colforsin has been researched along with glyburide in 104 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 1 (0.96) | 18.7374 |
1990's | 52 (50.00) | 18.2507 |
2000's | 44 (42.31) | 29.6817 |
2010's | 7 (6.73) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K | 1 |
Alibhai, KN; Huizinga, JD; Richardson, D | 1 |
Cooper, CW; Ishizuka, J; Murakami, M; Nickols, GA; Sumi, S; Thompson, JC; Townsend, CM | 1 |
Burnham, BL; Chick, WL; Clark, SA | 1 |
Ashcroft, SJ; Niki, I | 1 |
Greger, R; Kunzelmann, K; Lindeman, S; Lindeman, V; Pavenstädt, H; Späth, M | 1 |
Beggs, M; Beresford, G; Clarke, J; Espinal, J; Hammonds, P; Mertz, RJ | 1 |
Berg, M; Boyd, AE; Gaines, KL; Nelson, TY; Rajan, AS | 1 |
Chang, CH; Chang, TM; Chey, WY; Coy, DH | 1 |
Khan, SA; Mathews, WR; Meisheri, KD | 1 |
Hiramatsu, T; Kotlikoff, MI; Kume, H; Takagi, K | 1 |
Nakashima, M; Vanhoutte, PM | 1 |
Horie, M; Okada, Y; Sasayama, S; Tominaga, M | 1 |
Burns, DM; Howard, GA; Kawase, T; Roos, BA | 1 |
Horie, M; Okada, Y; Tominaga, M | 1 |
Maggi, CA; Morbidelli, L; Parenti, A; Santicioli, P; Ziche, M | 1 |
Devor, DC; Forrest, JN; Frizzell, RA; Suggs, WK | 1 |
Giuliani, S; Maggi, CA; Santicioli, P | 1 |
Kalsner, S | 1 |
Heath, BM; Terrar, DA | 1 |
Akatsuka, Y; Egashira, K; Katsuda, Y; Narishige, T; Shimokawa, H; Takeshita, A; Ueno, H | 1 |
Aizawa, T; Hashizume, K; Ishihara, F; Komatsu, M; Nishii, N; Sato, Y; Suzuki, N; Yamada, T | 1 |
Bonev, AD; Mawe, GM; Nelson, MT; Zhang, L | 1 |
Gao, Y; Nishimura, Y; Suzuki, A; Yoshida, K | 1 |
Baró, I; Berthon, B; Escande, D; Hongre, AS | 1 |
Bonev, AD; Brayden, JE; Nelson, MT; Quayle, JM | 1 |
Jackson, WF | 1 |
Ko, FN; Lin, CH; Lu, ST; Teng, CM; Wu, YC | 1 |
Faraci, FM; Heistad, DD; Kitazono, T | 1 |
Baró, I; Demolombe, S; Escande, D; Loussouarn, G; Mohammad-Panah, R | 1 |
Bridges, RJ; Devor, DC; Frizzell, RA; Singh, AK | 1 |
Gidday, JM; Maceren, RG; Meier, JA; Shah, AR; Zhu, Y | 1 |
Hüsken, BC; Pfaffendorf, M; van Zwieten, PA | 1 |
Baumlin, Y; Kessler, C; Linde, C; Löffler, C; Quast, U | 1 |
Illek, B; Machen, TE; Yankaskas, JR | 1 |
Huang, Y; Kwok, KH | 1 |
Chan, HC; Chung, YW; Fong, SK; So, SC; Wong, PY | 1 |
al-Nakkash, L; Cotton, CU | 1 |
Buus, C; Mulvany, MJ; Nilsson, H; Prieto, D | 1 |
Kocić, I | 1 |
Fullerton, DA; McIntyre, RC; Meldrum, DR; Sheridan, BC | 1 |
Becq, F; Chappe, V; Gola, M; Hanrahan, JW; Mettey, Y; Verrier, B; Vierfond, JM | 1 |
Ookuma, K; Ookuma, M; York, DA | 1 |
Edwards, RH; Grodsky, GM; Ma, YH | 1 |
Collins, R; Rodriguez-Pena, MS; Spiegel, AM; Woodard, C | 1 |
Benes, C; Creuzet, C; Fagard, R; Miyazaki, J; Roisin, MP; Van Tan, H | 1 |
Katusic, ZS; Onoue, H | 1 |
Burns, DM; Kawase, T | 1 |
Brahimi-Horn, MC; Capeau, J; Mailleau, C | 1 |
von der Weid, PY | 1 |
Hill, RJ; Magee, W; Masamune, H; Oleynek, JJ; Tracey, WR | 1 |
Becq, F; Cerutti, M; Chappe, V; Devauchelle, G; Gola, M; Julien, M; Verrier, B | 1 |
Argent, BE; Becq, F; Bulteau, L; Chappe, V; Dérand, R; Dormer, RL; Figarella, C; Galietta, LJ; Gola, M; Gray, MA; Joffre, M; Kammouni, W; Marvingt-Mounir, C; McPherson, MA; Merten, M; Métayé, T; Mettey, Y; Pereira, MM; Rogier, C; Sarrouilhe, D; Tarran, R; Verrier, B; Vierfond, JM; Zegarra-Moran, O | 1 |
Hourani, SM; Pearson, A; Tennant, JP | 1 |
Bridges, RJ; Devor, DC; Gerlach, AC; Gondor, M; Pilewski, JM; Singh, AK | 1 |
Elliott, RA; Hudman, D; Norman, RI | 1 |
Bottrill, FE; Hiley, CR; Omar, R; White, R | 1 |
Asai, M; Iwasaki, Y; Morishita, M; Mutsuga, N; Nomura, A; Oiso, Y; Saito, H; Yamamori, E; Yoshida, M | 1 |
Harvey, BJ; Urbach, V; Walsh, DE | 1 |
Beauwens, R; Boom, A; Frerotte, M; Golstein, PE; Sande, JV | 1 |
Chang, HY; Chen, CW; Hsiue, TR | 1 |
Becq, F; Bulteau, L; Dérand, R; Dormer, RL; Folli, C; Galietta, LJ; Joffre, M; Jougla, C; McNeilly, CM; Métayé, T; Mettey, Y; Morris, MR; Pereira, MM; Vierfond, JM; Zegarra-Moran, O | 1 |
Hein, TW; Kuo, L; Muthuchamy, M; Wang, W; Zoghi, B | 1 |
García de Boto, MJ; Hidalgo, A; Martínez, C; Sánchez, M | 1 |
Meadows, HJ; Randall, AD | 1 |
Akagawa, Y; Hirono, C; Iwasa, Y; Nakamoto, T; Shiba, Y; Sugita, M | 1 |
Van Helden, DF; von der Weid, PY; Zhao, J | 1 |
Barbry, P; Fischer, H; Fukuda, N; Illek, B; Matthay, MA; Sartori, C | 1 |
Al-Nakkash, L; Reinach, PS | 1 |
Bessard, G; Bréant, D; Caron, F; Corompt, E; Devillier, P | 1 |
Bonanno, JA; Sun, XC | 1 |
Bridges, RJ; Devor, DC; Frizzell, RA; Singh, AK; Singh, S; van Driessche, W | 1 |
Dura, E; Jijakli, H; Malaisse, WJ; Oguzhan, B; Sener, A; Zhang, HX | 1 |
Bai, C; Jiang, J; Koller, BH; Matthay, MA; Song, Y; Verkman, AS | 1 |
Butt, AG; Carter, DJ; Cheng, S; Hamilton, KL | 1 |
Lazrak, A; Matalon, S | 1 |
Clancy, JP; Cobb, BR; Fan, L; Kovacs, TE; Sorscher, EJ | 1 |
Harvey, JR; Vogalis, F | 1 |
Assef, YA; Damiano, AE; Ibarra, C; Kotsias, BA; Zotta, E | 1 |
Ishikawa, T; Ito, Y; Kondo, M; Kume, H; Nakayama, S; Sato, S; Shimokata, K; Son, M | 1 |
Berthiaume, Y; Brochiero, E; Dagenais, A; Leroy, C | 1 |
Becq, F; Bulteau-Pignoux, L; Dérand, R; Janet, T; Montoni, A; Moreau, B; Muller, JM | 1 |
Bendhack, LM; Callera, GE; Caperuto, LC; Carvalho, CR; Tostes, RC; Yeh, E | 1 |
