colforsin has been researched along with gamma-aminobutyric acid in 82 studies
Timeframe | Studies, this research(%) | All Research% |
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pre-1990 | 9 (10.98) | 18.7374 |
1990's | 31 (37.80) | 18.2507 |
2000's | 28 (34.15) | 29.6817 |
2010's | 13 (15.85) | 24.3611 |
2020's | 1 (1.22) | 2.80 |
Authors | Studies |
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Bauer, C; Caldwell, L; Kinnier, WJ; Lancaster, J; McMillan, B; Price, CH; Sweetnam, PM | 1 |
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J | 1 |
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K | 1 |
Eisenberg, HM; Hulsebosch, CE; Lu, Y; Morgan, B; Perez-Polo, JR; Pizzo, DP; Werrbach-Perez, K; Westlund, KN | 1 |
Blackstone, CD; Huganir, RL; Moss, SJ; Smart, TG | 1 |
Ishac, E; Li, C; White, G | 1 |
Hansson, E; Rönnbäck, L | 1 |
Abucham, J; Reichlin, S | 1 |
Wickelgren, WO; Womble, MD | 1 |
Mehta, AK; Ticku, MK | 1 |
Leonard, JP; Wickelgren, WO | 1 |
Heuschneider, G; Schwartz, RD | 1 |
Eimerl, S; Minc-Golomb, D; Schramm, M | 1 |
Barnes, EM; Hablitz, JJ; Tehrani, MH | 1 |
Starr, BS; Starr, MS | 1 |
Hill, DR | 1 |
Weiss, S | 1 |
Dowling, JE; O'Brien, DR | 1 |
Finger, W; Martin, C | 1 |
Cao, Z; Hosford, DA; Lin, FH; Lin, S; Wang, Y | 1 |
Amico, C; Cupello, A; Robello, M | 1 |
Desrues, L; Lamacz, M; Tonon, MC; Vaudry, H | 1 |
Cherubini, E; Sciancalepore, M | 1 |
Kirifides, ML; Lin, RC; Liu, W; Mouradian, RD; Sessler, FM; Waterhouse, BD | 1 |
Fisone, G; Greengard, P; Snyder, GL | 1 |
Bannon, MJ; Granneman, JG; Kapatos, G; Tian, Y | 1 |
Katsuki, H; Kawahara, F; Saito, H | 1 |
Giménez, C; Gomeza, J; Zafra, F | 1 |
Bowery, NG; Malcangio, M | 1 |
Gerschenfeld, HM; Llano, I | 1 |
Adam-Vizi, V; Baranyi, M; Chernaeva, L; Déri, Z; Vizi, ES; Zelles, T | 1 |
Cherubini, E; Sciancalepore, M; Strata, F | 1 |
Bonci, A; Williams, JT | 1 |
Li, A; Wang, HL; Wu, T | 1 |
Bickford, PC; Gould, TJ | 1 |
Obrietan, K; van den Pol, AN | 1 |
Corsi, L; De Blas, AL; Ghose, S; Grayson, DR; Neale, JH; Vicini, S; Wroblewska, B | 1 |
Barni, S; Castoldi, AF; Costa, LG; Manzo, L; Randine, G | 1 |
Bagley, EE; Christie, MJ; Vaughan, CW | 1 |
Konishi, S; Mitoma, H | 1 |
Estevez, AY; O'Regan, MH; Phillis, JW; Song, D | 1 |
Arias-Montaño, JA; Bahena-Trujillo, R | 1 |
Aghajanian, GK; Jolas, T; Nestler, EJ | 1 |
Konishi, S; Saitow, F; Satake, S; Yamada, J | 2 |
Franco, R; Pasantes-Morales, H; Quesada, O | 1 |
Li, P; Yang, XL | 1 |
Beltrán-Parrazal, L; Clapp, C; Martínez de la Escalera, G; Noris, G | 1 |
Maneuf, YP; McKnight, AT | 1 |
Fuentes, T; Galindo, A; García Estañ, J; Hernández, J; Vargas, ML | 1 |
Duffy, SN; Nguyen, PV | 1 |
Gómez-Villafuertes, R; Gualix, J; Miras-Portugal, MT; Pintor, J | 1 |
Deadwyler, SA; Hampson, RE; Weiner, JL; Zhuang, SY | 1 |
Mascia, FM; Olianas, MC; Onali, P | 1 |
Christie, MJ; Hack, SP; Vaughan, CW | 1 |
Bali, B; Kovács, KJ | 1 |
González-Maeso, J; Green, A; Koenig, JA; Wise, A | 1 |
Hinkle, DJ; Macdonald, RL | 1 |
Konishi, S; Rusakov, D; Saitow, F; Satake, S | 1 |
Fujita, T; Kumamoto, E; Yang, K | 1 |
Harvey, VL; Stephens, GJ | 1 |
Eliasson, L; Galvanovskis, J; MacDonald, PE; Obermüller, S; Rorsman, P; Vikman, J | 1 |
Hablitz, JJ; Wu, J | 1 |
de Novellis, V; Maione, S; Marabese, I; Mariani, L; Palazzo, E; Rodella, L; Rossi, F; Siniscalco, D | 1 |
Glitsch, M | 1 |
Aceves, J; Erlij, D; Florán, B; Florán, L; Gonzalez, B; Paz, F | 1 |
Ling, Z; Mao, R; Pipeleers, D; Van de Casteele, M; Wang, C | 1 |
Cho, YW; Hahm, ET; Lee, CH; Lee, JJ | 1 |
Ishida, K; Mitoma, H; Mizusawa, H | 1 |
Ballabio, M; Bonanno, G; Frasca, A; Fumagalli, F; Magnaghi, V; Parducz, A; Procacci, P; Racagni, G | 1 |
Chen, ZN; Li, CY; Shi, HB; Song, NY; Ye, HB; Yin, SK | 1 |
Carloni, P; Cherubini, E; Giorgetti, A; Griguoli, M; Maul, A; Nguyen, C | 1 |
Simeone, TA; White, HS; Wilcox, KS | 1 |
Di Prisco, S; Grilli, M; Marchi, M; Pittaluga, A; Summa, M; Usai, C | 1 |
Adan, RA; Meye, FJ; Ramakers, GM; Smidt, MP; van Zessen, R | 1 |
Cho, Y; Han, D; Heo, H; Joung, I; Kwon, YK; Yoo, M | 1 |
Ganguly, A; Lee, D | 1 |
Berretta, N; Bonito-Oliva, A; Castelli, V; Fisone, G; Giorgi, M; Ledonne, A; Mango, D; Mercuri, NB; Nisticò, R; Sancesario, G | 1 |
Bobeck, EN; Chen, Q; Ingram, SL; Morgan, MM | 1 |
Blake, CB; Smith, BN | 1 |
Danielsson, J; Emala, CW; Funayama, H; Gallos, G; Kim, B; Worgall, TS; Xu, D; Yim, PD; Zaidi, S | 1 |
Dai, S; Guo, Z; He, X; Hu, Z; Jiao, Z; Lu, M; Wang, H; Xu, D | 1 |
1 review(s) available for colforsin and gamma-aminobutyric acid
Article | Year |
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The role of receptor binding in drug discovery.
