colforsin has been researched along with clonidine in 83 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 25 (30.12) | 18.7374 |
1990's | 46 (55.42) | 18.2507 |
2000's | 11 (13.25) | 29.6817 |
2010's | 1 (1.20) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Cuddon, P; Fleming, A; Floto, RA; Goldsmith, P; Jahreiss, L; O'Kane, CJ; Pask, D; Rubinsztein, DC; Saiki, S; Sarkar, S; Siddiqi, FH; Ttofi, EK; Williams, A | 1 |
Bradley, ME; Buxton, IL; Keef, KD; Zhang, L | 1 |
Arner, P; Hellmér, J; Marcus, C; Sonnenfeld, T | 1 |
Chan, CB; MacPhail, RM | 1 |
Lin, W; McCook, EC; Seidler, FJ; Slotkin, TA | 1 |
Cheng, JT; Tsai, LH | 1 |
Arner, P; Engfeldt, P; Goldinger, M; Marcus, C | 1 |
McCook, EC; Nemeroff, CB; Seidler, FJ; Slotkin, TA | 1 |
Evinger, MJ; Meeley, MP; Regunathan, S; Reis, DJ | 1 |
Ball, SG; Ong, ML; Vaughan, PF | 1 |
Mori-Okamoto, J; Namii, Y; Tatsuno, J | 1 |
Amiel, C; Bernard, C; Ferrary, E; Friedlander, G; Sterkers, O | 1 |
Burnham, BL; Chick, WL; Clark, SA | 1 |
Osborne, NN | 1 |
Silverman, PB; Steketee, JD; Swann, AC | 1 |
Allard, WJ; Saperstein, R; Slater, EE; Strout, HV; Vicario, PP | 1 |
Cepelík, J; Hynie, S | 2 |
Breuiller, M; Ferré, F; Leroy, MJ; Litime, MH; Rouot, B | 1 |
Burton, MD; Johnson, DC; Kazemi, H | 1 |
Mulder, AH; Schoffelmeer, AN; Wierenga, EA | 1 |
Mobley, PL; Northam, WJ | 1 |
Shaikh, IM; Skala, JP | 1 |
Giudicelli, Y; Leneveu, MC; Pecquery, R | 1 |
Kilbinger, H; Racké, K; Schwörer, H | 1 |
Kotecha, N; Neild, TO | 1 |
Steketee, JD; Swann, AC | 1 |
Hariharan, S; Phillippe, M; Saunders, T | 1 |
García-Sáinz, JA; Martínez, OM | 1 |
Ullrich, S; Wollheim, CB | 2 |
Burnside, B; Dearry, A | 1 |
Ambrosini, A; Gatti, G; Meldolesi, J; Pozzan, T; Westhead, EW | 1 |
Bylund, DB; Ray-Prenger, C; Turner, JT | 1 |
Collin, JP; Martin, C; Voisin, P | 1 |
Baes, M; Denef, C; Swennen, L | 1 |
Edvinsson, L; Fredholm, BB; Jansen, I | 1 |
Neubig, RR; Szamraj, O | 1 |
Kawai, M; Kitamura, Y; Nomura, Y; Segawa, T | 1 |
Mulder, AH; Putters, J; Schoffelmeer, AN | 1 |
Burns, TW; Bylund, DB; Forte, LR; Langley, PE; Terry, BE | 1 |
Kawata, K; Kitamura, Y; Nomura, Y; Watanabe, H | 1 |
Biondi, C; Borasio, PG; Capuzzo, A; Ferretti, ME; Trevisani, A | 1 |
Dufrane, SP; Garcia-Morales, P; Malaisse, WJ; Sener, A; Valverde, I | 1 |
McMahon, KK; Schimmel, RJ | 1 |
Ogihara, M | 1 |
Bertaccini, G; Coruzzi, G; Poli, E; Pozzoli, C | 1 |
Jumblatt, JE | 1 |
Bausher, LP; Horio, B | 1 |
Arilla, E; Guijarro, LG; López-Sañudo, S; Prieto, JC; Puebla, L | 1 |
Pyne, NJ; Stevens, PA | 1 |
Aarab, L; Chabardès, D; Siaume-Perez, S | 1 |
Akerman, KE; Jansson, CC; Savola, JM | 1 |
Ernsberger, P; Furin, J; Liedtke, CM | 1 |
Aston-Jones, G; Shiekhattar, R | 1 |
Lo, SJ; Shih, YL | 1 |
Agresti, C; Bernardo, A; Levi, G; Patrizio, M; Petrucci, TC | 1 |
Brunner, HR; Grouzmann, E; Nicod, P; Thompson, N; Waeber, B; Waeber, G | 1 |
Bolaffi, JL; Grodsky, GM; Ma, YH; Rodd, GG | 1 |
Bausher, L; Horio, B; Matsui, H; Mead, A; Sears, M | 1 |
Arner, P; Dauzats, M; Hellström, L; Langin, D; Reynisdottir, S | 1 |
Lundquist, I; Salehi, A | 1 |
Arner, P; Hellström, L; Reynisdottir, S; Wahrenberg, H | 1 |
Deuson, TE; Sellke, FW; Stamler, A; Tofukuji, M; Wang, SY | 1 |
Hagström-Toft, E; Hellström, L; Reynisdottir, S; Rössner, S | 1 |
Gregory, DS; Hirota, A; Kiuchi, Y; Nii, H | 1 |
Robinson, NE; Zhang, XY; Zhu, FX | 1 |
Arrizurieta, E; Bertuccio, C; Ibarra, FR; Martin, RS; Paz, L; Pignataro, O; Toledo, J | 1 |
Coca-Prados, M; Ortego, J | 1 |
Akaike, N; Li, JS; Nabekura, J; Rhee, JS; Xu, TL | 1 |
Adachi, T; Nakao, S; Shingu, K; Shinomura, T | 1 |
Bobirnac, I; Gazi, L; Loetscher, E; Parsley, S; Schoeffter, P | 1 |
Kitazawa, T; Maezono, Y; Taneike, T | 1 |
Fujimoto, S; Hamamoto, Y; Ishida, H; Kajikawa, M; Mukai, E; Seino, Y; Takeda, T; Tsuji, K; Tsuura, Y; Yamada, Y | 1 |
Sugimoto, M; Uchida-Oka, N | 1 |
Alarcón, P; García-Sancho, J; Núñez, L | 1 |
Auman, JT; Seidler, FJ; Slotkin, TA; Tate, CA | 1 |
Greger, R; Herbst, M; Hescheler, J; Sasse, P; Ullrich, S; Yu, H | 1 |
Azad, SC; DeBock, F; Hapfelmeier, G; Kurz, J; Parsons, CG; Rammes, G; Zieglgänsberger, W | 1 |
Eglen, RM; Kendall, DA; Maclennan, SJ; Pinthong, D; Wilson, VG | 1 |
Beck, DR; Buvanendran, A; Kroin, JS; Topic, JE; Tuman, KJ; Watts, DE | 1 |
Cozzi, RR; Hovdestad, LR; Katoh, F; Marshall, WS; Watters, KD | 1 |
Bylund, DB; Montgomery, MD | 1 |
83 other study(ies) available for colforsin and clonidine
Article | Year |
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Novel targets for Huntington's disease in an mTOR-independent autophagy pathway.
