Page last updated: 2024-08-23

colforsin and carbostyril

colforsin has been researched along with carbostyril in 44 studies

Research

Studies (44)

TimeframeStudies, this research(%)All Research%
pre-19903 (6.82)18.7374
1990's9 (20.45)18.2507
2000's10 (22.73)29.6817
2010's19 (43.18)24.3611
2020's3 (6.82)2.80

Authors

AuthorsStudies
Hague, NL; Hunneyball, IM; Loh, E; Morgan, JP; Perreault, CL; Sim, MF1
Böhm, M; Erdmann, E; La Rosée, K; Schmidt, U; Schwinger, RH1
Andersson, KE; Lindgren, S1
Malik, KU; Williams, JL2
Andersson, KE; Belfrage, P; Degerman, E; Lindgren, S; Manganiello, VC1
Criscuoli, M; Del Monte, M; Subissi, A1
Arai, Y; Funayama, K; Kadowaki, S; Takahashi, K; Umezu, K; Yamada, N1
Imai, M; Shinkawa, T; Yamasaki, F; Yoshitomi, K1
Lee, HZ1
Maurice, DH; Palmer, D; Tsoi, K1
Carey, GB; Finnegan, RB1
Greenberg, AG; Kraemer, FB; Xue, B; Zemel, MB1
Absher, PM; Dunkerley, HA; Jimmo, SL; Maurice, DH; Netherton, SJ; Palmer, D; Raymond, DR; Russell, JC; Sage, EH; Tilley, DG; Vernon, RB1
Burris, KD; Kikuchi, T; Molinoff, PB; Molski, TF; Ryan, E; Tottori, K; Xu, C; Yocca, FD1
Kelly, C; Sawmiller, DR; Tarpey, SB; Thompson, WJ; Townsley, MI1
Guéguen, L; Laforest, MF; Pouliot, E; Richard, FJ1
Burris, KD; Kikuchi, T; Miwa, T; Mori, T; Stark, A; Tadori, Y; Tottori, K1
Carter, RL; Maurice, DH; Raymond, DR; Wilson, LS1
Ke, PQ; Liang, XY; Ren, Z; Shen, HW; Shu, YM; Wang, NN; Yao, SZ; Zeng, HT; Zhuang, GL1
Kawago, K; Matsuda, K; Nishio, T; Sano, Y; Uchiyama, M; Yamada, T1
Hayashi, H; Sudo, T1
Fujimaki-Aoba, K; Hokari, S; Takada, M1
Albuz, FK; Armstrong, DT; Gilchrist, RB; Lane, M; Sasseville, M; Thompson, JG1
Arnoletti, E; Baragli, A; Ghè, C; Ghigo, E; Granata, R; Muccioli, G1
Forbes, RA; Kikuchi, T; McQuade, RD; Tadori, Y1
Bolger, GB; Clancy, JP; Ehrhardt, A; Fan, L; Li, Y; Mitchell, LH; Naren, AP; Pyle, LC; Ren, A; Rowe, SM; Sorscher, EJ1
Calvert, AE; Chen, B; Meng, X; Nelin, LD1
Kikuchi, T; Tadori, Y1
Gilchrist, RB; Kelly, JM; Rose, RD; Sutton-McDowall, ML; Thompson, JG1
Dwinell, MB; Hauser, AD; Roy, I; Williams, CL; Wilson, JM; Zimmerman, NP1
Baulain, U; Diederich, M; Großfeld, R; Heinzmann, J; Herrmann, D; Lucas-Hahn, A; Niemann, H; Timmermann, B; Ulloa, SM1
Giembycz, MA; Johnson, M; Joshi, T; Newton, R1
Ahmady, A; Bedaiwy, M; Farghaly, T; Hussein, M; Khalifa, E; Mostafa, S1
Azari-Dolatabad, N; Hajian, M; Hosseini, SM; Nasr-Esfahani, MH; Ostadhosseini, S; Rahmani, HR1
Birket, SE; Chu, KK; Fernandez, CM; Grizzle, WE; Hanes, J; Houser, GH; Lin, V; Liu, L; Mazur, M; Rowe, SM; Shastry, S; Sloane, PA; Solomon, GM; Sorscher, EJ; Tearney, GJ1
Elahi, F; Hyun, SH; Lee, E; Lee, H; Lee, J; Lee, ST; Lee, Y; Park, B; Park, CK1
Elahi, F; Hyun, SH; Lee, E; Lee, H; Lee, J; Lee, ST1
Aban, I; Boyles, SE; Chaudhry, IG; Chua, M; Gentzsch, M; Guimbellot, JS; Jaspers, I; Leach, JM; Quinney, NL1
Boyles, SE; Cholon, DM; Gentzsch, M; Martino, MEB; Quinney, NL; Ribeiro, CMP1
Bijvelds, MJC; Bose, SJ; Bot, AGM; Cai, Z; de Jonge, HR; Liu, J; Sheppard, DN; Wang, Y1
Brown, M; Chansaenroj, A; Doriguzzi, N; Nagashima, J; Songsasen, N; Thongkittidilok, C1
Becq, F; Cantereau, A; Froux, L; Llinares, J1
Beekman, JM; Graeber, SY; Hirtz, S; Kruisselbrink, E; Mall, MA; van der Ent, CK; van Mourik, P; Vonk, AM1

