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colforsin and gamma-aminobutyric acid

colforsin has been researched along with gamma-aminobutyric acid in 82 studies

Research

Studies (82)

TimeframeStudies, this research(%)All Research%
pre-19909 (10.98)18.7374
1990's31 (37.80)18.2507
2000's28 (34.15)29.6817
2010's13 (15.85)24.3611
2020's1 (1.22)2.80

Authors

AuthorsStudies
Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Eisenberg, HM; Hulsebosch, CE; Lu, Y; Morgan, B; Perez-Polo, JR; Pizzo, DP; Werrbach-Perez, K; Westlund, KN1
Blackstone, CD; Huganir, RL; Moss, SJ; Smart, TG1
Ishac, E; Li, C; White, G1
Hansson, E; Rönnbäck, L1
Abucham, J; Reichlin, S1
Wickelgren, WO; Womble, MD1
Mehta, AK; Ticku, MK1
Leonard, JP; Wickelgren, WO1
Heuschneider, G; Schwartz, RD1
Eimerl, S; Minc-Golomb, D; Schramm, M1
Barnes, EM; Hablitz, JJ; Tehrani, MH1
Starr, BS; Starr, MS1
Hill, DR1
Weiss, S1
Dowling, JE; O'Brien, DR1
Finger, W; Martin, C1
Cao, Z; Hosford, DA; Lin, FH; Lin, S; Wang, Y1
Amico, C; Cupello, A; Robello, M1
Desrues, L; Lamacz, M; Tonon, MC; Vaudry, H1
Cherubini, E; Sciancalepore, M1
Kirifides, ML; Lin, RC; Liu, W; Mouradian, RD; Sessler, FM; Waterhouse, BD1
Fisone, G; Greengard, P; Snyder, GL1
Bannon, MJ; Granneman, JG; Kapatos, G; Tian, Y1
Katsuki, H; Kawahara, F; Saito, H1
Giménez, C; Gomeza, J; Zafra, F1
Bowery, NG; Malcangio, M1
Gerschenfeld, HM; Llano, I1
Adam-Vizi, V; Baranyi, M; Chernaeva, L; Déri, Z; Vizi, ES; Zelles, T1
Cherubini, E; Sciancalepore, M; Strata, F1
Bonci, A; Williams, JT1
Li, A; Wang, HL; Wu, T1
Bickford, PC; Gould, TJ1
Obrietan, K; van den Pol, AN1
Corsi, L; De Blas, AL; Ghose, S; Grayson, DR; Neale, JH; Vicini, S; Wroblewska, B1
Barni, S; Castoldi, AF; Costa, LG; Manzo, L; Randine, G1
Bagley, EE; Christie, MJ; Vaughan, CW1
Konishi, S; Mitoma, H1
Estevez, AY; O'Regan, MH; Phillis, JW; Song, D1
Arias-Montaño, JA; Bahena-Trujillo, R1
Aghajanian, GK; Jolas, T; Nestler, EJ1
Konishi, S; Saitow, F; Satake, S; Yamada, J2
Franco, R; Pasantes-Morales, H; Quesada, O1
Li, P; Yang, XL1
Beltrán-Parrazal, L; Clapp, C; Martínez de la Escalera, G; Noris, G1
Maneuf, YP; McKnight, AT1
Fuentes, T; Galindo, A; García Estañ, J; Hernández, J; Vargas, ML1
Duffy, SN; Nguyen, PV1
Gómez-Villafuertes, R; Gualix, J; Miras-Portugal, MT; Pintor, J1
Deadwyler, SA; Hampson, RE; Weiner, JL; Zhuang, SY1
Mascia, FM; Olianas, MC; Onali, P1
Christie, MJ; Hack, SP; Vaughan, CW1
Bali, B; Kovács, KJ1
González-Maeso, J; Green, A; Koenig, JA; Wise, A1
Hinkle, DJ; Macdonald, RL1
Konishi, S; Rusakov, D; Saitow, F; Satake, S1
Fujita, T; Kumamoto, E; Yang, K1
Harvey, VL; Stephens, GJ1
Eliasson, L; Galvanovskis, J; MacDonald, PE; Obermüller, S; Rorsman, P; Vikman, J1
Hablitz, JJ; Wu, J1
de Novellis, V; Maione, S; Marabese, I; Mariani, L; Palazzo, E; Rodella, L; Rossi, F; Siniscalco, D1
Glitsch, M1
Aceves, J; Erlij, D; Florán, B; Florán, L; Gonzalez, B; Paz, F1
Ling, Z; Mao, R; Pipeleers, D; Van de Casteele, M; Wang, C1
Cho, YW; Hahm, ET; Lee, CH; Lee, JJ1
Ishida, K; Mitoma, H; Mizusawa, H1
Ballabio, M; Bonanno, G; Frasca, A; Fumagalli, F; Magnaghi, V; Parducz, A; Procacci, P; Racagni, G1
Chen, ZN; Li, CY; Shi, HB; Song, NY; Ye, HB; Yin, SK1
Carloni, P; Cherubini, E; Giorgetti, A; Griguoli, M; Maul, A; Nguyen, C1
Simeone, TA; White, HS; Wilcox, KS1
Di Prisco, S; Grilli, M; Marchi, M; Pittaluga, A; Summa, M; Usai, C1
Adan, RA; Meye, FJ; Ramakers, GM; Smidt, MP; van Zessen, R1
Cho, Y; Han, D; Heo, H; Joung, I; Kwon, YK; Yoo, M1
Ganguly, A; Lee, D1
Berretta, N; Bonito-Oliva, A; Castelli, V; Fisone, G; Giorgi, M; Ledonne, A; Mango, D; Mercuri, NB; Nisticò, R; Sancesario, G1
Bobeck, EN; Chen, Q; Ingram, SL; Morgan, MM1
Blake, CB; Smith, BN1
Danielsson, J; Emala, CW; Funayama, H; Gallos, G; Kim, B; Worgall, TS; Xu, D; Yim, PD; Zaidi, S1
Dai, S; Guo, Z; He, X; Hu, Z; Jiao, Z; Lu, M; Wang, H; Xu, D1