Topics: Animals; Drug Design; Humans; Receptors, Drug | 1993 |
81 other study(ies) available for colforsin and gamma-aminobutyric acid
Article | Year |
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Chemical genetics reveals a complex functional ground state of neural stem cells.
Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells | 2007 |
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship | 2010 |
Effects of nerve growth factor and acetyl-L-carnitine arginyl amide on the human neuronal line HCN-1A.
Topics: 1-Methyl-3-isobutylxanthine; Acetylcarnitine; Animals; Arginine; Brain Chemistry; Cell Differentiation; Cell Line; Colforsin; gamma-Aminobutyric Acid; Humans; Immunohistochemistry; Mice; Nerve Growth Factors; Neurofilament Proteins; Neurons | 1992 |
Functional modulation of GABAA receptors by cAMP-dependent protein phosphorylation.
Topics: Animals; Cell Line; Cells, Cultured; Colforsin; Cyclic AMP; Electric Conductivity; gamma-Aminobutyric Acid; Immunosorbent Techniques; Kinetics; Mice; Mutagenesis, Site-Directed; Neurons; Peptide Mapping; Phosphorylation; Protein Kinases; Rats; Receptors, GABA-A; Recombinant Proteins; Transfection; Zinc | 1992 |
1,9-Dideoxyforskolin does not mimic all cAMP and protein kinase A independent effects of forskolin on GABA activated ion currents in adult rat sensory neurons.
Topics: Animals; Colforsin; Cyclic AMP; Electric Conductivity; gamma-Aminobutyric Acid; Ion Channels; Neurons, Afferent; Protein Kinases; Rats; Rats, Inbred Strains | 1992 |
Receptor regulation of the glutamate, GABA and taurine high-affinity uptake into astrocytes in primary culture.
Topics: Animals; Animals, Newborn; Aspartic Acid; Astrocytes; Biological Transport; Cells, Cultured; Cerebral Cortex; Cholera Toxin; Colforsin; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Isoproterenol; Kinetics; Phenylephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Serotonin; Serotonin; Taurine; Virulence Factors, Bordetella | 1991 |
Regulation of cholecystokinin octapeptide secretion by rat cerebral cortical cells in primary culture.
Topics: Animals; Calcium; Cells, Cultured; Cerebral Cortex; Colforsin; Embryo, Mammalian; GABA Antagonists; gamma-Aminobutyric Acid; Membrane Potentials; Neurotransmitter Agents; Potassium; Rats; Sincalide; Tetrodotoxin; Verapamil; Veratridine | 1991 |
Inhibition of a cAMP-dependent Ca-activated K conductance by forskolin prolongs Ca action potential duration in lamprey sensory neurons.
Topics: Action Potentials; Animals; Calcium Chloride; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; In Vitro Techniques; Lampreys; Neurons, Afferent; Potassium; Potassium Channels; Spinal Cord; Tetrodotoxin | 1990 |
gamma-Aminobutyric acidA receptor desensitization in mice spinal cord cultured neurons: lack of involvement of protein kinases A and C.
Topics: Animals; Cells, Cultured; Chloride Channels; Colforsin; Female; gamma-Aminobutyric Acid; Male; Membrane Proteins; Mice; Mice, Inbred C57BL; Neurons; Protein Kinase C; Protein Kinase Inhibitors; Protein Kinases; Receptors, GABA-A; Spinal Cord | 1990 |
Prolongation of calcium action potentials by gamma-aminobutyric acid in primary sensory neurones of lamprey.
Topics: Action Potentials; Animals; Calcium; Colforsin; Fishes; gamma-Aminobutyric Acid; In Vitro Techniques; Ion Channels; Lampreys; Neurons, Afferent; Tetrodotoxin; Time Factors | 1986 |
cAMP and forskolin decrease gamma-aminobutyric acid-gated chloride flux in rat brain synaptoneurosomes.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Brain; Bucladesine; Chloride Channels; Chlorides; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; In Vitro Techniques; Membrane Proteins; Muscimol; Rats; Synaptosomes | 1989 |
Cysteine sulfinic acid-induced release of D-[3H]aspartate and [14C]GABA in hippocampus slices: the role of sodium channels and cAMP.
Topics: 1-Methyl-3-isobutylxanthine; Amino Acids; Animals; Aspartic Acid; Calcium; Cnidarian Venoms; Colforsin; Cysteine; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Male; Neurotoxins; Neurotransmitter Agents; Rats; Sodium Channels; Tetrodotoxin | 1989 |
cAMP increases the rate of GABAA receptor desensitization in chick cortical neurons.
