Page last updated: 2024-08-23

colforsin and 1,9-dideoxyforskolin

colforsin has been researched along with 1,9-dideoxyforskolin in 109 studies

Research

Studies (109)

TimeframeStudies, this research(%)All Research%
pre-19909 (8.26)18.7374
1990's81 (74.31)18.2507
2000's16 (14.68)29.6817
2010's3 (2.75)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abe, A; Karaki, H1
Felíu, JE; Herias, M; Olea, J; Pereda, C; Rossi, I1
Gauthier, C; Soustre, H1
Bringhurst, FR; Fukayama, S; Tashjian, AH1
Ganetzky, B; Stern, M1
Hirst, BH; Hunter, J; McEwan, GT; Simmons, NL1
Olianas, MC; Onali, P1
Díaz, M; Gill, DR; Higgins, CF; Hyde, SC; Sepúlveda, FV; Valverde, MA1
Ishac, E; Li, C; White, G1
De Luca, M; Galietta, LJ; Mastrocola, T; Romeo, G; Rugolo, M1
Appel, NM; De Souza, EB; Laurenza, A; Robbins, JD; Seamon, KB; Simpson, IA1
Chan, JY; Chan, SH; Fu, MJ; Lin, KS1
Corrèze, C; Delemer, B; Dib, K; Haye, B; Jacquemin, C; Saunier, B1
Farkas, EM; Papachristou, DN; Patel, YC; Zingg, HH1
Morris, DI; Ruoho, AE; Seamon, KB; Speicher, LA; Tew, KD1
Hirst, BH; Hunter, J; Simmons, NL2
Wadler, S; Yang, CP1
Doi, K; Matsunaga, T; Mori, N1
Boutjdir, M; Fischmeister, R; Hanf, R; Méry, PF; Shrier, A1
Aronstam, RS; Daly, JW; Nishizawa, Y; Seamon, KB1
Baidan, LV; Fertel, RH; Wood, JD; Xia, Y1
Anderson, RJ; Breckon, R; Colston, D1
Crooks, JR; Keogh, DP; Mitchell, MJ; Smith, SL1
Elders, MJ; Hu, LM; Kemp, SF; Peng, CF; Smith, WG1
McMorris, FA; Raible, DW1
Bonvallet, R; Lemtiri-Chlieh, F; Rougier, O1
Baxter, DA; Byrne, JH1
Sitkovsky, MV; Takayama, H; Trenn, G1
Aldrich, RW; Garber, SS; Hoshi, T1
White, MM1
Harris-Warrick, RM1
Wickelgren, WO; Womble, MD1
Wadler, S; Wiernik, PH1
Adams, M; Boarder, MR; Marriott, D1
McGee, R; McHugh, EM1
Habberfield, AD; Joost, HG; Laurenza, A; Seamon, KB; Simpson, IA1
Alexander, SP; Hernández, F; Kendall, DA1
Fan, P1
Kuzhikandathil, EV; Molloy, GR1
Eltze, M1
Ambrosio, C; Barbaccia, ML; Massotti, M; Roscetti, G; Trabucchi, M1
Craig, CG; Temple, SD; White, TD1
Bellé, R; Cormier, P; Drewing, S; Minella, O; Mulner-Lorillon, O; Poulhe, R; Schmalzing, G1
Alvaro, D; Boyer, JL; Cho, W; Mennone, A1
Furukata, K; Hosokami, T; Ide, S; Iimori, T; Ikegami, S; Sasaki, T; Senda, M1
Reich, H; Sei, Y1
Gean, PW; Huang, CC1
Díaz, M; Higgins, CF; Rucăreanu, C; Sepúlveda, FV; Valverde, MA1
Sorota, S1
Gill, DR; Higgins, CF; Hyde, SC; McNaughton, PA; Mintenig, GM; Sardini, A; Sepúlveda, FV; Valverde, MA1
Cook, SA; Lichtman, AH; Martin, BR; Welch, SP1
Alton, EW; Geddes, DM; Munkonge, FM; Osborne, LR1
Basile, A; Gusovsky, F; Sei, Y; Skolnick, P; Takemura, M1
De Greef, C; Droogmans, G; Eggermont, J; Nilius, B; Raeymaekers, L; Sehrer, J; Viana, F1