Reviews

1 review(s) available for colforsin and carbostyril

ArticleYear
[Pharmacology of antipsychotics at human dopamine D2 and D3 receptors].
    Nihon shinkei seishin yakurigaku zasshi = Japanese journal of psychopharmacology, 2012, Volume: 32, Issue:1

    Topics: Antipsychotic Agents; Aripiprazole; Cells, Cultured; Colforsin; Dopamine D2 Receptor Antagonists; Humans; Piperazines; Quinolones; Receptors, Dopamine D2; Receptors, Dopamine D3; Schizophrenia

2012

Other Studies

43 other study(ies) available for colforsin and carbostyril

ArticleYear
Differential inotropic effects of flosequinan in ventricular muscle from normal ferrets versus patients with end-stage heart failure.
    British journal of pharmacology, 1992, Volume: 106, Issue:3

    Topics: Animals; Calcium; Colforsin; Dose-Response Relationship, Drug; Ferrets; Heart Failure; Heart Ventricles; Humans; In Vitro Techniques; Male; Milrinone; Myocardial Contraction; Pyridones; Quinolines; Quinolones; Stimulation, Chemical; Vasodilator Agents

1992
Effect of the phosphodiesterase inhibitor UK 61260 on human myocardial inotropy and diastolic relaxation.
    Journal of cardiovascular pharmacology, 1992, Volume: 19, Issue:6

    Topics: Adult; Colforsin; Electric Stimulation; Female; Heart; Humans; Imidazoles; In Vitro Techniques; Isometric Contraction; Male; Middle Aged; Myocardial Contraction; Papillary Muscles; Phosphodiesterase Inhibitors; Quinolones; Receptors, Adrenergic, beta

1992
Comparison of the effects of milrinone and OPC 3911 with those of isoprenaline, forskolin and dibutyryl-cAMP in rat aorta.
    General pharmacology, 1991, Volume: 22, Issue:4

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Aorta, Thoracic; Bucladesine; Calcium; Colforsin; In Vitro Techniques; Isoproterenol; Male; Milrinone; Phenylephrine; Phosphodiesterase Inhibitors; Potassium; Pyridones; Quinolones; Rats; Rats, Inbred Strains; Vasodilation

1991
Forskolin stimulates prostaglandin synthesis in rabbit heart by a mechanism that requires calcium and is independent of cyclic AMP.
    Circulation research, 1990, Volume: 67, Issue:5

    Topics: 6-Ketoprostaglandin F1 alpha; Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Diltiazem; Epoprostenol; Heart; In Vitro Techniques; Myocardium; Phenylisopropyladenosine; Phosphoric Diester Hydrolases; Prostaglandins; Quinolones; Rabbits; Stimulation, Chemical

1990
Inhibitory modulation by cAMP of isoproterenol-induced prostacyclin synthesis in rabbit heart.
    The American journal of physiology, 1989, Volume: 257, Issue:4 Pt 2

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; 6-Ketoprostaglandin F1 alpha; Adenylyl Cyclase Inhibitors; Animals; Blood Pressure; Colforsin; Cyclic AMP; Epoprostenol; Heart; Heart Rate; In Vitro Techniques; Isoproterenol; Male; Myocardium; Phenylisopropyladenosine; Platelet Aggregation Inhibitors; Quinolones; Rabbits; Thionucleotides