Topics: Animals; Autophagy; Calcium Channels, L-Type; Clonidine; Cyclic AMP; Humans; Huntington Disease; Imidazoline Receptors; Minoxidil; Protein Kinases; Signal Transduction; TOR Serine-Threonine Kinases; Type C Phospholipases; Verapamil | 2008 |
Action of alpha 2A-adrenergic receptors in circular smooth muscle of canine proximal colon.
Topics: Adenylate Cyclase Toxin; Animals; Binding, Competitive; Cell Membrane; Clonidine; Colforsin; Colon; Dogs; Epinephrine; Female; In Vitro Techniques; Isoproterenol; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Oxymetazoline; Pertussis Toxin; Prazosin; Receptors, Adrenergic, alpha; Tetrodotoxin; Virulence Factors, Bordetella; Yohimbine | 1992 |
Mechanisms for differences in lipolysis between human subcutaneous and omental fat cells.
Topics: Abdomen; Adenosine Deaminase; Adipose Tissue; Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Bucladesine; Catecholamines; Clonidine; Colforsin; Dose-Response Relationship, Drug; Female; Humans; Lipolysis; Male; Middle Aged; Norepinephrine; Omentum; Radioligand Assay; Receptors, Adrenergic, beta; Skin; Xanthines | 1992 |
Functional characterization of alpha-adrenoceptors on pancreatic islets of fa/fa Zucker rats.
Topics: Animals; Cells, Cultured; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Epinephrine; Female; Glucose; Insulin; Islets of Langerhans; Obesity; Prazosin; Rats; Rats, Zucker; Receptors, Adrenergic, alpha; Yohimbine | 1992 |
Overexpression of alpha 2-adrenergic receptors in fetal rat heart: receptors in search of a function.
Topics: Adenylyl Cyclases; Animals; Animals, Newborn; Clonidine; Colforsin; Fetal Heart; Gestational Age; In Vitro Techniques; Isoproterenol; Myocardium; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Yohimbine | 1992 |
Pharmacological characterization of alpha 2-adrenoceptors in isolated jejunum of rabbits.
Topics: Animals; Clonidine; Colforsin; GTP-Binding Proteins; Guanabenz; In Vitro Techniques; Jejunum; Muscle Contraction; Norepinephrine; Rabbits; Receptors, Adrenergic, alpha | 1992 |
Effects of lipolytic and antilipolytic agents on glucose transport in human fat cells.
Topics: Adenylyl Cyclase Inhibitors; Adipose Tissue; Anti-Inflammatory Agents, Non-Steroidal; Biological Transport; Bucladesine; Cells, Cultured; Clonidine; Colforsin; Dinoprostone; Dose-Response Relationship, Drug; Drug Interactions; Glucose; Humans; Insulin; Lipolysis; Niacin; Phenylisopropyladenosine; Xanthines | 1991 |
Species differences in alpha 2-adrenergic regulation of platelet adenylate cyclase.
Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adult; Alprostadil; Animals; Blood Platelets; Clonidine; Colforsin; Down-Regulation; Humans; Male; Rabbits; Radioimmunoassay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Species Specificity; Statistics as Topic; Yohimbine | 1991 |
Effects of clonidine and other imidazole-receptor binding agents on second messenger systems and calcium influx in bovine adrenal chromaffin cells.
Topics: Adrenal Glands; Animals; Calcium; Cattle; Cells, Cultured; Clonidine; Colforsin; Cyclic AMP; Cyclic GMP; Inositol Phosphates; Receptors, Drug; Second Messenger Systems; Signal Transduction | 1991 |
Regulation of noradrenaline release from rat occipital cortex tissue chops by alpha 2-adrenergic agonists.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Brimonidine Tartrate; Bucladesine; Clonidine; Colforsin; Cyclic AMP; Histological Techniques; Male; Norepinephrine; Occipital Lobe; Quinoxalines; Rats; Rats, Inbred Strains | 1991 |
Subtypes of adrenergic receptors and intracellular mechanisms involved in modulatory effects of noradrenaline on glutamate.
