Page last updated: 2024-08-23

colforsin and alpha-aminopyridine

colforsin has been researched along with alpha-aminopyridine in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19909 (34.62)18.7374
1990's3 (11.54)18.2507
2000's3 (11.54)29.6817
2010's9 (34.62)24.3611
2020's2 (7.69)2.80

Authors

AuthorsStudies
Blinks, JR; Endoh, M; Taira, N; Yanagisawa, T1
Ahn, HS; Eardley, D; Prioli, N; Watkins, R1
Simpson, LL1
Alberts, P; Ogren, VR1
Bowyer, JF; Weiner, N1
Renit-Soria, J; Stinnakre, J; Van Renterghem, C1
Bali, JP; Choquet, A; Galleyrand, JC; Magous, R1
Cox, RT; Walker, RJ1
Komajda, M1
Clarke, W; Kung, HF; Kung, MP; Maayani, S; Zhuang, ZP1
Bobirnac, I; Bruinvels, AT; Danzeisen, M; Gazi, L; Geisse, S; Hoyer, D; Schoeffter, P; Schüpbach, E; Sommer, B; Tricklebank, M1
Assié, MB; Cosi, C; Koek, W1
Assié, MB; Colpaert, FC; Cosi, C; Koek, W; Patoiseau, JF; Pauwels, PJ; Vacher, B1
Cutz, E; Farragher, SM; Fu, XW; Pan, J; Wang, D; Wong, V1
Chung, C; Dubé, D; Friesen, RW; Huang, Z; Kwok, E; Laliberté, F; Liu, S; Tota, MR; Veilleux, A; Young, A; Zhang, L1
Beume, R; Hirrle, A; Marx, D; Tenor, H; Wohlsen, A1
Basma, H; Fahrid, M; Gunji, Y; Holz, O; Kanaji, N; Liu, X; Magnussen, H; Michalski, J; Muller, KC; Nakanishi, M; Nelson, A; Nogel, S; Rabe, KF; Rennard, SI; Sato, T; Toews, ML; Wang, X1
Bond, M; Cui, MZ; Duggirala, A; Hewer, RC; Hindmarch, CC; Kimura, TE; Newby, AC1
Becq, F; Boinot, C; Ferru-Clément, R; Jollivet Souchet, M1
Bond, M; Duggirala, A; Johnson, JL; Kimura, TE; Newby, AC; Sala-Newby, GB; Wu, YJ1
Carrillo, JJ; Lin, HV; Wang, J1
Aban, I; Boyles, SE; Chaudhry, IG; Chua, M; Gentzsch, M; Guimbellot, JS; Jaspers, I; Leach, JM; Quinney, NL1
Boyles, SE; Cholon, DM; Gentzsch, M; Martino, MEB; Quinney, NL; Ribeiro, CMP1
Bijvelds, MJC; Bose, SJ; Bot, AGM; Cai, Z; de Jonge, HR; Liu, J; Sheppard, DN; Wang, Y1
Hanrahan, JW; Luo, Y; Thomas, DY; Turner, MJ1
Beekman, JM; Graeber, SY; Hirtz, S; Kruisselbrink, E; Mall, MA; van der Ent, CK; van Mourik, P; Vonk, AM1

Other Studies

26 other study(ies) available for colforsin and alpha-aminopyridine

ArticleYear
Effects of new inotropic agents on cyclic nucleotide metabolism and calcium transients in canine ventricular muscle.
    Circulation, 1986, Volume: 73, Issue:3 Pt 2

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Aequorin; Aminopyridines; Amrinone; Animals; Calcium; Carbachol; Cardiotonic Agents; Colforsin; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Enoximone; Female; Imidazoles; Male; Milrinone; Myocardial Contraction; Myocardium; Nifedipine; Nucleotides, Cyclic; Pyrazines; Pyridones; Quinolines; Time Factors

1986
Effects of several newer cardiotonic drugs on cardiac cyclic AMP metabolism.
    Biochemical pharmacology, 1986, Apr-01, Volume: 35, Issue:7

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; 3',5'-Cyclic-GMP Phosphodiesterases; Adenylyl Cyclases; Aminopyridines; Amrinone; Animals; Cardiotonic Agents; Colforsin; Cyclic AMP; Enoximone; Guinea Pigs; Hydrolysis; Imidazoles; Isoenzymes; Milrinone; Myocardial Contraction; Myocardium; Phosphodiesterase Inhibitors; Pyridones