Reviews

1 review(s) available for colforsin and gamma-aminobutyric acid

ArticleYear
The role of receptor binding in drug discovery.
    Journal of natural products, 1993, Volume: 56, Issue:4

    Topics: Animals; Drug Design; Humans; Receptors, Drug

1993

Other Studies

81 other study(ies) available for colforsin and gamma-aminobutyric acid

ArticleYear
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
Effects of nerve growth factor and acetyl-L-carnitine arginyl amide on the human neuronal line HCN-1A.
    International journal of developmental neuroscience : the official journal of the International Society for Developmental Neuroscience, 1992, Volume: 10, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Acetylcarnitine; Animals; Arginine; Brain Chemistry; Cell Differentiation; Cell Line; Colforsin; gamma-Aminobutyric Acid; Humans; Immunohistochemistry; Mice; Nerve Growth Factors; Neurofilament Proteins; Neurons

1992
Functional modulation of GABAA receptors by cAMP-dependent protein phosphorylation.
    Science (New York, N.Y.), 1992, Jul-31, Volume: 257, Issue:5070

    Topics: Animals; Cell Line; Cells, Cultured; Colforsin; Cyclic AMP; Electric Conductivity; gamma-Aminobutyric Acid; Immunosorbent Techniques; Kinetics; Mice; Mutagenesis, Site-Directed; Neurons; Peptide Mapping; Phosphorylation; Protein Kinases; Rats; Receptors, GABA-A; Recombinant Proteins; Transfection; Zinc

1992
1,9-Dideoxyforskolin does not mimic all cAMP and protein kinase A independent effects of forskolin on GABA activated ion currents in adult rat sensory neurons.
    Brain research, 1992, Jul-17, Volume: 586, Issue:1

    Topics: Animals; Colforsin; Cyclic AMP; Electric Conductivity; gamma-Aminobutyric Acid; Ion Channels; Neurons, Afferent; Protein Kinases; Rats; Rats, Inbred Strains

1992
Receptor regulation of the glutamate, GABA and taurine high-affinity uptake into astrocytes in primary culture.
    Brain research, 1991, May-10, Volume: 548, Issue:1-2

    Topics: Animals; Animals, Newborn; Aspartic Acid; Astrocytes; Biological Transport; Cells, Cultured; Cerebral Cortex; Cholera Toxin; Colforsin; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Isoproterenol; Kinetics; Phenylephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin; Taurine; Virulence Factors, Bordetella

1991
Regulation of cholecystokinin octapeptide secretion by rat cerebral cortical cells in primary culture.
    Endocrinology, 1991, Volume: 129, Issue:6

    Topics: Animals; Calcium; Cells, Cultured; Cerebral Cortex; Colforsin; Embryo, Mammalian; GABA Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Neurotransmitter Agents; Potassium; Rats; Sincalide; Tetrodotoxin; Verapamil; Veratridine

1991
Inhibition of a cAMP-dependent Ca-activated K conductance by forskolin prolongs Ca action potential duration in lamprey sensory neurons.
    Brain research, 1990, Jun-04, Volume: 518, Issue:1-2

    Topics: Action Potentials; Animals; Calcium Chloride; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; In Vitro Techniques; Lampreys; Neurons, Afferent; Potassium; Potassium Channels; Spinal Cord; Tetrodotoxin

1990
gamma-Aminobutyric acidA receptor desensitization in mice spinal cord cultured neurons: lack of involvement of protein kinases A and C.
    Molecular pharmacology, 1990, Volume: 38, Issue:5

    Topics: Animals; Cells, Cultured; Chloride Channels; Colforsin; Female; gamma-Aminobutyric Acid; Male; Membrane Proteins; Mice; Mice, Inbred C57BL; Neurons; Protein Kinase C; Protein Kinase Inhibitors; Protein Kinases; Receptors, GABA-A; Spinal Cord

1990
Prolongation of calcium action potentials by gamma-aminobutyric acid in primary sensory neurones of lamprey.
    The Journal of physiology, 1986, Volume: 375

    Topics: Action Potentials; Animals; Calcium; Colforsin; Fishes; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Channels; Lampreys; Neurons, Afferent; Tetrodotoxin; Time Factors

1986
cAMP and forskolin decrease gamma-aminobutyric acid-gated chloride flux in rat brain synaptoneurosomes.
    Proceedings of the National Academy of Sciences of the United States of America, 1989, Volume: 86, Issue:8

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Brain; Bucladesine; Chloride Channels; Chlorides; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Proteins; Muscimol; Rats; Synaptosomes

1989
Cysteine sulfinic acid-induced release of D-[3H]aspartate and [14C]GABA in hippocampus slices: the role of sodium channels and cAMP.
    Brain research, 1989, Jun-26, Volume: 490, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Amino Acids; Animals; Aspartic Acid; Calcium; Cnidarian Venoms; Colforsin; Cysteine; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Neurotoxins; Neurotransmitter Agents; Rats; Sodium Channels; Tetrodotoxin

1989
cAMP increases the rate of GABAA receptor desensitization in chick cortical neurons.
    Synapse (New York, N.Y.), 1989, Volume: 4, Issue:2

    Topics: Animals; Cells, Cultured; Cerebral Cortex; Chick Embryo; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; Receptors, GABA-A

1989
Circling evoked by intranigral SKF 38393: a GABA-mediated D-1 response?
    Pharmacology, biochemistry, and behavior, 1989, Volume: 32, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Colforsin; Dopamine Agents; Dose-Response Relationship, Drug; Drug Synergism; gamma-Aminobutyric Acid; Male; Motor Activity; Nipecotic Acids; Pentobarbital; Rats; Rats, Inbred Strains; Substantia Nigra

