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colforsin and glycine

colforsin has been researched along with glycine in 59 studies

Research

Studies (59)

TimeframeStudies, this research(%)All Research%
pre-19901 (1.69)18.7374
1990's25 (42.37)18.2507
2000's24 (40.68)29.6817
2010's9 (15.25)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Randic, M; Rusin, KI; Ryu, PD1
Brosnan, JT; Collett, VM; Hall, B; Jois, M1
Braun, W; Reymann, A; Woermann, C1
Soderling, TR; Tan, SE; Wenthold, RJ1
Cavanni, P; Ferraguti, F; Mugnaini, M; Pinnola, V; Trist, D; Van Amsterdam, FT1
Chetkovich, DM; Sweatt, JD1
Baker, SR; Goldsworthy, J; Johnson, BG; Salhoff, CR; Schoepp, DD1
Caciagli, F; Casabona, G; Ciccarelli, R; De Bernardis, E; Di Iorio, P; L'Episcopo, MR; Nicoletti, F; Shinozaki, H1
Jane, D; Jones, A; Jones, P; Kemp, M; Pook, P; Roberts, P; Sunter, D; Udvarhelyi, P; Watkins, J1
Ishida, M; Kataoka, K; Nakamura, Y; Saitoh, T; Shinozaki, H; Tsuji, K1
Arilla, E; Puebla, L1
Bedingfield, JS; Jane, DE; Kemp, MC; Roberts, PJ; Tse, HW; Watkins, JC1
Bockaert, J; Manahan-Vaughan, D; Pin, JP; Reiser, M; Reymann, KG; Riedel, G; Wilsch, V1
Alexander, SP; Kendall, DA; Neil, KE1
Dowd, LA; Robinson, MB1
Glitsch, M; Llano, I; Marty, A1
Belagaje, R; Burnett, JP; Johnson, BG; Mayne, NG; Monn, JA; Salhoff, CR; Schoepp, DD; Wright, RA; Wu, S1
Henderson, PJ; McDonald, TP; Walmsley, AR1
Maccaferri, G; McBain, CJ; Tóth, K1
Adam, G; Cartmell, J; Chaboz, S; Henningsen, R; Kemp, JA; Klingelschmidt, A; Metzler, V; Monsma, F; Mutel, V; Schaffhauser, H; Wichmann, J1
Han, Y; Slaughter, MM1
Balázs, R; Chun, Y; Cotman, CW; Miller, S; O'Toole, J1
Akaike, N; Li, JS; Nabekura, J; Rhee, JS; Xu, TL1
Battaglia, G; Bruno, V; Flor, PJ; Gasparini, F; Hess, SD; Inderbitzin, W; Johnson, EC; Kuhn, R; Laurie, D; Leonhardt, T; Lukic, S; Nicoletti, F; Portet, C; Sauer, D; Schmutz, M; Sommer, B; Urwyler, S; Varney, MA1
Estevez, AY; O'Regan, MH; Phillis, JW; Song, D1
Akaike, N; Nabekura, J; Omura, T1
Hirouchi, M; Itoh, Y; Kimura, K; Oka, M; Ukai, Y1
Casabona, G; Copani, A; Di Giorgi Gerevini, V; Mutel, V; Nicoletti, F; Nicosia, A; Romano, C; Storto, M1
Evans, DI; Jones, RS; Woodhall, G1
Howson, PA; Jane, DE; Kingston, AE; Schoepp, DD; Thomas, NK; Wright, RA1
Fujimori, S; Hinoi, E; Nakamura, Y; Yoneda, Y1
Li, P; Yang, XL1
Kirchgessner, AL; Ouedraogo, R; Tong, Q1
Becq, F; Bulteau-Pignoux, L; Derand, R2
Chesnoy-Marchais, D1
Johnson, SW; Shen, KZ1
Foster, AC; Naeve, GS; Selkirk, JV1
Irifune, M; Nishikawa, T; Ohnishi, Y; Sato, T; Tanaka, K; Teramoto, T1
López-Vera, E; Pérez-León, JA; Salceda, R1
Inoue, M; Kawamura, Y; Kudo, Y; Manita, S; Miyakawa, H; Nakamura, T1
Konishi, S; Rusakov, D; Saitow, F; Satake, S1
Fujita, T; Kumamoto, E; Yang, K1
Akaike, N; Katsurabayashi, S; Kubota, H; Moorhouse, AJ1
de Novellis, V; Maione, S; Marabese, I; Mariani, L; Palazzo, E; Rodella, L; Rossi, F; Siniscalco, D1
Brose, N; Gibson, HE; Jones, S; Morton, AJ; Reim, K1
Chen, JF; Cunha, RA; Domenici, MR; Grò, MC; Martire, A; Pepponi, R; Popoli, P; Rebola, N; Schwarzschild, MA; Tebano, MT1
Glitsch, M1
Hasegawa, H; Inoue, A; Kohno, M; Miyazaki, T; Muraoka, M; Oka, K; Yasukawa, M1
Cho, JH; Choi, BJ; Choi, IS; Jang, IS; Kim, J; Kim, SJ; Lee, JJ; Nakamura, M; Park, HM1
Jang, IS; Nakamura, M1
Chen, ZN; Li, CY; Shi, HB; Song, NY; Ye, HB; Yin, SK1
Alzheimer, C; Wess, J; Zheng, F1
Bückers, J; Chapman, ER; Dean, C; Engelhardt, J; Hell, SW; Jackson, MB; Kamin, D; Liu, H; Stahlberg, MA; Staudt, T; Vingill, S1
Di Prisco, S; Grilli, M; Marchi, M; Pittaluga, A; Summa, M; Usai, C1
Colbert, CM; Eskin, A; Pita-Almenar, JD; Zou, S1
Edlund, A; Eliasson, L; Esguerra, JL; Flodström-Tullberg, M; Wendt, A1
Clauss, WG; Fronius, M; Vitzthum, C1