1989
Relaxant effects of the selective phosphodiesterase inhibitors milrinone and OPC 3911 on isolated human mesenteric vessels.
    Pharmacology & toxicology, 1989, Volume: 64, Issue:5

    Topics: Adult; Aged; Calcium Channel Blockers; Colforsin; Female; Humans; In Vitro Techniques; Isoproterenol; Male; Middle Aged; Milrinone; Muscle, Smooth, Vascular; Norepinephrine; Ouabain; Phosphodiesterase Inhibitors; Potassium; Pyridones; Quinolones; Splanchnic Circulation; Vasodilator Agents

1989
Effects of anti-asthma drugs on PAF-induced death in mice.
    Prostaglandins, 1988, Volume: 36, Issue:6

    Topics: Adrenalectomy; Adrenergic beta-Agonists; Animals; Asthma; Bronchodilator Agents; Colforsin; Dexamethasone; Dose-Response Relationship, Drug; Histamine Antagonists; Mice; Models, Biological; Nedocromil; Phthalazines; Platelet Activating Factor; Pyridazines; Quinolones; Serotonin Antagonists

1988
Effect of a major metabolite of the antiallergic drug repirinast on phosphodiesterase and adenylate cyclase activities.
    Arzneimittel-Forschung, 1995, Volume: 45, Issue:1

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclase Inhibitors; Animals; Colforsin; Cromolyn Sodium; Exudates and Transudates; Histamine H1 Antagonists; Histamine Release; In Vitro Techniques; Lung; Male; Peritoneal Cavity; Phosphodiesterase Inhibitors; Quinolones; Rats; Rats, Wistar; Theophylline

1995
Effects of amiloride and a novel diuretic, 7-chloro-2,3-dihydro-1-(2-methylbenzoyl)-4(1H)-quinolinone-4-oxime-o-su lfonic acid, potassium salt (M17055), on calcium transport in the rabbit connecting tubule.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:3

    Topics: Amiloride; Animals; Calcium; Calcium-Binding Proteins; Cell Membrane Permeability; Colforsin; Diuretics; In Vitro Techniques; Intracellular Fluid; Kidney Tubules; Male; Nephrons; Oximes; Parathyroid Hormone; Quinolones; Rabbits; Sodium

1993
Inhibitory effect of 2-phenyl-4-quinolone on serotonin-mediated changes in the morphology and permeability of endothelial monolayers.
    European journal of pharmacology, 1997, Sep-24, Volume: 335, Issue:2-3

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Biological Transport; Cattle; Cell Size; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic GMP; Endothelium; Enzyme Inhibitors; Gap Junctions; Myocardium; Nitroprusside; Permeability; Protein Kinase C; Quinolones; Rats; Serotonin; Serum Albumin; Staurosporine; Tetradecanoylphorbol Acetate

1997
Synergistic inhibition of vascular smooth muscle cell migration by phosphodiesterase 3 and phosphodiesterase 4 inhibitors.
    Circulation research, 1998, May-04, Volume: 82, Issue:8

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenine; Animals; Aorta; Becaplermin; Cell Movement; Cells, Cultured; Colforsin; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Drug Synergism; Humans; Kinetics; Muscle, Smooth, Vascular; Phosphodiesterase Inhibitors; Platelet-Derived Growth Factor; Proto-Oncogene Proteins c-sis; Quinolones; Rats; Recombinant Proteins

1998
Characterization of cyclic AMP efflux from swine adipocytes in vitro.
    Obesity research, 1998, Volume: 6, Issue:4

    Topics: Adipocytes; Adrenergic beta-Agonists; Animals; Antimycin A; Cells, Cultured; Colforsin; Cyclic AMP; Isoproterenol; Probenecid; Quinolones; Swine; Swine, Miniature; Xanthines

1998
Mechanism of intracellular calcium ([Ca2+]i) inhibition of lipolysis in human adipocytes.
    FASEB journal : official publication of the Federation of American Societies for Experimental Biology, 2001, Volume: 15, Issue:13

