Page last updated: 2024-08-23

colforsin and buspirone

colforsin has been researched along with buspirone in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19906 (50.00)18.7374
1990's1 (8.33)18.2507
2000's5 (41.67)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Nomura, Y; Okada, F; Tokumitsu, Y1
Cornfield, LJ; Martin, AR; Nelson, DL; Taylor, EW1
Hyslop, DK; Maayani, S; Smith, DW; Yocca, FD1
Bockaert, J; Bouhelal, R; Cory, RN; Dumuis, A; Sebben, M1
De Vivo, M; Maayani, S1
Hsu, KS; Huang, CC; Liang, YC1
Beneytez, ME; Benhamu, B; Caicoya, AG; Delgado, M; Fuentes, JA; López-Rodríguez, ML; Manzanares, J; Morcillo, MJ; Pozo, MA; Rubia, FJ1
Assié, MB; Colpaert, FC; Cosi, C; Koek, W; Patoiseau, JF; Pauwels, PJ; Vacher, B1
Borsini, F; Cassano, GB; Giromella, A; Lucacchini, A; Marazziti, D; Mayer, N; Mazzoni, MR; Naccarato, AG; Palego, L1
Lisinicchia, JG; Watts, VJ1
Bönisch, H; Brüss, M; Göthert, M; Kostanian, A1

Other Studies

12 other study(ies) available for colforsin and buspirone

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Pertussis toxin attenuates 5-hydroxytryptamine1A receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in rat hippocampal membranes.
    Journal of neurochemistry, 1989, Volume: 52, Issue:5

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Buspirone; Cell Membrane; Colforsin; GTP-Binding Proteins; Hippocampus; Male; Membrane Proteins; Molecular Weight; Pertussis Toxin; Pyrimidines; Rats; Rats, Inbred Strains; Receptors, Serotonin; Serotonin; Tetrahydronaphthalenes; Virulence Factors, Bordetella

1989
MDL 73005EF: partial agonist at the 5-HT1A receptor negatively linked to adenylate cyclase.
    European journal of pharmacology, 1989, Dec-07, Volume: 173, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenosine Triphosphate; Adenylyl Cyclase Inhibitors; Animals; Buspirone; Colforsin; Cyclic AMP; Dioxins; Hippocampus; In Vitro Techniques; Male; Membranes; Pindolol; Rats; Rats, Inbred Strains; Receptors, Serotonin; Spiro Compounds; Tetrahydronaphthalenes; Tryptamines

1989
BMY 7378, a buspirone analog with high affinity, selectivity and low intrinsic activity at the 5-HT1A receptor in rat and guinea pig hippocampal membranes.
    European journal of pharmacology, 1987, Jun-04, Volume: 137, Issue:2-3

    Topics: Adenylyl Cyclases; Animals; Anti-Anxiety Agents; Buspirone; Colforsin; Guinea Pigs; Hippocampus; In Vitro Techniques; Piperazines; Pyrimidines; Rats; Receptors, Serotonin; Species Specificity; Structure-Activity Relationship

1987
Piperazine derivatives including the putative anxiolytic drugs, buspirone and ipsapirone, are agonists at 5-HT1A receptors negatively coupled with adenylate cyclase in hippocampal neurons.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 335, Issue:5

    Topics: Adenylyl Cyclases; Animals; Anti-Anxiety Agents; Buspirone; Cells, Cultured; Colforsin; Guinea Pigs; Hippocampus; In Vitro Techniques; Male; Neurons; Pyrimidines; Receptors, Serotonin

1987
Characterization of the 5-hydroxytryptamine1a receptor-mediated inhibition of forskolin-stimulated adenylate cyclase activity in guinea pig and rat hippocampal membranes.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Buspirone; Colforsin; Dose-Response Relationship, Drug; Guinea Pigs; Hippocampus; Indoles; Lisuride; Mathematics; Pyrimidines; Rats; Receptors, Serotonin; Tetrahydronaphthalenes

1986
A role for extracellular adenosine in time-dependent reversal of long-term potentiation by low-frequency stimulation at hippocampal CA1 synapses.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Nov-15, Volume: 19, Issue:22

    Topics: Adenosine; Animals; Buspirone; Colforsin; Cyclic AMP; Electric Stimulation; Enzyme Inhibitors; Excitatory Postsynaptic Potentials; Hippocampus; In Vitro Techniques; Least-Squares Analysis; Long-Term Potentiation; Male; Neurons; Piperazines; Purinergic P1 Receptor Antagonists; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Synapses; Synaptic Transmission; Theobromine; Thionucleotides; Time Factors; Xanthines

1999
Biochemical, electrophysiological and neurohormonal studies with B-20991, a selective 5-HT1A receptor agonist.
    Pharmacology, 2001, Volume: 62, Issue:4

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Body Temperature; Buspirone; Colforsin; Corticosterone; Cyclic AMP; Dendrites; Dose-Response Relationship, Drug; Electrophysiology; HeLa Cells; Humans; Imidazoles; Male; Mice; Neurons; Piperazines; Pyridines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2001
5-HT1A receptor activation and antidepressant-like effects: F 13714 has high efficacy and marked antidepressant potential.
    European journal of pharmacology, 2001, May-25, Volume: 420, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminopyridines; Animals; Antidepressive Agents; Binding, Competitive; Buspirone; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); HeLa Cells; Humans; Male; Motor Activity; Piperazines; Piperidines; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming

2001
Region-dependent effects of flibanserin and buspirone on adenylyl cyclase activity in the human brain.
    The international journal of neuropsychopharmacology, 2002, Volume: 5, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Aged; Aged, 80 and over; Benzimidazoles; Binding, Competitive; Brain; Buspirone; Colforsin; Dose-Response Relationship, Drug; Female; Hippocampus; Humans; Male; Middle Aged; Piperazines; Prefrontal Cortex; Raphe Nuclei; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2002
Sensitization of adenylate cyclase by short-term activation of 5-HT1A receptors.
    Cellular signalling, 2003, Volume: 15, Issue:12

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Adenylyl Cyclases; Animals; Arachidonic Acid; Buspirone; Calcimycin; CHO Cells; Colforsin; Cricetinae; Cricetulus; Cyclic AMP; Cycloheximide; Dose-Response Relationship, Drug; Flavonoids; Humans; Indoles; Indomethacin; Maleimides; Pertussis Toxin; Phorbol Esters; Piperazines; Pyridines; Receptor, Serotonin, 5-HT1A; Serotonin; Serotonin 5-HT1 Receptor Agonists; Serotonin 5-HT1 Receptor Antagonists; Time Factors; Tryptamines

2003
The naturally occurring Arg219Leu variant of the human 5-HT1A receptor: impairment of signal transduction.
    Pharmacogenetics and genomics, 2005, Volume: 15, Issue:4

    Topics: Anti-Anxiety Agents; Arginine; Buspirone; Cell Line; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Genetic Variation; Humans; Inhibitory Concentration 50; Leucine; Pharmacogenetics; Piperazines; Protein Binding; Receptor, Serotonin, 5-HT1A; Serotonin Antagonists; Signal Transduction; Transfection

2005