Chidekel, A; Ramesh Babu, PB; Shaffer, TH; Utidjian, L | 1 |
Joo, NS; Lee, DJ; Rustagi, A; Wine, JJ; Winges, KM | 1 |
Finkbeiner, WF; Muanprasat, C; Nielson, DW; Pedemonte, N; Salinas, DB; Verkman, AS | 1 |
Basavappa, S; Coon, S; Sundaram, U; Vulapalli, SR; Yule, D; Zhang, H | 1 |
Chemtob, S; Clyman, RI; Fouron, JC; Ginzinger, D; Kajino, H; Marrache, AM; Moss, TJ; Roman, C; Seidner, SR; Vazquez-Tello, A; Waleh, N | 1 |
Findlay, IA; Li, H; Sheppard, DN | 1 |
Borba, PF; Jacobus, AP; Loss, ES; Rodrigues, DO; Wassermann, GF | 1 |
Becq, F; Norez, C; Robert, R | 1 |
Szkudelski, T | 1 |
Ameen, N; Melvin, JE; Vidyasagar, S; Zhang, H | 1 |
Becq, F; Guibert, C; Norez, C; Robert, R; Savineau, JP | 1 |
Chen, X; Tian, YM; Xing, Y; Xue, H; Yan, M; Yang, N; Zhu, JX | 1 |
Clancy, JP; Cormet-Boyaka, E; Fan, L; Kirk, KL; Maloney, K; Musgrove, L; Rennolds, J; Sztul, E; Tower, C | 1 |
Eguchi, S; Kawano, T; Mawatari, K; Nakajo, N; Nakaya, Y; Oshita, S; Takahashi, A; Tanaka, K; Yasui, S | 1 |
Britton, F; Dixon, R; Hwang, S; Sanders, K; Ward, S | 1 |
Al-Nakkash, L; Batia, L; Bhakta, M; Hale, N; Jensen, J; Peterson, A; Sears, S; Skinner, R | 1 |
Ballard, HJ; Cai, W; Lu, L; Tu, J | 1 |
Deachapunya, C; Poonyachoti, S | 1 |
Gurgul-Convey, E; Kaminski, MT; Lenzen, S | 1 |
Lenzen, S; Teraoku, H | 1 |
104 other study(ies) available for colforsin and glyburide
Article | Year |
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Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship | 2010 |
On the pharmacological and physiological role of glibenclamide-sensitive potassium channels in colonic smooth muscle.
Topics: Animals; Benzopyrans; Carbachol; Colforsin; Colon; Cromakalim; Dogs; Drug Interactions; Electric Stimulation; Female; Gallopamil; Glyburide; Male; Muscle Contraction; Muscle, Smooth; Potassium Channels; Pyrroles; Stereoisomerism | 1992 |
Role of extracellular magnesium in insulin secretion from rat insulinoma cells.
Topics: Animals; Calcium; Cell Line; Colforsin; Glyburide; Glyceraldehyde; Insulin; Insulin Secretion; Insulinoma; Kinetics; Magnesium; Pancreatic Neoplasms; Potassium Chloride; Rats; Tumor Cells, Cultured; Verapamil | 1992 |
Modulation of glucose-induced insulin secretion from a rat clonal beta-cell line.
Topics: 1-Methyl-3-isobutylxanthine; Alanine; Animals; Carbachol; Cell Line; Clone Cells; Clonidine; Colforsin; Dose-Response Relationship, Drug; Glucose; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Potassium; Rats; Stereoisomerism | 1990 |
Possible involvement of protein phosphorylation in the regulation of the sulphonylurea receptor of a pancreatic beta-cell line, HIT T15.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Adenosine Triphosphatases; Adenosine Triphosphate; Animals; ATP-Binding Cassette Transporters; Cell Line; Cell Membrane; Colforsin; Diazoxide; Glyburide; Humans; Insulin; Insulin Secretion; Islets of Langerhans; Isoquinolines; Phosphorylation; Piperazines; Potassium Channels; Potassium Channels, Inwardly Rectifying; Protein Kinase Inhibitors; Proteins; Receptors, Drug; Rubidium; Sulfonylurea Receptors; Tetradecanoylphorbol Acetate | 1991 |
Effect of depolarizing and hyperpolarizing agents on the membrane potential difference of primary cultures of rabbit aorta vascular smooth muscle cells.
Topics: Animals; Aorta; Benzopyrans; Cattle; Cells, Cultured; Colforsin; Cromakalim; Glyburide; Membrane Potentials; Muscle, Smooth, Vascular; Nucleotides; Pyrroles; Rabbits | 1991 |
Insulin-secreting beta-cells possess specific receptors for interleukin-1 beta.
Topics: Calcium; Cell Line; Colforsin; Diglycerides; Glucose; Glyburide; Homeostasis; Insulin; Insulin Secretion; Interleukin-1; Islets of Langerhans; Receptors, Immunologic; Receptors, Interleukin-1; Second Messenger Systems | 1990 |
Increased cytosolic calcium. A signal for sulfonylurea-stimulated insulin release from beta cells.
Topics: Animals; Calcium; Cells, Cultured; Colforsin; Cricetinae; Cyclic AMP; Glyburide; Insulin; Islets of Langerhans; Tolbutamide; Verapamil | 1987 |
Galanin inhibits cholecystokinin secretion in STC-1 cells.
Topics: Adenylate Cyclase Toxin; Animals; Bombesin; Cell Line; Cholecystokinin; Colforsin; Cyclic AMP; Galanin; Glyburide; Kinetics; Mice; Neuroendocrine Tumors; Neuropeptides; Neurotransmitter Agents; Pituitary Adenylate Cyclase-Activating Polypeptide; Potassium Channel Blockers; Potassium Chloride; Rats; Tumor Cells, Cultured; Virulence Factors, Bordetella | 1995 |
Role of calcium-activated K+ channels in vasodilation induced by nitroglycerine, acetylcholine and nitric oxide.
Topics: Acetylcholine; Adenosine Triphosphate; Animals; Calcium; Charybdotoxin; Colforsin; Drug Interactions; Glyburide; Guanidines; Mesenteric Arteries; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Nitroglycerin; Norepinephrine; Peptides; Pinacidil; Potassium; Potassium Channels; Rabbits; Scorpion Venoms; Vasodilation; Vasodilator Agents | 1993 |
Role of calcium-activated potassium channels in the relaxation of tracheal smooth muscles by forskolin.