Other Studies

59 other study(ies) available for colforsin and glycine

ArticleYear
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
Modulation of excitatory amino acid responses in rat dorsal horn neurons by tachykinins.
    Journal of neurophysiology, 1992, Volume: 68, Issue:1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Amino Acids; Animals; Calcium; Cesium; Colforsin; Glycine; Ibotenic Acid; In Vitro Techniques; N-Methylaspartate; Neurokinin A; Neurons; Peptides; Phorbol Esters; Quisqualic Acid; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Spinal Cord; Substance P; Tachykinins

1992
Flux through glycine cleavage system in isolated hepatocytes: effects of glucagon, cAMP, and calcium.
    Biochemistry and cell biology = Biochimie et biologie cellulaire, 1990, Volume: 68, Issue:2

    Topics: Animals; Bucladesine; Calcium; Colforsin; Cyclic AMP; Glucagon; Glycine; In Vitro Techniques; Liver; Male; Rats; Rats, Inbred Strains; Theophylline

1990
Proabsorptive properties of forskolin: disposition of glycine, leucine and lysine in rat jejunum.
    Naunyn-Schmiedeberg's archives of pharmacology, 1986, Volume: 334, Issue:1

    Topics: Animals; Biological Transport, Active; Colforsin; Cyclic AMP; Glycine; In Vitro Techniques; Intestinal Absorption; Intestinal Mucosa; Jejunum; Leucine; Lysine; Male; Proteins; Rats; Rats, Inbred Strains

1986
Phosphorylation of AMPA-type glutamate receptors by calcium/calmodulin-dependent protein kinase II and protein kinase C in cultured hippocampal neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1994, Volume: 14, Issue:3 Pt 1

    Topics: alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Colforsin; Cyclic AMP-Dependent Protein Kinases; Glutamates; Glutamic Acid; Glycine; Hippocampus; Intracellular Signaling Peptides and Proteins; Ionomycin; Membrane Proteins; Myristoylated Alanine-Rich C Kinase Substrate; Phosphorylation; Protein Kinase C; Proteins; Rats; Receptors, Glutamate; Receptors, N-Methyl-D-Aspartate; Tetradecanoylphorbol Acetate

1994
Pharmacological analysis of carboxyphenylglycines at metabotropic glutamate receptors.
    European journal of pharmacology, 1994, Sep-15, Volume: 269, Issue:1

    Topics: Adenylyl Cyclases; Animals; Benzoates; CHO Cells; Colforsin; Computer Simulation; Cricetinae; Cricetulus; Cyclic AMP; Dose-Response Relationship, Drug; Glycine; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, Kainic Acid; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Stereoisomerism

1994
nMDA receptor activation increases cyclic AMP in area CA1 of the hippocampus via calcium/calmodulin stimulation of adenylyl cyclase.
    Journal of neurochemistry, 1993, Volume: 61, Issue:5

    Topics: 2-Amino-5-phosphonovalerate; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenylyl Cyclases; Animals; Ascorbic Acid; Calcium; Calmodulin; Cell Membrane; Colforsin; Cyclic AMP; Deoxyadenosines; Dopamine; Enzyme Activation; Evoked Potentials; Glycine; Hippocampus; In Vitro Techniques; Isoproterenol; Kinetics; Models, Neurological; N-Methylaspartate; Pyramidal Tracts; Quinoxalines; Rats; Receptors, N-Methyl-D-Aspartate; Sulfonamides; Theophylline; Trifluoperazine

1993
3,5-dihydroxyphenylglycine is a highly selective agonist for phosphoinositide-linked metabotropic glutamate receptors in the rat hippocampus.
    Journal of neurochemistry, 1994, Volume: 63, Issue:2

    Topics: Aging; Amino Acids, Dicarboxylic; Animals; Animals, Newborn; Colforsin; Cyclic AMP; Cycloleucine; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Glycine; Hippocampus; In Vitro Techniques; Kinetics; Male; Neurotoxins; Phosphatidylinositols; Rats; Rats, Sprague-Dawley; Receptors, Glutamate; Resorcinols; Second Messenger Systems

1994
Interaction between metabotropic receptors and purinergic transmission in rat hippocampal slices.
    Brain research, 1994, May-09, Volume: 645, Issue:1-2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Colforsin; Cycloleucine; Cyclopropanes; Glycine; Hippocampus; In Vitro Techniques; Male; Neurotoxins; Purines; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Synaptic Transmission