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; 8-Bromo Cyclic Adenosine Monophosphate; Adipocytes; Androstadienes; Bucladesine; Calcium; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Dose-Response Relationship, Drug; Humans; Insulin; Isoproterenol; Lipolysis; Phosphodiesterase Inhibitors; Phosphorylation; Potassium Chloride; Quinolones; Sterol Esterase; Wortmannin; Xanthines

2001
Altered phosphodiesterase 3-mediated cAMP hydrolysis contributes to a hypermotile phenotype in obese JCR:LA-cp rat aortic vascular smooth muscle cells: implications for diabetes-associated cardiovascular disease.
    Diabetes, 2002, Volume: 51, Issue:4

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Animals; Aorta; Cell Membrane; Cell Movement; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Cytosol; Diabetes Mellitus, Type 2; Hydrolysis; Muscle, Smooth, Vascular; Obesity; Phenotype; Phosphodiesterase Inhibitors; Quinolones; Rats; Rats, Mutant Strains

2002
Aripiprazole, a novel antipsychotic, is a high-affinity partial agonist at human dopamine D2 receptors.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 302, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Antipsychotic Agents; Aripiprazole; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; GTP-Binding Proteins; Humans; Piperazines; Quinolones; Radioligand Assay; Receptors, Dopamine D2; Signal Transduction; Spiperone

2002
Phosphodiesterase 3 activity is reduced in dog lung following pacing-induced heart failure.
    American journal of physiology. Lung cellular and molecular physiology, 2003, Volume: 284, Issue:5

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Animals; Capillaries; Capillary Permeability; Colforsin; Cyclic AMP; Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Dogs; Heart Failure; Hydrolysis; Lung; Pacemaker, Artificial; Phosphodiesterase Inhibitors; Pulmonary Circulation; Quinolones; Reverse Transcriptase Polymerase Chain Reaction

2003
Fundamental significance of specific phosphodiesterases in the control of spontaneous meiotic resumption in porcine oocytes.
    Molecular reproduction and development, 2005, Volume: 70, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Analysis of Variance; Animals; Chorionic Gonadotropin; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Combinations; Female; Gonadotropins, Equine; Meiosis; Oocytes; Phosphodiesterase Inhibitors; Quinolones; Sus scrofa

2005
Aripiprazole's low intrinsic activities at human dopamine D2L and D2S receptors render it a unique antipsychotic.
    European journal of pharmacology, 2005, May-16, Volume: 515, Issue:1-3

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Binding, Competitive; Cell Membrane; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; DNA, Complementary; Dopamine; Dopamine Agonists; Dopamine Antagonists; Haloperidol; Humans; Lisuride; Piperazines; Piperidines; Quinolones; Raclopride; Radioligand Assay; Receptors, Dopamine D2; Risperidone; Transfection; Tritium

2005
Numerous distinct PKA-, or EPAC-based, signalling complexes allow selective phosphodiesterase 3 and phosphodiesterase 4 coordination of cell adhesion.
    Cellular signalling, 2007, Volume: 19, Issue:12

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenylyl Cyclases; Cell Adhesion; Cell Line; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Enzyme Activators; Guanine Nucleotide Exchange Factors; Humans; Multiprotein Complexes; Peptide Fragments; Phosphodiesterase 3 Inhibitors; Phosphodiesterase Inhibitors; Protein Structure, Tertiary; Quinolones; Signal Transduction; Transfection

2007
Effects of cilostamide and forskolin on the meiotic resumption and embryonic development of immature human oocytes.
    Human reproduction (Oxford, England), 2008, Volume: 23, Issue:3

    Topics: Adenylyl Cyclases; Adult; Cells, Cultured; Colforsin; Drug Synergism; Embryonic Development; Female; Gap Junctions; Humans; Meiosis; Oocytes; Phosphodiesterase Inhibitors; Quinolones

2008
Effects of arginine vasotocin and vasopressin receptor antagonists on Na+ and Cl- transport in the isolated skin of two frog species, Hyla japonica and Rana nigromaculata.
    General and comparative endocrinology, 2008, May-15, Volume: 157, Issue:1