Topics: Acebutolol; Albuterol; Animals; Cells, Cultured; Cerebellum; Chick Embryo; Clonidine; Colforsin; Electric Conductivity; Ethanolamines; Glutamates; Glutamic Acid; Isoproterenol; Membrane Potentials; Neurons; Norepinephrine; Prazosin; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Tolazoline; Yohimbine | 1991 |
Antidiuretic hormone stimulation of adenylate cyclase in semicircular canal epithelium.
Topics: Adenylyl Cyclases; Adrenergic alpha-Agonists; Animals; Calcitonin; Clonidine; Colforsin; Cyclic AMP; Dinoprostone; Endolymph; Epithelium; Glucagon; Isoproterenol; Norepinephrine; Organ Culture Techniques; Parathyroid Hormone; Rana esculenta; Semicircular Canals; Vasopressins; Vasotocin | 1991 |
Modulation of glucose-induced insulin secretion from a rat clonal beta-cell line.
Topics: 1-Methyl-3-isobutylxanthine; Alanine; Animals; Carbachol; Cell Line; Clone Cells; Clonidine; Colforsin; Dose-Response Relationship, Drug; Glucose; Glyburide; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Potassium; Rats; Stereoisomerism | 1990 |
Inhibition of cAMP production by alpha 2-adrenoceptor stimulation in rabbit retina.
Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Clonidine; Colforsin; Cyclic AMP; GTP-Binding Proteins; In Vitro Techniques; Pertussis Toxin; Phosphoric Diester Hydrolases; Quinoxalines; Rabbits; Retina; Vasoactive Intestinal Peptide; Virulence Factors, Bordetella | 1991 |
Noradrenergic receptor mechanisms in neophobia.
Topics: Adenylyl Cyclases; Animals; Anxiety; Behavior, Animal; Clonidine; Colforsin; Dopamine beta-Hydroxylase; Environment; Isoproterenol; Male; Norepinephrine; Oxidopamine; Phenylephrine; Prosencephalon; Rats; Rats, Inbred Strains; Receptors, Adrenergic | 1992 |
The function but not the expression of rat liver inhibitory guanine nucleotide binding protein is altered in streptozotocin-induced diabetes.
Topics: Adenylyl Cyclases; Amino Acid Sequence; Animals; Antibody Specificity; Cell Membrane; Clonidine; Colforsin; Diabetes Mellitus, Experimental; GTP-Binding Proteins; Immunoblotting; Liver; Male; Molecular Sequence Data; Molecular Weight; Rats | 1991 |
Inhibitory effects of clonidine and dopamine on adenylate cyclase of rabbit ciliary processes.
Topics: Adenylyl Cyclase Inhibitors; Animals; Ciliary Body; Clonidine; Colforsin; Dopamine; In Vitro Techniques; Isoproterenol; Rabbits; Receptors, Adrenergic, alpha | 1990 |
Functional coupling of the alpha 2-adrenergic receptor-adenylate cyclase complex in the pregnant human myometrium.
Topics: Adenosine Diphosphate Ribose; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Adult; Binding, Competitive; Clonidine; Colforsin; Cyclic AMP; Dioxanes; Drug Interactions; Electrophoresis, Polyacrylamide Gel; Female; GTP-Binding Proteins; Humans; Idazoxan; Myometrium; Norepinephrine; Pertussis Toxin; Pregnancy; Pregnancy Trimester, Third; Receptors, Adrenergic, alpha; Virulence Factors, Bordetella; Yohimbine | 1990 |
Adrenergic and cholinergic interaction in central ventilatory control.
Topics: Acetylcholine; Animals; Atropine; Cardiovascular Physiological Phenomena; Cardiovascular System; Clonidine; Colforsin; Cyclic AMP; Dogs; Isoproterenol; Medulla Oblongata; Propanolamines; Receptors, Adrenergic; Receptors, Cholinergic; Respiration; Respiratory Center; Second Messenger Systems; Yohimbine | 1990 |
Inhibitory effects of neuropeptide Y on adenylate cyclase of rabbit ciliary processes.
Topics: Adenylyl Cyclase Inhibitors; Animals; Ciliary Body; Clonidine; Colforsin; Isoproterenol; Neuropeptide Y; Rabbits; Vasoactive Intestinal Peptide | 1990 |
Role of adenylate cyclase in presynaptic alpha 2-adrenoceptor- and mu-opioid receptor-mediated inhibition of [3H]noradrenaline release from rat brain cortex slices.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Animals; Bucladesine; Cadmium; Calcimycin; Cerebral Cortex; Clonidine; Colforsin; Cyclic AMP; Electric Stimulation; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Morphine; Norepinephrine; Phentolamine; Pyrrolidinones; Rats; Receptors, Adrenergic, alpha; Receptors, Opioid; Receptors, Opioid, mu; Rolipram | 1986 |
Clonidine inhibits the isoproterenol-induced desensitization of the beta noradrenergic activated adenylate cyclase system in astrocytes.
Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Astrocytes; Clonidine; Colforsin; Cyclic AMP; Enzyme Activation; Isoproterenol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1987 |
Alpha 2-adrenergic receptors in brown adipose tissue of infant rats--II. Studies on function and regulation.
Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adipose Tissue, Brown; Animals; Clonidine; Colforsin; Hydroxydopamines; Kinetics; Lipolysis; Oxidopamine; Pertussis Toxin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Sympathectomy, Chemical; Virulence Factors, Bordetella; Yohimbine | 1988 |
Influence of androgenic status on the alpha 2/beta-adrenergic control of lipolysis in white fat cells: predominant alpha 2-antilipolytic response in testosterone-treated-castrated hamsters.
