Page last updated: 2024-08-23

colforsin and butaclamol

colforsin has been researched along with butaclamol in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19902 (22.22)18.7374
1990's3 (33.33)18.2507
2000's3 (33.33)29.6817
2010's1 (11.11)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
Hayashi, S; Kato, A; Mizuno, K; Morita, A; Nakata, E; Ohashi, K; Yamamura, K1
Lovenberg, TW; Mailman, RB; Nichols, DE; Roth, RH1
Lam, DM; Pachter, JA1
Hall, DA; Strange, PG1
Chen, LJ; Dong, ZJ; Guo, X; Han, YF; Jin, GZ1
Fu, D; Javitch, JA; Lin, H; Strange, PG; Wilson, J1
Akam, E; Strange, PG1

Other Studies

9 other study(ies) available for colforsin and butaclamol

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: de
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Analgesics; Animals; Benzimidazoles; Drug Design; Drug Evaluation, Preclinical; Humans; Microsomes, Liver; Neuralgia; Nociceptin Receptor; Pyrroles; Rats; Receptors, Opioid; Structure-Activity Relationship

2010
D1 dopamine receptors of NS20Y neuroblastoma cells are functionally similar to rat striatal D1 receptors.
    Journal of neurochemistry, 1991, Volume: 57, Issue:5

    Topics: Benzazepines; Butaclamol; Carbachol; Cell Line; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine; Dopamine Agents; Flupenthixol; Kinetics; Neuroblastoma; Oxotremorine; Phenanthridines; Radioligand Assay; Receptors, Dopamine; Receptors, Dopamine D1; Sulpiride; Tubocurarine

1991
Interactions between vasoactive intestinal peptide and dopamine in the rabbit retina: stimulation of a common adenylate cyclase.
    Journal of neurochemistry, 1986, Volume: 46, Issue:1

    Topics: Adenylyl Cyclases; Animals; Butaclamol; Chickens; Colforsin; Cyclic AMP; Dopamine; Dose-Response Relationship, Drug; Drug Interactions; Ergolines; Metoclopramide; Quinpirole; Rabbits; Receptors, Cell Surface; Receptors, Dopamine; Receptors, Vasoactive Intestinal Peptide; Retina; Sodium Fluoride; Vasoactive Intestinal Peptide

1986
Evidence that antipsychotic drugs are inverse agonists at D2 dopamine receptors.
    British journal of pharmacology, 1997, Volume: 121, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Butaclamol; CHO Cells; Colforsin; Cricetinae; Cyclic AMP; Dopamine Agonists; Receptors, Dopamine D2

1997
Dual actions of (-)-stepholidine on the dopamine receptor-mediated adenylate cyclase activity in rat corpus striatum.
    Life sciences, 1997, Volume: 61, Issue:4

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Benzazepines; Berberine; Butaclamol; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Female; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Synaptosomes

1997
Mechanisms of inverse agonism of antipsychotic drugs at the D(2) dopamine receptor: use of a mutant D(2) dopamine receptor that adopts the activated conformation.
    Journal of neurochemistry, 2001, Volume: 77, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Antipsychotic Agents; Apomorphine; Binding, Competitive; Bromocriptine; Butaclamol; Chlorpromazine; CHO Cells; Clozapine; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; GTP-Binding Proteins; Haloperidol; Humans; Macromolecular Substances; Mutagenesis, Site-Directed; Phenethylamines; Piperidines; Protein Binding; Protein Conformation; Radioligand Assay; Receptors, Dopamine D2; Recombinant Fusion Proteins; Sodium; Spiperone; Structure-Activity Relationship; Sulpiride; Transfection; Tyramine

2001
Inverse agonist properties of atypical antipsychotic drugs.
    Biochemical pharmacology, 2004, Jun-01, Volume: 67, Issue:11

    Topics: Animals; Antipsychotic Agents; Butaclamol; CHO Cells; Clozapine; Colforsin; Cricetinae; Cyclic AMP; Drug Interactions; Female; Humans; Receptors, Dopamine D2; Risperidone; Sodium

2004