Topics: Animals; Apamin; Calcium; Carbachol; Charybdotoxin; Colforsin; Cyclic AMP; Drug Interactions; Electrophysiology; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Nifedipine; Potassium Channel Blockers; Potassium Channels; Scorpion Venoms; Trachea | 1994 |
Isoproterenol causes hyperpolarization through opening of ATP-sensitive potassium channels in vascular smooth muscle of the canine saphenous vein.
Topics: Animals; Atenolol; Charybdotoxin; Colforsin; Dogs; Female; Glyburide; Ion Channel Gating; Isoproterenol; Male; Membrane Potentials; Muscle, Smooth, Vascular; Ouabain; Potassium Channels; Propanolamines; Receptors, Adrenergic, beta; Saphenous Vein; Scorpion Venoms; Yohimbine | 1995 |
Glibenclamide, an ATP-sensitive K+ channel blocker, inhibits cardiac cAMP-activated Cl- conductance.
Topics: Animals; Chloride Channels; Colforsin; Cyclic AMP; Electrophysiology; Glyburide; Guinea Pigs; Heart; In Vitro Techniques; Isoproterenol; Male; Myocardium; Phosphorylation | 1995 |
Diverse actions of calcitonin gene-related peptide on intracellular free Ca2+ concentrations in UMR 106 osteoblastic cells.
Topics: Adenosine Triphosphate; Animals; Bone Neoplasms; Calcitonin; Calcitonin Gene-Related Peptide; Calcium; Colforsin; Dose-Response Relationship, Drug; Egtazic Acid; Fura-2; Glyburide; Guanidines; Osteoblasts; Osteosarcoma; Pinacidil; Potassium; Potassium Channels; Rats; Spectrometry, Fluorescence; Tumor Cells, Cultured; Vasodilator Agents | 1995 |
Additional similarity of cardiac cAMP-activated Cl- channels to CFTR Cl- channels.
Topics: Animals; Blotting, Northern; Chloride Channels; Colforsin; Cyclic AMP; Cystic Fibrosis; Glyburide; Guinea Pigs; Heart; RNA, Messenger | 1994 |
Calcitonin gene-related peptide selectively increases cAMP levels in the guinea-pig ureter.
Topics: Animals; Benzopyrans; Calcitonin Gene-Related Peptide; Colforsin; Cromakalim; Cyclic AMP; Cyclic GMP; Drug Interactions; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Membrane Potentials; Potassium Channels; Pyrroles; Ureter | 1995 |
cAMP-activated Cl- channels in primary cultures of spiny dogfish (Squalus acanthias) rectal gland.
Topics: Animals; Cells, Cultured; Chloride Channels; Colforsin; Cyclic AMP; Dogfish; Electrophysiology; Glyburide; Iodides; Salt Gland | 1995 |
Multiple mechanisms in the smooth muscle relaxant action of calcitonin gene-related peptide (CGRP) in the guinea-pig ureter.
Topics: Action Potentials; Animals; Arginine; Benzopyrans; Calcitonin Gene-Related Peptide; Colforsin; Cromakalim; Dose-Response Relationship, Drug; Electric Stimulation; Glyburide; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Nitroarginine; Parasympatholytics; Pyrroles; Ureter | 1994 |
Propranolol antagonizes coronary artery relaxation by a potassium channel opener.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Biological Transport; Cattle; Colforsin; Coronary Vessels; Cyclic AMP; Drug Interactions; Glyburide; Guanidines; Guinea Pigs; In Vitro Techniques; Muscle Relaxation; Muscle, Smooth; Muscle, Smooth, Vascular; Nitroprusside; Pinacidil; Potassium Channels; Propranolol; Rubidium Radioisotopes; Trachea; Vasodilator Agents | 1994 |
Effect of glibenclamide, forskolin, and isoprenaline on the parallel activation of KATP and reduction of IK by cromakalim in cardiac myocytes.
Topics: Animals; Benzopyrans; Cells, Cultured; Colforsin; Cromakalim; Glyburide; Guinea Pigs; Isoproterenol; Myocardium; Potassium Channels; Pyrroles; Sodium-Potassium-Exchanging ATPase; Vasodilator Agents | 1994 |
ATP sensitive potassium channels are involved in adenosine A2 receptor mediated coronary vasodilatation in the dog.
Topics: Acetylcholine; Adenosine; Adenosine Triphosphate; Adenosine-5'-(N-ethylcarboxamide); Animals; Colforsin; Coronary Circulation; Dogs; Dose-Response Relationship, Drug; Glyburide; Guanidines; Ion Channel Gating; Pinacidil; Potassium Channels; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P2; Theophylline; Vasodilator Agents; Xanthines | 1994 |
Insulin secretion by the pancreatic beta cell of aged rats.
Topics: Aging; Animals; Colforsin; Dose-Response Relationship, Drug; Glucose; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Male; Nifedipine; Potassium; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate | 1994 |
Protein kinase A mediates activation of ATP-sensitive K+ currents by CGRP in gallbladder smooth muscle.
Topics: Adenosine Triphosphate; Animals; Calcitonin Gene-Related Peptide; Colforsin; Cyclic AMP-Dependent Protein Kinases; Electrophysiology; Ethers, Cyclic; Female; Gallbladder; Glyburide; Guanosine Diphosphate; Guinea Pigs; Male; Muscle, Smooth; Okadaic Acid; Phosphoric Monoester Hydrolases; Potassium Channels; Thionucleotides | 1994 |
Relaxant effects of calcitonin gene-related peptide on isolated small renal arteries in stroke-prone spontaneously hypertensive rats.
Topics: Acetylcholine; Animals; Calcitonin Gene-Related Peptide; Colforsin; Dose-Response Relationship, Drug; Glyburide; Hypertension; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Renal Artery | 1994 |
Effects of sulphonylureas on cAMP-stimulated Cl- transport via the cystic fibrosis gene product in human epithelial cells.
Topics: Adenosine Triphosphate; Blood Proteins; Cell Line; Chloride Channels; Colforsin; Cyclic AMP; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Diazoxide; Electrophysiology; Glyburide; Humans; Sulfonylurea Compounds; Tolbutamide | 1994 |
Calcitonin gene-related peptide activated ATP-sensitive K+ currents in rabbit arterial smooth muscle via protein kinase A.
Topics: Adenosine Triphosphate; Adenylyl Cyclases; Animals; Biotransformation; Calcitonin Gene-Related Peptide; Calcium; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electrophysiology; Enzyme Activation; Glyburide; In Vitro Techniques; Mesenteric Arteries; Muscle, Smooth, Vascular; Potassium Channels; Rabbits; Signal Transduction; Vasodilation | 1994 |
Arteriolar tone is determined by activity of ATP-sensitive potassium channels.
Topics: Adenosine Triphosphate; Animals; Arterioles; Benzopyrans; Bucladesine; Colforsin; Cricetinae; Cromakalim; Epoprostenol; Glyburide; Guanidines; Isoproterenol; Male; Mesocricetus; Methacholine Chloride; Muscle Tonus; Muscle, Smooth, Vascular; Muscles; Nitroprusside; Pinacidil; Potassium Channels; Pyrroles; Quaternary Ammonium Compounds; Vasoconstriction; Vasodilation; Vasodilator Agents | 1993 |
The relaxant actions on guinea-pig trachealis of atherosperminine isolated from Fissistigma glaucescens.