1994
Antagonism of presynaptically mediated depressant responses and cyclic AMP-coupled metabotropic glutamate receptors.
    European journal of pharmacology, 1994, Jan-15, Volume: 266, Issue:2

    Topics: Aminobutyrates; Animals; Animals, Newborn; Benzoates; Cerebral Cortex; Colforsin; Cyclic AMP; Cycloleucine; Electrophysiology; Glycine; Guinea Pigs; Neurotoxins; Rats; Receptors, Metabotropic Glutamate; Synaptic Transmission

1994
Novel agonists for metabotropic glutamate receptors: trans- and cis-2-(2-carboxy-3-methoxymethylcyclopropyl)glycine (trans- and cis-MCG-I).
    Neuropharmacology, 1995, Volume: 34, Issue:8

    Topics: Animals; Animals, Newborn; Cells, Cultured; Colforsin; Cyclic AMP; Electrophysiology; Excitatory Amino Acid Agonists; Glycine; In Vitro Techniques; Male; Quisqualic Acid; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Reflex; Spinal Cord; Synapses

1995
Glycine increases the number of somatostatin receptors and somatostatin-mediated inhibition of the adenylate cyclase system in the rat hippocampus.
    Journal of neuroscience research, 1996, Feb-01, Volume: 43, Issue:3

    Topics: Adenylyl Cyclase Inhibitors; Animals; Cell Membrane; Cerebral Cortex; Cerebral Ventricles; Colforsin; Frontal Lobe; Glycine; Guanylyl Imidodiphosphate; Hippocampus; Injections, Intraventricular; Kinetics; Parietal Lobe; Rats; Rats, Wistar; Receptors, Somatostatin; Somatostatin; Strychnine; Time Factors; Up-Regulation

1996
Structure-activity relationships for a series of phenylglycine derivatives acting at metabotropic glutamate receptors (mGluRs).
    British journal of pharmacology, 1995, Volume: 116, Issue:8

    Topics: Amino Acids, Dicarboxylic; Aminobutyrates; Animals; Animals, Newborn; Anti-Inflammatory Agents, Non-Steroidal; Cerebral Cortex; Colforsin; Cyclic AMP; Cycloleucine; Glycine; Inositol Phosphates; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Structure-Activity Relationship

1995
Physiological and pharmacological profile of trans-azetidine-2,4-dicarboxylic acid: metabotropic glutamate receptor agonism and effects on long-term potentiation.
    Neuroscience, 1996, Volume: 72, Issue:4

    Topics: Animals; Azetidinecarboxylic Acid; Benzoates; Cells, Cultured; Colforsin; Cyclic AMP; Epithelial Cells; Epithelium; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Hippocampus; Hydrolysis; Inositol Phosphates; Kidney; Long-Term Potentiation; Male; N-Methylaspartate; Organ Culture Techniques; Patch-Clamp Techniques; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Swine; Temperature; Transfection

1996
Coupling of metabotropic glutamate receptors to phosphoinositide mobilisation and inhibition of cyclic AMP generation in the guinea-pig cerebellum.
    British journal of pharmacology, 1996, Volume: 118, Issue:2

    Topics: 2-Chloroadenosine; Animals; Cerebellum; Colforsin; Cyclic AMP; Cycloleucine; Female; Glutamic Acid; Glycine; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Phosphatidylinositols; Receptors, Metabotropic Glutamate; Resorcinols

1996
Rapid stimulation of EAAC1-mediated Na+-dependent L-glutamate transport activity in C6 glioma cells by phorbol ester.
    Journal of neurochemistry, 1996, Volume: 67, Issue:2

    Topics: Adenylyl Cyclases; Amiloride; Amino Acid Transport System X-AG; Animals; Aspartic Acid; ATP-Binding Cassette Transporters; Calcimycin; Carrier Proteins; Colforsin; Enzyme Inhibitors; Ethers, Cyclic; Excitatory Amino Acid Transporter 3; Glioma; Glutamate Plasma Membrane Transport Proteins; Glutamates; Glycine; Kinetics; Okadaic Acid; Phosphoric Monoester Hydrolases; Protein Kinase C; Rats; Sodium; Sodium-Potassium-Exchanging ATPase; Symporters; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured

1996
Glutamate as a candidate retrograde messenger at interneurone-Purkinje cell synapses of rat cerebellum.
    The Journal of physiology, 1996, Dec-01, Volume: 497 ( Pt 2)

    Topics: 2-Amino-5-phosphonovalerate; Alanine; Animals; Benzoates; Colforsin; Cyclopropanes; Electrophysiology; Excitatory Amino Acid Antagonists; Glutamic Acid; Glycine; Interneurons; Kinetics; Presynaptic Terminals; Purkinje Cells; Quinoxalines; Rats; Receptors, Metabotropic Glutamate; Synapses; Synaptic Transmission; Tetrodotoxin

1996
The novel metabotropic glutamate receptor agonist 2R,4R-APDC potentiates stimulation of phosphoinositide hydrolysis in the rat hippocampus by 3,5-dihydroxyphenylglycine: evidence for a synergistic interaction between group 1 and group 2 receptors.
    Neuropharmacology, 1996, Volume: 35, Issue:12

