Page last updated: 2024-08-23

colforsin and baclofen

colforsin has been researched along with baclofen in 34 studies

Research

Studies (34)

TimeframeStudies, this research(%)All Research%
pre-19908 (23.53)18.7374
1990's13 (38.24)18.2507
2000's12 (35.29)29.6817
2010's1 (2.94)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Creveling, CR; Daly, JW; Lewandowski, GA; McNeal, ET1
Bellows, DS; Clarke, ID; Diamandis, P; Dirks, PB; Graham, J; Jamieson, LG; Ling, EK; Sacher, AG; Tyers, M; Ward, RJ; Wildenhain, J1
de Koning, HP; Huchedé, B; Jenks, BG; Roubos, EW1
Kamatchi, GL; Ticku, MK1
Wojcik, WJ; Xu, J1
Dolphin, AC; McGuirk, SM; Scott, RH1
Costa, E; Paez, X; Ulivi, M; Wojcik, WJ1
Boar, BR; Cross, AJ; Green, AR; Robinson, TN; Toczek, JM1
Hill, DR1
Barbaccia, ML; Costa, E; Szekely, AM1
Enna, SJ; Ferkany, JW; Scherer, RW1
Desrues, L; Lamacz, M; Tonon, MC; Vaudry, H1
Fisone, G; Greengard, P; Snyder, GL1
Bowery, NG; Malcangio, M1
González, MP; Oset-Gasque, MJ; Parramón, M1
Andrade, R1
Bowery, NG; Knight, AR1
Itoh, Y; Kimura, K; Oka, M; Shimidzu, T; Ukai, Y; Yoshikuni, Y1
Hashimoto, T; Kuriyama, K1
Olianas, MC; Onali, P1
Barilà, B; Cupello, A; Robello, M1
Bao, GB; Ma, L; Pei, G; Pu, L1
Snead, OC1
Beltrán-Parrazal, L; Clapp, C; Martínez de la Escalera, G; Noris, G1
Becú-Villalobos, D; Bianchi, M; Chamson-Reig, A; Libertun, C; Lux-Lantos, V; Pignataro, O; Rey-Roldán, E1
Gómez-Villafuertes, R; Gualix, J; Miras-Portugal, MT; Pintor, J1
Mascia, FM; Olianas, MC; Onali, P1
Ballabio, M; Cavarretta, IT; Froestl, W; Lambert, JJ; Magnaghi, V; Melcangi, RC; Zucchi, I1
Harvey, VL; Stephens, GJ1
Novotny, J; Stöhr, J; Svoboda, P1
Ivenshitz, M; Segal, M1
Desrayaud, S; Gjoni, T; Imobersteg, S; Urwyler, S1
Fujita, T; Oka, M; Wada, M; Wu, Q; Yamamoto, A1
Di Prisco, S; Grilli, M; Marchi, M; Pittaluga, A; Summa, M; Usai, C1

Other Studies

34 other study(ies) available for colforsin and baclofen

ArticleYear
[3H]Batrachotoxinin A 20 alpha-benzoate binding to voltage-sensitive sodium channels: a rapid and quantitative assay for local anesthetic activity in a variety of drugs.
    Journal of medicinal chemistry, 1985, Volume: 28, Issue:3

    Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Batrachotoxins; Calcium Channel Blockers; Cyclic AMP; Guinea Pigs; Histamine H1 Antagonists; In Vitro Techniques; Ion Channels; Neurotoxins; Sodium; Tranquilizing Agents; Tritium

1985
Chemical genetics reveals a complex functional ground state of neural stem cells.
    Nature chemical biology, 2007, Volume: 3, Issue:5

    Topics: Animals; Cell Survival; Cells, Cultured; Mice; Molecular Structure; Neoplasms; Neurons; Pharmaceutical Preparations; Sensitivity and Specificity; Stem Cells

2007
Dynamics of cyclic-AMP efflux in relation to alpha-MSH secretion from melanotrope cells of Xenopus laevis.
    Life sciences, 1992, Volume: 51, Issue:21

    Topics: 1-Methyl-3-isobutylxanthine; alpha-MSH; Amphibian Proteins; Animals; Baclofen; Calcium; Colforsin; Corticotropin-Releasing Hormone; Cyclic AMP; Dopamine; In Vitro Techniques; Peptide Hormones; Peptides; Pituitary Gland; Xenopus laevis

1992
GABAB receptor activation inhibits Ca2(+)-activated 86Rb-efflux in cultured spinal cord neurons via G-protein mechanism.
    Brain research, 1990, Jan-08, Volume: 506, Issue:2