Topics: Animals; Cells, Cultured; Cerebral Cortex; Chick Embryo; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; Receptors, GABA-A | 1989 |
Circling evoked by intranigral SKF 38393: a GABA-mediated D-1 response?
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Colforsin; Dopamine Agents; Dose-Response Relationship, Drug; Drug Synergism; gamma-Aminobutyric Acid; Male; Motor Activity; Nipecotic Acids; Pentobarbital; Rats; Rats, Inbred Strains; Substantia Nigra | 1989 |
GABAB receptor modulation of adenylate cyclase activity in rat brain slices.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Baclofen; Brain; Cerebral Cortex; Colforsin; Cyclic AMP; Diterpenes; gamma-Aminobutyric Acid; In Vitro Techniques; Nipecotic Acids; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A | 1985 |
Forskolin attenuates the evoked release of [3H]GABA from striatal neurons in primary culture.
Topics: Animals; Bucladesine; Cells, Cultured; Colforsin; Corpus Striatum; Cyclic AMP; gamma-Aminobutyric Acid; Mice; Thionucleotides | 1988 |
Dopaminergic regulation of GABA release from the intact goldfish retina.
Topics: Animals; Calcium; Colforsin; Cyclic AMP; Cyprinidae; Dopamine; gamma-Aminobutyric Acid; Glutamates; Glutamic Acid; Goldfish; In Vitro Techniques; Retina; Synaptic Transmission | 1985 |
Presynaptic effect of gamma-aminobutyric acid on the inhibitory nerve and nerve terminals in the crayfish neuromuscular junction.
Topics: Action Potentials; Animals; Astacoidea; Colforsin; gamma-Aminobutyric Acid; In Vitro Techniques; Neural Inhibition; Neuromuscular Junction; Peripheral Nerves; Serotonin | 1989 |
GABAB receptor-mediated effects in synaptosomes of lethargic (lh/lh) mice.
Topics: Animals; Calcium; Cerebral Cortex; Colforsin; Cyclic AMP; Epilepsy; Epilepsy, Absence; gamma-Aminobutyric Acid; Hybridization, Genetic; Male; Mice; Mice, Inbred Strains; Potassium Chloride; Receptors, GABA-B; Synaptosomes; Thalamus | 1995 |
Regulation of GABAA receptor in cerebellar granule cells in culture: differential involvement of kinase activities.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Cells, Cultured; Cerebellum; Chloride Channels; Colforsin; Cyclic AMP; Cytoplasmic Granules; Electrophysiology; gamma-Aminobutyric Acid; Kinetics; Membrane Potentials; Membrane Proteins; Phosphorylation; Phosphotransferases; Picrotoxin; Protein Kinase Inhibitors; Protein Kinases; Rats; Rats, Wistar; Receptors, GABA-A | 1993 |
Mechanism of action of gamma-aminobutyric acid on frog melanotrophs.
Topics: Adenylyl Cyclases; Animals; Baclofen; Calcium; Calcium Channels; Colforsin; Cyclic AMP; GABA-A Receptor Agonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Inositol Phosphates; Male; Melanocyte-Stimulating Hormones; Models, Biological; Pituitary Gland, Posterior; Rana ridibunda; Receptors, GABA-A; Receptors, GABA-B; Signal Transduction; Taurine | 1995 |
Protein kinase A-dependent increase in frequency of miniature GABAergic currents in rat CA3 hippocampal neurons.
Topics: Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electric Conductivity; gamma-Aminobutyric Acid; Hippocampus; In Vitro Techniques; Kynurenic Acid; Neurons; Patch-Clamp Techniques; Protein Kinase Inhibitors; Rats; Rats, Wistar; Tetrodotoxin; Thionucleotides | 1995 |
Noradrenergic enhancement of GABA-induced input resistance changes in layer V regular spiking pyramidal neurons of rat somatosensory cortex.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Colforsin; Electrophysiology; gamma-Aminobutyric Acid; In Vitro Techniques; Isoproterenol; Membrane Potentials; Microelectrodes; Muscimol; Norepinephrine; Pyramidal Cells; Rats; Somatosensory Cortex | 1995 |
Phosphorylation of DARPP-32 is regulated by GABA in rat striatum and substantia nigra.
Topics: Animals; Baclofen; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine and cAMP-Regulated Phosphoprotein 32; GABA Antagonists; gamma-Aminobutyric Acid; Male; Nerve Tissue Proteins; Phosphoproteins; Phosphorylation; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, GABA; Substantia Nigra | 1994 |
Dopamine and gamma-aminobutyric acid transporters: differential regulation by agents that promote phosphorylation.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Carrier Proteins; Colforsin; Dopamine; Dopamine Plasma Membrane Transport Proteins; Ethers, Cyclic; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Membrane Glycoproteins; Membrane Proteins; Membrane Transport Proteins; Neostriatum; Nerve Tissue Proteins; Okadaic Acid; Organic Anion Transporters; Phorbol Esters; Phosphoprotein Phosphatases; Phosphorylation; Rats; Rats, Sprague-Dawley; Signal Transduction; Synaptosomes | 1994 |
Inhibition by 5-HT7 receptor stimulation of GABAA receptor-activated current in cultured rat suprachiasmatic neurones.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cell Membrane; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; gamma-Aminobutyric Acid; Membrane Potentials; Neurons; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, Serotonin; Ritanserin; Serotonin; Suprachiasmatic Nucleus | 1994 |
Cellular distribution and regulation by cAMP of the GABA transporter (GAT-1) mRNA.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Animals, Newborn; Astrocytes; Base Sequence; Bucladesine; Carrier Proteins; Cells, Cultured; Cerebral Cortex; Cloning, Molecular; Colforsin; Cyclic AMP; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Gene Expression Regulation; Glial Fibrillary Acidic Protein; Immunohistochemistry; Kinetics; Membrane Proteins; Membrane Transport Proteins; Molecular Sequence Data; Neuroglia; Oligodeoxyribonucleotides; Organic Anion Transporters; Rats; Rats, Wistar; RNA, Messenger; Tetradecanoylphorbol Acetate; Time Factors | 1994 |
GABAB receptor-mediated inhibition of forskolin-stimulated cyclic AMP accumulation in rat spinal cord.