    Topics: Animals; Antidiuretic Hormone Receptor Antagonists; Anura; Benzazepines; Biological Transport; Chlorides; Colforsin; Dose-Response Relationship, Drug; Electrophysiology; Female; In Vitro Techniques; Male; Piperidines; Quinolones; Receptors, Vasopressin; Skin; Sodium; Species Specificity; Time Factors; Vasotocin

2008
Effects of the cAMP-elevating agents cilostamide, cilostazol and forskolin on the phosphorylation of Akt and GSK-3beta in platelets.
    Thrombosis and haemostasis, 2009, Volume: 102, Issue:2

    Topics: Animals; Binding Sites; Blood Platelets; Cilostazol; Colforsin; Collagen; Cyclic AMP; Glycogen Synthase Kinase 3; Glycogen Synthase Kinase 3 beta; In Vitro Techniques; Isoquinolines; Phosphatidylinositol 3-Kinases; Phosphorylation; Platelet Aggregation; Platelet Aggregation Inhibitors; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Quinolones; Rats; Rats, Sprague-Dawley; Serine; Sulfonamides; Tetrazoles

2009
Effects of arginine vasotocin and mesotocin on the activation and development of amiloride-blockable short-circuit current across larval, adult, and cultured larval bullfrog skins.
    Journal of comparative physiology. B, Biochemical, systemic, and environmental physiology, 2010, Volume: 180, Issue:3

    Topics: Adrenal Cortex Hormones; Amiloride; Animals; Antidiuretic Hormone Receptor Antagonists; Benzazepines; Colforsin; Electrophysiological Phenomena; Epithelial Sodium Channel Blockers; Epithelial Sodium Channels; Epithelium; Gene Expression; Larva; Oxytocin; Piperidines; Quinolones; Rana catesbeiana; Receptors, Oxytocin; Receptors, Pituitary Hormone; Receptors, Vasopressin; Skin; Vasotocin

2010
Simulated physiological oocyte maturation (SPOM): a novel in vitro maturation system that substantially improves embryo yield and pregnancy outcomes.
    Human reproduction (Oxford, England), 2010, Volume: 25, Issue:12

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Blastocyst; Cattle; Cell Communication; Cells, Cultured; Chorionic Gonadotropin; Colforsin; Culture Media, Serum-Free; Cumulus Cells; Cyclic AMP; Embryo Implantation; Embryo, Mammalian; Embryonic Development; Female; Fertilization in Vitro; Follicle Stimulating Hormone; Gap Junctions; Mice; Oocytes; Oogenesis; Pregnancy; Pregnancy Outcome; Quinolones

2010
Acylated and unacylated ghrelin attenuate isoproterenol-induced lipolysis in isolated rat visceral adipocytes through activation of phosphoinositide 3-kinase γ and phosphodiesterase 3B.
    Biochimica et biophysica acta, 2011, Volume: 1811, Issue:6

    Topics: Acylation; Adipocytes; Adrenergic beta-Agonists; Animals; Benzimidazoles; Blotting, Western; Cells, Cultured; Class Ib Phosphatidylinositol 3-Kinase; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Dose-Response Relationship, Drug; Drug Interactions; Ghrelin; Glycerol; Intra-Abdominal Fat; Isoproterenol; Lipolysis; Male; Phosphodiesterase Inhibitors; Phosphoinositide-3 Kinase Inhibitors; Proto-Oncogene Proteins c-akt; Quinolones; Quinoxalines; Rats; Rats, Wistar; Thiazolidinediones

2011
Functional potencies of dopamine agonists and antagonists at human dopamine D₂ and D₃ receptors.
    European journal of pharmacology, 2011, Volume: 666, Issue:1-3

    Topics: Animals; Aripiprazole; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Humans; Piperazines; Quinolones; Receptors, Dopamine D2; Receptors, Dopamine D3

2011
Regulatory domain phosphorylation to distinguish the mechanistic basis underlying acute CFTR modulators.
    American journal of physiology. Lung cellular and molecular physiology, 2011, Volume: 301, Issue:4

    Topics: Aminophenols; Animals; Blotting, Western; Cell Line; Chlorocebus aethiops; Colforsin; Cresols; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Diffusion Chambers, Culture; Dimerization; Enzyme-Linked Immunosorbent Assay; Gene Expression; High-Throughput Screening Assays; Humans; Ion Channel Gating; Ion Transport; Lentivirus; Membrane Transport Modulators; Mice; Mutation; Phosphorylation; Protein Structure, Tertiary; Pyrazoles; Quinolones; Retroviridae; Transduction, Genetic