    Topics: Aging; Animals; Animals, Newborn; Brain; Cloning, Molecular; Colforsin; Cyclic AMP; Cycloleucine; Drug Synergism; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Hippocampus; Humans; Inositol; Kinetics; Neuroprotective Agents; Phosphatidylinositols; Proline; Quisqualic Acid; Rats; Receptors, Metabotropic Glutamate; Recombinant Proteins; Resorcinols; Second Messenger Systems

1996
Asparagine 394 in putative helix 11 of the galactose-H+ symport protein (GalP) from Escherichia coli is associated with the internal binding site for cytochalasin B and sugar.
    The Journal of biological chemistry, 1997, Jun-13, Volume: 272, Issue:24

    Topics: Amino Acid Sequence; Asparagine; Binding Sites; Biological Transport; Calcium-Binding Proteins; Carrier Proteins; Catalysis; Colforsin; Cytochalasin B; Escherichia coli; Galactose; Glucose; Glycine; Humans; Kinetics; Molecular Sequence Data; Monosaccharide Transport Proteins; Periplasmic Binding Proteins

1997
Target-specific expression of presynaptic mossy fiber plasticity.
    Science (New York, N.Y.), 1998, Feb-27, Volume: 279, Issue:5355

    Topics: Afferent Pathways; Animals; Colforsin; Cyclic AMP; Cycloleucine; Cyclopropanes; Electric Stimulation; Excitatory Postsynaptic Potentials; Glycine; Hippocampus; In Vitro Techniques; Interneurons; Long-Term Potentiation; Mossy Fibers, Hippocampal; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Synaptic Transmission

1998
Characterization of [3H]-(2S,2'R,3'R)-2-(2',3'-dicarboxy-cyclopropyl)glycine ([3H]-DCG IV) binding to metabotropic mGlu2 receptor-transfected cell membranes.
    British journal of pharmacology, 1998, Volume: 123, Issue:3

    Topics: Animals; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cyclopropanes; Glycine; Guanosine 5'-O-(3-Thiotriphosphate); Protein Binding; Rats; Receptors, Metabotropic Glutamate; Recombinant Proteins; Sulfur Radioisotopes; Transfection; Tritium

1998
Protein kinases modulate two glycine currents in salamander retinal ganglion cells.
    The Journal of physiology, 1998, May-01, Volume: 508 ( Pt 3)

    Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Ambystoma; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Glycine; Glycine Agents; Isoquinolines; Kinetics; Kynurenic Acid; Membrane Potentials; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Protein Kinase C; Retinal Ganglion Cells; Strychnine; Sulfonamides

1998
Metabotropic glutamate receptor agonists potentiate cyclic AMP formation induced by forskolin or beta-adrenergic receptor activation in cerebral cortical astrocytes in culture.
    Journal of neurochemistry, 1998, Volume: 70, Issue:6

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Animals, Newborn; Astrocytes; Cells, Cultured; Colforsin; Cyclic AMP; Cycloleucine; Drug Synergism; Estrenes; Excitatory Amino Acid Agonists; Glycine; Neocortex; Phosphodiesterase Inhibitors; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Adrenergic, beta; Receptors, Metabotropic Glutamate; Resorcinols; Signal Transduction; Type C Phospholipases; Up-Regulation

1998
Alpha2-adrenoceptor-mediated enhancement of glycine response in rat sacral dorsal commissural neurons.
    Neuroscience, 1999, Volume: 89, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adrenergic alpha-Agonists; Animals; Bucladesine; Clonidine; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Electrophysiology; Glycine; Glycine Agents; GTP-Binding Proteins; Ion Channel Gating; Isoproterenol; Lumbosacral Region; Neurons, Afferent; Nociceptors; Norepinephrine; Pertussis Toxin; Phenylephrine; Phosphodiesterase Inhibitors; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Strychnine; Virulence Factors, Bordetella

1999
(R,S)-4-phosphonophenylglycine, a potent and selective group III metabotropic glutamate receptor agonist, is anticonvulsive and neuroprotective in vivo.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:3

    Topics: Animals; Anticonvulsants; Brain; Cell Line; Cell Membrane; Colforsin; Corpus Striatum; Cyclic AMP; Electroshock; Glutamic Acid; Glycine; Humans; Kinetics; Male; Mice; Mice, Inbred Strains; N-Methylaspartate; Neuroprotective Agents; Phosphatidylinositols; Protein Isoforms; Quinolinic Acid; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Recombinant Proteins; Second Messenger Systems; Seizures; Structure-Activity Relationship

1999
Hyposmotically induced amino acid release from the rat cerebral cortex: role of phospholipases and protein kinases.
    Brain research, 1999, Oct-09, Volume: 844, Issue:1-2