1989
GABAB receptor modulation of adenylate cyclase activity in rat brain slices.
    British journal of pharmacology, 1985, Volume: 84, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Baclofen; Brain; Cerebral Cortex; Colforsin; Cyclic AMP; Diterpenes; gamma-Aminobutyric Acid; In Vitro Techniques; Nipecotic Acids; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Forskolin attenuates the evoked release of [3H]GABA from striatal neurons in primary culture.
    Brain research, 1988, Oct-25, Volume: 463, Issue:1

    Topics: Animals; Bucladesine; Cells, Cultured; Colforsin; Corpus Striatum; Cyclic AMP; gamma-Aminobutyric Acid; Mice; Thionucleotides

1988
Dopaminergic regulation of GABA release from the intact goldfish retina.
    Brain research, 1985, Dec-23, Volume: 360, Issue:1-2

    Topics: Animals; Calcium; Colforsin; Cyclic AMP; Cyprinidae; Dopamine; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Goldfish; In Vitro Techniques; Retina; Synaptic Transmission

1985
Presynaptic effect of gamma-aminobutyric acid on the inhibitory nerve and nerve terminals in the crayfish neuromuscular junction.
    Neuroscience letters, 1989, Feb-13, Volume: 97, Issue:1-2

    Topics: Action Potentials; Animals; Astacoidea; Colforsin; gamma-Aminobutyric Acid; In Vitro Techniques; Neural Inhibition; Neuromuscular Junction; Peripheral Nerves; Serotonin

1989
GABAB receptor-mediated effects in synaptosomes of lethargic (lh/lh) mice.
    Journal of neurochemistry, 1995, Volume: 65, Issue:5

    Topics: Animals; Calcium; Cerebral Cortex; Colforsin; Cyclic AMP; Epilepsy; Epilepsy, Absence; gamma-Aminobutyric Acid; Hybridization, Genetic; Male; Mice; Mice, Inbred Strains; Potassium Chloride; Receptors, GABA-B; Synaptosomes; Thalamus

1995
Regulation of GABAA receptor in cerebellar granule cells in culture: differential involvement of kinase activities.
    Neuroscience, 1993, Volume: 53, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Cells, Cultured; Cerebellum; Chloride Channels; Colforsin; Cyclic AMP; Cytoplasmic Granules; Electrophysiology; gamma-Aminobutyric Acid; Kinetics; Membrane Potentials; Membrane Proteins; Phosphorylation; Phosphotransferases; Picrotoxin; Protein Kinase Inhibitors; Protein Kinases; Rats; Rats, Wistar; Receptors, GABA-A

1993
Mechanism of action of gamma-aminobutyric acid on frog melanotrophs.
    Journal of molecular endocrinology, 1995, Volume: 14, Issue:1

    Topics: Adenylyl Cyclases; Animals; Baclofen; Calcium; Calcium Channels; Colforsin; Cyclic AMP; GABA-A Receptor Agonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Inositol Phosphates; Male; Melanocyte-Stimulating Hormones; Models, Biological; Pituitary Gland, Posterior; Rana ridibunda; Receptors, GABA-A; Receptors, GABA-B; Signal Transduction; Taurine

1995
Protein kinase A-dependent increase in frequency of miniature GABAergic currents in rat CA3 hippocampal neurons.
    Neuroscience letters, 1995, Mar-03, Volume: 187, Issue:2

    Topics: Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electric Conductivity; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Kynurenic Acid; Neurons; Patch-Clamp Techniques; Protein Kinase Inhibitors; Rats; Rats, Wistar; Tetrodotoxin; Thionucleotides

1995
Noradrenergic enhancement of GABA-induced input resistance changes in layer V regular spiking pyramidal neurons of rat somatosensory cortex.
    Brain research, 1995, Mar-27, Volume: 675, Issue:1-2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Colforsin; Electrophysiology; gamma-Aminobutyric Acid; In Vitro Techniques; Isoproterenol; Membrane Potentials; Microelectrodes; Muscimol; Norepinephrine; Pyramidal Cells; Rats; Somatosensory Cortex

1995
Phosphorylation of DARPP-32 is regulated by GABA in rat striatum and substantia nigra.
    Journal of neurochemistry, 1994, Volume: 63, Issue:5

    Topics: Animals; Baclofen; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine and cAMP-Regulated Phosphoprotein 32; GABA Antagonists; gamma-Aminobutyric Acid; Male; Nerve Tissue Proteins; Phosphoproteins; Phosphorylation; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, GABA; Substantia Nigra

1994
Dopamine and gamma-aminobutyric acid transporters: differential regulation by agents that promote phosphorylation.
    Neuroscience letters, 1994, May-23, Volume: 173, Issue:1-2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Carrier Proteins; Colforsin; Dopamine; Dopamine Plasma Membrane Transport Proteins; Ethers, Cyclic; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Glycoproteins; Membrane Proteins; Membrane Transport Proteins; Neostriatum; Nerve Tissue Proteins; Okadaic Acid; Organic Anion Transporters; Phorbol Esters; Phosphoprotein Phosphatases; Phosphorylation; Rats; Rats, Sprague-Dawley; Signal Transduction; Synaptosomes

1994
Inhibition by 5-HT7 receptor stimulation of GABAA receptor-activated current in cultured rat suprachiasmatic neurones.
    The Journal of physiology, 1994, Jul-01, Volume: 478 ( Pt 1)

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cell Membrane; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Membrane Potentials; Neurons; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Serotonin; Ritanserin; Serotonin; Suprachiasmatic Nucleus

1994
Cellular distribution and regulation by cAMP of the GABA transporter (GAT-1) mRNA.
    Brain research. Molecular brain research, 1994, Volume: 21, Issue:1-2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Astrocytes; Base Sequence; Bucladesine; Carrier Proteins; Cells, Cultured; Cerebral Cortex; Cloning, Molecular; Colforsin; Cyclic AMP; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Gene Expression Regulation; Glial Fibrillary Acidic Protein; Immunohistochemistry; Kinetics; Membrane Proteins; Membrane Transport Proteins; Molecular Sequence Data; Neuroglia; Oligodeoxyribonucleotides; Organic Anion Transporters; Rats; Rats, Wistar; RNA, Messenger; Tetradecanoylphorbol Acetate; Time Factors

