Page last updated: 2024-08-23

colforsin and idazoxan

colforsin has been researched along with idazoxan in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19902 (11.11)18.7374
1990's13 (72.22)18.2507
2000's2 (11.11)29.6817
2010's1 (5.56)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Dieudonne, MN; Giudicelli, Y; Pecquery, R1
Bitran, JA; Chen, G; Gusovsky, F; Manji, HK; Potter, WZ1
Medgett, IC; Rajanayagam, MA; Rand, MJ1
Carpéné, C; Galitzky, J; Lafontan, M; Langin, D; Larrouy, D1
Breuiller, M; Ferré, F; Leroy, MJ; Litime, MH; Rouot, B1
Galzin, AM; Langer, SZ; Ramdine, R1
Lafontan, M; Langin, D; Paris, H; Stillings, MR1
Bouloumie, A; Galitzky, J; Lafontan, M; Langin, D; Remaury, A; Tavernier, G; Valet, P1
Cooke, HJ; Wood, JD; Zafirov, DH1
Baba, A; Kawai, N; Moroji, T; Yamamoto, H; Yamamoto, T1
Lee, A; Lynch, KR; Rosin, DL; Talley, E1
Goldstein, I; Huang, YH; Moreland, RB; Traish, AM1
Correze, C; Dib, K; el Jamali, A; Lambert, B; Wrisez, F1
Farley, JT; Klimek, V; Ordway, GA; Zhang, W; Zhu, MY1
Bobirnac, I; Gazi, L; Loetscher, E; Parsley, S; Schoeffter, P1
Akerman, KE; Jansson, CC; Kukkonen, JP1
Akerman, KE; Holmqvist, T; Kukkonen, JP; Näsman, J1
Amodeo, FS; Brummett, CM; Hong, EK; Janda, AM; Lydic, R1

Other Studies

18 other study(ies) available for colforsin and idazoxan

ArticleYear
Characteristics of the alpha 2/beta-adrenoceptor-coupled adenylate cyclase system and their relationship with adrenergic responsiveness in hamster fat cells from different anatomical sites.
    European journal of biochemistry, 1992, Apr-15, Volume: 205, Issue:2

    Topics: Adenylyl Cyclases; Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Colforsin; Cricetinae; Dioxanes; Epididymis; Epinephrine; GTP-Binding Proteins; Idazoxan; Isoproterenol; Kinetics; Lipolysis; Macromolecular Substances; Male; Mesocricetus; Organ Specificity; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Skin; Theophylline

1992
Idazoxan down-regulates beta-adrenoceptors on C6 glioma cells in vitro.
    European journal of pharmacology, 1992, Nov-02, Volume: 227, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Autoradiography; Cholera Toxin; Colforsin; Cyclic AMP; Dioxanes; Down-Regulation; Glioma; Idazoxan; Isoproterenol; Protein Kinase C; Rats; Receptors, Adrenergic, beta; Tumor Cells, Cultured

1992
Vasoconstrictor responses of rat tail artery to sympathetic nerve stimulation contain a component due to activation of postjunctional beta- or alpha 2-adrenoceptors.
    European journal of pharmacology, 1990, Feb-20, Volume: 177, Issue:1-2

    Topics: Adenylyl Cyclases; Adrenergic beta-Antagonists; Animals; Calcium; Colforsin; Dioxanes; Electric Stimulation; Idazoxan; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Neurotransmitter Agents; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Regional Blood Flow; Sympathetic Nervous System; Tail; Vasoconstriction

1990
Non-adrenergic sites for imidazolines are not directly involved in the alpha 2-adrenergic antilipolytic effect of UK 14304 in rat adipocytes.
    Biochemical pharmacology, 1990, Aug-01, Volume: 40, Issue:3