    Topics: Acetophenones; Alanine; Amino Acids; Animals; Arachidonic Acids; Aspartic Acid; Brain Edema; Cerebral Cortex; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dimethyl Sulfoxide; Enzyme Inhibitors; Estrenes; Ethanolamines; Fatty Acids, Unsaturated; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Hypotonic Solutions; Male; Osmotic Pressure; Phosphodiesterase Inhibitors; Phospholipases A; Phospholipases A2; Protein Kinase C; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Serine; Solvents; Taurine; Water-Electrolyte Balance

1999
Intracellular pathways of V(1) and V(2) receptors activated by arginine vasopressin in rat hippocampal neurons.
    The Journal of biological chemistry, 1999, Nov-12, Volume: 274, Issue:46

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Arginine Vasopressin; Benzazepines; Calcium; Calcium-Calmodulin-Dependent Protein Kinase Type 2; Calcium-Calmodulin-Dependent Protein Kinases; Colforsin; Cyclic AMP-Dependent Protein Kinases; Deamino Arginine Vasopressin; Egtazic Acid; Enzyme Inhibitors; Glycine; Hippocampus; Neurons; Oligopeptides; Patch-Clamp Techniques; Peptide Fragments; Protein Kinase C; Pyrrolidonecarboxylic Acid; Rats; Receptors, Vasopressin

1999
Role of metabotropic glutamate receptor subclasses in modulation of adenylyl cyclase activity by a nootropic NS-105.
    European journal of pharmacology, 2000, Jan-03, Volume: 387, Issue:1

    Topics: Adenylyl Cyclases; Animals; Benzoates; Cells, Cultured; Cerebral Cortex; Colforsin; Cyclic AMP; Excitatory Amino Acid Antagonists; Fetus; Gene Expression Regulation; Glycine; Male; Membranes; Neurons; Nootropic Agents; Oligodeoxyribonucleotides, Antisense; Oligonucleotides; Piperidines; Proline; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; RNA, Messenger

2000
Reducing conditions differentially affect the functional and structural properties of group-I and -II metabotropic glutamate receptors.
    Brain research, 2000, Jun-09, Volume: 867, Issue:1-2

    Topics: Amino Acids, Dicarboxylic; Animals; Anticonvulsants; Carbachol; Cell Membrane; Cerebellum; CHO Cells; Cholinergic Agonists; Colforsin; Cricetinae; Cyclic AMP; Cycloleucine; Cyclopropanes; Dimerization; Dithiothreitol; Excitatory Amino Acid Agonists; Glycine; Hippocampus; Humans; Kidney; Neurons; Neuroprotective Agents; Quisqualic Acid; Rats; Receptors, Metabotropic Glutamate; Signal Transduction

2000
Differential actions of PKA and PKC in the regulation of glutamate release by group III mGluRs in the entorhinal cortex.
    Journal of neurophysiology, 2001, Volume: 85, Issue:2

    Topics: Adenine; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyclopentanes; Entorhinal Cortex; Enzyme Activation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Glycine; In Vitro Techniques; Indoles; Isoquinolines; Male; Maleimides; Presynaptic Terminals; Protein Kinase C; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Sulfonamides; Tricarboxylic Acids

2001
(S)-3,4-DCPG, a potent and selective mGlu8a receptor agonist, activates metabotropic glutamate receptors on primary afferent terminals in the neonatal rat spinal cord.
    Neuropharmacology, 2001, Volume: 40, Issue:3

    Topics: Animals; Animals, Newborn; Benzoates; Cell Line; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Humans; In Vitro Techniques; Membrane Potentials; Neurons, Afferent; Presynaptic Terminals; Rats; Receptors, Metabotropic Glutamate; Spinal Cord; Stereoisomerism; Substrate Specificity

2001
Group III metabotropic glutamate receptors in rat cultured calvarial osteoblasts.
    Biochemical and biophysical research communications, 2001, Feb-23, Volume: 281, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Aminobutyrates; Animals; Animals, Newborn; Cells, Cultured; Colforsin; Cyclic AMP; Gene Expression; Glycine; Male; Osteoblasts; Protein Isoforms; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Skull

2001
Forskolin modulation of desensitization at GABA(A) and glycine receptors is not mediated by cAMP-dependent protein kinase in isolated carp amacrine-like cells.
    Pflugers Archiv : European journal of physiology, 2001, Volume: 441, Issue:6

    Topics: Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; gamma-Aminobutyric Acid; Glycine; Goldfish; Isoquinolines; Membrane Potentials; Patch-Clamp Techniques; Receptors, GABA-A; Receptors, Glycine; Retina; Sulfonamides

2001
Localization and function of group III metabotropic glutamate receptors in rat pancreatic islets.
    American journal of physiology. Endocrinology and metabolism, 2002, Volume: 282, Issue:6

    Topics: Animals; Benzoates; Cell Membrane; Colforsin; Cyclic AMP; Cytoplasmic Granules; DNA Primers; Excitatory Amino Acid Antagonists; Female; Gene Expression; Glucagon; Glutamic Acid; Glycine; Islets of Langerhans; Microscopy, Immunoelectron; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Reverse Transcriptase Polymerase Chain Reaction; Synaptophysin; Tissue Distribution

2002
The cystic fibrosis mutation G551D alters the non-Michaelis-Menten behavior of the cystic fibrosis transmembrane conductance regulator (CFTR) channel and abolishes the inhibitory Genistein binding site.
    The Journal of biological chemistry, 2002, Sep-27, Volume: 277, Issue:39