2011
Pharmacologic agents elevating cAMP prevent arginase II expression and proliferation of pulmonary artery smooth muscle cells.
    American journal of respiratory cell and molecular biology, 2012, Volume: 47, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenylyl Cyclases; Arginase; Cell Hypoxia; Cell Proliferation; Cells, Cultured; Colforsin; Cyclic AMP; Enzyme Induction; Humans; Myocytes, Smooth Muscle; Phosphodiesterase 3 Inhibitors; Pulmonary Artery; Quinolones; Signal Transduction

2012
Regulation of sheep oocyte maturation using cAMP modulators.
    Theriogenology, 2013, Jan-01, Volume: 79, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Embryo, Mammalian; Embryonic Development; Female; Follicle Stimulating Hormone; In Vitro Oocyte Maturation Techniques; Oocytes; Oogenesis; Osmolar Concentration; Phosphodiesterase Inhibitors; Quality Control; Quinolones; Sheep

2013
Cyclic AMP regulates the migration and invasion potential of human pancreatic cancer cells.
    Molecular carcinogenesis, 2015, Volume: 54, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Amides; Apoptosis; Carcinoma, Pancreatic Ductal; Cell Line, Tumor; Cell Movement; Cell Proliferation; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Deoxycytidine; Enzyme Inhibitors; Gemcitabine; Humans; Neoplasm Invasiveness; Pancreatic Neoplasms; Phosphodiesterase Inhibitors; Pyridines; Quinolones; rho GTP-Binding Proteins; rhoA GTP-Binding Protein; rhoC GTP-Binding Protein; Vasodilator Agents

2015
Effects of different oocyte retrieval and in vitro maturation systems on bovine embryo development and quality.
    Zygote (Cambridge, England), 2015, Volume: 23, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Blastocyst; Cattle; Colforsin; Culture Media; DNA Methylation; Female; Fertilization in Vitro; Gene Expression Regulation, Developmental; In Vitro Oocyte Maturation Techniques; Male; Oocyte Retrieval; Quinolones

2015
The long-acting β2 -adrenoceptor agonist, indacaterol, enhances glucocorticoid receptor-mediated transcription in human airway epithelial cells in a gene- and agonist-dependent manner.
    British journal of pharmacology, 2015, Volume: 172, Issue:10

    Topics: Adrenergic beta-2 Receptor Agonists; Benzodioxoles; Cells, Cultured; Colforsin; Dexamethasone; Drug Interactions; Epithelial Cells; Humans; Indans; Ligands; Quinolones; Receptors, Glucocorticoid; Respiratory Mucosa; Response Elements; Steroids; Transcriptional Activation; Transfection

2015
The effect of temporary meiotic attenuation on the in vitro maturation outcome of bovine oocytes.
    In vitro cellular & developmental biology. Animal, 2015, Volume: 51, Issue:7

    Topics: Animals; Blastocyst; Cattle; Cells, Cultured; Colforsin; Culture Media; Female; Fertilization in Vitro; Follicle Stimulating Hormone; In Vitro Oocyte Maturation Techniques; Luteinizing Hormone; Male; Meiosis; Oocytes; Purines; Quinolones; Roscovitine; Time Factors

2015
Effects of cilostamide and/or forskolin on the meiotic resumption and development competence of growing ovine oocytes selected by brilliant cresyl blue staining.
    Theriogenology, 2016, Volume: 85, Issue:8

    Topics: Animals; Colforsin; Embryonic Development; In Vitro Oocyte Maturation Techniques; Meiosis; Oocytes; Oxazines; Quinolones; Sheep

2016
Combination therapy with cystic fibrosis transmembrane conductance regulator modulators augment the airway functional microanatomy.
    American journal of physiology. Lung cellular and molecular physiology, 2016, 05-15, Volume: 310, Issue:10

    Topics: Amiloride; Aminophenols; Animals; Cells, Cultured; Chloride Channel Agonists; Colforsin; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Drug Evaluation, Preclinical; Drug Therapy, Combination; Humans; Membrane Potentials; Mice; Mutation, Missense; NIH 3T3 Cells; Quinolones