    Topics: Adenylate Cyclase Toxin; Animals; Baclofen; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; GTP-Binding Proteins; Mice; Mice, Inbred C57BL; Pertussis Toxin; Receptors, GABA-A; Rubidium Radioisotopes; Spinal Cord; Virulence Factors, Bordetella

1990
Gamma aminobutyric acid B receptor-mediated inhibition of adenylate cyclase in cultured cerebellar granule cells: blockade by islet-activating protein.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 239, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Adenylate Cyclase Toxin; Adenylyl Cyclase Inhibitors; Animals; Autoradiography; Baclofen; Bicuculline; Cerebellum; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Pertussis Toxin; Rats; Receptors, GABA-A; Time Factors; Virulence Factors, Bordetella

1986
An investigation into the mechanisms of inhibition of calcium channel currents in cultured sensory neurones of the rat by guanine nucleotide analogues and (-)-baclofen.
    British journal of pharmacology, 1989, Volume: 97, Issue:1

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Baclofen; Calcium Channels; Cells, Cultured; Cholera Toxin; Colforsin; Culture Techniques; Electrophysiology; Enzyme Activation; Guanine Nucleotides; Guanosine 5'-O-(3-Thiotriphosphate); Guanosine Triphosphate; Neurons, Afferent; Protein Kinase C; Rats; Thionucleotides; Type C Phospholipases

1989
Islet-activating protein inhibits the beta-adrenergic receptor facilitation elicited by gamma-aminobutyric acidB receptors.
    Journal of neurochemistry, 1989, Volume: 53, Issue:3

    Topics: Adenosine Diphosphate Ribose; Animals; Baclofen; Cerebral Cortex; Colforsin; Cyclic AMP; Drug Synergism; GTP-Binding Proteins; Hippocampus; Isoproterenol; Male; Pertussis Toxin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, beta; Receptors, GABA-A; Virulence Factors, Bordetella

1989
Effects of the putative antagonists phaclofen and delta-aminovaleric acid on GABAB receptor biochemistry.
    British journal of pharmacology, 1989, Volume: 98, Issue:3

    Topics: Amino Acids; Amino Acids, Neutral; Animals; Baclofen; Cerebral Cortex; Colforsin; Cyclic AMP; In Vitro Techniques; Isoproterenol; Kinetics; Male; Proteins; Radioligand Assay; Rats; Receptors, GABA-A

1989
GABAB receptor modulation of adenylate cyclase activity in rat brain slices.
    British journal of pharmacology, 1985, Volume: 84, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Baclofen; Brain; Cerebral Cortex; Colforsin; Cyclic AMP; Diterpenes; gamma-Aminobutyric Acid; In Vitro Techniques; Nipecotic Acids; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, GABA-A

1985
Effect of a protracted antidepressant treatment on signal transduction and [3H](-)-baclofen binding at GABAB receptors.
    The Journal of pharmacology and experimental therapeutics, 1987, Volume: 243, Issue:1

    Topics: Adenylyl Cyclases; Animals; Anthracenes; Baclofen; Cerebral Cortex; Colforsin; Desipramine; Drug Administration Schedule; Imipramine; Injections, Intraperitoneal; Kinetics; Male; Maprotiline; Rats; Rats, Inbred Strains; Receptors, GABA-A

1987
Evidence for pharmacologically distinct subsets of GABAB receptors.
    Brain research bulletin, 1988, Volume: 21, Issue:3

    Topics: Animals; Baclofen; Binding, Competitive; Colforsin; Cyclic AMP; In Vitro Techniques; Isoproterenol; Male; Propylamines; Rats; Rats, Inbred Strains; Receptors, GABA-A

1988
Mechanism of action of gamma-aminobutyric acid on frog melanotrophs.
    Journal of molecular endocrinology, 1995, Volume: 14, Issue:1

    Topics: Adenylyl Cyclases; Animals; Baclofen; Calcium; Calcium Channels; Colforsin; Cyclic AMP; GABA-A Receptor Agonists; GABA-B Receptor Agonists; gamma-Aminobutyric Acid; In Vitro Techniques; Inositol Phosphates; Male; Melanocyte-Stimulating Hormones; Models, Biological; Pituitary Gland, Posterior; Rana ridibunda; Receptors, GABA-A; Receptors, GABA-B; Signal Transduction; Taurine

1995
Phosphorylation of DARPP-32 is regulated by GABA in rat striatum and substantia nigra.
    Journal of neurochemistry, 1994, Volume: 63, Issue:5