Topics: Analgesics; Animals; Animals, Newborn; Baclofen; Capsaicin; Colforsin; Cyclic AMP; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Norepinephrine; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Cord | 1993 |
Beta-adrenergic enhancement of inhibitory synaptic activity in rat cerebellar stellate and Purkinje cells.
Topics: Action Potentials; Animals; Cerebellum; Colforsin; gamma-Aminobutyric Acid; In Vitro Techniques; Isoproterenol; Kinetics; Norepinephrine; Purkinje Cells; Rats; Receptors, Adrenergic, beta; Synapses; Tetrodotoxin | 1993 |
Transmitter release by non-receptor activation of the alpha-subunit of guanine nucleotide regulatory protein in rat striatal slices.
Topics: 3,4-Dihydroxyphenylacetic Acid; Acetylcholine; Adrenergic Uptake Inhibitors; Aluminum Chloride; Aluminum Compounds; Animals; Calcium; Chlorides; Colforsin; Corpus Striatum; Dopamine; Dopamine Uptake Inhibitors; Drug Synergism; Egtazic Acid; Enzyme Inhibitors; Ethylmaleimide; gamma-Aminobutyric Acid; GTP-Binding Proteins; Male; Monoamine Oxidase Inhibitors; Neomycin; Nomifensine; Pargyline; Phosphatidylinositol Diacylglycerol-Lyase; Phosphoric Diester Hydrolases; Rats; Rats, Wistar; Reserpine; Ruthenium Red; Signal Transduction; Sodium Fluoride; Stimulation, Chemical; Synaptosomes; Type C Phospholipases | 1995 |
Cyclic AMP-dependent modulation of giant depolarizing potentials by metabotropic glutamate receptors in the rat hippocampus.
Topics: Animals; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; Hippocampus; Kynurenic Acid; Membrane Potentials; Quisqualic Acid; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate | 1995 |
Increased probability of GABA release during withdrawal from morphine.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Action Potentials; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dopamine; Dopamine Antagonists; Enzyme Activation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Guinea Pigs; Interneurons; Morphine; Nerve Tissue Proteins; Organophosphorus Compounds; Patch-Clamp Techniques; Phorbol 12,13-Dibutyrate; Picrotoxin; Receptors, GABA-A; Salicylamides; Serotonin; Signal Transduction; Staurosporine; Strychnine; Substance Withdrawal Syndrome; Tegmentum Mesencephali; Thionucleotides | 1997 |
Vasoactive intestinal polypeptide enhances the GABAergic synaptic transmission in cultured hippocampal neurons.
Topics: 2-Amino-5-phosphonovalerate; 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Cadmium Chloride; Calcium Channel Blockers; Carcinogens; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Hippocampus; Neurons; Patch-Clamp Techniques; Rats; Synaptic Transmission; Tetrodotoxin; Vasoactive Intestinal Peptide | 1997 |
Age-related deficits in the cerebellar beta adrenergic signal transduction cascade in Fischer 344 rats.
Topics: Aging; Animals; Cerebellum; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; Male; Rats; Rats, Inbred F344; Receptors, Adrenergic, beta; Signal Transduction | 1997 |
GABA activity mediating cytosolic Ca2+ rises in developing neurons is modulated by cAMP-dependent signal transduction.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenine; Adenylyl Cyclase Inhibitors; Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cytosol; Electric Stimulation; Embryo, Mammalian; Enzyme Inhibitors; gamma-Aminobutyric Acid; Hypothalamus, Middle; Isoquinolines; Neurons; Rats; Rats, Sprague-Dawley; Signal Transduction; Sulfonamides; Synapses; Tetrodotoxin; Thionucleotides | 1997 |
N-acetylaspartylglutamate stimulates metabotropic glutamate receptor 3 to regulate expression of the GABA(A) alpha6 subunit in cerebellar granule cells.
Topics: Animals; Cells, Cultured; Cerebellum; Colforsin; Cyclic AMP; Dipeptides; Electric Conductivity; Furosemide; gamma-Aminobutyric Acid; Ion Channel Gating; Neurons; Polymerase Chain Reaction; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Receptors, Metabotropic Glutamate; RNA, Messenger; Transcription, Genetic | 1997 |
Ethanol selectively interferes with the trophic action of NMDA and carbachol on cultured cerebellar granule neurons undergoing apoptosis.
Topics: Animals; Apoptosis; Carbachol; Cell Survival; Cells, Cultured; Central Nervous System Depressants; Cerebellum; Colforsin; Drug Interactions; Ethanol; Excitatory Amino Acid Agonists; gamma-Aminobutyric Acid; Microscopy, Electron; Muscarinic Agonists; N-Methylaspartate; Neurons; Potassium; Rats; Rats, Sprague-Dawley | 1998 |
Inhibition by adenosine receptor agonists of synaptic transmission in rat periaqueductal grey neurons.