Feltz, A; Zerr, P1
Roberts, PJ; Toms, NJ1
Björnsson, OG; Gibbons, GF; Sparks, CE; Sparks, JD1
Barajas-López, C1
Kirk, J; Kirk, K1
Katz, S; Mok, W; Phaneuf, S; Salari, H; Wong, S1
Dover, PJ; McCaig, CD1
Chou, CY; Shen, MR; Wu, SN1
Kim, KT; Park, TJ1
Argent, BE; Chambers, JA; Gray, MA; Harris, A; Mathews, CJ; Verdon, B; Wardle, CJ; Winpenny, JP1
Chiu, CT; Fan, LW; Tsao, HL; Yang, C; Yu, SM1
Becherer, U; Feltz, A; Rodeau, JL; Zerr, P1
Hewlett, EL; Login, IS1
Asai, T; McDonald, TF; Pelzer, S1
Krouse, ME; Law, TC; Luckie, DB; Sikic, BI; Wine, JJ1
Tokimasa, T1
Buczko, E; Dufau, ML; Khanum, A1
Galietta, LJ; Romano, L; Rossi, GA; Sacco, O; Zegarra-Moran, O1
Cikós, T; Kalthoff, H; Krull, NB; Ungefroren, H1
Bucher, B; Côrtes, SF; Lemos, VS; Takeda, K1
Gandía, L; García, AG; Ramirez-Lavergne, C; Trifaró, JM; Villarroya, M; Vitale, ML1
Miranda, D; Morán, J; Pasantes-Morales, H; Sánchez Olea, R1
Miranda, D; Morán, J; Pasantes-Morales, H; Peña-Segura, C1
Chen, Y; Herness, MS; Sun, XD1
Bhatnagar, A; Dhir, P; Srivastava, SK; Wang, LF1
Chang, YH; Chern, Y; Ching, YH; Conti, M; Lai, HL; Lee, YC1
Cid, LP; Eguiguren, AL; Sepúlveda, FV; Stutzin, A1
Komatsu, N; Muramatsu, T; Oda, T1
Khan, M; Pahan, K; Singh, I1
Ambikapathy, S; Bond, TD; Mohammad, S; Valverde, MA1
Al-Dahan, MI; Jalilian Tehrani, MH; Thalmann, RH1
Christofi, FL; Jamaleddin, AJ; Liu, CY; Zhang, H1
DePinho, RA; Eisen, AM; Gallo, V; Ghiani, CA; Knutson, PL; McBain, CJ; Yuan, X1
d'Alcantara, P; Schiffmann, SN; Swillens, S1
Darszon, A; de la Vega-Beltrán, JL; Espinosa, F; Gasque, G; López-González, I; Serrano, CJ; Treviño, CL1
Garfield, RE; Okawa, T; Saade, GR; Syal, AS; Vedernikov, YP1
Morales-Mulia, M; Morán, J; Pasantes-Morales, H1
Bottrill, FE; Hiley, CR; Omar, R; White, R1
Brès, V; Duvoid, A; Hurbin, A; Hussy, N; Moos, FC; Orcel, H; Rabié, A1
Lock, H; Valverde, MA1
Evans, DI; Jones, RS; Woodhall, G1
Liu, LA; Shi, LJ; Wang, CA1
Hescheler, J; Lenka, N; Su, J; Ullrich, S; Yu, H1
Anderson, AE; Mayne, A; Pfaffinger, PJ; Schrader, LA; Sweatt, JD1
Battaglia, M; Bernardi, P; Fassetta, M; Gentile, A; Gramaglia, D; Petronilli, V; Ranzato, L; Rasola, A1
Ding, X; Staudinger, JL1
Di Carlo, A; Macchia, V; Mariano, A; Terracciano, D1
Altrup, U; Ure, A1
Asakawa, Y; Hagiwara, H; Hashimoto, T; Hoshi, T; Kudou, M; Suzuki, T; Takeuchi, F1
Ahluwalia, J1
Huang, XZ; Jin, D; Kim, DH; Lee, KJ; Li, JH; Qi, XF; Song, SB; Teng, YC; Yoon, YS1
Blum, AE; Dubyak, GR; Walsh, BC1
Campochiaro, PA; Gong, YY; Hackett, SF; Iwase, T; Lu, L; Seidel, CP; Stevens, RK; Wang, X1
Acosta-Gómez, EI; Angel-Chavez, LI; Castro, E; Cruzblanca, H; Morales-Avalos, M1