    Topics: Animals; Baclofen; Colforsin; Corpus Striatum; Cyclic AMP; Dopamine and cAMP-Regulated Phosphoprotein 32; GABA Antagonists; gamma-Aminobutyric Acid; Male; Nerve Tissue Proteins; Phosphoproteins; Phosphorylation; Radioimmunoassay; Rats; Rats, Sprague-Dawley; Receptors, GABA; Substantia Nigra

1994
GABAB receptor-mediated inhibition of forskolin-stimulated cyclic AMP accumulation in rat spinal cord.
    Neuroscience letters, 1993, Aug-20, Volume: 158, Issue:2

    Topics: Analgesics; Animals; Animals, Newborn; Baclofen; Capsaicin; Colforsin; Cyclic AMP; GABA-A Receptor Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Norepinephrine; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Spinal Cord

1993
GABAB receptors modulate catecholamine secretion in chromaffin cells by a mechanism involving cyclic AMP formation.
    British journal of pharmacology, 1993, Volume: 110, Issue:4

    Topics: Adenylate Cyclase Toxin; Animals; Baclofen; Calcium; Catecholamines; Cattle; Cells, Cultured; Cholera Toxin; Chromaffin Granules; Colforsin; Cyclic AMP; Organophosphorus Compounds; Pertussis Toxin; Receptors, GABA-B; Virulence Factors, Bordetella

1993
Enhancement of beta-adrenergic responses by Gi-linked receptors in rat hippocampus.
    Neuron, 1993, Volume: 10, Issue:1

    Topics: Adenylyl Cyclases; Animals; Baclofen; Colforsin; Electric Conductivity; Electrophysiology; GTP-Binding Proteins; Hippocampus; Male; Norepinephrine; Potassium Channels; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, beta; Receptors, GABA-A; Receptors, Serotonin

1993
The pharmacology of adenylyl cyclase modulation by GABAB receptors in rat brain slices.
    Neuropharmacology, 1996, Volume: 35, Issue:6

    Topics: Adenylyl Cyclases; Animals; Baclofen; Brain; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Male; Norepinephrine; Rats; Rats, Wistar; Receptors, GABA-B

1996
Involvement of metabotropic glutamate receptors in Gi- and Gs-dependent modulation of adenylate cyclase activity induced by a novel cognition enhancer NS-105 in rat brain.
    Brain research, 1997, Apr-18, Volume: 754, Issue:1-2

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Adrenergic alpha-Agonists; Alanine; Animals; Baclofen; Brimonidine Tartrate; Cell Membrane; Cerebral Cortex; Cholera Toxin; Cognition; Colforsin; Cyclic AMP; Cycloleucine; Excitatory Amino Acid Antagonists; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); In Vitro Techniques; Isoproterenol; Kinetics; Male; Manganese; Pertussis Toxin; Piperidines; Proline; Quinoxalines; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Receptors, Neurotransmitter; Virulence Factors, Bordetella; Yohimbine

1997
In vivo evidence that GABA(B) receptors are negatively coupled to adenylate cyclase in rat striatum.
    Journal of neurochemistry, 1997, Volume: 69, Issue:1

    Topics: Adenylyl Cyclases; Adrenergic beta-Agonists; Animals; Baclofen; Colforsin; Corpus Striatum; Cyclic AMP; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Isoproterenol; Locomotion; Male; Organophosphorus Compounds; Rats; Rats, Wistar; Receptors, GABA-B; Signal Transduction

1997
GABA(B) receptor-mediated stimulation of adenylyl cyclase activity in membranes of rat olfactory bulb.
    British journal of pharmacology, 1999, Volume: 126, Issue:3

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Baclofen; Calcium; Calmodulin; Colforsin; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; GABA Agonists; GABA Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; In Vitro Techniques; Indomethacin; Injections, Intraventricular; Male; Membranes; Neuropeptides; Neuroprotective Agents; Olfactory Bulb; Organophosphorus Compounds; Pertussis Toxin; Phosphinic Acids; Phospholipases A; Phospholipids; Pituitary Adenylate Cyclase-Activating Polypeptide; Propanolamines; Propylamines; Quinacrine; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Transducin; Virulence Factors, Bordetella

1999
GABA(B) receptor activation protects GABA(A) receptor from cyclic AMP-dependent down-regulation in rat cerebellar granule cells.
    Neuroscience, 1999, Volume: 93, Issue:3