Topics: Alkaloids; Animals; Benzopyrans; Calcium; Calmodulin; Colforsin; Cromakalim; Cyclic AMP; Cyclic GMP; Egtazic Acid; Epithelium; Female; Glyburide; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Nifedipine; Nitroprusside; Phenanthrenes; Plants, Medicinal; Propranolol; Pyrroles; Theophylline; Trachea; Vasodilator Agents | 1993 |
Effect of norepinephrine on rat basilar artery in vivo.
Topics: Animals; Arginine; Basilar Artery; Colforsin; Glyburide; Male; NG-Nitroarginine Methyl Ester; Norepinephrine; Rats; Rats, Sprague-Dawley; Vasodilation | 1993 |
Expression of CFTR controls cAMP-dependent activation of epithelial K+ currents.
Topics: Calcium; Cell Line; Charybdotoxin; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Epithelium; Glyburide; Humans; Ionomycin; Kinetics; Membrane Potentials; Pancreas; Patch-Clamp Techniques; Potassium Channels; Recombinant Proteins; Thionucleotides; Transfection | 1996 |
Modulation of Cl- secretion by benzimidazolones. II. Coordinate regulation of apical GCl and basolateral GK.
Topics: Animals; Benzimidazoles; Bumetanide; Calcium; Carbachol; Cell Line; Cell Membrane; Charybdotoxin; Chloride Channels; Chlorides; Chlorophenols; Colforsin; Drug Synergism; Glyburide; Kinetics; Membrane Potentials; Patch-Clamp Techniques; Time Factors | 1996 |
KATP channels mediate adenosine-induced hyperemia in retina.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenosine Triphosphate; Adenylyl Cyclases; Animals; Benzopyrans; Colforsin; Cromakalim; Cyclic AMP; Dose-Response Relationship, Drug; Fluorescein Angiography; Glyburide; Hyperemia; Muscle, Smooth, Vascular; Potassium Channel Blockers; Potassium Channels; Pyrroles; Regional Blood Flow; Retinal Vessels; Second Messenger Systems; Signal Transduction; Swine; Vasodilation; Vasodilator Agents | 1996 |
Contribution of ATP-sensitive potassium channels to beta-adrenoceptor-mediated responses.
Topics: Adenosine Triphosphate; Animals; Bisoprolol; Colforsin; Dose-Response Relationship, Drug; Glyburide; In Vitro Techniques; Isoproterenol; Male; Muscle, Smooth, Vascular; Potassium Channels; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Vasoconstriction | 1997 |
Activators of protein kinase A induce a glibenclamide-sensitive 86Rb+ efflux in rat isolated aorta.
Topics: Animals; Aorta; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Glyburide; Male; Rats; Rats, Sprague-Dawley; Rubidium | 1997 |
cAMP and genistein stimulate HCO3- conductance through CFTR in human airway epithelia.
Topics: Adenosine Triphosphate; Bicarbonates; Cell Membrane; Chlorides; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Electric Conductivity; Enzyme Inhibitors; Genistein; Glyburide; Humans; Isoflavones; Lung; ortho-Aminobenzoates; Phosphoric Monoester Hydrolases; Tumor Cells, Cultured | 1997 |
Effects of putative K+ channel blockers on beta-adrenoceptor-mediated vasorelaxation of rat mesenteric artery.
Topics: Adenosine Triphosphate; Adrenergic beta-Agonists; Animals; Barium; Benzopyrans; Calcium; Charybdotoxin; Colforsin; Cromakalim; Cyclic AMP; Dose-Response Relationship, Drug; Fenoterol; Glyburide; Isoproterenol; Male; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phenylephrine; Potassium Channel Blockers; Pyrroles; Rats; Rats, Sprague-Dawley; Vasoconstrictor Agents; Vasodilator Agents | 1997 |
Stimulation of anion secretion by beta-adrenoceptors in the mouse endometrial epithelium.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adrenergic Agonists; Adrenergic Antagonists; Animals; Anions; Cells, Cultured; Chloride Channels; Colforsin; Cyclic AMP; Endometrium; Epinephrine; Epithelium; Female; Glyburide; Imines; Ion Transport; Isoproterenol; Mice; Propranolol; Receptors, Adrenergic, beta | 1997 |
Bovine pancreatic duct cells express cAMP- and Ca(2+)-activated apical membrane Cl- conductances.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Adenosine Triphosphate; Animals; Anions; Calcium; Cattle; Cell Line; Cells, Cultured; Chelating Agents; Chloride Channels; Chlorides; Colforsin; Cyclic AMP; Egtazic Acid; Epithelial Cells; Epithelium; Glyburide; Ionomycin; Kinetics; Membrane Potentials; ortho-Aminobenzoates; Pancreatic Ducts; Theophylline | 1997 |
Interactions between neuropeptide Y and the adenylate cyclase pathway in rat mesenteric small arteries: role of membrane potential.
Topics: 4-Aminopyridine; Acetylcholine; Adenylyl Cyclases; Animals; Charybdotoxin; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dichlororibofuranosylbenzimidazole; Gadolinium; Glyburide; In Vitro Techniques; Isoproterenol; Male; Membrane Potentials; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Neuropeptide Y; Nifedipine; Potassium Channels; Rats; Rats, Wistar; Thionucleotides | 1997 |
Pretreatment with rimalkalim changes the adrenergic responsiveness of isolated guinea pig papillary muscle.
Topics: Animals; Bucladesine; Cardiotonic Agents; Chromans; Colforsin; Enzyme Inhibitors; Female; Glyburide; Guinea Pigs; Male; Metoprolol; Muscle Relaxants, Central; Papillary Muscles; Phenylephrine; Potassium Channels; Pyrrolidines; Sympathetic Nervous System; Thapsigargin | 1997 |
KATP channels contribute to beta- and adenosine receptor-mediated pulmonary vasorelaxation.
Topics: Acetylcholine; Adenosine; Adenylyl Cyclases; Animals; ATP-Binding Cassette Transporters; Colforsin; Cromakalim; Cyclic AMP; Cyclic GMP; Glyburide; In Vitro Techniques; Isoproterenol; KATP Channels; Kinetics; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pulmonary Artery; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, Purinergic P1; Tolbutamide; Vasodilation | 1997 |
Structural basis for specificity and potency of xanthine derivatives as activators of the CFTR chloride channel.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Glyburide; Iodides; Ion Transport; Patch-Clamp Techniques; Recombinant Proteins; Structure-Activity Relationship; Xanthines | 1998 |
Effects of leptin on insulin secretion from isolated rat pancreatic islets.
Topics: Animals; Calcium; Colforsin; Enzyme Activation; Glucose; Glyburide; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Leptin; Male; Mice; Protein Kinase C; Proteins; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate | 1998 |
Chronic sympathetic innervation of islets in transgenic mice results in differential desensitization of alpha-adrenergic inhibition of insulin secretion.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Glucose; Colforsin; Female; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Mice, Inbred C57BL; Mice, Transgenic; Nerve Growth Factors; Phentolamine; Promoter Regions, Genetic; Rats; Receptors, Adrenergic, alpha; Recombinant Fusion Proteins; Reference Values; Sympathetic Nervous System; Time Factors | 1997 |
Decreased insulin content and secretion in RIN 1046-38 cells overexpressing alpha 2-adrenergic receptors.
