; Fenfluramine; Hippocampus; In Vitro Techniques; Isoproterenol; Kainic Acid; Membrane Potentials; Norepinephrine; Pyramidal Cells; Rats; Rats, Wistar; Serotonin; Serotonin Agents

2009
Relationship between increase in astrocytic GLT-1 glutamate transport and late-LTP.
    Learning & memory (Cold Spring Harbor, N.Y.), 2012, Nov-19, Volume: 19, Issue:12

    Topics: Alanine Transaminase; Analysis of Variance; Animals; Animals, Newborn; Aspartic Acid; Astrocytes; Biophysics; Biotinylation; Cells, Cultured; Colforsin; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Amino Acid Transporter 1; Excitatory Amino Acid Transporter 2; Excitatory Postsynaptic Potentials; Flow Cytometry; Glial Fibrillary Acidic Protein; Glutamates; Glutamic Acid; Glycine; Hippocampus; In Vitro Techniques; Indoles; Kainic Acid; Long-Term Potentiation; Male; Neurons; Protein Transport; Quinoxalines; Rats; Rats, Sprague-Dawley; Sodium Channel Blockers; Tetrodotoxin; Valine

2012