    Topics: Adenylate Cyclase Toxin; Adenylyl Cyclases; Animals; Baclofen; Cerebellar Cortex; Chloride Channels; Colforsin; Cyclic AMP; Down-Regulation; Enzyme Activation; GABA Agonists; Ion Channel Gating; Ion Transport; Muscimol; Nerve Tissue Proteins; Patch-Clamp Techniques; Pertussis Toxin; Rats; Rats, Wistar; Receptors, GABA-A; Receptors, GABA-B; Signal Transduction; Virulence Factors, Bordetella

1999
Acute desensitization of nociceptin/orphanin FQ inhibition of voltage-gated calcium channels in freshly dissociated hippocampal neurons.
    The European journal of neuroscience, 1999, Volume: 11, Issue:10

    Topics: Animals; Baclofen; Barium; Calcium; Calcium Channel Blockers; Calcium Channels, P-Type; Carcinogens; Cells, Cultured; Colforsin; Electrophysiology; Extracellular Space; GABA Agonists; Hippocampus; Ion Channel Gating; Membrane Potentials; Nociceptin; Opioid Peptides; Patch-Clamp Techniques; Peptide Fragments; Protein Kinase C; Pyramidal Cells; Rats; Rats, Sprague-Dawley; Tetradecanoylphorbol Acetate; Tetrodotoxin

1999
Evidence for a G protein-coupled gamma-hydroxybutyric acid receptor.
    Journal of neurochemistry, 2000, Volume: 75, Issue:5

    Topics: Adenylyl Cyclases; Animals; Baclofen; Brain; Brain Chemistry; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Enzyme Activation; Enzyme Inhibitors; Female; GABA Agonists; GTP Phosphohydrolases; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Male; Rats; Rats, Sprague-Dawley; Receptors, Cell Surface; Receptors, Presynaptic; Sodium Oxybate; Subcellular Fractions

2000
GABA inhibition of immortalized gonadotropin-releasing hormone neuronal excitability involves GABA(A) receptors negatively coupled to cyclic adenosine monophosphate formation.
    Endocrine, 2001, Volume: 14, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Baclofen; Bicuculline; Calcium; Calcium Channels; Cell Line, Transformed; Cell Membrane; Colforsin; Cyclic AMP; gamma-Aminobutyric Acid; Gonadotropin-Releasing Hormone; Kinetics; Muscimol; Neurons; Potassium; Receptors, GABA-A

2001
GABA(B) receptors in anterior pituitary cells. Mechanism of action coupled to endocrine effects.
    Neuroendocrinology, 2001, Volume: 73, Issue:5

    Topics: Animals; Baclofen; Barium Compounds; Calcium; Calcium Channel Blockers; Cells, Cultured; Chlorides; Colforsin; Cyclic AMP; Dopamine; Female; Luteinizing Hormone; Pertussis Toxin; Pituitary Gland, Anterior; Potassium Channel Blockers; Potassium Chloride; Proestrus; Prolactin; Rats; Receptors, GABA-B; Tetraethylammonium; Thyrotropin-Releasing Hormone; Virulence Factors, Bordetella

2001
GABAB receptor-mediated presynaptic potentiation of ATP ionotropic receptors in rat midbrain synaptosomes.
    Neuropharmacology, 2003, Volume: 44, Issue:3

    Topics: Adenosine Triphosphate; Animals; Baclofen; Calcium; Colforsin; Competitive Bidding; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Fura-2; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; Glial Fibrillary Acidic Protein; Immunohistochemistry; In Vitro Techniques; Mesencephalon; Muscimol; Nerve Tissue Proteins; Picrotoxin; Rats; Receptors, GABA-B; Receptors, Purinergic P2; Receptors, Purinergic P2X; Synaptosomes; Time Factors

2003
Positive regulation of GABA(B) receptors dually coupled to cyclic AMP by the allosteric agent CGP7930.
    European journal of pharmacology, 2003, Jun-20, Volume: 471, Issue:2

    Topics: Adenylyl Cyclases; Allosteric Regulation; Animals; Baclofen; Calmodulin; Colforsin; Corpus Striatum; Corticotropin-Releasing Hormone; Cyclic AMP; Cytoplasmic Granules; Drug Synergism; Frontal Lobe; gamma-Aminobutyric Acid; Gene Expression; Male; Olfactory Bulb; Phenols; Rats; Rats, Sprague-Dawley; Receptors, GABA; Receptors, GABA-B; Signal Transduction

2003
GABAB receptors in Schwann cells influence proliferation and myelin protein expression.
    The European journal of neuroscience, 2004, Volume: 19, Issue:10