Topics: Animals; Antibodies, Monoclonal; Carbachol; Cell Line; Colforsin; Cyclic AMP; Fluorescent Antibody Technique, Indirect; Gastric Inhibitory Polypeptide; Gene Expression; Glucose; Glyburide; GTP-Binding Protein alpha Subunits, Gi-Go; Humans; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Mice; Pertussis Toxin; Potassium Chloride; Receptors, Adrenergic, alpha; Transfection; Virulence Factors, Bordetella | 1997 |
Rapid activation and nuclear translocation of mitogen-activated protein kinases in response to physiological concentration of glucose in the MIN6 pancreatic beta cell line.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium-Calmodulin-Dependent Protein Kinases; Cell Line; Cell Nucleus; Colforsin; Egtazic Acid; Enzyme Activation; Glucose; Glyburide; Hypoglycemic Agents; Islets of Langerhans; Kainic Acid; Mice; Mice, Transgenic; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Mitogen-Activated Protein Kinases; Nifedipine; Potassium; Receptors, Glutamate | 1998 |
The effect of subarachnoid hemorrhage on mechanisms of vasodilation mediated by cyclic adenosine monophosphate.
Topics: 4-Aminopyridine; Adenylyl Cyclases; Animals; Basilar Artery; Charybdotoxin; Colforsin; Cyclic AMP; Disease Models, Animal; Dogs; Endothelium, Vascular; Enzyme Activation; Female; Glyburide; Ischemic Attack, Transient; Male; Potassium Channel Blockers; Potassium Channels; Subarachnoid Hemorrhage; Vasodilation; Vasodilator Agents | 1998 |
Calcitonin gene-related peptide stimulates potassium efflux through adenosine triphosphate-sensitive potassium channels and produces membrane hyperpolarization in osteoblastic UMR106 cells.
Topics: Adenosine Triphosphate; Animals; Calcitonin Gene-Related Peptide; Colforsin; Enzyme Inhibitors; Glyburide; Guanidines; Isoquinolines; Membrane Potentials; Osteoblasts; Osteosarcoma; Pinacidil; Potassium; Potassium Channel Blockers; Potassium Channels; Protein Kinase Inhibitors; Rats; Sulfonamides; Tetraethylammonium; Tumor Cells, Cultured | 1998 |
Interrelationship between the Na+/glucose cotransporter and CFTR in Caco-2 cells: relevance to cystic fibrosis.
Topics: Biological Transport; Caco-2 Cells; Calcium Channel Blockers; Cell Differentiation; Chlorides; Colforsin; Cyclic AMP; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Dose-Response Relationship, Drug; Enzyme Inhibitors; Glucose; Glyburide; Glycoconjugates; Humans; Ion Channel Gating; Membrane Glycoproteins; Monosaccharide Transport Proteins; ortho-Aminobenzoates; Phlorhizin; Sodium; Sodium-Glucose Transporter 1; Thionucleotides | 1998 |
ATP-sensitive K+ channels in smooth muscle cells of guinea-pig mesenteric lymphatics: role in nitric oxide and beta-adrenoceptor agonist-induced hyperpolarizations.
Topics: Adenosine Triphosphate; Adrenergic beta-Agonists; Animals; Colforsin; Cyclic GMP; Enzyme Inhibitors; Glyburide; Guanylate Cyclase; Guinea Pigs; Isoproterenol; Isoquinolines; Membrane Potentials; Mesenteric Arteries; Muscle, Smooth, Vascular; Nitric Oxide; Potassium Channel Blockers; Potassium Channels; Protein Kinase Inhibitors; Receptors, Adrenergic, beta; Sulfonamides | 1998 |
Selective activation of adenosine A3 receptors with N6-(3-chlorobenzyl)-5'-N-methylcarboxamidoadenosine (CB-MECA) provides cardioprotection via KATP channel activation.
Topics: Adenosine; Adenylyl Cyclases; Animals; Anti-Arrhythmia Agents; Binding, Competitive; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Decanoic Acids; Dose-Response Relationship, Drug; Glyburide; Hydroxy Acids; Hypoglycemic Agents; Myocardial Reperfusion Injury; Myocardium; Perfusion; Potassium Channels; Rabbits; Receptor, Adenosine A3; Receptors, Purinergic P1; Xanthines | 1998 |
Cystic fibrosis transmembrane conductance regulator (CFTR) confers glibenclamide sensitivity to outwardly rectifying chloride channel (ORCC) in Hi-5 insect cells.
Topics: 1-Methyl-3-isobutylxanthine; 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; Animals; ATP-Binding Cassette Transporters; beta-Galactosidase; Calcium Channels; Cells, Cultured; Chlorides; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Genetic Vectors; Glyburide; Humans; Ion Channel Gating; Moths; Nucleopolyhedroviruses; Patch-Clamp Techniques; Recombinant Fusion Proteins; Spodoptera; Xanthines | 1999 |
Development of substituted Benzo[c]quinolizinium compounds as novel activators of the cystic fibrosis chloride channel.
Topics: Animals; CHO Cells; Cilia; Colforsin; Cricetinae; Cystic Fibrosis Transmembrane Conductance Regulator; Drug Design; Female; Glyburide; Humans; Male; Membrane Potentials; Mice; Mice, Inbred BALB C; Mice, Knockout; Molecular Structure; Nasal Mucosa; Patch-Clamp Techniques; Quinolines; Quinolizines; Recombinant Proteins; Structure-Activity Relationship; Transfection | 1999 |
Effects of noradrenaline, the calcium ionophore A23187, forskolin, sodium nitroprusside and glibenclamide on the degradation of extracellular adenosine 5'-triphosphate by the rat isolated vas deferens.
Topics: 5'-Nucleotidase; Adenosine Diphosphate; Adenosine Monophosphate; Adenosine Triphosphate; Animals; Calcimycin; Colforsin; Glyburide; Inosine; Male; Nitroprusside; Norepinephrine; Rats; Rats, Wistar; Time Factors; Vas Deferens | 1999 |
Stimulation of Cl(-) secretion by chlorzoxazone.
Topics: Amiloride; Anions; Bronchi; Bumetanide; Cell Membrane; Cells, Cultured; Charybdotoxin; Chlorine; Chlorzoxazone; Colforsin; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Drug Interactions; Epithelium; Glyburide; Humans; Isoproterenol; Nasal Mucosa; Nystatin; Potassium Channel Blockers; Rubidium; Zoxazolamine | 2000 |
K(ATP) channels mediate the beta(2)-adrenoceptor agonist-induced relaxation of rat detrusor muscle.
Topics: Adenosine Triphosphate; Adrenergic beta-Agonists; Animals; Clenbuterol; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Electric Stimulation; Female; Glyburide; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Pinacidil; Potassium Channels; Rats; Rats, Wistar; Urinary Bladder; Vasodilator Agents | 2000 |
Interaction of cyclic AMP modulating agents with levcromakalim in the relaxation of rat isolated mesenteric artery.
Topics: Adenosine-5'-(N-ethylcarboxamide); Animals; Bucladesine; Colforsin; Cromakalim; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Glyburide; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; Rats; Rats, Wistar; Thionucleotides; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents | 2000 |
Antidiabetic sulfonylurea enhances secretagogue-induced adrenocorticotropin secretion and proopiomelanocortin gene expression in vitro.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenocorticotropic Hormone; Animals; Cell Line; Clone Cells; Colforsin; Diazoxide; Diuretics; Gene Expression; Glyburide; Hypoglycemic Agents; Plasmids; Pro-Opiomelanocortin; Promoter Regions, Genetic; Rats; Reverse Transcriptase Polymerase Chain Reaction; Sodium Chloride Symporter Inhibitors; Stimulation, Chemical; Sulfonylurea Compounds | 2000 |
CFTR regulation of intracellular calcium in normal and cystic fibrosis human airway epithelia.