2016
Cilostamide and forskolin treatment during pre-IVM improves preimplantation development of cloned embryos by influencing meiotic progression and gap junction communication in pigs.
    Theriogenology, 2016, Volume: 86, Issue:3

    Topics: Adjuvants, Immunologic; Animals; Blastocyst; Bucladesine; Colforsin; Dose-Response Relationship, Drug; Embryo Culture Techniques; Embryo Transfer; Female; Gap Junctions; In Vitro Oocyte Maturation Techniques; Meiosis; Phosphodiesterase Inhibitors; Quinolones; Swine

2016
Supplement of cilostamide in growth medium improves oocyte maturation and developmental competence of embryos derived from small antral follicles in pigs.
    Theriogenology, 2017, Mar-15, Volume: 91

    Topics: Animals; Colforsin; Embryo Culture Techniques; Embryo, Mammalian; Embryonic Development; Female; In Vitro Oocyte Maturation Techniques; Oocytes; Ovarian Follicle; Quinolones; Swine

2017
Nasospheroids permit measurements of CFTR-dependent fluid transport.
    JCI insight, 2017, 11-16, Volume: 2, Issue:22

    Topics: Aminophenols; Aminopyridines; Benzodioxoles; Biological Transport; Colforsin; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Drug Combinations; Humans; Mutation; Nasal Mucosa; Particle Size; Precision Medicine; Quinolones; Spheroids, Cellular

2017
The cystic fibrosis airway milieu enhances rescue of F508del in a pre-clinical model.
    The European respiratory journal, 2018, Volume: 52, Issue:6

    Topics: Aminophenols; Aminopyridines; Benzodioxoles; Bronchi; Cell Line; Colforsin; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Epithelial Cells; Humans; Inflammation; Mutation; Quinolones; Respiratory System

2018
Differential thermostability and response to cystic fibrosis transmembrane conductance regulator potentiators of human and mouse F508del-CFTR.
    American journal of physiology. Lung cellular and molecular physiology, 2019, 07-01, Volume: 317, Issue:1

    Topics: Adenosine Triphosphate; Aminophenols; Aminopyridines; Animals; Base Sequence; Benzodioxoles; Chloride Channel Agonists; CHO Cells; Colforsin; Cricetulus; Cyclic AMP-Dependent Protein Kinases; Cystic Fibrosis Transmembrane Conductance Regulator; Gene Expression; Genistein; Ion Transport; Mice; NIH 3T3 Cells; Patch-Clamp Techniques; Protein Stability; Quinolones; Sequence Deletion; Species Specificity; Temperature; Transgenes

2019
Cilostamide and forskolin maintain gap junction function of incubated dog follicles.
    Theriogenology, 2020, Jan-15, Volume: 142

    Topics: Animals; Cells, Cultured; Colforsin; Dogs; Female; Gap Junctions; Meiosis; Oocytes; Oogenesis; Ovarian Follicle; Quinolones

2020
Quantitative phase imaging to study transmembrane water fluxes regulated by CFTR and AQP3 in living human airway epithelial CFBE cells and CHO cells.
    PloS one, 2020, Volume: 15, Issue:5

    Topics: Aminophenols; Animals; Aquaporin 3; Biological Transport, Active; Biophysical Phenomena; Bronchi; Cell Line; Chloride Channel Agonists; CHO Cells; Colforsin; Cricetulus; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Epithelial Cells; Humans; Microscopy, Interference; Mutant Proteins; Osmosis; Quinolones; Respiratory Mucosa; RNA, Messenger; Water

2020
Comparison of Organoid Swelling and
    American journal of respiratory and critical care medicine, 2020, 12-01, Volume: 202, Issue:11

    Topics: Adolescent; Adult; Aminophenols; Aminopyridines; Benzodioxoles; Child; Chlorides; Colforsin; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Drug Combinations; Edema; Female; Forced Expiratory Volume; Homozygote; Humans; In Vitro Techniques; Male; Membrane Potentials; Middle Aged; Nasal Mucosa; Organoids; Precision Medicine; Prospective Studies; Quinolones; Rectum; Sweat; Treatment Outcome; Vital Capacity; Young Adult

2020