Topics: 1-Methyl-3-isobutylxanthine; Adipose Tissue; Animals; Brimonidine Tartrate; Clonidine; Colforsin; Cricetinae; Cyclic AMP; Epinephrine; Isoproterenol; Lipolysis; Male; Mesocricetus; Niacin; Orchiectomy; Phentolamine; Propranolol; Quinoxalines; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Testosterone | 1988 |
Adrenergic modulation of the release of 5-hydroxytryptamine from the vascularly perfused ileum of the guinea-pig.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Clonidine; Colforsin; Guinea Pigs; Hydroxyindoleacetic Acid; Ileum; Isoproterenol; Male; Naphthyridines; Perfusion; Phosphodiesterase Inhibitors; Serotonin | 1988 |
A study of the phasic response of arterioles of the guinea pig small intestine to prolonged exposure to norepinephrine.
Topics: 1-Methyl-3-isobutylxanthine; 8-Bromo Cyclic Adenosine Monophosphate; Animals; Arterioles; Clonidine; Colforsin; Cyclic GMP; Dose-Response Relationship, Drug; Guinea Pigs; Intestine, Small; Isoproterenol; Membrane Potentials; Norepinephrine; Oxidation-Reduction; Propranolol; Temperature; Theophylline; Vasoconstriction; Yohimbine | 1989 |
Subacute noradrenergic agonist infusions in vivo increase Na+, K+-ATPase and ouabain binding in rat cerebral cortex.
Topics: Animals; Brain; Cerebral Cortex; Clonidine; Colforsin; Hydroxydopamines; Isoproterenol; Male; Norepinephrine; Ouabain; Oxidopamine; Phenylephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Sodium-Potassium-Exchanging ATPase | 1989 |
Absence of alpha-2 adrenergic effects on cAMP production in a genital tract smooth muscle cell line.
Topics: Animals; Cell Line, Transformed; Clonidine; Colforsin; Cricetinae; Cyclic AMP; Epinephrine; Genital Neoplasms, Male; Isoproterenol; Leiomyosarcoma; Male; Muscle, Smooth; Norepinephrine; Propranolol; Receptors, Adrenergic, alpha; Tumor Cells, Cultured; Vas Deferens | 1989 |
Functional alpha 2-adrenoceptors in rat adipocytes: inhibition of cyclic AMP accumulation.
Topics: Adenylate Cyclase Toxin; Adipose Tissue; Animals; Brimonidine Tartrate; Clonidine; Colforsin; Cricetinae; Cyclic AMP; Male; Pertussis Toxin; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Virulence Factors, Bordetella | 1989 |
GTP-dependent inhibition of insulin secretion by epinephrine in permeabilized RINm5F cells. Lack of correlation between insulin secretion and cyclic AMP levels.
Topics: Adenylate Cyclase Toxin; Calcium; Cell Line; Cell Membrane Permeability; Clonidine; Colforsin; Cyclic AMP; Epinephrine; Ethers; Guanosine Triphosphate; Insulin; Insulin Secretion; Ionomycin; Kinetics; Models, Biological; Pertussis Toxin; Propranolol; Virulence Factors, Bordetella | 1988 |
Stimulation of distinct D2 dopaminergic and alpha 2-adrenergic receptors induces light-adaptive pigment dispersion in teleost retinal pigment epithelium.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Benzazepines; Clonidine; Colforsin; Dopamine; Ergolines; Fishes; Light; Pigment Epithelium of Eye; Quinpirole; Receptors, Adrenergic, alpha; Receptors, Dopamine; Receptors, Dopamine D2; Retinal Pigments | 1988 |
Second-messenger control of catecholamine release from PC12 cells. Role of muscarinic receptors and nerve-growth-factor-induced cell differentiation.
Topics: Adrenal Gland Neoplasms; Animals; Carbachol; Catecholamines; Cell Differentiation; Clonidine; Colforsin; Cyclic AMP; Dopamine; Ethers; Ionomycin; Nerve Growth Factors; Pheochromocytoma; Phorbol Esters; Potassium; Rats; Receptors, Muscarinic; Tumor Cells, Cultured | 1988 |
Alpha 2-adrenergic receptors in the human cell line, HT29. Characterization with the full agonist radioligand [3H]UK-14,304 and inhibition of adenylate cyclase.
Topics: Adenocarcinoma; Adenylyl Cyclase Inhibitors; Adrenergic alpha-Agonists; Brimonidine Tartrate; Cell Line; Clonidine; Colforsin; Colonic Neoplasms; Dose-Response Relationship, Drug; Guanosine Triphosphate; Humans; Kinetics; Magnesium; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha; Vasoactive Intestinal Peptide; Yohimbine | 1985 |
Alpha 2-adrenergic regulation of arylalkylamine N-acetyltransferase in organ-cultured chick pineal gland: characterization with agonists and modulation of experimentally stimulated enzyme activity.
Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Acetyltransferases; Adrenergic alpha-Agonists; Animals; Arylamine N-Acetyltransferase; Bucladesine; Chickens; Cholera Toxin; Circadian Rhythm; Clonidine; Colforsin; Organ Culture Techniques; Pineal Gland; Potassium Chloride; Receptors, Adrenergic, alpha | 1987 |
Beta-adrenergic stimulation of adenosine-3',5'-monophosphate (c-AMP) accumulation and of prolactin and growth hormone secretion in rat anterior pituitary cell cultures.
Topics: Animals; Cells, Cultured; Clonidine; Colforsin; Cyclic AMP; Dexamethasone; Diterpenes; Female; Growth Hormone; Isoproterenol; Pituitary Gland, Anterior; Prolactin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta | 1985 |
Neuropeptide Y is a potent inhibitor of cyclic AMP accumulation in feline cerebral blood vessels.
Topics: Animals; Cats; Cerebral Arteries; Clonidine; Colforsin; Cyclic AMP; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Nerve Tissue Proteins; Neuropeptide Y; Vascular Resistance | 1985 |
Large-scale purification of alpha 2-adrenergic receptor-enriched membranes from human platelets. Persistent association of guanine nucleotides with nonpurified membranes.