Topics: Adenosine Triphosphate; Calcium; Cell Line; Cells, Cultured; Colforsin; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Epithelial Cells; Glyburide; Hexokinase; Humans; Intracellular Fluid; Lung; Mutation; Nucleotides; ortho-Aminobenzoates; Receptors, Purinergic; Suramin; Temperature | 2000 |
Inhibition of basolateral cAMP permeability in the toad urinary bladder.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; ATP-Binding Cassette Transporters; Bufo marinus; Calcium Channel Blockers; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Epithelium; Glyburide; In Vitro Techniques; Membrane Fluidity; ortho-Aminobenzoates; Osmosis; Permeability; Pinacidil; Potassium Channels; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Receptors; Urinary Bladder; Vasodilator Agents; Vasopressins; Water | 2000 |
Mechanism of adenosine-induced vasodilation in rat diaphragm microcirculation.
Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Blood Flow Velocity; Colforsin; Diaphragm; Dose-Response Relationship, Drug; Glyburide; Laser-Doppler Flowmetry; Male; Microcirculation; Potassium Channel Blockers; Potassium Channels; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Vasodilation; Vasodilator Agents | 2000 |
Properties of CFTR activated by the xanthine derivative X-33 in human airway Calu-3 cells.
Topics: 1-Methyl-3-isobutylxanthine; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Biological Transport; Caffeine; Calcium Channel Blockers; Chlorides; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Dose-Response Relationship, Drug; Glyburide; Hypoglycemic Agents; In Vitro Techniques; Iodides; Iodine Radioisotopes; Membrane Potentials; Membrane Proteins; ortho-Aminobenzoates; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Phosphorylation; Respiratory Mucosa; Theophylline; Xanthines | 2000 |
Functional and molecular characterization of receptor subtypes mediating coronary microvascular dilation to adenosine.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Animals; Antihypertensive Agents; Blotting, Western; Colforsin; Coronary Vessels; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Enzyme-Linked Immunosorbent Assay; Female; Glyburide; Heart; Hypoglycemic Agents; In Situ Hybridization; Male; Microcirculation; Myocardium; Peptides; Phenethylamines; Potassium Channel Blockers; Purinergic P1 Receptor Antagonists; Receptors, Purinergic P1; Reverse Transcriptase Polymerase Chain Reaction; Stress, Physiological; Swine; Thionucleotides; Tissue Distribution; Triazines; Triazoles | 2001 |
Involvement of K(ATP) channels in diethylstilbestrol-induced relaxation in rat aorta.
Topics: Animals; Aorta; Colforsin; Cyclic AMP; Diazoxide; Diethylstilbestrol; Dose-Response Relationship, Drug; Eflornithine; Glyburide; In Vitro Techniques; Indoles; Male; Muscle, Smooth, Vascular; Norepinephrine; Papaverine; Potassium Channels; Rats; Rats, Wistar; Spermine; Tamoxifen; Tetraethylammonium; Vasoconstriction; Vasodilation; Vasodilator Agents | 2001 |
Functional characterisation of human TASK-3, an acid-sensitive two-pore domain potassium channel.
Topics: 1-Methyl-3-isobutylxanthine; Acids; Animals; Barium Compounds; Bupivacaine; Cell Line; Cesium; Chlorides; Colforsin; Dose-Response Relationship, Drug; Female; Gene Expression; Glyburide; Halothane; Humans; Kinetics; Membrane Potentials; Oocytes; Potassium; Potassium Channels; Potassium Channels, Tandem Pore Domain; Pregnanediones; Tetradecanoylphorbol Acetate; Tetraethylammonium; Time Factors; Xenopus | 2001 |
Gramicidin-perforated patch analysis on HCO3- secretion through a forskolin-activated anion channel in rat parotid intralobular duct cells.
Topics: Amiloride; Animals; Anions; Bicarbonates; Bumetanide; Chlorides; Colforsin; Glyburide; Gramicidin; In Vitro Techniques; Male; Membrane Potentials; Methazolamide; Parotid Gland; Patch-Clamp Techniques; Rats; Rats, Wistar | 2001 |
Nitric oxide decreases pacemaker activity in lymphatic vessels of guinea pig mesentery.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetylcholine; Animals; Biological Clocks; Calcium; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Enzyme Inhibitors; Female; Glyburide; Guinea Pigs; In Vitro Techniques; Lymphatic System; Male; Membrane Potentials; Mesentery; Muscle, Smooth; Nitric Oxide; Nitric Oxide Donors; Vasodilator Agents | 2001 |
Partial restoration of defective chloride conductance in DeltaF508 CF mice by trimethylamine oxide.
Topics: Animals; Apigenin; Chloride Channels; Colforsin; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Dose-Response Relationship, Drug; Electric Conductivity; Electrophysiology; Flavonoids; Glyburide; Methylamines; Mice; Oxidants; Rectum; Reference Values | 2001 |
Activation of a CFTR-mediated chloride current in a rabbit corneal epithelial cell line.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Cell Line; Chlorides; Colforsin; Cornea; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Epithelial Cells; Gene Expression; Genistein; Glyburide; Patch-Clamp Techniques; Phosphodiesterase Inhibitors; Rabbits; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger | 2001 |
Relaxation and modulation of cyclic AMP production in response to atrial natriuretic peptides in guinea pig tracheal smooth muscle.
Topics: Adenylyl Cyclases; Animals; Apamin; Atrial Natriuretic Factor; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Glyburide; Guanylate Cyclase; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Natriuretic Peptide, C-Type; Nitroprusside; Oxadiazoles; Peptide Fragments; Peptides; Phosphodiesterase Inhibitors; Potassium Channel Blockers; Quinoxalines; Rolipram; Trachea | 2001 |
Expression, localization, and functional evaluation of CFTR in bovine corneal endothelial cells.
Topics: Angiogenesis Inhibitors; Animals; Bicarbonates; Cattle; Cell Membrane Permeability; Cell Polarity; Cells, Cultured; Chlorides; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Endothelium, Corneal; Enzyme Inhibitors; Fluoresceins; Fluorescent Antibody Technique, Indirect; Fluorescent Dyes; Genistein; Glyburide; Hydrogen-Ion Concentration; Hypoglycemic Agents; Nitrobenzoates; Quinolinium Compounds | 2002 |
Transepithelial impedance analysis of chloride secretion.
Topics: Angiogenesis Inhibitors; Anti-Arrhythmia Agents; Cell Line; Chlorides; Colforsin; Electric Impedance; Electrophysiology; Epithelial Cells; Glyburide; Humans; Nitrobenzoates; Time Factors | 2002 |
Insulinotropic action of amino acids at their physiological concentrations: I. Experiments in incubated islets.
Topics: Amino Acids; Animals; Calcium; Cells, Cultured; Colforsin; Cytochalasin B; Female; Glucose; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Rats; Rats, Wistar; Theophylline | 2002 |
Pleural surface fluorescence measurement of Na+ and Cl- transport across the air space-capillary barrier.