1986
Use of pharmacologic antagonists to deduce commonalities of biologic activity among clostridial neurotoxins.
    The Journal of pharmacology and experimental therapeutics, 1988, Volume: 245, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; Acetylcholine; Amifampridine; Aminopyridines; Ammonium Chloride; Animals; Botulinum Toxins; Calcium; Cholera Toxin; Colforsin; Female; Guanidine; Guanidines; In Vitro Techniques; Methylamines; Mice; Neuromuscular Junction; Neurotoxins; Tetanus Toxin; Theophylline

1988
Interaction of forskolin with the effect of atropine on [3H]acetylcholine secretion in guinea-pig ileum myenteric plexus.
    The Journal of physiology, 1988, Volume: 395

    Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Aminopyridines; Animals; Atropine; Colforsin; Cyclic GMP; Drug Interactions; Guinea Pigs; Ileum; In Vitro Techniques; Myenteric Plexus; Neuromuscular Junction

1988
K+ channel and adenylate cyclase involvement in regulation of Ca2+-evoked release of [3H]dopamine from synaptosomes.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 248, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; Adenylate Cyclase Toxin; Adenylyl Cyclases; Aminopyridines; Animals; Calcium; Colforsin; Dopamine; Ergolines; Ethylmaleimide; In Vitro Techniques; Pertussis Toxin; Potassium Channels; Quinpirole; Rats; Synaptosomes; Tetraethylammonium Compounds; Virulence Factors, Bordetella

1989
beta-Adrenergic induced K+ current in Xenopus oocytes: role of cAMP, inhibition by muscarinic agents.
    Proceedings of the Royal Society of London. Series B, Biological sciences, 1985, Jan-22, Volume: 223, Issue:1232

    Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Adenosine; Aminobenzoates; Aminopyridines; Animals; Atropine; Calcimycin; Colforsin; Cyclic AMP; Diterpenes; Female; Isoproterenol; Oocytes; Phosphodiesterase Inhibitors; Potassium; Receptors, Adrenergic, beta; Tetraethylammonium Compounds; Xenopus laevis

1985
[Is forskolin a stimulant of gastric secretion?].
    Comptes rendus des seances de la Societe de biologie et de ses filiales, 1988, Volume: 182, Issue:3

    Topics: Aminopyridines; Animals; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Gastric Acid; Gastrins; Histamine; Parietal Cells, Gastric; Rabbits; Rats

1988
An analysis of the inhibitory responses of dopamine and octopamine on Helix central neurons.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1988, Volume: 91, Issue:2

    Topics: 4-Aminopyridine; Adenylyl Cyclase Inhibitors; Aminopyridines; Animals; Bucladesine; Colforsin; Dopamine; Evoked Potentials; Helix, Snails; Imines; Membrane Potentials; Neuromuscular Depolarizing Agents; Neurons; Octopamine; Potassium Channels

1988
[New cardiotonic agents].
    Annales de cardiologie et d'angeiologie, 1985, Volume: 34, Issue:10

    Topics: Aminopyridines; Amrinone; Cardiotonic Agents; Colforsin; Deoxyepinephrine; Humans; Imidazoles; Levodopa; Milrinone; Practolol; Prenalterol; Propanolamines; Pyridones; Quinazolines; Xamoterol

1985
A potential 5-HT1A receptor antagonist: p-MPPI.
    Life sciences, 1994, Volume: 55, Issue:19

    Topics: Adenylyl Cyclases; Aminopyridines; Animals; Binding, Competitive; Colforsin; Guanosine Triphosphate; Hippocampus; In Vitro Techniques; Iodine Radioisotopes; Kinetics; Ligands; Piperazines; Rats; Receptors, Serotonin; Serotonin Antagonists; Stimulation, Chemical

1994
The agonist activities of the putative antipsychotic agents, L-745,870 and U-101958 in HEK293 cells expressing the human dopamine D4.4 receptor.
    British journal of pharmacology, 1998, Volume: 124, Issue:5

    Topics: Aminopyridines; Antipsychotic Agents; Cell Line; Clozapine; Colforsin; Cyclic AMP; Dopamine; Dopamine Agonists; Dopamine Antagonists; Humans; Kidney; Piperidines; Pyridines; Pyrroles; Raclopride; Receptors, Dopamine D2; Receptors, Dopamine D4; Recombinant Proteins; Salicylamides; Spiperone

1998
Correlation between low/high affinity ratios for 5-HT(1A) receptors and intrinsic activity.
    European journal of pharmacology, 1999, Dec-10, Volume: 386, Issue:1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminopyridines; Animals; Colforsin; GTP-Binding Protein alpha Subunits, Gi-Go; Guanylyl Imidodiphosphate; HeLa Cells; Hippocampus; Humans; In Vitro Techniques; Male; Membranes; Pertussis Toxin; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Virulence Factors, Bordetella

