Page last updated: 2024-08-23

colforsin and diazepam

colforsin has been researched along with diazepam in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19903 (23.08)18.7374
1990's7 (53.85)18.2507
2000's2 (15.38)29.6817
2010's1 (7.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Hashemi, FS; Niles, LP1
Adler-Graschinsky, E; Elgoyhen, B1
Kojima, I; Ogata, E; Shibata, H1
Collado, MC; Hernández, J; Martinez, E; Peñafiel, R1
Chapal, J; Loubatières-Mariani, MM; Manteghetti, M; Petit, P1
Neu, JM; Niles, LP; Tenn, CC1
Niles, LP; Tenn, CC1
Chugun, A; Gomi, H; Hara, Y; Kaigo, H; Kondo, H; Minami, I; Nishimura, H; Watanabe, H1
Niles, LP; Wang, J1
Fuentes, T; Galindo, A; García Estañ, J; Hernández, J; Vargas, ML1
Fukuda, K; Hashiguchi, M; Hisano, T; Iwasaki, Y; Sato, M; Segawa, H; Uetsuki, N; Uga, H1

Other Studies

13 other study(ies) available for colforsin and diazepam

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
Pharmacological inhibition of forskolin-stimulated adenylate cyclase activity in rat brain by melatonin, its analogs, and diazepam.
    Biochemical pharmacology, 1990, Dec-15, Volume: 40, Issue:12

    Topics: Adenylyl Cyclases; Animals; Benzodiazepinones; Brain; Brain Mapping; Cell Membrane; Colforsin; Corpus Striatum; Diazepam; Dose-Response Relationship, Drug; Enzyme Activation; Flumazenil; In Vitro Techniques; Male; Melatonin; Rats; Rats, Inbred Strains

1990
Diminution by benzodiazepines of the chronotropic responses to noradrenaline in rat isolated atria.
    European journal of pharmacology, 1989, May-30, Volume: 164, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Anti-Anxiety Agents; Benzodiazepinones; Clonazepam; Colforsin; Cyclic AMP; Diazepam; Female; Flumazenil; Heart; Heart Rate; In Vitro Techniques; Isoquinolines; Male; Myocardium; Norepinephrine; Rats; Rats, Inbred Strains

1989
Diazepam inhibits potassium-induced aldosterone secretion in adrenal glomerulosa cell.
    Biochemical and biophysical research communications, 1986, Mar-28, Volume: 135, Issue:3

    Topics: Adrenal Glands; Aldosterone; Animals; Cattle; Colforsin; Diazepam; Dose-Response Relationship, Drug; Potassium; Receptors, GABA-A; Secretory Rate

1986
Diazepam potentiates the positive inotropic effect of isoprenaline in rat ventricle strips: role of cyclic AMP.
    European journal of pharmacology, 1995, Aug-25, Volume: 282, Issue:1-3

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Bucladesine; Cardiotonic Agents; Colforsin; Cyclic AMP; Diazepam; Drug Synergism; Electric Stimulation; Female; Heart Ventricles; In Vitro Techniques; Isoproterenol; Male; Rats; Rats, Sprague-Dawley

1995
[Research of the mechanism of the inhibition of insulin secretion induced by a peripheral benzodiazepine: 4'-chlordiazepam].
    Comptes rendus des seances de la Societe de biologie et de ses filiales, 1993, Volume: 187, Issue:4

    Topics: Animals; Bucladesine; Colforsin; Convulsants; Diazepam; Insulin; Insulin Antagonists; Insulin Secretion; Islets of Langerhans; Male; Rats; Rats, Wistar; Theophylline

1993
PK 11195 blockade of benzodiazepine-induced inhibition of forskolin-stimulated adenylate cyclase activity in the striatum.
    British journal of pharmacology, 1996, Volume: 119, Issue:2

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Benzodiazepines; Benzodiazepinones; Colforsin; Corpus Striatum; Diazepam; Drug Interactions; Flumazenil; GABA-A Receptor Antagonists; Guanosine Triphosphate; Indoles; Isoquinolines; Kinetics; Male; Pertussis Toxin; Rats; Rats, Sprague-Dawley; Stimulation, Chemical; Virulence Factors, Bordetella

1996
Sensitization of G protein-coupled benzodiazepine receptors in the striatum of 6-hydroxydopamine-lesioned rats.
    Journal of neurochemistry, 1997, Volume: 69, Issue:5

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Colforsin; Corpus Striatum; Diazepam; GTP-Binding Proteins; Guanosine Triphosphate; Kinetics; Male; Oxidopamine; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, GABA-A; Signal Transduction; Substantia Nigra; Tritium

1997
Diazepam potentiates the positive inotropic effects of histamine and forskolin in guinea-pig papillary muscles.
    Journal of veterinary pharmacology and therapeutics, 1998, Volume: 21, Issue:5

    Topics: Anesthetics, Intravenous; Animals; Colforsin; Cyclic AMP; Diazepam; Drug Interactions; Guinea Pigs; Histamine; Myocardial Contraction; Papillary Muscles; Stimulation, Chemical

1998
Diazepam inhibits forskolin-stimulated adenylyl cyclase activity in human tumour cells.
    Pharmacology & toxicology, 1999, Volume: 85, Issue:4

    Topics: Adenylyl Cyclase Inhibitors; Anti-Anxiety Agents; Breast Neoplasms; Cell Membrane; Colforsin; Diazepam; Dose-Response Relationship, Drug; Drug Interactions; Humans; Melanoma; Tumor Cells, Cultured

1999
Synergistic interaction of diazepam with 3',5'-cyclic adenosine monophosphate-elevating agents on rat aortic rings.
    European journal of pharmacology, 2001, Oct-05, Volume: 428, Issue:2

    Topics: Animals; Aorta, Thoracic; Colforsin; Cyclic AMP; Diazepam; Dose-Response Relationship, Drug; Drug Synergism; Enzyme Inhibitors; Female; Flumazenil; GABA Modulators; gamma-Aminobutyric Acid; In Vitro Techniques; Isoproterenol; Isoquinolines; Male; Milrinone; Muscle Relaxants, Central; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Phenylephrine; Rats; Rats, Sprague-Dawley; Vasoconstriction; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

2001
Potentiation of proopiomelanocortin gene expression in cultured pituitary cells by benzodiazepines.
    Anesthesiology, 2003, Volume: 98, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Anti-Anxiety Agents; Cells, Cultured; Colforsin; Diazepam; Gene Expression Regulation; Genes, Reporter; Kinetics; Luciferases; Mice; Midazolam; Pro-Opiomelanocortin; Transfection

2003