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding Sites; Binding, Competitive; Brimonidine Tartrate; Bucladesine; Cell Membrane; Colforsin; Dioxanes; Idazoxan; Kinetics; Lipolysis; Phentolamine; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1990
Functional coupling of the alpha 2-adrenergic receptor-adenylate cyclase complex in the pregnant human myometrium.
    The Journal of clinical endocrinology and metabolism, 1990, Volume: 70, Issue:5

    Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adult; Binding, Competitive; Clonidine; Colforsin; Cyclic AMP; Dioxanes; Drug Interactions; Electrophoresis, Polyacrylamide Gel; Female; GTP-Binding Proteins; Humans; Idazoxan; Myometrium; Norepinephrine; Pertussis Toxin; Pregnancy; Pregnancy Trimester, Third; Receptors, Adrenergic, alpha; Virulence Factors, Bordetella; Yohimbine

1990
Involvement of adenylate cyclase and protein kinase C in the alpha 2-adrenoceptor-mediated inhibition of noradrenaline and 5-hydroxytryptamine release in rat hypothalamic slices.
    Naunyn-Schmiedeberg's archives of pharmacology, 1989, Volume: 340, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Antihypertensive Agents; Brimonidine Tartrate; Colforsin; Dioxanes; Electric Stimulation; Hypothalamus; Idazoxan; In Vitro Techniques; Male; Norepinephrine; Phorbol 12,13-Dibutyrate; Protein Kinase C; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin

1989
[3H]RX821002: a new tool for the identification of alpha 2A-adrenoceptors.
    European journal of pharmacology, 1989, Aug-11, Volume: 167, Issue:1

    Topics: Adrenergic alpha-Antagonists; Binding, Competitive; Catecholamines; Cell Membrane; Colforsin; Cyclic AMP; Dioxanes; Dioxins; Humans; Idazoxan; Kinetics; Radioligand Assay; Receptors, Adrenergic, alpha; Tumor Cells, Cultured; Yohimbine

1989
Molecular mechanisms underlying regional variations of catecholamine-induced lipolysis in rat adipocytes.
    The American journal of physiology, 1995, Volume: 268, Issue:6 Pt 1

    Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Base Sequence; Brimonidine Tartrate; Bucladesine; Catecholamines; Cell Membrane; Cells, Cultured; Colforsin; Cyclic AMP; Dioxanes; DNA Primers; Epididymis; Gene Expression; Idazoxan; Isoproterenol; Lipase; Lipolysis; Male; Molecular Sequence Data; Organ Specificity; Polymerase Chain Reaction; Propanolamines; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, beta-1; Receptors, Adrenergic, beta-2; RNA, Messenger; Skin

1995
Elevation of cAMP facilitates noradrenergic transmission in submucous neurons of guinea pig ileum.
    The American journal of physiology, 1993, Volume: 264, Issue:3 Pt 1

    Topics: 1-Methyl-3-isobutylxanthine; Adrenergic alpha-Antagonists; Animals; Colforsin; Cyclic AMP; Dioxanes; Electric Stimulation; Ganglia; Guinea Pigs; Idazoxan; Ileum; Membrane Potentials; Microelectrodes; Neurons; Norepinephrine; Phentolamine; Receptors, Purinergic; Synaptic Transmission; Yohimbine

1993
Inhibitory effect of idazoxan on forskolin-stimulated adenylate cyclase activity through 5-hydroxytryptamine1A receptors.
    Arzneimittel-Forschung, 1994, Volume: 44, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Adrenergic alpha-Antagonists; Animals; Colforsin; Dioxanes; Hippocampus; Idazoxan; In Vitro Techniques; Male; Membranes; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Serotonin

1994
Characterization of alpha 2A-adrenergic receptors in GT1 neurosecretory cells.
    Neuroendocrinology, 1995, Volume: 62, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blotting, Northern; Cell Line; Colforsin; Dioxanes; Idazoxan; Immunohistochemistry; Male; Mice; Mice, Inbred C57BL; Neurons; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha

1995
Expression of functional alpha2-adrenergic receptor subtypes in human corpus cavernosum and in cultured trabecular smooth muscle cells.
    Receptors & signal transduction, 1997, Volume: 7, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Binding, Competitive; Brimonidine Tartrate; Cells, Cultured; Colforsin; Cyclic AMP; Humans; Idazoxan; Male; Muscle Contraction; Muscle, Smooth; Penis; Quinoxalines; Radioisotopes; Receptors, Adrenergic, alpha-2; Ribonucleases; RNA, Messenger; Yohimbine

1997
Sodium saccharin inhibits adenylyl cyclase activity in non-taste cells.
    Cellular signalling, 1997, Volume: 9, Issue:6

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adipocytes; Adrenergic alpha-Agonists; Animals; Astrocytes; Brimonidine Tartrate; Carcinogens; Cell Fractionation; Cell Membrane; Cerebral Cortex; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; GTP-Binding Proteins; Idazoxan; Male; Pertussis Toxin; Phenylisopropyladenosine; Quinoxalines; Rats; Rats, Wistar; Saccharin; Signal Transduction; Swine; Taste; Thyroid Gland; Virulence Factors, Bordetella

1997
alpha2C adrenoceptors inhibit adenylyl cyclase in mouse striatum: potential activation by dopamine.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:3

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adrenergic alpha-Antagonists; alpha-Methyltyrosine; Animals; Cell Line; Colforsin; Corpus Striatum; Crosses, Genetic; Cyclic AMP; Dopamine; Enzyme Activation; Homozygote; Idazoxan; In Vitro Techniques; Kinetics; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Mice, Knockout; Norepinephrine; Rats; Receptors, Adrenergic, alpha-2; Recombinant Proteins; Reserpine; Transfection

1999
Functional alpha2C-adrenoceptors in human neuroblastoma SH-SY5Y cells.
    European journal of pharmacology, 1999, May-07, Volume: 372, Issue:1

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Brimonidine Tartrate; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Guanfacine; Humans; Idazoxan; Isoquinolines; Neuroblastoma; Oxymetazoline; Piperazines; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured; Yohimbine

1999
Agonist trafficking of G(i/o)-mediated alpha(2A)-adrenoceptor responses in HEL 92.1.7 cells.
    British journal of pharmacology, 2001, Volume: 132, Issue:7

    Topics: Adrenergic Agonists; Adrenergic Antagonists; Biological Transport; Calcium; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Epinephrine; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Idazoxan; Pertussis Toxin; Propranolol; Receptors, Adrenergic, alpha-2; Tumor Cells, Cultured; Virulence Factors, Bordetella; Yohimbine

2001
Different roles for Gi and Go proteins in modulation of adenylyl cyclase type-2 activity.
    Journal of neurochemistry, 2002, Volume: 83, Issue:6

    Topics: Adenylyl Cyclases; Animals; Binding, Competitive; Cell Line; Colforsin; Cyclic AMP; Enzyme Activation; Enzyme Activators; Enzyme Inhibitors; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gs; Guanosine 5'-O-(3-Thiotriphosphate); Heterotrimeric GTP-Binding Proteins; Humans; Idazoxan; Pertussis Toxin; Protein Kinase C; Receptors, Adrenergic, alpha-2; Signal Transduction; Spodoptera; Tetradecanoylphorbol Acetate

2002
Perineural dexmedetomidine added to ropivacaine for sciatic nerve block in rats prolongs the duration of analgesia by blocking the hyperpolarization-activated cation current.
    Anesthesiology, 2011, Volume: 115, Issue:4

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Amides; Analgesia; Anesthetics, Local; Animals; Behavior, Animal; Colforsin; Cyclic Nucleotide-Gated Cation Channels; Dexmedetomidine; Dose-Response Relationship, Drug; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; Hypnotics and Sedatives; Idazoxan; Male; Nerve Block; Pain Measurement; Potassium Channel Blockers; Potassium Channels; Prazosin; Pyrimidines; Rats; Rats, Sprague-Dawley; Ropivacaine; Sciatic Nerve

2011