    Topics: Animals; Binding Sites; CHO Cells; Colforsin; Cricetinae; Cystic Fibrosis Transmembrane Conductance Regulator; Dose-Response Relationship, Drug; Genistein; Glutathione Transferase; Glycine; Iodides; Kinetics; Models, Chemical; Patch-Clamp Techniques; Protein Binding; Time Factors

2002
Potentiation of glycine responses by dideoxyforskolin and tamoxifen in rat spinal neurons.
    The European journal of neuroscience, 2003, Volume: 17, Issue:4

    Topics: Alkaloids; Animals; Anticarcinogenic Agents; Benzophenanthridines; Calcium; Cells, Cultured; Colforsin; Dose-Response Relationship, Drug; Drug Synergism; Embryo, Mammalian; Enzyme Inhibitors; Extracellular Space; Glycine; Membrane Potentials; Neurons; Patch-Clamp Techniques; Phenanthridines; Rats; Receptors, GABA-A; Spinal Cord; Tamoxifen; Time Factors; Zinc

2003
Group II metabotropic glutamate receptor modulation of excitatory transmission in rat subthalamic nucleus.
    The Journal of physiology, 2003, Dec-01, Volume: 553, Issue:Pt 2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; 2-Amino-5-phosphonovalerate; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; 6-Cyano-7-nitroquinoxaline-2,3-dione; Adenylyl Cyclase Inhibitors; Amino Acids; Amino Acids, Dicarboxylic; Animals; Colforsin; Cyclopropanes; Electric Stimulation; Electrophysiology; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Glycine; Imines; In Vitro Techniques; Isoquinolines; Male; Picrotoxin; Protein Kinase C; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Subthalamic Nucleus; Sulfonamides; Synaptic Transmission; Tetradecanoylphorbol Acetate; Xanthenes

2003
Comparative pharmacology of the activity of wild-type and G551D mutated CFTR chloride channel: effect of the benzimidazolone derivative NS004.
    The Journal of membrane biology, 2003, Jul-15, Volume: 194, Issue:2

    Topics: Animals; Benzimidazoles; Chlorophenols; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cystic Fibrosis Transmembrane Conductance Regulator; Dose-Response Relationship, Drug; Glycine; Ion Channel Gating; Membrane Potentials; Mutagenesis, Site-Directed; Mutation; Structure-Activity Relationship

2003
Blockade of excitatory amino acid transporters in the rat hippocampus results in enhanced activation of group I and group III metabotropic glutamate receptors.
    Neuropharmacology, 2003, Volume: 45, Issue:7

    Topics: Animals; Aspartic Acid; Benzoates; Colforsin; Cyclic AMP; Excitatory Amino Acid Antagonists; Excitatory Amino Acid Transporter 1; Excitatory Amino Acid Transporter 2; Glycine; Hippocampus; In Vitro Techniques; Inositol 1,4,5-Trisphosphate; Male; Methoxyhydroxyphenylglycol; Pyridines; Quisqualic Acid; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate

2003
Inhibitory effects of group II mGluR-related drugs on memory performance in mice.
    Physiology & behavior, 2004, Volume: 80, Issue:5

    Topics: Amino Acids; Animals; Anticonvulsants; Avoidance Learning; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclopropanes; Dose-Response Relationship, Drug; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Glycine; Isoquinolines; Male; Memory; Mice; Reaction Time; Receptors, Metabotropic Glutamate; Rolipram; Signal Transduction; Sulfonamides; Tetradecanoylphorbol Acetate; Xanthenes

2004
Pharmacological properties of glycine transport in the frog retina.
    Neurochemical research, 2004, Volume: 29, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Amoxapine; Animals; Biological Transport; Colforsin; Glycine; Ranidae; Retina; Sarcosine; Tetradecanoylphorbol Acetate

2004
Glutamate release increases during mossy-CA3 LTP but not during Schaffer-CA1 LTP.
    The European journal of neuroscience, 2004, Volume: 19, Issue:6

    Topics: 2-Amino-5-phosphonovalerate; Animals; Animals, Newborn; Aspartic Acid; Calcium; Colforsin; Coloring Agents; Cyclopropanes; Dose-Response Relationship, Radiation; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Glycine; Hippocampus; In Vitro Techniques; Kynurenic Acid; Long-Term Potentiation; Magnesium; Male; Mossy Fibers, Hippocampal; Neuroglia; Rats; Rats, Sprague-Dawley; Time Factors

2004
AMPA receptor-mediated presynaptic inhibition at cerebellar GABAergic synapses: a characterization of molecular mechanisms.
    The European journal of neuroscience, 2004, Volume: 19, Issue:9

    Topics: Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Benzoxazines; Calcium; Calcium Channel Blockers; Cerebellum; Chelating Agents; Colforsin; Cyclopropanes; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Morpholines; Naphthalenes; Neural Inhibition; Neurons; Piperidines; Presynaptic Terminals; Pyrazoles; Rats; Rats, Wistar; Receptors, AMPA; Ryanodine; Synapses; Triazines; Triazoles