    Topics: Animals; Baclofen; Blotting, Northern; Blotting, Western; Bromodeoxyuridine; Cell Division; Cells, Cultured; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; GABA Antagonists; Hypoxanthine Phosphoribosyltransferase; Immunohistochemistry; Indoles; Membrane Proteins; Myelin Proteins; Protein Isoforms; Rats; Rats, Sprague-Dawley; Receptors, GABA-B; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Schwann Cells; Sciatic Nerve; Tetrazolium Salts; Time Factors

2004
Mechanism of GABA receptor-mediated inhibition of spontaneous GABA release onto cerebellar Purkinje cells.
    The European journal of neuroscience, 2004, Volume: 20, Issue:3

    Topics: Action Potentials; Age Factors; Animals; Baclofen; Barium; Cadmium; Calcium; Cerebellum; Colforsin; Drug Interactions; Enzyme Inhibitors; Exotoxins; GABA Agonists; GABA Antagonists; gamma-Aminobutyric Acid; In Vitro Techniques; Male; Mice; Neural Inhibition; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Purkinje Cells; Receptors, GABA-A; Ruthenium Red; Synaptic Transmission; Tetrodotoxin

2004
Characterization of [3H]-forskolin binding sites in young and adult rat brain cortex: identification of suramin as a competitive inhibitor of [3H]-forskolin binding.
    Canadian journal of physiology and pharmacology, 2005, Volume: 83, Issue:7

    Topics: Adrenergic beta-Agonists; Aging; Animals; Baclofen; Binding, Competitive; Cell Membrane; Cerebral Cortex; Colforsin; GABA Agonists; Guanylyl Imidodiphosphate; Isoproterenol; Magnesium; Male; Rats; Rats, Wistar; Receptors, Drug; Suramin

2005
Simultaneous NMDA-dependent long-term potentiation of EPSCs and long-term depression of IPSCs in cultured rat hippocampal neurons.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2006, Jan-25, Volume: 26, Issue:4

    Topics: 2-Amino-5-phosphonovalerate; Animals; Baclofen; Calcium; Cells, Cultured; Colforsin; Cyclic AMP; Evoked Potentials; Hippocampus; Long-Term Potentiation; Long-Term Synaptic Depression; Neuronal Plasticity; Neurons; Nitric Oxide; Nitric Oxide Synthase; Nitroarginine; Patch-Clamp Techniques; Phosphinic Acids; Propanolamines; Quinoxalines; Rats; Receptors, GABA-B; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Tetrodotoxin; Thionucleotides; Time Factors

2006
The positive allosteric modulator GS39783 enhances GABA(B) receptor-mediated inhibition of cyclic AMP formation in rat striatum in vivo.
    Journal of neurochemistry, 2006, Volume: 96, Issue:5

    Topics: Animals; Baclofen; Colforsin; Corpus Striatum; Cyclic AMP; Cyclopentanes; Dose-Response Relationship, Drug; Drug Interactions; GABA Agonists; GABA Antagonists; Male; Microdialysis; Phosphinic Acids; Pyrimidines; Radioimmunoassay; Rats; Rats, Wistar; Receptors, GABA-A; Time Factors

2006
Functional expression of metabotropic GABAB receptors in primary cultures of astrocytes from rat cerebral cortex.
    Biochemical and biophysical research communications, 2006, Mar-17, Volume: 341, Issue:3

    Topics: Adenylyl Cyclase Inhibitors; Adenylyl Cyclases; Animals; Astrocytes; Baclofen; Cell Membrane; Cells, Cultured; Cerebral Cortex; Colforsin; Gene Expression Regulation; Guanosine Triphosphate; Rats; Receptors, GABA-B; RNA, Messenger

2006
Presynaptic mGlu7 receptors control GABA release in mouse hippocampus.
    Neuropharmacology, 2013, Volume: 66

    Topics: Adenylyl Cyclase Inhibitors; Aminobutyrates; Animals; Baclofen; Benzhydryl Compounds; Benzoates; Benzylamines; Colforsin; Dose-Response Relationship, Drug; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Exocytosis; GABA Antagonists; gamma-Aminobutyric Acid; Glycine; Hippocampus; Imines; Mice; Phosphinic Acids; Potassium Chloride; Pyridones; Receptors, GABA-B; Receptors, Metabotropic Glutamate; Synaptosomes; Syntaxin 1; Vesicular Inhibitory Amino Acid Transport Proteins

2013