1994
GABAB receptor-mediated inhibition of forskolin-stimulated cyclic AMP accumulation in rat spinal cord.
    Neuroscience letters, 1993, Aug-20, Volume: 158, Issue:2

    Topics: Analgesics; Animals; Animals, Newborn; Baclofen; Capsaicin; Colforsin; Cyclic AMP; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Norepinephrine; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Cord

1993
Beta-adrenergic enhancement of inhibitory synaptic activity in rat cerebellar stellate and Purkinje cells.
    The Journal of physiology, 1993, Volume: 468

    Topics: Action Potentials; Animals; Cerebellum; Colforsin; gamma-Aminobutyric Acid; In Vitro Techniques; Isoproterenol; Kinetics; Norepinephrine; Purkinje Cells; Rats; Receptors, Adrenergic, beta; Synapses; Tetrodotoxin

1993
Transmitter release by non-receptor activation of the alpha-subunit of guanine nucleotide regulatory protein in rat striatal slices.
    Journal of neuroscience research, 1995, Oct-01, Volume: 42, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Acetylcholine; Adrenergic Uptake Inhibitors; Aluminum Chloride; Aluminum Compounds; Animals; Calcium; Chlorides; Colforsin; Corpus Striatum; Dopamine; Dopamine Uptake Inhibitors; Drug Synergism; Egtazic Acid; Enzyme Inhibitors; Ethylmaleimide; gamma-Aminobutyric Acid; GTP-Binding Proteins; Male; Monoamine Oxidase Inhibitors; Neomycin; Nomifensine; Pargyline; Phosphatidylinositol Diacylglycerol-Lyase; Phosphoric Diester Hydrolases; Rats; Rats, Wistar; Reserpine; Ruthenium Red; Signal Transduction; Sodium Fluoride; Stimulation, Chemical; Synaptosomes; Type C Phospholipases

1995
Cyclic AMP-dependent modulation of giant depolarizing potentials by metabotropic glutamate receptors in the rat hippocampus.
    The Journal of physiology, 1995, Nov-15, Volume: 489 ( Pt 1)

    Topics: Animals; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; Hippocampus; Kynurenic Acid; Membrane Potentials; Quisqualic Acid; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate

1995
Increased probability of GABA release during withdrawal from morphine.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Jan-15, Volume: 17, Issue:2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dopamine; Dopamine Antagonists; Enzyme Activation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Interneurons; Morphine; Nerve Tissue Proteins; Organophosphorus Compounds; Patch-Clamp Techniques; Phorbol 12,13-Dibutyrate; Picrotoxin; Receptors, GABA-A; Salicylamides; Serotonin; Signal Transduction; Staurosporine; Strychnine; Substance Withdrawal Syndrome; Tegmentum Mesencephali; Thionucleotides

1997
Vasoactive intestinal polypeptide enhances the GABAergic synaptic transmission in cultured hippocampal neurons.
    Brain research, 1997, Jan-23, Volume: 746, Issue:1-2

    Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Cadmium Chloride; Calcium Channel Blockers; Carcinogens; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hippocampus; Neurons; Patch-Clamp Techniques; Rats; Synaptic Transmission; Tetrodotoxin; Vasoactive Intestinal Peptide

1997
Age-related deficits in the cerebellar beta adrenergic signal transduction cascade in Fischer 344 rats.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:2

    Topics: Aging; Animals; Cerebellum; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta; Signal Transduction

1997
GABA activity mediating cytosolic Ca2+ rises in developing neurons is modulated by cAMP-dependent signal transduction.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1997, Jun-15, Volume: 17, Issue:12

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenine; Adenylyl Cyclase Inhibitors; Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cytosol; Electric Stimulation; Embryo, Mammalian; Enzyme Inhibitors; gamma-Aminobutyric Acid; Hypothalamus, Middle; Isoquinolines; Neurons; Rats; Rats, Sprague-Dawley; Signal Transduction; Sulfonamides; Synapses; Tetrodotoxin; Thionucleotides

1997
N-acetylaspartylglutamate stimulates metabotropic glutamate receptor 3 to regulate expression of the GABA(A) alpha6 subunit in cerebellar granule cells.
    Journal of neurochemistry, 1997, Volume: 69, Issue:6

    Topics: Animals; Cells, Cultured; Cerebellum; Colforsin; Cyclic AMP; Dipeptides; Electric Conductivity; Furosemide; gamma-Aminobutyric Acid; Ion Channel Gating; Neurons; Polymerase Chain Reaction; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Metabotropic Glutamate; RNA, Messenger; Transcription, Genetic

1997
Ethanol selectively interferes with the trophic action of NMDA and carbachol on cultured cerebellar granule neurons undergoing apoptosis.
    Brain research. Developmental brain research, 1998, Dec-07, Volume: 111, Issue:2

    Topics: Animals; Apoptosis; Carbachol; Cell Survival; Cells, Cultured; Central Nervous System Depressants; Cerebellum; Colforsin; Drug Interactions; Ethanol; Excitatory Amino Acid Agonists; gamma-Aminobutyric Acid; Microscopy, Electron; Muscarinic Agonists; N-Methylaspartate; Neurons; Potassium; Rats; Rats, Sprague-Dawley

1998
Inhibition by adenosine receptor agonists of synaptic transmission in rat periaqueductal grey neurons.
    The Journal of physiology, 1999, Apr-01, Volume: 516 ( Pt 1)

    Topics: Action Potentials; Adenosine; Animals; Colforsin; gamma-Aminobutyric Acid; Glutamic Acid; In Vitro Techniques; Membrane Potentials; Neurons; Patch-Clamp Techniques; Periaqueductal Gray; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Synaptic Transmission

1999
Monoaminergic long-term facilitation of GABA-mediated inhibitory transmission at cerebellar synapses.
    Neuroscience, 1999, Volume: 88, Issue:3