Topics: Adenylyl Cyclases; Blood Platelets; Cell Fractionation; Cell Membrane; Centrifugation, Density Gradient; Clonidine; Colforsin; Epinephrine; Guanosine Diphosphate; Guanosine Triphosphate; Humans; Norepinephrine; Receptors, Adrenergic, beta; Tritium; Yohimbine | 1986 |
Alpha 2-adrenoceptor-GTP binding regulatory protein-adenylate cyclase system in cerebral cortical membranes of adult and senescent rats.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Aging; Animals; Cerebral Cortex; Clonidine; Colforsin; Epinephrine; Female; GTP-Binding Proteins; Guanosine Triphosphate; Kinetics; Male; Membranes; NAD; Pertussis Toxin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Virulence Factors, Bordetella | 1986 |
Activation of presynaptic alpha 2-adrenoceptors attenuates the inhibitory effect of mu-opioid receptor agonists on noradrenaline release from brain slices.
Topics: Animals; Brain Chemistry; Cadmium; Clonidine; Colforsin; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; In Vitro Techniques; Male; Morphine; Norepinephrine; Phentolamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Opioid; Receptors, Opioid, mu | 1986 |
Comparative effects of forskolin and isoproterenol on the cyclic AMP content of human adipocytes.
Topics: Adipose Tissue; Clonidine; Colforsin; Cyclic AMP; Epinephrine; Humans; Isoproterenol | 1987 |
Effects of pertussis toxin on the alpha 2-adrenoceptor-inhibitory GTP-binding protein-adenylate cyclase system in rat brain: pharmacological and neurochemical studies.
Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Brain Chemistry; Clonidine; Colforsin; Epinephrine; GTP-Binding Proteins; Injections, Intraventricular; Kinetics; Male; Motor Activity; Pertussis Toxin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Virulence Factors, Bordetella | 1987 |
Modulation of synaptic transmission in mammalian sympathetic ganglia: effects of catecholamines, prostaglandins and cyclic nucleotides.
Topics: Animals; Catecholamines; Clonidine; Colforsin; Cyclic AMP; Dinoprostone; Diterpenes; Enkephalin, Methionine; Ganglia, Sympathetic; Guinea Pigs; Kinetics; Phenylephrine; Prostaglandins E; Synaptic Transmission | 1984 |
Inhibitory effect of clonidine upon adenylate cyclase activity, cyclic AMP production, and insulin release in rat pancreatic islets.
Topics: Adenylyl Cyclases; Animals; Clonidine; Colforsin; Cyclic AMP; Diterpenes; Insulin; Insulin Secretion; Islets of Langerhans; Rats; Secretory Rate | 1984 |
Islet cyclic AMP levels are not lowered during alpha 2-adrenergic inhibition of insulin release.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Antihypertensive Agents; Clonidine; Colforsin; Cyclic AMP; Diterpenes; Epinephrine; Glucose; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Male; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Yohimbine | 1984 |
Inhibition of forskolin activated adenylate cyclase in hamster adipocyte membranes with prostaglandin E1 and clonidine.
Topics: Adenylyl Cyclases; Adipose Tissue; Alprostadil; Animals; Antihypertensive Agents; Cell Membrane; Clonidine; Colforsin; Cricetinae; Diterpenes; Enzyme Activation; Kinetics; Male; Mesocricetus; Prostaglandins E | 1982 |
Expression of alpha 2-receptor-mediated responses by insulin in primary culture of rat hepatocytes.
Topics: Animals; Cells, Cultured; Clonidine; Colforsin; Cyclic AMP; Cycloheximide; Drug Interactions; Glucagon; Glucose; Insulin; Liver; Male; Oxymetazoline; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Time Factors | 1995 |
Histamine H3-receptor-induced inhibition of duodenal cholinergic transmission is independent of intracellular cyclic AMP and GMP.
Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; Adenosine; Animals; Clonidine; Colforsin; Cyclic AMP; Cyclic GMP; Duodenum; Guinea Pigs; Histamine Agonists; In Vitro Techniques; Male; Methylhistamines; Parasympathetic Nervous System; Receptors, Histamine H3; Signal Transduction; Synaptic Transmission | 1993 |
Prejunctional alpha 2-adrenoceptors and adenylyl cyclase regulation in the rabbit iris-ciliary body.
Topics: Adenylyl Cyclases; Animals; Axons; Chromatography, High Pressure Liquid; Ciliary Body; Clonidine; Colforsin; Cyclic AMP; Ethylmaleimide; GTP-Binding Proteins; Iris; Rabbits; Receptors, Adrenergic, alpha-2; Signal Transduction; Sympathetic Nervous System; Tyrosine 3-Monooxygenase | 1994 |
Regulation of cyclic AMP production in adult human ciliary processes.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Child; Ciliary Body; Clonidine; Colforsin; Cyclic AMP; Endothelins; Humans; Isoproterenol; Stimulation, Chemical; Vasoactive Intestinal Peptide | 1995 |
Alpha-2 adrenoceptors modulate the somatostatinergic system and G protein levels in the rat hippocampus.
Topics: Adenosine Diphosphate; Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Clonidine; Colforsin; GTP-Binding Proteins; Hippocampus; Kinetics; Male; Membranes; Pertussis Toxin; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Somatostatin; Virulence Factors, Bordetella; Yohimbine | 1995 |
The inhibition of adenylyl cyclase activity in isolated lung membranes by muscarinic and alpha-adrenoceptor agonists: role of G-protein alpha and beta gamma sub-units.