2004
Adenosine inhibits GABAergic and glycinergic transmission in adult rat substantia gelatinosa neurons.
    Journal of neurophysiology, 2004, Volume: 92, Issue:5

    Topics: 4-Aminopyridine; 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Animals; Colforsin; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Neurons; Pain; Phorbol 12,13-Dibutyrate; Potassium Channel Blockers; Potassium Channels; Rats; Substantia Gelatinosa; Synaptic Transmission

2004
Differential modulation of evoked and spontaneous glycine release from rat spinal cord glycinergic terminals by the cyclic AMP/protein kinase A transduction cascade.
    Journal of neurochemistry, 2004, Volume: 91, Issue:3

    Topics: Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Glycine; In Vitro Techniques; Membrane Potentials; Neural Inhibition; Neurons; Patch-Clamp Techniques; Phosphoric Diester Hydrolases; Presynaptic Terminals; Rats; Rats, Wistar; Sacrococcygeal Region; Signal Transduction; Spinal Cord

2004
Differential roles of mGlu8 receptors in the regulation of glutamate and gamma-aminobutyric acid release at periaqueductal grey level.
    Neuropharmacology, 2005, Volume: 49 Suppl 1

    Topics: Alanine; Aminobutyrates; Analysis of Variance; Animals; Benzoates; Colforsin; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Immunohistochemistry; Isoquinolines; Male; Microdialysis; Microscopy, Immunoelectron; Periaqueductal Gray; Phosphoserine; Protein Kinase Inhibitors; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Sulfonamides; Time Factors

2005
A similar impairment in CA3 mossy fibre LTP in the R6/2 mouse model of Huntington's disease and in the complexin II knockout mouse.
    The European journal of neuroscience, 2005, Volume: 22, Issue:7

    Topics: 2-Amino-5-phosphonovalerate; Adaptor Proteins, Vesicular Transport; Age Factors; Animals; Anticonvulsants; Colforsin; Cyclopropanes; Disease Models, Animal; Dose-Response Relationship, Drug; Dose-Response Relationship, Radiation; Drug Interactions; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glycine; Hippocampus; Huntington Disease; In Vitro Techniques; Long-Term Potentiation; Mice; Mice, Knockout; Mossy Fibers, Hippocampal; Nerve Tissue Proteins; Patch-Clamp Techniques; Time Factors

2005
Adenosine A2A receptors and metabotropic glutamate 5 receptors are co-localized and functionally interact in the hippocampus: a possible key mechanism in the modulation of N-methyl-D-aspartate effects.
    Journal of neurochemistry, 2005, Volume: 95, Issue:4

    Topics: Adenosine; Adenosine A2 Receptor Agonists; Animals; Bicuculline; Blotting, Western; Colforsin; Disks Large Homolog 4 Protein; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Embryo, Mammalian; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Postsynaptic Potentials; Female; Fluorescent Antibody Technique; GABA Antagonists; Glycine; Hippocampus; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Membrane Proteins; N-Methylaspartate; Neurons; Patch-Clamp Techniques; Phenethylamines; Phenylacetates; Pregnancy; Presynaptic Terminals; Pyridines; Qa-SNARE Proteins; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Adenosine A2; Receptors, Metabotropic Glutamate; Synaptophysin; Vesicular Glutamate Transport Protein 1

2005
Selective inhibition of spontaneous but not Ca2+ -dependent release machinery by presynaptic group II mGluRs in rat cerebellar slices.
    Journal of neurophysiology, 2006, Volume: 96, Issue:1

    Topics: Action Potentials; Animals; Cadmium; Calcium; Calcium Channels; Cerebellum; Colforsin; Cyclopropanes; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Interneurons; N-Methylaspartate; Nickel; Patch-Clamp Techniques; Presynaptic Terminals; Purkinje Cells; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Synaptic Vesicles

2006
Identification of N-arachidonylglycine as the endogenous ligand for orphan G-protein-coupled receptor GPR18.
    Biochemical and biophysical research communications, 2006, Sep-01, Volume: 347, Issue:3

    Topics: Animals; Arachidonic Acids; Calcium; Cell Line; Colforsin; Cricetinae; Cyclic AMP; Glycine; Humans; Ligands; Receptors, G-Protein-Coupled

2006
Cyclic AMP-mediated long-term facilitation of glycinergic transmission in developing spinal dorsal horn neurons.
    Journal of neurochemistry, 2009, Volume: 110, Issue:5

    Topics: Animals; Animals, Newborn; Cell Differentiation; Colforsin; Cyclic AMP; Glycine; Inhibitory Postsynaptic Potentials; Long-Term Potentiation; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Receptors, Glycine; Substantia Gelatinosa; Synaptic Transmission

2009
GlyT-2 mediates the forskolin-induced increase of glycinergic transmission.
    Neuroreport, 2010, Apr-21, Volume: 21, Issue:6

    Topics: Animals; Colforsin; Glycine; Glycine Plasma Membrane Transport Proteins; Inhibitory Postsynaptic Potentials; Neural Inhibition; Neurons; Neurotransmitter Agents; Organ Culture Techniques; Posterior Horn Cells; Rats; Rats, Sprague-Dawley; Substantia Gelatinosa