1999
5-HT1A receptor activation and antidepressant-like effects: F 13714 has high efficacy and marked antidepressant potential.
    European journal of pharmacology, 2001, May-25, Volume: 420, Issue:2-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Aminopyridines; Animals; Antidepressive Agents; Binding, Competitive; Buspirone; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Guanosine 5'-O-(3-Thiotriphosphate); HeLa Cells; Humans; Male; Motor Activity; Piperazines; Piperidines; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Serotonin Antagonists; Serotonin Receptor Agonists; Swimming

2001
Neuroepithelial bodies in mammalian lung express functional serotonin type 3 receptor.
    American journal of physiology. Lung cellular and molecular physiology, 2001, Volume: 281, Issue:4

    Topics: Aminopyridines; Animals; Calcium; Chemoreceptor Cells; Colforsin; Cricetinae; Dose-Response Relationship, Drug; Gene Expression; Humans; Immunohistochemistry; In Situ Hybridization; Indoles; Ion Channel Gating; Ketanserin; Lung; Mammals; Membrane Potentials; Mesocricetus; Mice; Mice, Inbred C57BL; Patch-Clamp Techniques; Piperazines; Rabbits; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Respiratory Mucosa; RNA, Messenger; Serotonin; Serotonin Antagonists; Tropisetron

2001
Dynamic activation of cystic fibrosis transmembrane conductance regulator by type 3 and type 4D phosphodiesterase inhibitors.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:2

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Adenylyl Cyclases; Aminopyridines; Benzamides; Biotransformation; Blotting, Western; Cell Line; Chlorides; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclopropanes; Cystic Fibrosis Transmembrane Conductance Regulator; Enzyme Activation; Humans; Iodine Radioisotopes; Isoquinolines; Phosphodiesterase Inhibitors; Sulfonamides

2005
Effect of cyclic AMP-elevating agents on airway ciliary beat frequency in central and lateral airways in rat precision-cut lung slices.
    European journal of pharmacology, 2010, Jun-10, Volume: 635, Issue:1-3

    Topics: Aminopyridines; Animals; Benzamides; Colforsin; Cyclic AMP; Cyclopropanes; Dissection; Enzyme Inhibitors; Female; In Vitro Techniques; Lung; Mucociliary Clearance; Phosphodiesterase 4 Inhibitors; Prostaglandins; Rats; Rats, Wistar; Rolipram; Terbutaline; Time Factors

2010
Attenuation of inhibitory prostaglandin E2 signaling in human lung fibroblasts is mediated by phosphodiesterase 4.
    American journal of respiratory cell and molecular biology, 2012, Volume: 47, Issue:6

    Topics: Adrenergic beta-2 Receptor Agonists; Albuterol; Aminopyridines; Benzamides; Cells, Cultured; Chemotaxis; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Cyclopropanes; Dinoprostone; Fibroblasts; Fibronectins; Gene Expression; Humans; Iloprost; Isoenzymes; Lung; Phosphodiesterase 4 Inhibitors; Pulmonary Disease, Chronic Obstructive; Receptors, Epoprostenol; Receptors, Prostaglandin; Receptors, Prostaglandin E, EP2 Subtype; Rolipram; Second Messenger Systems

2012
Inhibition of Egr1 expression underlies the anti-mitogenic effects of cAMP in vascular smooth muscle cells.
    Journal of molecular and cellular cardiology, 2014, Volume: 72

    Topics: Adenosine; Aminopyridines; Animals; Cell Proliferation; Colforsin; Cyclic AMP; Cyclic AMP Response Element-Binding Protein; Cyclic AMP-Dependent Protein Kinases; Early Growth Response Protein 1; Epoprostenol; ets-Domain Protein Elk-1; Gene Expression Regulation; Guanine Nucleotide Exchange Factors; Human Umbilical Vein Endothelial Cells; Male; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Organ Specificity; Primary Cell Culture; Protein Binding; rac1 GTP-Binding Protein; Rats; Rats, Sprague-Dawley; Serum Response Factor; Signal Transduction

2014
Searching for combinations of small-molecule correctors to restore f508del-cystic fibrosis transmembrane conductance regulator function and processing.
    The Journal of pharmacology and experimental therapeutics, 2014, Volume: 350, Issue:3