Topics: Action Potentials; Adenosine; Animals; Colforsin; gamma-Aminobutyric Acid; Glutamic Acid; In Vitro Techniques; Membrane Potentials; Neurons; Patch-Clamp Techniques; Periaqueductal Gray; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Synaptic Transmission | 1999 |
Monoaminergic long-term facilitation of GABA-mediated inhibitory transmission at cerebellar synapses.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Cerebellum; Colforsin; Cyclic AMP; Electric Stimulation; Enzyme Inhibitors; Evoked Potentials; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Isoquinolines; Long-Term Potentiation; Methiothepin; Neuronal Plasticity; Norepinephrine; Propranolol; Protein Kinase Inhibitors; Purkinje Cells; Rats; Rats, Wistar; Receptors, GABA; Serotonin; Sulfonamides; Synapses; Synaptic Transmission; Tetrodotoxin; Thionucleotides | 1999 |
Hyposmotically induced amino acid release from the rat cerebral cortex: role of phospholipases and protein kinases.
Topics: Acetophenones; Alanine; Amino Acids; Animals; Arachidonic Acids; Aspartic Acid; Brain Edema; Cerebral Cortex; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dimethyl Sulfoxide; Enzyme Inhibitors; Estrenes; Ethanolamines; Fatty Acids, Unsaturated; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Hypotonic Solutions; Male; Osmotic Pressure; Phosphodiesterase Inhibitors; Phospholipases A; Phospholipases A2; Protein Kinase C; Pyrrolidinones; Rats; Rats, Sprague-Dawley; Serine; Solvents; Taurine; Water-Electrolyte Balance | 1999 |
[3H] gamma-aminobutyric acid transport in rat substantia nigra pars reticulata synaptosomes: pharmacological characterization and phorbol ester-induced inhibition.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Basal Ganglia; beta-Alanine; Biological Transport; Carcinogens; Colforsin; Enzyme Inhibitors; GABA Agents; gamma-Aminobutyric Acid; Nipecotic Acids; Proline; Protein Kinase C; Rats; Rats, Wistar; Staurosporine; Substantia Nigra; Synaptosomes; Tetradecanoylphorbol Acetate; Tritium | 1999 |
Chronic morphine increases GABA tone on serotonergic neurons of the dorsal raphe nucleus: association with an up-regulation of the cyclic AMP pathway.
Topics: Adenylyl Cyclases; Analgesics, Opioid; Animals; Cardiovascular Agents; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electrophysiology; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Inhibitors; Excitatory Amino Acid Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Isoquinolines; Male; Membrane Potentials; Morphine; N-Methylaspartate; Neural Inhibition; Periaqueductal Gray; Phenylephrine; Pyrimidines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Serotonin; Substance Withdrawal Syndrome; Sulfonamides; Sympathomimetics; Tetrazoles; Tetrodotoxin; Thionucleotides | 2000 |
Synaptic activation of AMPA receptors inhibits GABA release from cerebellar interneurons.
Topics: Animals; Cell Membrane; Cerebellum; Chelating Agents; Colforsin; Egtazic Acid; Electric Stimulation; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Microelectrodes; Nerve Fibers; Neural Inhibition; Patch-Clamp Techniques; Purkinje Cells; Rats; Rats, Wistar; Receptors, AMPA; Synapses | 2000 |
Efflux of osmolyte amino acids during isovolumic regulation in hippocampal slices.
Topics: Amino Acids; Animals; Aspartic Acid; Biological Transport; Chloride Channels; Colforsin; Cyclooxygenase Inhibitors; gamma-Aminobutyric Acid; Hippocampus; Hypotonic Solutions; Male; Neurons; Niflumic Acid; Nitrobenzoates; Organ Culture Techniques; Osmolar Concentration; Potassium; Rats; Rats, Wistar; Rubidium Radioisotopes; Taurine; Tritium; Water; Water-Electrolyte Balance | 2000 |
beta-adrenergic receptor-mediated presynaptic facilitation of inhibitory GABAergic transmission at cerebellar interneuron-Purkinje cell synapses.
Topics: Action Potentials; Adrenergic beta-Agonists; Animals; Cerebellum; Colforsin; Electric Stimulation; gamma-Aminobutyric Acid; In Vitro Techniques; Interneurons; Isoproterenol; Neural Inhibition; Norepinephrine; Presynaptic Terminals; Protein Isoforms; Purkinje Cells; Rats; Rats, Wistar; Receptors, Adrenergic, beta; Synapses; Synaptic Transmission | 2000 |
Forskolin modulation of desensitization at GABA(A) and glycine receptors is not mediated by cAMP-dependent protein kinase in isolated carp amacrine-like cells.
Topics: Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; gamma-Aminobutyric Acid; Glycine; Goldfish; Isoquinolines; Membrane Potentials; Patch-Clamp Techniques; Receptors, GABA-A; Receptors, Glycine; Retina; Sulfonamides | 2001 |
GABA inhibition of immortalized gonadotropin-releasing hormone neuronal excitability involves GABA(A) receptors negatively coupled to cyclic adenosine monophosphate formation.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Baclofen; Bicuculline; Calcium; Calcium Channels; Cell Line, Transformed; Cell Membrane; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Kinetics; Muscimol; Neurons; Potassium; Receptors, GABA-A | 2001 |
Block by gabapentin of the facilitation of glutamate release from rat trigeminal nucleus following activation of protein kinase C or adenylyl cyclase.
Topics: Acetates; Adenylyl Cyclases; Amines; Analgesics; Animals; Colforsin; Cyclohexanecarboxylic Acids; Dose-Response Relationship, Drug; Enzyme Activation; Gabapentin; gamma-Aminobutyric Acid; Glutamic Acid; In Vitro Techniques; Male; Potassium; Protein Kinase C; Rats; Tetradecanoylphorbol Acetate; Trigeminal Nuclei; Tritium | 2001 |
Synergistic interaction of diazepam with 3',5'-cyclic adenosine monophosphate-elevating agents on rat aortic rings.
Topics: Animals; Aorta, Thoracic; Colforsin; Cyclic AMP; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Female; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; In Vitro Techniques; Isoproterenol; Isoquinolines; Male; Milrinone; Muscle Relaxants, Central; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Rats; Rats, Sprague-Dawley; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents | 2001 |
Postsynaptic application of a peptide inhibitor of cAMP-dependent protein kinase blocks expression of long-lasting synaptic potentiation in hippocampal neurons.