2010
Protein kinase A and C signaling induces bilirubin potentiation of GABA/glycinergic synaptic transmission in rat ventral cochlear nucleus neurons.
    Brain research, 2010, Aug-12, Volume: 1348

    Topics: Animals; Animals, Newborn; Antioxidants; Benzophenanthridines; Bilirubin; Cochlear Nucleus; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Isoquinolines; Neural Inhibition; Neurons; Patch-Clamp Techniques; Phorbol Esters; Protein Kinase C; Rats; Signal Transduction; Sulfonamides; Synaptic Transmission

2010
M2 muscarinic acetylcholine receptors regulate long-term potentiation at hippocampal CA3 pyramidal cell synapses in an input-specific fashion.
    Journal of neurophysiology, 2012, Volume: 108, Issue:1

    Topics: Animals; Anthracenes; Anticonvulsants; Biophysical Phenomena; Bungarotoxins; CA3 Region, Hippocampal; Colforsin; Cyclopropanes; Electric Stimulation; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; GABA Antagonists; Gallamine Triethiodide; Glycine; In Vitro Techniques; Long-Term Potentiation; Mice; Mice, Knockout; Nerve Net; Nicotinic Antagonists; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Pyramidal Cells; Receptor, Muscarinic M2; Synapses; Time Factors

2012
Distinct subsets of Syt-IV/BDNF vesicles are sorted to axons versus dendrites and recruited to synapses by activity.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Apr-18, Volume: 32, Issue:16

    Topics: Activated-Leukocyte Cell Adhesion Molecule; Animals; Animals, Newborn; Axons; Brain-Derived Neurotrophic Factor; Cells, Cultured; Coculture Techniques; Colforsin; Dendrites; Disks Large Homolog 4 Protein; Embryo, Mammalian; Excitatory Amino Acid Agents; Excitatory Postsynaptic Potentials; Female; Glycine; Hippocampus; Humans; Intracellular Signaling Peptides and Proteins; Luminescent Proteins; Male; Membrane Proteins; Mice; Mice, Knockout; Microtubule-Associated Proteins; Neurons; Patch-Clamp Techniques; Rats; Receptors, AMPA; Sodium Channel Blockers; Synapses; Synaptic Vesicles; Synaptophysin; Synaptotagmins; Tetrodotoxin; Time Factors; Transfection; Vesicular Glutamate Transport Protein 1; Vesicular Inhibitory Amino Acid Transport Proteins

2012
Presynaptic mGlu7 receptors control GABA release in mouse hippocampus.
    Neuropharmacology, 2013, Volume: 66

    Topics: Adenylyl Cyclase Inhibitors; Aminobutyrates; Animals; Baclofen; Benzhydryl Compounds; Benzoates; Benzylamines; Colforsin; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Exocytosis; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Hippocampus; Imines; Mice; Phosphinic Acids; Potassium Chloride; Pyridones; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Synaptosomes; Syntaxin 1; Vesicular Inhibitory Amino Acid Transport Proteins

2013
Relationship between increase in astrocytic GLT-1 glutamate transport and late-LTP.
    Learning & memory (Cold Spring Harbor, N.Y.), 2012, Nov-19, Volume: 19, Issue:12

    Topics: Alanine Transaminase; Analysis of Variance; Animals; Animals, Newborn; Aspartic Acid; Astrocytes; Biophysics; Biotinylation; Cells, Cultured; Colforsin; Electric Stimulation; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Excitatory Amino Acid Transporter 1; Excitatory Amino Acid Transporter 2; Excitatory Postsynaptic Potentials; Flow Cytometry; Glial Fibrillary Acidic Protein; Glutamates; Glutamic Acid; Glycine; Hippocampus; In Vitro Techniques; Indoles; Kainic Acid; Long-Term Potentiation; Male; Neurons; Protein Transport; Quinoxalines; Rats; Rats, Sprague-Dawley; Sodium Channel Blockers; Tetrodotoxin; Valine

2012
CFTR and Anoctamin 1 (ANO1) contribute to cAMP amplified exocytosis and insulin secretion in human and murine pancreatic beta-cells.
    BMC medicine, 2014, May-28, Volume: 12

    Topics: Animals; Anoctamin-1; Calcium; Calcium Channels; Chloride Channels; Colforsin; Cyclic AMP; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Exocytosis; Glucagon-Like Peptide 1; Glycine; Humans; Hydrazines; Insulin-Secreting Cells; Insulins; Ion Channels; Mice; Neoplasm Proteins; Patch-Clamp Techniques

2014
Mechanosensitive activation of CFTR by increased cell volume and hydrostatic pressure but not shear stress.
    Biochimica et biophysica acta, 2015, Volume: 1848, Issue:11 Pt A

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Cell Size; Chlorides; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Epithelium; Female; Glycine; Humans; Hydrazines; Hydrostatic Pressure; Ion Channel Gating; Lung; Membrane Potentials; Mutation; Oocytes; Patch-Clamp Techniques; Shear Strength; Stress, Mechanical; Xenopus laevis

2015