Topics: Acridines; Animals; Aquaporin 1; Aquaporin 5; Aquaporins; Biological Transport; Blood-Air Barrier; Carrier Proteins; Chlorides; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Fluorescent Dyes; Glyburide; In Vitro Techniques; Membrane Proteins; Mice; Mice, Inbred Strains; Mice, Knockout; Organic Chemicals; Pleura; Sodium | 2003 |
Methoxsalen stimulates electrogenic Cl- secretion in the mouse jejunum.
Topics: Animals; Barium; Bumetanide; Chlorine; Colforsin; Dose-Response Relationship, Drug; Glyburide; In Vitro Techniques; Intestinal Mucosa; Ion Transport; Jejunum; Male; Methoxsalen; Mice; Patch-Clamp Techniques; Potassium Channels; Reference Values; Sensitivity and Specificity | 2002 |
cAMP-induced changes of apical membrane potentials of confluent H441 monolayers.
Topics: Amiloride; Cell Culture Techniques; Cell Line; Cell Membrane; Chlorides; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Epithelial Sodium Channels; Glyburide; Humans; Kinetics; Lung; Membrane Potentials; Patch-Clamp Techniques; Respiratory Mucosa; Sodium Channels | 2003 |
Adenosine receptors and phosphodiesterase inhibitors stimulate Cl- secretion in Calu-3 cells.
Topics: Adenosine Deaminase; Anions; Cell Line; Chlorine; Cilostazol; Colforsin; Cyclic AMP; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Electrophysiology; Epithelium; Glyburide; Humans; Hypoglycemic Agents; Milrinone; Mutation; Papaverine; Phosphodiesterase Inhibitors; Piperazines; Purines; Receptors, Purinergic P1; Rolipram; Sildenafil Citrate; Sulfones; Tetrazoles; Time Factors | 2003 |
Altered excitability of intestinal neurons in primary culture caused by acute oxidative stress.
Topics: Action Potentials; Animals; Caffeine; Calcium; Cell Culture Techniques; Central Nervous System Stimulants; Clotrimazole; Colforsin; Duodenum; Enzyme Activators; Female; Glyburide; Guinea Pigs; Hydrogen Peroxide; Male; Membrane Potentials; Neurons; Oxidative Stress; Patch-Clamp Techniques; Potassium Channel Blockers; Potassium Channels; Tetraethylammonium | 2003 |
CFTR in K562 human leukemic cells.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Antibodies; Cell Membrane; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Glyburide; Hematopoietic Stem Cells; Homeostasis; Humans; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Membrane Potentials; RNA, Messenger; Tumor Cells, Cultured | 2003 |
ATP release triggered by activation of the Ca2+-activated K+ channel in human airway Calu-3 cells.
Topics: Adenosine Diphosphate; Adenosine Triphosphate; Benzimidazoles; Bumetanide; Calcium; Cell Size; Charybdotoxin; Chlorzoxazone; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Cytosol; Epithelial Cells; Glyburide; Humans; Ionomycin; Isoproterenol; Luciferases; Lung; Potassium Channels, Calcium-Activated; Potassium Chloride; Purinergic P2 Receptor Antagonists; Receptors, Purinergic P2Y1 | 2004 |
Molecular identity and function in transepithelial transport of K(ATP) channels in alveolar epithelial cells.
Topics: Amiloride; Animals; ATP-Binding Cassette Transporters; Base Sequence; Colforsin; DNA; DNA Primers; Glyburide; Kinetics; Male; Pinacidil; Potassium Channels; Potassium Channels, Inwardly Rectifying; Pulmonary Alveoli; Rats; Rats, Sprague-Dawley; Receptors, Drug; Respiratory Mucosa; Reverse Transcriptase Polymerase Chain Reaction; Sulfonylurea Receptors | 2004 |
Activation of VPAC1 receptors by VIP and PACAP-27 in human bronchial epithelial cells induces CFTR-dependent chloride secretion.
Topics: Bronchi; Cell Line; Chlorides; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Epithelial Cells; Glyburide; Humans; Hypoglycemic Agents; Iodides; Neuropeptides; Pituitary Adenylate Cyclase-Activating Polypeptide; Receptors, Pituitary Adenylate Cyclase-Activating Polypeptide; Receptors, Pituitary Hormone; Receptors, Vasoactive Intestinal Peptide; Receptors, Vasoactive Intestinal Polypeptide, Type I; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Vasoactive Intestinal Peptide | 2004 |
Changes in the vascular beta-adrenoceptor-activated signalling pathway in 2Kidney-1Clip hypertensive rats.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Aorta, Thoracic; Caffeine; Calcium-Transporting ATPases; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Gene Expression; Glyburide; Hypertension, Renovascular; Isoproterenol; Kidney; Male; Membrane Proteins; Muscle, Smooth, Vascular; Phenylephrine; Potassium Channels; Rats; Rats, Wistar; Receptors, Adrenergic, beta; RNA, Messenger; Sarcolemma; Signal Transduction; Thapsigargin; Vasoconstriction; Vasodilation | 2004 |
Regulation of apical surface fluid and protein secretion in human airway epithelial cell line Calu-3.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Anti-Arrhythmia Agents; Body Fluids; Cell Line; Cell Polarity; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Dinoprost; Epithelial Cells; Glyburide; Humans; Muramidase; Oxytocics; Respiratory Mucosa; Stilbenes; Tetradecanoylphorbol Acetate | 2004 |
Regulation of antiprotease and antimicrobial protein secretion by airway submucosal gland serous cells.
Topics: alpha 1-Antichymotrypsin; alpha 1-Antitrypsin; Amino Acid Sequence; Animals; Anti-Inflammatory Agents; Cell Division; Cell Line; Chromatography, High Pressure Liquid; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Electrophoresis, Polyacrylamide Gel; Enzyme-Linked Immunosorbent Assay; Epithelial Cells; Glyburide; Humans; Mass Spectrometry; Molecular Sequence Data; Muramidase; Potassium Channels; Protease Inhibitors; Respiratory Mucosa; Reverse Transcriptase Polymerase Chain Reaction; Sequence Homology, Amino Acid; Serine Endopeptidases; Sodium; Spectrometry, Mass, Electrospray Ionization; Swine; Time Factors | 2004 |
CFTR involvement in nasal potential differences in mice and pigs studied using a thiazolidinone CFTR inhibitor.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amiloride; Animals; Benzoates; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Diuretics; Female; Glyburide; Hypoglycemic Agents; Male; Membrane Potentials; Mice; Mice, Inbred CFTR; Nasal Mucosa; Sus scrofa; Thiazoles; Thiazolidines | 2004 |
Chloride channels in the small intestinal cell line IEC-18.
Topics: Animals; Calcium Signaling; Cell Line; Chloride Channels; Chlorides; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Cytosol; Epithelial Cells; Extracellular Fluid; Fluorescent Antibody Technique; Fura-2; Glyburide; Intestine, Small; Ionomycin; Membrane Potentials; Nitrobenzoates; Osmolar Concentration; Patch-Clamp Techniques; Radioisotopes; Rats | 2005 |
Prostaglandin E2--mediated relaxation of the ductus arteriosus: effects of gestational age on g protein-coupled receptor expression, signaling, and vasomotor control.
Topics: 16,16-Dimethylprostaglandin E2; 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenylyl Cyclases; Alprostadil; Animals; Biphenyl Compounds; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dinoprostone; Ductus Arteriosus; Enzyme Activation; Female; Gestational Age; Glyburide; Indomethacin; Isometric Contraction; NG-Nitroarginine Methyl Ester; Nitroprusside; Papio; Potassium Channels; Pregnancy; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP2 Subtype; Receptors, Prostaglandin E, EP3 Subtype; Receptors, Prostaglandin E, EP4 Subtype; Sheep; Signal Transduction; Sodium Fluoride; Thionucleotides; Vasomotor System | 2004 |
The relationship between cell proliferation, Cl- secretion, and renal cyst growth: a study using CFTR inhibitors.