    Topics: 1-Deoxynojirimycin; Aminopyridines; Benzamides; Benzodioxoles; Cell Survival; Colforsin; Cystic Fibrosis Transmembrane Conductance Regulator; Dose-Response Relationship, Drug; HeLa Cells; Humans; Thiazoles

2014
cAMP-induced actin cytoskeleton remodelling inhibits MKL1-dependent expression of the chemotactic and pro-proliferative factor, CCN1.
    Journal of molecular and cellular cardiology, 2015, Volume: 79

    Topics: Actin Cytoskeleton; Adenosine; Aminopyridines; Animals; Carotid Arteries; Cell Proliferation; Chemotaxis; Colforsin; Cyclic AMP; Cysteine-Rich Protein 61; Epoprostenol; Humans; Male; Mitogens; Models, Biological; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Rats, Sprague-Dawley; rho-Associated Kinases; rhoA GTP-Binding Protein; Serum Response Factor; Trans-Activators; Transcription Factors; Transcription, Genetic

2015
GPR142 Agonists Stimulate Glucose-Dependent Insulin Secretion via Gq-Dependent Signaling.
    PloS one, 2016, Volume: 11, Issue:4

    Topics: Aminopyridines; Animals; Colforsin; Cyclic AMP; Gene Expression Regulation; Glucose; HEK293 Cells; Humans; Insulin; Insulin Secretion; Islets of Langerhans; Male; Mice; Mice, Inbred C57BL; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Phosphorylation; Primary Cell Culture; Protein Subunits; Pyrazoles; Receptors, G-Protein-Coupled; Recombinant Proteins; Signal Transduction; Tryptophan

2016
Nasospheroids permit measurements of CFTR-dependent fluid transport.
    JCI insight, 2017, 11-16, Volume: 2, Issue:22

    Topics: Aminophenols; Aminopyridines; Benzodioxoles; Biological Transport; Colforsin; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Drug Combinations; Humans; Mutation; Nasal Mucosa; Particle Size; Precision Medicine; Quinolones; Spheroids, Cellular

2017
The cystic fibrosis airway milieu enhances rescue of F508del in a pre-clinical model.
    The European respiratory journal, 2018, Volume: 52, Issue:6

    Topics: Aminophenols; Aminopyridines; Benzodioxoles; Bronchi; Cell Line; Colforsin; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Epithelial Cells; Humans; Inflammation; Mutation; Quinolones; Respiratory System

2018
Differential thermostability and response to cystic fibrosis transmembrane conductance regulator potentiators of human and mouse F508del-CFTR.
    American journal of physiology. Lung cellular and molecular physiology, 2019, 07-01, Volume: 317, Issue:1

    Topics: Adenosine Triphosphate; Aminophenols; Aminopyridines; Animals; Base Sequence; Benzodioxoles; Chloride Channel Agonists; CHO Cells; Colforsin; Cricetulus; Cyclic AMP-Dependent Protein Kinases; Cystic Fibrosis Transmembrane Conductance Regulator; Gene Expression; Genistein; Ion Transport; Mice; NIH 3T3 Cells; Patch-Clamp Techniques; Protein Stability; Quinolones; Sequence Deletion; Species Specificity; Temperature; Transgenes

2019
The dual phosphodiesterase 3/4 inhibitor RPL554 stimulates rare class III and IV CFTR mutants.
    American journal of physiology. Lung cellular and molecular physiology, 2020, 05-01, Volume: 318, Issue:5

    Topics: Aminopyridines; Animals; Benzodioxoles; Bronchi; Cell Line; Colforsin; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 3; Cyclic Nucleotide Phosphodiesterases, Type 4; Cystic Fibrosis Transmembrane Conductance Regulator; Humans; Isoquinolines; Mutation; Phosphodiesterase 3 Inhibitors; Phosphodiesterase 4 Inhibitors; Primary Cell Culture; Pyrimidinones; Rats; Rats, Inbred F344; Thyroid Epithelial Cells; Transgenes

2020
Comparison of Organoid Swelling and
    American journal of respiratory and critical care medicine, 2020, 12-01, Volume: 202, Issue:11

    Topics: Adolescent; Adult; Aminophenols; Aminopyridines; Benzodioxoles; Child; Chlorides; Colforsin; Cystic Fibrosis; Cystic Fibrosis Transmembrane Conductance Regulator; Drug Combinations; Edema; Female; Forced Expiratory Volume; Homozygote; Humans; In Vitro Techniques; Male; Membrane Potentials; Middle Aged; Nasal Mucosa; Organoids; Precision Medicine; Prospective Studies; Quinolones; Rectum; Sweat; Treatment Outcome; Vital Capacity; Young Adult

2020