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Cerebellum; Colforsin; Cyclic AMP; Electric Stimulation; Enzyme Inhibitors; Evoked Potentials; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Isoquinolines; Long-Term Potentiation; Methiothepin; Neuronal Plasticity; Norepinephrine; Propranolol; Protein Kinase Inhibitors; Purkinje Cells; Rats; Rats, Wistar; Receptors, GABA; Serotonin; Sulfonamides; Synapses; Synaptic Transmission; Tetrodotoxin; Thionucleotides

1999
Hyposmotically induced amino acid release from the rat cerebral cortex: role of phospholipases and protein kinases.
    Brain research, 1999, Oct-09, Volume: 844, Issue:1-2

    Topics: Acetophenones; Alanine; Amino Acids; Animals; Arachidonic Acids; Aspartic Acid; Brain Edema; Cerebral Cortex; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dimethyl Sulfoxide; Enzyme Inhibitors; Estrenes; Ethanolamines; Fatty Acids, Unsaturated; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Hypotonic Solutions; Male; Osmotic Pressure; Phosphodiesterase Inhibitors; Phospholipases A; Phospholipases A2; Protein Kinase C; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Serine; Solvents; Taurine; Water-Electrolyte Balance

1999
[3H] gamma-aminobutyric acid transport in rat substantia nigra pars reticulata synaptosomes: pharmacological characterization and phorbol ester-induced inhibition.
    Neuroscience letters, 1999, Oct-22, Volume: 274, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Basal Ganglia; beta-Alanine; Biological Transport; Carcinogens; Colforsin; Enzyme Inhibitors; GABA Agents; gamma-Aminobutyric Acid; Nipecotic Acids; Proline; Protein Kinase C; Rats; Rats, Wistar; Staurosporine; Substantia Nigra; Synaptosomes; Tetradecanoylphorbol Acetate; Tritium

1999
Chronic morphine increases GABA tone on serotonergic neurons of the dorsal raphe nucleus: association with an up-regulation of the cyclic AMP pathway.
    Neuroscience, 2000, Volume: 95, Issue:2

    Topics: Adenylyl Cyclases; Analgesics, Opioid; Animals; Cardiovascular Agents; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Inhibitors; Excitatory Amino Acid Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Isoquinolines; Male; Membrane Potentials; Morphine; N-Methylaspartate; Neural Inhibition; Periaqueductal Gray; Phenylephrine; Pyrimidines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Serotonin; Substance Withdrawal Syndrome; Sulfonamides; Sympathomimetics; Tetrazoles; Tetrodotoxin; Thionucleotides

2000
Synaptic activation of AMPA receptors inhibits GABA release from cerebellar interneurons.
    Nature neuroscience, 2000, Volume: 3, Issue:6

    Topics: Animals; Cell Membrane; Cerebellum; Chelating Agents; Colforsin; Egtazic Acid; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Microelectrodes; Nerve Fibers; Neural Inhibition; Patch-Clamp Techniques; Purkinje Cells; Rats; Rats, Wistar; Receptors, AMPA; Synapses

2000
Efflux of osmolyte amino acids during isovolumic regulation in hippocampal slices.
    Journal of neuroscience research, 2000, Sep-15, Volume: 61, Issue:6

    Topics: Amino Acids; Animals; Aspartic Acid; Biological Transport; Chloride Channels; Colforsin; Cyclooxygenase Inhibitors; gamma-Aminobutyric Acid; Hippocampus; Hypotonic Solutions; Male; Neurons; Niflumic Acid; Nitrobenzoates; Organ Culture Techniques; Osmolar Concentration; Potassium; Rats; Rats, Wistar; Rubidium Radioisotopes; Taurine; Tritium; Water; Water-Electrolyte Balance

2000
beta-adrenergic receptor-mediated presynaptic facilitation of inhibitory GABAergic transmission at cerebellar interneuron-Purkinje cell synapses.
    Journal of neurophysiology, 2000, Volume: 84, Issue:4

    Topics: Action Potentials; Adrenergic beta-Agonists; Animals; Cerebellum; Colforsin; Electric Stimulation; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Isoproterenol; Neural Inhibition; Norepinephrine; Presynaptic Terminals; Protein Isoforms; Purkinje Cells; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Synapses; Synaptic Transmission

2000
Forskolin modulation of desensitization at GABA(A) and glycine receptors is not mediated by cAMP-dependent protein kinase in isolated carp amacrine-like cells.
    Pflugers Archiv : European journal of physiology, 2001, Volume: 441, Issue:6

    Topics: Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; gamma-Aminobutyric Acid; Glycine; Goldfish; Isoquinolines; Membrane Potentials; Patch-Clamp Techniques; Receptors, GABA-A; Receptors, Glycine; Retina; Sulfonamides

2001
GABA inhibition of immortalized gonadotropin-releasing hormone neuronal excitability involves GABA(A) receptors negatively coupled to cyclic adenosine monophosphate formation.
    Endocrine, 2001, Volume: 14, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Baclofen; Bicuculline; Calcium; Calcium Channels; Cell Line, Transformed; Cell Membrane; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Kinetics; Muscimol; Neurons; Potassium; Receptors, GABA-A

2001
Block by gabapentin of the facilitation of glutamate release from rat trigeminal nucleus following activation of protein kinase C or adenylyl cyclase.
    British journal of pharmacology, 2001, Volume: 134, Issue:2

    Topics: Acetates; Adenylyl Cyclases; Amines; Analgesics; Animals; Colforsin; Cyclohexanecarboxylic Acids; Dose-Response Relationship, Drug; Enzyme Activation; Gabapentin; gamma-Aminobutyric Acid; Glutamic Acid; In Vitro Techniques; Male; Potassium; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate; Trigeminal Nuclei; Tritium

2001
Synergistic interaction of diazepam with 3',5'-cyclic adenosine monophosphate-elevating agents on rat aortic rings.
    European journal of pharmacology, 2001, Oct-05, Volume: 428, Issue:2

    Topics: Animals; Aorta, Thoracic; Colforsin; Cyclic AMP; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Female; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; In Vitro Techniques; Isoproterenol; Isoquinolines; Male; Milrinone; Muscle Relaxants, Central; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Rats; Rats, Sprague-Dawley; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