Topics: Animals; Carrier Proteins; Cells, Cultured; Chromosome Pairing; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electric Conductivity; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Hippocampus; Intracellular Signaling Peptides and Proteins; Kinetics; Long-Term Potentiation; Mice; Mice, Inbred C57BL; Patch-Clamp Techniques; Peptide Fragments; Pyramidal Cells; Synaptic Transmission; Thionucleotides | 2003 |
GABAB receptor-mediated presynaptic potentiation of ATP ionotropic receptors in rat midbrain synaptosomes.
Topics: Adenosine Triphosphate; Animals; Baclofen; Calcium; Colforsin; Competitive Bidding; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Fura-2; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Immunohistochemistry; In Vitro Techniques; Mesencephalon; Muscimol; Nerve Tissue Proteins; Picrotoxin; Rats; Receptors, GABA-B; Receptors, Purinergic P2; Receptors, Purinergic P2X; Synaptosomes; Time Factors | 2003 |
Functional significance of cannabinoid-mediated, depolarization-induced suppression of inhibition (DSI) in the hippocampus.
Topics: Action Potentials; Animals; Benzoxazines; Calcium Channel Blockers; Cannabinoid Receptor Modulators; Cannabinoids; Colforsin; Electric Stimulation; Enzyme Activators; Enzyme Inhibitors; gamma-Aminobutyric Acid; Hippocampus; Interneurons; Lidocaine; Male; Marine Toxins; Morpholines; Naphthalenes; Neural Inhibition; omega-Conotoxin GVIA; Oxazoles; Patch-Clamp Techniques; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug; Receptors, GABA-A; Sodium Channel Blockers | 2003 |
Positive regulation of GABA(B) receptors dually coupled to cyclic AMP by the allosteric agent CGP7930.
Topics: Adenylyl Cyclases; Allosteric Regulation; Animals; Baclofen; Calmodulin; Colforsin; Corpus Striatum; Corticotropin-Releasing Hormone; Cyclic AMP; Cytoplasmic Granules; Drug Synergism; Frontal Lobe; gamma-Aminobutyric Acid; Gene Expression; Male; Olfactory Bulb; Phenols; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-B; Signal Transduction | 2003 |
Modulation of GABA release during morphine withdrawal in midbrain neurons in vitro.
Topics: Action Potentials; Adenosine; Affinity Labels; Animals; Colforsin; Cyclic AMP; Dipyridamole; Dose-Response Relationship, Drug; Drug Interactions; Enkephalins; Enzyme Inhibitors; gamma-Aminobutyric Acid; In Vitro Techniques; Isoquinolines; Male; Mesencephalon; Mice; Mice, Inbred C57BL; Morphine; Morphine Dependence; Naloxone; Narcotic Antagonists; Narcotics; Neural Inhibition; Neurons; Patch-Clamp Techniques; Periaqueductal Gray; Probenecid; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Substance Withdrawal Syndrome; Sulfonamides; Synaptic Transmission; Thioinosine; Time Factors; Uricosuric Agents; Vasodilator Agents; Xanthines | 2003 |
GABAergic control of neuropeptide gene expression in parvocellular neurons of the hypothalamic paraventricular nucleus.
Topics: Animals; Animals, Newborn; Arginine Vasopressin; Autoradiography; Bicuculline; Cell Count; Colforsin; Corticotropin-Releasing Hormone; Female; GABA Antagonists; gamma-Aminobutyric Acid; Gene Expression; Glutamate Decarboxylase; Immunohistochemistry; In Situ Hybridization; Isoenzymes; Male; Microinjections; Microscopy, Immunoelectron; Neurons; Neuropeptides; Organ Culture Techniques; Paraventricular Hypothalamic Nucleus; Potassium; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; RNA, Messenger | 2003 |
Agonist-induced desensitization and endocytosis of heterodimeric GABAB receptors in CHO-K1 cells.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Bacterial Proteins; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dimerization; Dose-Response Relationship, Drug; Endocytosis; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; gamma-Aminobutyric Acid; Gene Expression; Green Fluorescent Proteins; Humans; Luminescent Proteins; Microscopy, Confocal; Protein Subunits; Receptors, GABA-B; Recombinant Proteins; Time Factors | 2003 |
Beta subunit phosphorylation selectively increases fast desensitization and prolongs deactivation of alpha1beta1gamma2L and alpha1beta3gamma2L GABA(A) receptor currents.
Topics: Cell Line; Colforsin; Culture Media, Serum-Free; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electric Conductivity; gamma-Aminobutyric Acid; Humans; Kinetics; Mutation; Patch-Clamp Techniques; Phosphoprotein Phosphatases; Phosphorylation; Protein Subunits; Receptors, GABA-A; Serine | 2003 |
AMPA receptor-mediated presynaptic inhibition at cerebellar GABAergic synapses: a characterization of molecular mechanisms.
Topics: Action Potentials; alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid; Animals; Benzothiadiazines; Benzoxazines; Calcium; Calcium Channel Blockers; Cerebellum; Chelating Agents; Colforsin; Cyclopropanes; Drug Interactions; Egtazic Acid; Enzyme Inhibitors; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Morpholines; Naphthalenes; Neural Inhibition; Neurons; Piperidines; Presynaptic Terminals; Pyrazoles; Rats; Rats, Wistar; Receptors, AMPA; Ryanodine; Synapses; Triazines; Triazoles | 2004 |
Adenosine inhibits GABAergic and glycinergic transmission in adult rat substantia gelatinosa neurons.