Topics: Adenosine Diphosphate Ribose; Adenylyl Cyclase Inhibitors; Adrenergic alpha-Agonists; Animals; Cholera Toxin; Clonidine; Colforsin; GTP-Binding Proteins; Guanine Nucleotides; Guanylyl Imidodiphosphate; Guinea Pigs; In Vitro Techniques; Lung; Male; Membranes; Methacholine Chloride; Muscarinic Agonists; Norepinephrine; Protein Conformation | 1995 |
The activation of protein kinase C prevents PGE2-induced inhibition of AVP-dependent cAMP accumulation in the rat outer medullary collecting tubule.
Topics: Acetylcholine; Adrenergic alpha-Agonists; Animals; Arginine Vasopressin; Clonidine; Colforsin; Cyclic AMP; Dinoprostone; Enzyme Activation; Kidney Medulla; Kidney Tubules, Collecting; Male; Osmolar Concentration; Protein Kinase C; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate | 1993 |
Different sensitivity of alpha 2A-C10 and alpha 2C-C4 receptor subtypes in coupling to inhibition of cAMP accumulation.
Topics: Adenine; Adenylyl Cyclases; Adrenergic alpha-Antagonists; Clonidine; Colforsin; Cyclic AMP; Fibroblasts; Humans; Imidazoles; Kinetics; Medetomidine; Norepinephrine; Receptors, Adrenergic, alpha-2; Tetradecanoylphorbol Acetate; Transfection; Yohimbine | 1994 |
Alpha 2-adrenergic, but not imidazole, agonists activate NaCl cotransport in rabbit tracheal epithelial cells.
Topics: Adrenergic alpha-Agonists; Animals; Antihypertensive Agents; Carrier Proteins; Cells, Cultured; Chloride-Bicarbonate Antiporters; Clonidine; Colforsin; Cyclic AMP; Drug Interactions; Epithelial Cells; Epithelium; Guanabenz; Imidazoles; Imidazoline Receptors; Iodine Radioisotopes; Isoproterenol; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Receptors, Drug; Second Messenger Systems; Sodium Chloride Symporters; Symporters; Thromboxane-A Synthase; Trachea | 1993 |
Modulation of opiate responses in brain noradrenergic neurons by the cyclic AMP cascade: changes with chronic morphine.
Topics: Animals; Clonidine; Colforsin; Cyclic AMP; Drug Synergism; Endorphins; Locus Coeruleus; Morphine; Neurons; Norepinephrine; Rats; Rats, Sprague-Dawley; Time Factors | 1993 |
Induction of cell expansion of goldfish melanocytoma cells (GMM-1) by epinephrine and dexamethasone requires external calcium.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Calcium; Cell Line; Cell Size; Clonidine; Colforsin; Dexamethasone; Diglycerides; Egtazic Acid; Epinephrine; Goldfish; Melanoma; Nifedipine; Receptors, Adrenergic; Tumor Cells, Cultured; Yohimbine | 1993 |
Human immunodeficiency virus coat protein gp120 inhibits the beta-adrenergic regulation of astroglial and microglial functions.
Topics: Adenylyl Cyclases; Animals; Animals, Newborn; Astrocytes; Cells, Cultured; Cerebral Cortex; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Glial Fibrillary Acidic Protein; Glioma; HIV Envelope Protein gp120; Humans; Isoproterenol; Kinetics; Mesoderm; Phosphoproteins; Phosphorylation; Propranolol; Rats; Receptors, Adrenergic, beta; Recombinant Proteins; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha; Vimentin | 1993 |
Neuropeptide Y expression and regulation in a differentiated rat insulin-secreting cell line.
Topics: Adenylyl Cyclases; Animals; Cell Differentiation; Clonidine; Colforsin; Cyclic AMP; Enzyme Activation; Enzyme-Linked Immunosorbent Assay; Gene Expression Regulation, Neoplastic; Glucagon; Glucagon-Like Peptide 1; Glucagon-Like Peptides; Insulin; Insulin Secretion; Insulinoma; Neuropeptide Y; Pancreatic Neoplasms; Peptide Fragments; Protein Kinase C; Rats; Receptors, Neuropeptide Y; Tumor Cells, Cultured | 1993 |
Opposite, phase-dependent effects of 3,4,5-trimethoxybenzoic acid 8-(diethylamino) octyl ester or tetracaine on islet function during three phases of glucose-stimulated insulin secretion.
Topics: Animals; Clonidine; Colforsin; Gallic Acid; Glucose; Insulin; Insulin Secretion; Islets of Langerhans; Male; Pertussis Toxin; Rats; Tetracaine; Virulence Factors, Bordetella | 1993 |
Regulation and bioelectrical effects of cyclic adenosine monophosphate production in the ciliary epithelial bilayer.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Aqueous Humor; Ciliary Body; Clonidine; Colforsin; Cyclic AMP; Electrophysiology; Isoproterenol; Male; Membrane Potentials; Pigment Epithelium of Eye; Rabbits; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Timolol; Vasoactive Intestinal Peptide | 1996 |
Adipocyte lipolysis in normal weight subjects with obesity among first-degree relatives.
Topics: Adipocytes; Adrenergic beta-Agonists; Adult; Body Mass Index; Bucladesine; Clonidine; Colforsin; Diabetes Mellitus, Type 2; Dobutamine; Dose-Response Relationship, Drug; Female; Glycerol; Humans; Isoproterenol; Lipolysis; Male; Norepinephrine; Nuclear Family; Obesity; Pedigree; Receptors, Adrenergic, beta; RNA, Messenger; Sterol Esterase; Sympathomimetics; Terbutaline | 1996 |
Modulation of islet G-proteins, alpha-glucosidehydrolase inhibition and insulin release stimulated by various secretagogues.