2001
Postsynaptic application of a peptide inhibitor of cAMP-dependent protein kinase blocks expression of long-lasting synaptic potentiation in hippocampal neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Feb-15, Volume: 23, Issue:4

    Topics: Animals; Carrier Proteins; Cells, Cultured; Chromosome Pairing; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electric Conductivity; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Intracellular Signaling Peptides and Proteins; Kinetics; Long-Term Potentiation; Mice; Mice, Inbred C57BL; Patch-Clamp Techniques; Peptide Fragments; Pyramidal Cells; Synaptic Transmission; Thionucleotides

2003
GABAB receptor-mediated presynaptic potentiation of ATP ionotropic receptors in rat midbrain synaptosomes.
    Neuropharmacology, 2003, Volume: 44, Issue:3

    Topics: Adenosine Triphosphate; Animals; Baclofen; Calcium; Colforsin; Competitive Bidding; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Fura-2; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Immunohistochemistry; In Vitro Techniques; Mesencephalon; Muscimol; Nerve Tissue Proteins; Picrotoxin; Rats; Receptors, GABA-B; Receptors, Purinergic P2; Receptors, Purinergic P2X; Synaptosomes; Time Factors

2003
Functional significance of cannabinoid-mediated, depolarization-induced suppression of inhibition (DSI) in the hippocampus.
    Journal of neurophysiology, 2003, Volume: 90, Issue:1

    Topics: Action Potentials; Animals; Benzoxazines; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Cannabinoids; Colforsin; Electric Stimulation; Enzyme Activators; Enzyme Inhibitors; gamma-Aminobutyric Acid; Hippocampus; Interneurons; Lidocaine; Male; Marine Toxins; Morpholines; Naphthalenes; Neural Inhibition; omega-Conotoxin GVIA; Oxazoles; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Receptors, GABA-A; Sodium Channel Blockers

2003
Positive regulation of GABA(B) receptors dually coupled to cyclic AMP by the allosteric agent CGP7930.
    European journal of pharmacology, 2003, Jun-20, Volume: 471, Issue:2

    Topics: Adenylyl Cyclases; Allosteric Regulation; Animals; Baclofen; Calmodulin; Colforsin; Corpus Striatum; Corticotropin-Releasing Hormone; Cyclic AMP; Cytoplasmic Granules; Drug Synergism; Frontal Lobe; gamma-Aminobutyric Acid; Gene Expression; Male; Olfactory Bulb; Phenols; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-B; Signal Transduction

2003
Modulation of GABA release during morphine withdrawal in midbrain neurons in vitro.
    Neuropharmacology, 2003, Volume: 45, Issue:5

    Topics: Action Potentials; Adenosine; Affinity Labels; Animals; Colforsin; Cyclic AMP; Dipyridamole; Dose-Response Relationship, Drug; Drug Interactions; Enkephalins; Enzyme Inhibitors; gamma-Aminobutyric Acid; In Vitro Techniques; Isoquinolines; Male; Mesencephalon; Mice; Mice, Inbred C57BL; Morphine; Morphine Dependence; Naloxone; Narcotic Antagonists; Narcotics; Neural Inhibition; Neurons; Patch-Clamp Techniques; Periaqueductal Gray; Probenecid; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Substance Withdrawal Syndrome; Sulfonamides; Synaptic Transmission; Thioinosine; Time Factors; Uricosuric Agents; Vasodilator Agents; Xanthines

2003
GABAergic control of neuropeptide gene expression in parvocellular neurons of the hypothalamic paraventricular nucleus.
    The European journal of neuroscience, 2003, Volume: 18, Issue:6

    Topics: Animals; Animals, Newborn; Arginine Vasopressin; Autoradiography; Bicuculline; Cell Count; Colforsin; Corticotropin-Releasing Hormone; Female; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression; Glutamate Decarboxylase; Immunohistochemistry; In Situ Hybridization; Isoenzymes; Male; Microinjections; Microscopy, Immunoelectron; Neurons; Neuropeptides; Organ Culture Techniques; Paraventricular Hypothalamic Nucleus; Potassium; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; RNA, Messenger

2003
Agonist-induced desensitization and endocytosis of heterodimeric GABAB receptors in CHO-K1 cells.
    European journal of pharmacology, 2003, Nov-14, Volume: 481, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Bacterial Proteins; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dimerization; Dose-Response Relationship, Drug; Endocytosis; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression; Green Fluorescent Proteins; Humans; Luminescent Proteins; Microscopy, Confocal; Protein Subunits; Receptors, GABA-B; Recombinant Proteins; Time Factors

2003
Beta subunit phosphorylation selectively increases fast desensitization and prolongs deactivation of alpha1beta1gamma2L and alpha1beta3gamma2L GABA(A) receptor currents.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2003, Dec-17, Volume: 23, Issue:37

    Topics: Cell Line; Colforsin; Culture Media, Serum-Free; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electric Conductivity; gamma-Aminobutyric Acid; Humans; Kinetics; Mutation; Patch-Clamp Techniques; Phosphoprotein Phosphatases; Phosphorylation; Protein Subunits; Receptors, GABA-A; Serine

2003
AMPA receptor-mediated presynaptic inhibition at cerebellar GABAergic synapses: a characterization of molecular mechanisms.
    The European journal of neuroscience, 2004, Volume: 19, Issue:9

    Topics: Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Benzoxazines; Calcium; Calcium Channel Blockers; Cerebellum; Chelating Agents; Colforsin; Cyclopropanes; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Morpholines; Naphthalenes; Neural Inhibition; Neurons; Piperidines; Presynaptic Terminals; Pyrazoles; Rats; Rats, Wistar; Receptors, AMPA; Ryanodine; Synapses; Triazines; Triazoles

2004
Adenosine inhibits GABAergic and glycinergic transmission in adult rat substantia gelatinosa neurons.
    Journal of neurophysiology, 2004, Volume: 92, Issue:5