Topics: 4-Aminopyridine; 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Animals; Colforsin; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Neurons; Pain; Phorbol 12,13-Dibutyrate; Potassium Channel Blockers; Potassium Channels; Rats; Substantia Gelatinosa; Synaptic Transmission | 2004 |
Mechanism of GABA receptor-mediated inhibition of spontaneous GABA release onto cerebellar Purkinje cells.
Topics: Action Potentials; Age Factors; Animals; Baclofen; Barium; Cadmium; Calcium; Cerebellum; Colforsin; Drug Interactions; Enzyme Inhibitors; Exotoxins; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Neural Inhibition; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Purkinje Cells; Receptors, GABA-A; Ruthenium Red; Synaptic Transmission; Tetrodotoxin | 2004 |
Regulated exocytosis and kiss-and-run of synaptic-like microvesicles in INS-1 and primary rat beta-cells.
Topics: Animals; Calcium; Calcium Channels; Cell Line, Tumor; Cell Membrane; Cell-Free System; Colforsin; Exocytosis; gamma-Aminobutyric Acid; Glucose; Insulinoma; Islets of Langerhans; Rats; Secretory Vesicles | 2005 |
Cooperative activation of D1 and D2 dopamine receptors enhances a hyperpolarization-activated inward current in layer I interneurons.
Topics: Action Potentials; Animals; Benzazepines; Cations; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dopamine; Dopamine Agonists; Dopamine Antagonists; gamma-Aminobutyric Acid; Interneurons; Ion Transport; Membrane Potentials; Neocortex; Patch-Clamp Techniques; Peptide Fragments; Prefrontal Cortex; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2 | 2005 |
Differential roles of mGlu8 receptors in the regulation of glutamate and gamma-aminobutyric acid release at periaqueductal grey level.
Topics: Alanine; Aminobutyrates; Analysis of Variance; Animals; Benzoates; Colforsin; Dose-Response Relationship, Drug; Drug Combinations; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Immunohistochemistry; Isoquinolines; Male; Microdialysis; Microscopy, Immunoelectron; Periaqueductal Gray; Phosphoserine; Protein Kinase Inhibitors; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Sulfonamides; Time Factors | 2005 |
Selective inhibition of spontaneous but not Ca2+ -dependent release machinery by presynaptic group II mGluRs in rat cerebellar slices.
Topics: Action Potentials; Animals; Cadmium; Calcium; Calcium Channels; Cerebellum; Colforsin; Cyclopropanes; Excitatory Postsynaptic Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Glycine; Interneurons; N-Methylaspartate; Nickel; Patch-Clamp Techniques; Presynaptic Terminals; Purkinje Cells; Rats; Rats, Sprague-Dawley; Receptors, Metabotropic Glutamate; Synaptic Vesicles | 2006 |
Adenosine A2A receptor stimulation decreases GAT-1-mediated GABA uptake in the globus pallidus of the rat.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine; Adenosine A2 Receptor Agonists; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Data Interpretation, Statistical; Enzyme Inhibitors; GABA Plasma Membrane Transport Proteins; gamma-Aminobutyric Acid; Globus Pallidus; In Vitro Techniques; Isoquinolines; Male; Okadaic Acid; Phenethylamines; Rats; Rats, Wistar; Sulfonamides; Synapses; Triazines; Triazoles | 2006 |
Glucagon-like peptide-1 stimulates GABA formation by pancreatic beta-cells at the level of glutamate decarboxylase.
Topics: Adenylyl Cyclases; Animals; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Enzyme Activation; gamma-Aminobutyric Acid; Glucagon-Like Peptide 1; Glutamate Decarboxylase; Insulin-Secreting Cells; Isoenzymes; Male; Rats; Rats, Wistar | 2007 |
Serotonergic modulation of GABAergic and glutamatergic synaptic transmission in mechanically isolated rat medial preoptic area neurons.
Topics: Animals; Colforsin; Evoked Potentials; gamma-Aminobutyric Acid; Glutamic Acid; Neurons; Patch-Clamp Techniques; Preoptic Area; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Synaptic Transmission | 2008 |
Reversibility of cerebellar GABAergic synapse impairment induced by anti-glutamic acid decarboxylase autoantibodies.
Topics: Aged; Animals; Animals, Newborn; Cerebellar Ataxia; Cerebellum; Colforsin; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Humans; Immunoglobulin G; In Vitro Techniques; Inhibitory Postsynaptic Potentials; Patch-Clamp Techniques; Rats; Synapses | 2008 |
GABA synthesis in Schwann cells is induced by the neuroactive steroid allopregnanolone.
Topics: Anesthetics; Animals; Cells, Cultured; Chromatography, High Pressure Liquid; Colforsin; Computational Biology; CREB-Binding Protein; Cyclic AMP; gamma-Aminobutyric Acid; Gene Expression Regulation; Glutamate Decarboxylase; Phosphorylation; Pregnanolone; Rats; Rats, Sprague-Dawley; RNA, Messenger; Schwann Cells; Sciatic Nerve; Signal Transduction; Time Factors; Up-Regulation | 2010 |
Protein kinase A and C signaling induces bilirubin potentiation of GABA/glycinergic synaptic transmission in rat ventral cochlear nucleus neurons.
Topics: Animals; Animals, Newborn; Antioxidants; Benzophenanthridines; Bilirubin; Cochlear Nucleus; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; gamma-Aminobutyric Acid; Glycine; In Vitro Techniques; Isoquinolines; Neural Inhibition; Neurons; Patch-Clamp Techniques; Phorbol Esters; Protein Kinase C; Rats; Signal Transduction; Sulfonamides; Synaptic Transmission | 2010 |
Nicotine blocks the hyperpolarization-activated current Ih and severely impairs the oscillatory behavior of oriens-lacunosum moleculare interneurons.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Analysis of Variance; Animals; Biological Clocks; Cardiovascular Agents; Colforsin; Cyclic Nucleotide-Gated Cation Channels; Dihydro-beta-Erythroidine; Dose-Response Relationship, Drug; Electric Stimulation; Excitatory Amino Acid Antagonists; Female; gamma-Aminobutyric Acid; Green Fluorescent Proteins; Hippocampus; Hyperpolarization-Activated Cyclic Nucleotide-Gated Channels; In Vitro Techniques; Interneurons; Male; Mecamylamine; Mice; Mice, Transgenic; Models, Biological; Models, Molecular; Neural Inhibition; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Patch-Clamp Techniques; Potassium Channels; Pyrimidines; Somatostatin | 2010 |
cAMP-dependent protein kinase A activity modulates topiramate potentiation of GABA(A) receptors.