Topics: Animals; Benzoates; Cell Division; Cell Line; Chloride Channels; Chlorides; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Dogs; Electric Conductivity; Epithelium; Genistein; Glyburide; Ion Transport; Kidney Diseases, Cystic; Nitrobenzoates; Thiazoles; Thiazolidines | 2004 |
Isoproterenol opens K+(ATP) channels via a beta2-adrenoceptor-linked mechanism in Sertoli cells from immature rats.
Topics: Adrenergic beta-Agonists; Animals; ATP-Binding Cassette Transporters; Colforsin; Dose-Response Relationship, Drug; Electrophysiology; Glyburide; Hypoglycemic Agents; Ion Channel Gating; Isoproterenol; KATP Channels; Lanthanum; Male; Membrane Potentials; Patch-Clamp Techniques; Potassium Channels, Inwardly Rectifying; Rats; Rats, Wistar; Receptors, Adrenergic, beta-2; Sertoli Cells; Testosterone | 2005 |
Disruption of CFTR chloride channel alters mechanical properties and cAMP-dependent Cl- transport of mouse aortic smooth muscle cells.
Topics: Adrenergic beta-Agonists; Angiotensin II; Animals; Aorta, Thoracic; Benzoates; Cells, Cultured; Chlorides; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Genistein; Glyburide; In Vitro Techniques; Isoproterenol; Mice; Mice, Inbred CFTR; Muscle, Smooth, Vascular; ortho-Aminobenzoates; Quinolizines; Serotonin; Thiazoles; Thiazolidines; Vasoactive Intestinal Peptide; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents | 2005 |
Resveratrol inhibits insulin secretion from rat pancreatic islets.
Topics: Animals; Colforsin; Dose-Response Relationship, Drug; Glucose; Glutamine; Glyburide; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Leucine; Male; Phytoalexins; Rats; Rats, Wistar; Resveratrol; Sesquiterpenes; Stilbenes; Terpenes; Tetradecanoylphorbol Acetate; Time Factors | 2006 |
Acute inflammation alters bicarbonate transport in mouse ileum.
Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acute Disease; Adenylyl Cyclases; Animals; Antibodies, Monoclonal; Bicarbonates; CD3 Complex; Chloride-Bicarbonate Antiporters; Chlorides; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Diarrhea; Disease Models, Animal; Electric Conductivity; Enzyme Activation; Enzyme Activators; Glyburide; Ileum; Inflammatory Bowel Diseases; Intestinal Secretions; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Nitrobenzoates | 2007 |
Expression and function of cystic fibrosis transmembrane conductance regulator in rat intrapulmonary arteries.
Topics: Analysis of Variance; Animals; Cells, Cultured; Chloride Channels; Colforsin; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Genistein; Glyburide; Immunoprecipitation; Iodides; Male; Muscle, Smooth, Vascular; Phosphorylation; Pulmonary Artery; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; Vasodilation | 2007 |
Appearance of segmental discrepancy of anion transport in rat distal colon.
Topics: Adenylyl Cyclases; Animals; Anions; Biological Transport, Active; Colforsin; Colon; Cyclic AMP; Cystic Fibrosis Transmembrane Conductance Regulator; Enzyme Activators; Gene Expression; Glyburide; Male; Rats; Rats, Sprague-Dawley; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Sodium-Potassium-Chloride Symporters; Solute Carrier Family 12, Member 2 | 2007 |
Cystic fibrosis transmembrane conductance regulator trafficking is mediated by the COPI coat in epithelial cells.
Topics: Adenocarcinoma; Cell Line, Tumor; Cell Membrane; Coat Protein Complex I; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Endoplasmic Reticulum; Epithelial Cells; Gene Expression Regulation, Neoplastic; Glyburide; Golgi Apparatus; Humans; Recombinant Proteins; RNA, Neoplasm; RNA, Small Interfering | 2008 |
Effects of prostaglandin E1 on vascular ATP-sensitive potassium channels.
Topics: Algorithms; Alprostadil; Analysis of Variance; Animals; Aorta, Thoracic; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Glyburide; In Vitro Techniques; KATP Channels; Male; Patch-Clamp Techniques; Phenylephrine; Pinacidil; Protein Kinase Inhibitors; Rats; Rats, Wistar; Thionucleotides; Vasoconstriction; Vasodilation; Vasodilator Agents | 2007 |
Inhibitory effect of caffeine on pacemaker activity in the oviduct is mediated by cAMP-regulated conductances.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; ATP-Binding Cassette Transporters; Biological Clocks; Caffeine; Colforsin; Cyclic AMP; Drug Interactions; Female; Glyburide; KATP Channels; Membrane Potentials; Mice; Mice, Inbred BALB C; Muscle Contraction; Muscle, Smooth; Oviducts; Phosphodiesterase Inhibitors; Pinacidil; Potassium Channels, Inwardly Rectifying; Receptors, Drug; Sulfonylurea Receptors | 2011 |
Stimulation of murine intestinal secretion by daily genistein injections: gender-dependent differences.
Topics: Animals; Anticarcinogenic Agents; Chlorides; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Female; Genistein; Glyburide; Intestine, Small; Male; Mice; Mice, Inbred C57BL; Sex Factors | 2011 |
cAMP/protein kinase A activates cystic fibrosis transmembrane conductance regulator for ATP release from rat skeletal muscle during low pH or contractions.
Topics: 1-Methyl-3-isobutylxanthine; Adenosine Triphosphate; Animals; Benzoates; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cystic Fibrosis Transmembrane Conductance Regulator; Glyburide; Hydrogen-Ion Concentration; Lactic Acid; Male; Muscle Contraction; Muscle, Skeletal; Myoblasts; Rats; Rats, Sprague-Dawley; Signal Transduction; Sodium-Calcium Exchanger; Sodium-Hydrogen Exchangers; Thiazolidines | 2012 |
Activation of chloride secretion by isoflavone genistein in endometrial epithelial cells.
Topics: 1-Methyl-3-isobutylxanthine; Amiloride; Animals; Bumetanide; Cell Membrane Permeability; Cells, Cultured; Chlorides; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Egtazic Acid; Endometrium; Epithelial Cells; Estradiol; Female; Fulvestrant; Genistein; Glyburide; Swine; Uridine Triphosphate | 2013 |
Physiological characterization of the human EndoC-βH1 β-cell line.
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adenosine Diphosphate; Adenosine Triphosphate; Biological Transport; Calcium Channels; Cell Line; Colforsin; Founder Effect; Gene Expression; Glucokinase; Glucose; Glucose Transporter Type 1; Glucose Transporter Type 2; Glutamine; Glyburide; Humans; Insulin; Insulin-Secreting Cells; Keto Acids; Leucine; Mannoheptulose; Phosphorylation; Potassium Channels, Inwardly Rectifying | 2015 |
Dynamics of Insulin Secretion from EndoC-
Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Cell Line; Colforsin; Exocytosis; Glucose; Glyburide; Humans; Insulin; Insulin Secretion; Insulin-Secreting Cells; Mannoheptulose; Signal Transduction | 2017 |