    Topics: 4-Aminopyridine; 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Animals; Colforsin; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Neurons; Pain; Phorbol 12,13-Dibutyrate; Potassium Channel Blockers; Potassium Channels; Rats; Substantia Gelatinosa; Synaptic Transmission

2004
Mechanism of GABA receptor-mediated inhibition of spontaneous GABA release onto cerebellar Purkinje cells.
    The European journal of neuroscience, 2004, Volume: 20, Issue:3

    Topics: Action Potentials; Age Factors; Animals; Baclofen; Barium; Cadmium; Calcium; Cerebellum; Colforsin; Drug Interactions; Enzyme Inhibitors; Exotoxins; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Neural Inhibition; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Purkinje Cells; Receptors, GABA-A; Ruthenium Red; Synaptic Transmission; Tetrodotoxin

2004
Regulated exocytosis and kiss-and-run of synaptic-like microvesicles in INS-1 and primary rat beta-cells.
    Diabetes, 2005, Volume: 54, Issue:3

    Topics: Animals; Calcium; Calcium Channels; Cell Line, Tumor; Cell Membrane; Cell-Free System; Colforsin; Exocytosis; gamma-Aminobutyric Acid; Glucose; Insulinoma; Islets of Langerhans; Rats; Secretory Vesicles

2005
Cooperative activation of D1 and D2 dopamine receptors enhances a hyperpolarization-activated inward current in layer I interneurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Jul-06, Volume: 25, Issue:27

    Topics: Action Potentials; Animals; Benzazepines; Cations; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dopamine; Dopamine Agonists; Dopamine Antagonists; gamma-Aminobutyric Acid; Interneurons; Ion Transport; Membrane Potentials; Neocortex; Patch-Clamp Techniques; Peptide Fragments; Prefrontal Cortex; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2

2005
Differential roles of mGlu8 receptors in the regulation of glutamate and gamma-aminobutyric acid release at periaqueductal grey level.
    Neuropharmacology, 2005, Volume: 49 Suppl 1

    Topics: Alanine; Aminobutyrates; Analysis of Variance; Animals; Benzoates; Colforsin; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Immunohistochemistry; Isoquinolines; Male; Microdialysis; Microscopy, Immunoelectron; Periaqueductal Gray; Phosphoserine; Protein Kinase Inhibitors; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Sulfonamides; Time Factors

2005
Selective inhibition of spontaneous but not Ca2+ -dependent release machinery by presynaptic group II mGluRs in rat cerebellar slices.
    Journal of neurophysiology, 2006, Volume: 96, Issue:1

    Topics: Action Potentials; Animals; Cadmium; Calcium; Calcium Channels; Cerebellum; Colforsin; Cyclopropanes; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Interneurons; N-Methylaspartate; Nickel; Patch-Clamp Techniques; Presynaptic Terminals; Purkinje Cells; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Synaptic Vesicles

2006
Adenosine A2A receptor stimulation decreases GAT-1-mediated GABA uptake in the globus pallidus of the rat.
    Neuropharmacology, 2006, Volume: 51, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenosine A2 Receptor Agonists; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Data Interpretation, Statistical; Enzyme Inhibitors; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Globus Pallidus; In Vitro Techniques; Isoquinolines; Male; Okadaic Acid; Phenethylamines; Rats; Rats, Wistar; Sulfonamides; Synapses; Triazines; Triazoles

2006
Glucagon-like peptide-1 stimulates GABA formation by pancreatic beta-cells at the level of glutamate decarboxylase.
    American journal of physiology. Endocrinology and metabolism, 2007, Volume: 292, Issue:4

    Topics: Adenylyl Cyclases; Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Enzyme Activation; gamma-Aminobutyric Acid; Glucagon-Like Peptide 1; Glutamate Decarboxylase; Insulin-Secreting Cells; Isoenzymes; Male; Rats; Rats, Wistar

2007
Serotonergic modulation of GABAergic and glutamatergic synaptic transmission in mechanically isolated rat medial preoptic area neurons.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2008, Volume: 33, Issue:2

    Topics: Animals; Colforsin; Evoked Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Neurons; Patch-Clamp Techniques; Preoptic Area; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Synaptic Transmission

2008
Reversibility of cerebellar GABAergic synapse impairment induced by anti-glutamic acid decarboxylase autoantibodies.
    Journal of the neurological sciences, 2008, Aug-15, Volume: 271, Issue:1-2

    Topics: Aged; Animals; Animals, Newborn; Cerebellar Ataxia; Cerebellum; Colforsin; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Humans; Immunoglobulin G; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Patch-Clamp Techniques; Rats; Synapses

2008
GABA synthesis in Schwann cells is induced by the neuroactive steroid allopregnanolone.
    Journal of neurochemistry, 2010, Volume: 112, Issue:4

    Topics: Anesthetics; Animals; Cells, Cultured; Chromatography, High Pressure Liquid; Colforsin; Computational Biology; CREB-Binding Protein; Cyclic AMP; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamate Decarboxylase; Phosphorylation; Pregnanolone; Rats; Rats, Sprague-Dawley; RNA, Messenger; Schwann Cells; Sciatic Nerve; Signal Transduction; Time Factors; Up-Regulation

2010
Protein kinase A and C signaling induces bilirubin potentiation of GABA/glycinergic synaptic transmission in rat ventral cochlear nucleus neurons.
    Brain research, 2010, Aug-12, Volume: 1348

    Topics: Animals; Animals, Newborn; Antioxidants; Benzophenanthridines; Bilirubin; Cochlear Nucleus; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Isoquinolines; Neural Inhibition; Neurons; Patch-Clamp Techniques; Phorbol Esters; Protein Kinase C; Rats; Signal Transduction; Sulfonamides; Synaptic Transmission

2010
Nicotine blocks the hyperpolarization-activated current Ih and severely impairs the oscillatory behavior of oriens-lacunosum moleculare interneurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2010, Aug-11, Volume: 30, Issue:32