Topics: 1-Deoxynojirimycin; 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic alpha-Agonists; Animals; Cholera Toxin; Clonidine; Colforsin; Enzyme Inhibitors; Female; Glucosamine; Glucose; Glycoside Hydrolases; GTP-Binding Proteins; In Vitro Techniques; Insulin; Insulin Secretion; Islets of Langerhans; Mannoheptulose; Mice; Pertussis Toxin; Phosphodiesterase Inhibitors; Protein Kinase C; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella | 1996 |
Catecholamine-induced adipocyte lipolysis in human hyperthyroidism.
Topics: Adipocytes; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adult; Bucladesine; Clonidine; Colforsin; Dobutamine; Female; Humans; Hyperthyroidism; Lipolysis; Male; Middle Aged; Norepinephrine; Receptors, Adrenergic, beta; Terbutaline | 1997 |
Effects of blood and crystalloid cardioplegia on adrenergic and myogenic vascular mechanisms.
Topics: Animals; Blood; Cardioplegic Solutions; Clonidine; Colforsin; Coronary Circulation; Coronary Vessels; Female; Heart Arrest, Induced; Isoproterenol; Male; Myocardial Contraction; Nitroprusside; Potassium Compounds; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta; Swine | 1997 |
Lipolytic catecholamine resistance linked to alpha 2-adrenoceptor sensitivity--a metabolic predictor of weight loss in obese subjects.
Topics: Adenosine Deaminase; Adipose Tissue; Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adult; Biomarkers; Biopsy; Clonidine; Cohort Studies; Colforsin; Dobutamine; Dose-Response Relationship, Drug; Female; Glycerol; Humans; Isoproterenol; Lipolysis; Middle Aged; Norepinephrine; Obesity; Receptors, Adrenergic, alpha; Terbutaline; Time Factors; Weight Loss | 1997 |
Response and level of beta-adrenergic, vasoactive intestinal peptide, and PACAP receptors during the circadian cycle.
Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Aqueous Humor; Ciliary Body; Circadian Rhythm; Clonidine; Colforsin; Cyclic AMP; Isoproterenol; Ligands; Male; Rabbits; Receptors, Adrenergic, beta; Receptors, Pituitary Adenylate Cyclase-Activating Polypeptide; Receptors, Pituitary Hormone; Vasoactive Intestinal Peptide | 1997 |
Role of cAMP and neuronal K+ channels on alpha 2-AR-induced inhibition of ACh release in equine trachea.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Adrenergic alpha-Agonists; Animals; Calcium; Charybdotoxin; Clonidine; Colforsin; Cyclic AMP; Electric Stimulation; Horses; Neurons; Peptides; Potassium Channel Blockers; Potassium Channels; Receptors, Adrenergic, alpha; Trachea | 1998 |
Regulation of cell cyclic AMP in medullary thick ascending limb of Henle in a rat model of chronic renal failure.
Topics: 1-Methyl-3-isobutylxanthine; Adrenergic alpha-Agonists; Animals; Calcitonin; Cell Separation; Clonidine; Colforsin; Creatinine; Cyclic AMP; Disease Models, Animal; Dose-Response Relationship, Drug; Glomerular Filtration Rate; In Vitro Techniques; Kidney Failure, Chronic; Loop of Henle; Male; Osmolar Concentration; Rats; Rats, Wistar; Vasopressins | 1998 |
Molecular identification and coexpression of galanin and GalR-1 galanin receptor in the human ocular ciliary epithelium: differential modulation of their expression by the activation of alpha2- and beta2-adrenergic receptors in cultured ciliary epithelial
Topics: Adrenergic alpha-Agonists; Aqueous Humor; Cell Line; Ciliary Body; Clonidine; Colforsin; Culture Media, Serum-Free; Epithelial Cells; Fluorescent Antibody Technique; Galanin; Humans; Norepinephrine; Protein Precursors; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta; Receptors, Galanin; Receptors, Neuropeptide; RNA, Messenger; Tetradecanoylphorbol Acetate | 1998 |
Alpha2-adrenoceptor-mediated enhancement of glycine response in rat sacral dorsal commissural neurons.
Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adrenergic alpha-Agonists; Animals; Bucladesine; Clonidine; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Electrophysiology; Glycine; Glycine Agents; GTP-Binding Proteins; Ion Channel Gating; Isoproterenol; Lumbosacral Region; Neurons, Afferent; Nociceptors; Norepinephrine; Pertussis Toxin; Phenylephrine; Phosphodiesterase Inhibitors; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Strychnine; Virulence Factors, Bordetella | 1999 |
Clonidine inhibits and phorbol acetate activates glutamate release from rat spinal synaptoneurosomes.
Topics: 4-Aminopyridine; Adrenergic alpha-Agonists; Animals; Calcium; Clonidine; Colforsin; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Activation; Glutamate Dehydrogenase; Glutamic Acid; In Vitro Techniques; Male; Potassium Chloride; Protein Kinase C; Rats; Rats, Wistar; Spectrometry, Fluorescence; Spinal Cord; Synaptosomes; Tetradecanoylphorbol Acetate | 1999 |
Functional alpha2C-adrenoceptors in human neuroblastoma SH-SY5Y cells.
Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Brimonidine Tartrate; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Guanfacine; Humans; Idazoxan; Isoquinolines; Neuroblastoma; Oxymetazoline; Piperazines; Prazosin; Quinoxalines; Receptors, Adrenergic, alpha-2; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tumor Cells, Cultured; Yohimbine | 1999 |
The mechanisms of alpha(2)-adrenoceptor agonist-induced contraction in longitudinal muscle of the porcine uterus.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Animals; Brimonidine Tartrate; Calcium; Calcium Channel Blockers; Clonidine; Colforsin; Cyclic AMP; Female; Fluorescent Dyes; Fura-2; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Myometrium; Pertussis Toxin; Quinoxalines; Swine; Uterus; Verapamil; Virulence Factors, Bordetella | 2000 |
Augmentation of basal insulin release from rat islets by preexposure to a high concentration of glucose.