Topics: Animals; Anticonvulsants; Biophysics; Bucladesine; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Drug Interactions; Electric Stimulation; Fructose; gamma-Aminobutyric Acid; Humans; Isoquinolines; Larva; Membrane Potentials; Microinjections; Oocytes; Patch-Clamp Techniques; Protein Kinase Inhibitors; Protein Subunits; Receptors, GABA-A; Sulfonamides; Topiramate; Xenopus | 2011 |
Presynaptic mGlu7 receptors control GABA release in mouse hippocampus.
Topics: Adenylyl Cyclase Inhibitors; Aminobutyrates; Animals; Baclofen; Benzhydryl Compounds; Benzoates; Benzylamines; Colforsin; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Exocytosis; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Hippocampus; Imines; Mice; Phosphinic Acids; Potassium Chloride; Pyridones; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Synaptosomes; Syntaxin 1; Vesicular Inhibitory Amino Acid Transport Proteins | 2013 |
Morphine withdrawal enhances constitutive μ-opioid receptor activity in the ventral tegmental area.
Topics: Adenylyl Cyclases; Analgesics, Opioid; Analysis of Variance; Animals; Colforsin; Cyclic AMP; Dopaminergic Neurons; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enzyme Activators; Female; gamma-Aminobutyric Acid; Male; Mice; Mice, Inbred C57BL; Morphine; Pregnancy; Receptors, Opioid, mu; Substance Withdrawal Syndrome; Ventral Tegmental Area | 2012 |
Upregulation of TrkB by forskolin facilitated survival of MSC and functional recovery of memory deficient model rats.
Topics: Adenylyl Cyclases; Animals; Brain-Derived Neurotrophic Factor; Cell Survival; Colforsin; Disease Models, Animal; gamma-Aminobutyric Acid; Genetic Therapy; Humans; Male; Maze Learning; Memory; Memory Disorders; Mesenchymal Stem Cell Transplantation; Mesenchymal Stem Cells; Neurons; Rats; Rats, Sprague-Dawley; Receptor, trkB; Recovery of Function; Regeneration; Transduction, Genetic; Up-Regulation | 2013 |
Suppression of inhibitory GABAergic transmission by cAMP signaling pathway: alterations in learning and memory mutants.
Topics: Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Drosophila melanogaster; Drosophila Proteins; GABAergic Neurons; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Learning; Memory, Short-Term; Mushroom Bodies; Mutation; Neuronal Plasticity; Receptors, GABA; Signal Transduction; Synapses | 2013 |
Phosphodiesterase 10A controls D1-mediated facilitation of GABA release from striato-nigral projections under normal and dopamine-depleted conditions.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Colforsin; Corpus Striatum; Dopamine; Dopamine Agonists; Drug Interactions; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Mice; Neural Pathways; Oxidopamine; Papaverine; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Phosphorylation; Potassium; Receptors, Dopamine D1; Substantia Nigra | 2014 |
Contribution of adenylyl cyclase modulation of pre- and postsynaptic GABA neurotransmission to morphine antinociception and tolerance.
Topics: Adenine; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Analgesics, Opioid; Animals; Bicuculline; Colforsin; Drug Tolerance; Enzyme Activators; Enzyme Inhibitors; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; Inhibitory Postsynaptic Potentials; Male; Miniature Postsynaptic Potentials; Morphine; Nociception; Presynaptic Terminals; Rats, Sprague-Dawley; Receptors, GABA-A; Synaptic Transmission | 2014 |
cAMP-dependent insulin modulation of synaptic inhibition in neurons of the dorsal motor nucleus of the vagus is altered in diabetic mice.
Topics: Animals; Brain Stem; Brefeldin A; Colforsin; Cyclic AMP; Diabetes Mellitus, Experimental; Diabetes Mellitus, Type 1; Electric Stimulation; Female; gamma-Aminobutyric Acid; Glucose Transporter Type 4; Golgi Apparatus; Indinavir; Inhibitory Postsynaptic Potentials; Insulin; Male; Mice; Neural Inhibition; Protein Transport; Synaptic Transmission; Vagus Nerve | 2014 |
Airway Epithelial Cell Release of GABA is Regulated by Protein Kinase A.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Bronchoalveolar Lavage Fluid; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Enzyme Activators; Epithelial Cells; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Guanine Nucleotide Exchange Factors; Humans; Male; Methacholine Chloride; Mice; Mice, Inbred C57BL; Myocytes, Smooth Muscle; Platelet-Derived Growth Factor; Propranolol; Receptor Protein-Tyrosine Kinases; Respiratory Mucosa; Rifabutin; RNA, Messenger; Signal Transduction; Terbutaline | 2016 |
The upregulation of glutamate decarboxylase 67 against hippocampal excitability damage in male fetal rats by prenatal caffeine exposure.
Topics: Adenylyl Cyclases; Animals; Brain-Derived Neurotrophic Factor; Caffeine; Colforsin; Female; gamma-Aminobutyric Acid; Glutamate Decarboxylase; Glutamic Acid; Hippocampus; Hypothalamo-Hypophyseal System; Male; Pituitary-Adrenal System; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Rats, Wistar; Receptor, Adenosine A2A; Up-Regulation | 2022 |