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Analysis of Variance; Animals; Biological Clocks; Cardiovascular Agents; Colforsin; Cyclic Nucleotide-Gated Cation Channels; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Female; gamma-Aminobutyric Acid; Green Fluorescent Proteins; Hippocampus; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Interneurons; Male; Mecamylamine; Mice; Mice, Transgenic; Models, Biological; Models, Molecular; Neural Inhibition; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Patch-Clamp Techniques; Potassium Channels; Pyrimidines; Somatostatin

2010
cAMP-dependent protein kinase A activity modulates topiramate potentiation of GABA(A) receptors.
    Epilepsy research, 2011, Volume: 96, Issue:1-2

    Topics: Animals; Anticonvulsants; Biophysics; Bucladesine; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Fructose; gamma-Aminobutyric Acid; Humans; Isoquinolines; Larva; Membrane Potentials; Microinjections; Oocytes; Patch-Clamp Techniques; Protein Kinase Inhibitors; Protein Subunits; Receptors, GABA-A; Sulfonamides; Topiramate; Xenopus

2011
Presynaptic mGlu7 receptors control GABA release in mouse hippocampus.
    Neuropharmacology, 2013, Volume: 66

    Topics: Adenylyl Cyclase Inhibitors; Aminobutyrates; Animals; Baclofen; Benzhydryl Compounds; Benzoates; Benzylamines; Colforsin; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Exocytosis; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Hippocampus; Imines; Mice; Phosphinic Acids; Potassium Chloride; Pyridones; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Synaptosomes; Syntaxin 1; Vesicular Inhibitory Amino Acid Transport Proteins

2013
Morphine withdrawal enhances constitutive μ-opioid receptor activity in the ventral tegmental area.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Nov-14, Volume: 32, Issue:46

    Topics: Adenylyl Cyclases; Analgesics, Opioid; Analysis of Variance; Animals; Colforsin; Cyclic AMP; Dopaminergic Neurons; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Activators; Female; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Morphine; Pregnancy; Receptors, Opioid, mu; Substance Withdrawal Syndrome; Ventral Tegmental Area

2012
Upregulation of TrkB by forskolin facilitated survival of MSC and functional recovery of memory deficient model rats.
    Biochemical and biophysical research communications, 2013, Feb-22, Volume: 431, Issue:4

    Topics: Adenylyl Cyclases; Animals; Brain-Derived Neurotrophic Factor; Cell Survival; Colforsin; Disease Models, Animal; gamma-Aminobutyric Acid; Genetic Therapy; Humans; Male; Maze Learning; Memory; Memory Disorders; Mesenchymal Stem Cell Transplantation; Mesenchymal Stem Cells; Neurons; Rats; Rats, Sprague-Dawley; Receptor, trkB; Recovery of Function; Regeneration; Transduction, Genetic; Up-Regulation

2013
Suppression of inhibitory GABAergic transmission by cAMP signaling pathway: alterations in learning and memory mutants.
    The European journal of neuroscience, 2013, Volume: 37, Issue:9

    Topics: Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Drosophila melanogaster; Drosophila Proteins; GABAergic Neurons; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Learning; Memory, Short-Term; Mushroom Bodies; Mutation; Neuronal Plasticity; Receptors, GABA; Signal Transduction; Synapses

2013
Phosphodiesterase 10A controls D1-mediated facilitation of GABA release from striato-nigral projections under normal and dopamine-depleted conditions.
    Neuropharmacology, 2014, Volume: 76 Pt A

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Colforsin; Corpus Striatum; Dopamine; Dopamine Agonists; Drug Interactions; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Mice; Neural Pathways; Oxidopamine; Papaverine; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Phosphorylation; Potassium; Receptors, Dopamine D1; Substantia Nigra

2014
Contribution of adenylyl cyclase modulation of pre- and postsynaptic GABA neurotransmission to morphine antinociception and tolerance.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2014, Volume: 39, Issue:9

    Topics: Adenine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Analgesics, Opioid; Animals; Bicuculline; Colforsin; Drug Tolerance; Enzyme Activators; Enzyme Inhibitors; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Male; Miniature Postsynaptic Potentials; Morphine; Nociception; Presynaptic Terminals; Rats, Sprague-Dawley; Receptors, GABA-A; Synaptic Transmission

2014
cAMP-dependent insulin modulation of synaptic inhibition in neurons of the dorsal motor nucleus of the vagus is altered in diabetic mice.
    American journal of physiology. Regulatory, integrative and comparative physiology, 2014, Sep-15, Volume: 307, Issue:6

    Topics: Animals; Brain Stem; Brefeldin A; Colforsin; Cyclic AMP; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 1; Electric Stimulation; Female; gamma-Aminobutyric Acid; Glucose Transporter Type 4; Golgi Apparatus; Indinavir; Inhibitory Postsynaptic Potentials; Insulin; Male; Mice; Neural Inhibition; Protein Transport; Synaptic Transmission; Vagus Nerve

2014
Airway Epithelial Cell Release of GABA is Regulated by Protein Kinase A.
    Lung, 2016, Volume: 194, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bronchoalveolar Lavage Fluid; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activators; Epithelial Cells; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Guanine Nucleotide Exchange Factors; Humans; Male; Methacholine Chloride; Mice; Mice, Inbred C57BL; Myocytes, Smooth Muscle; Platelet-Derived Growth Factor; Propranolol; Receptor Protein-Tyrosine Kinases; Respiratory Mucosa; Rifabutin; RNA, Messenger; Signal Transduction; Terbutaline

2016
The upregulation of glutamate decarboxylase 67 against hippocampal excitability damage in male fetal rats by prenatal caffeine exposure.
    Environmental toxicology, 2022, Volume: 37, Issue:11

    Topics: Adenylyl Cyclases; Animals; Brain-Derived Neurotrophic Factor; Caffeine; Colforsin; Female; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Glutamic Acid; Hippocampus; Hypothalamo-Hypophyseal System; Male; Pituitary-Adrenal System; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Wistar; Receptor, Adenosine A2A; Up-Regulation

2022