Topics: Adenosine Triphosphate; Adrenergic alpha-Agonists; Animals; Calcium; Cell Membrane Permeability; Cells, Cultured; Clonidine; Colforsin; Diazoxide; Dose-Response Relationship, Drug; Electroporation; Glucose; Guanosine Diphosphate; Insulin; Insulin Secretion; Intracellular Fluid; Islets of Langerhans; Male; Mannoheptulose; Mycophenolic Acid; Oligomycins; Potassium; Rats; Rats, Wistar; Tetradecanoylphorbol Acetate; Thionucleotides | 2000 |
Norepinephrine induces apoptosis in skin melanophores by attenuating cAMP-PKA signals via alpha2-adrenoceptors in the medaka, Oryzias latipes.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Apoptosis; Clonidine; Colforsin; Culture Techniques; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cysteine Proteinase Inhibitors; Isoquinolines; Melanophores; Norepinephrine; Oligopeptides; Oryzias; Phenylephrine; Prazosin; Protein Isoforms; Receptors, Adrenergic, alpha-2; Signal Transduction; Skin; Skin Pigmentation; Sulfonamides; Yohimbine | 2001 |
Direct actions of adrenergic agents on rat anterior pituitary cells.
Topics: Adrenergic Agents; Adrenocorticotropic Hormone; Animals; Calcium; Cells, Cultured; Clonidine; Colforsin; Corticotropin-Releasing Hormone; Culture Media; Epinephrine; Follicle Stimulating Hormone; Growth Hormone; Growth Hormone-Releasing Hormone; Isoproterenol; Luteinizing Hormone; Male; Phenylephrine; Pituitary Gland, Anterior; Prazosin; Prolactin; Propranolol; Rats; Thyrotropin | 2001 |
Beta-adrenoceptor-mediated cell signaling in the neonatal heart and liver: responses to terbutaline.
Topics: Animals; Animals, Newborn; Body Weight; Clonidine; Colforsin; Down-Regulation; Female; GTP-Binding Proteins; Heart; Isoproterenol; Liver; Male; Membrane Proteins; Organ Size; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Signal Transduction; Sodium Fluoride; Terbutaline | 2001 |
Membrane potential dependent modulations of calcium oscillations in insulin-secreting INS-1 cells.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Calcium Signaling; Cell Line; Clonidine; Colforsin; Diazoxide; Enzyme Inhibitors; Epinephrine; Fluorescent Dyes; Fura-2; Glucose; Hypoglycemic Agents; Insulin; Insulin Secretion; Islets of Langerhans; Membrane Potentials; Mice; Patch-Clamp Techniques; Potassium Channels; Prazosin; Receptors, Adrenergic, alpha-2; Thapsigargin; Tolbutamide | 2002 |
Alpha2-adrenoreceptor activation inhibits LTP and LTD in the basolateral amygdala: involvement of Gi/o-protein-mediated modulation of Ca2+-channels and inwardly rectifying K+-channels in LTD.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclase Inhibitors; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Amygdala; Animals; Barium; Cadmium; Calcium Channel Blockers; Calcium Channels; Clonidine; Colforsin; Cyclic Nucleotide Phosphodiesterases, Type 4; Electric Stimulation; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Heterotrimeric GTP-Binding Proteins; Imines; In Vitro Techniques; Isoquinolines; Long-Term Potentiation; Long-Term Synaptic Depression; Membrane Potentials; Mice; Norepinephrine; omega-Agatoxin IVA; omega-Conotoxins; Patch-Clamp Techniques; Pertussis Toxin; Piperazines; Potassium Channel Blockers; Potassium Channels, Inwardly Rectifying; Pyridines; Receptors, Adrenergic, alpha-2; Serotonin Antagonists; Sulfonamides; Yohimbine | 2003 |
No evidence for activation of alpha(2)-adrenoceptors by methanolic extracts of bovine brain and lung containing clonidine-displacing substance.
Topics: Adrenergic alpha-Agonists; Animals; Brain Chemistry; Brimonidine Tartrate; Cattle; Clonidine; Colforsin; Cyclic AMP; Guinea Pigs; In Vitro Techniques; Lung; Male; Methanol; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Swine; Tissue Extracts; Vas Deferens; Veins | 2003 |
Clonidine prolongation of lidocaine analgesia after sciatic nerve block in rats Is mediated via the hyperpolarization-activated cation current, not by alpha-adrenoreceptors.
Topics: Adrenergic alpha-Agonists; Anesthetics, Local; Animals; Clonidine; Colforsin; Dose-Response Relationship, Drug; Drug Synergism; Epinephrine; In Vitro Techniques; Ion Channels; Lidocaine; Male; Nerve Block; Pyrimidines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha; Sciatic Nerve | 2004 |
CFTR Cl- channel functional regulation by phosphorylation of focal adhesion kinase at tyrosine 407 in osmosensitive ion transporting mitochondria rich cells of euryhaline killifish.
Topics: Animals; Clonidine; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Electrophysiology; Focal Adhesion Protein-Tyrosine Kinases; Fundulidae; Hypertonic Solutions; Hypotonic Solutions; Ion Transport; Isoproterenol; Microscopy, Electron, Transmission; Microscopy, Immunoelectron; Mitochondria; Phosphorylation; Protein Transport; Sympatholytics; Sympathomimetics; Tyrosine | 2009 |
Lack of effect of the alpha2C-adrenoceptor Del322-325 polymorphism on inhibition of cyclic AMP production in HEK293 cells.
Topics: Adenylyl Cyclases; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Binding, Competitive; Brimonidine Tartrate; Cell Line; Clonidine; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Activators; Humans; Linear Models; Norepinephrine; Polymorphism, Genetic; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha-2; Signal Transduction; Transfection | 2010 |