Other Studies

109 other study(ies) available for colforsin and 1,9-dideoxyforskolin

ArticleYear
Calcium channel blocker-like action of 1,9-dideoxyforskolin in vascular smooth muscle.
    Japanese journal of pharmacology, 1992, Volume: 60, Issue:4

    Topics: Animals; Aorta, Thoracic; Calcium; Calcium Channel Blockers; Colforsin; Cytosol; Fura-2; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium; Rats; Rats, Wistar

1992
Fructose 2,6-bisphosphate levels and modulation of glycolysis by histamine, cholecystokinin, and forskolin in isolated rabbit gastric glands.
    Metabolism: clinical and experimental, 1992, Volume: 41, Issue:3

    Topics: 3-O-Methylglucose; Animals; Colforsin; Cyclic AMP; Fructosediphosphates; Gastric Mucosa; Glucose; Glycolysis; Histamine; In Vitro Techniques; Kinetics; Lactates; Methylglucosides; Pepsinogens; Phosphofructokinase-2; Phosphotransferases; Rabbits; Sincalide

1992
Forskolin effects on slow inward current and phasic tension of frog atrial fibres: modulation by adenosine and phosphodiesterase inhibitors.
    European journal of pharmacology, 1992, Feb-13, Volume: 225, Issue:2

    Topics: Adenosine; Animals; Calcium Channels; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Electric Stimulation; Heart Atria; In Vitro Techniques; Myocardial Contraction; Phosphodiesterase Inhibitors; Propranolol; Rana esculenta; Rana ridibunda; Stimulation, Chemical

1992
Forskolin-induced homologous desensitization via an adenosine 3',5'-monophosphate-dependent mechanism(s) in human osteoblast-like SaOS-2 cells.
    Endocrinology, 1992, Volume: 131, Issue:4

    Topics: Adenylate Cyclase Toxin; Cell Line; Cholera Toxin; Colforsin; Cyclic AMP; Drug Combinations; Drug Tolerance; Enzyme Activation; Hormones; Humans; Osteoblasts; Parathyroid Hormone; Pertussis Toxin; Protein Kinases; Virulence Factors, Bordetella

1992
Identification and characterization of inebriated, a gene affecting neuronal excitability in Drosophila.
    Journal of neurogenetics, 1992, Volume: 8, Issue:3

    Topics: Animals; Chromosome Mapping; Colforsin; Drosophila; Electrodes; Mutagenesis; Nerve Endings; Neurons; Phenotype; Potassium Channels; Quinidine; Synapses; Synaptic Transmission; Synaptosomes

1992
Volume-activated Cl- secretion and transepithelial vinblastine secretion mediated by P-glycoprotein are not correlated in cultured human T84 intestinal epithelial layers.
    FEBS letters, 1992, Jun-15, Volume: 304, Issue:2-3

    Topics: 4-Acetamido-4'-isothiocyanatostilbene-2,2'-disulfonic Acid; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Chloride Channels; Chlorides; Colforsin; Humans; Intestinal Mucosa; Membrane Glycoproteins; Membrane Proteins; Tumor Cells, Cultured; Vinblastine

1992
Is forskolin stimulation of rat striatal tyrosine hydroxylase dependent on adenylate cyclase activation?
    Neuroscience letters, 1992, Oct-12, Volume: 145, Issue:2

    Topics: Adenylyl Cyclases; Animals; Colforsin; Corpus Striatum; Cyclic AMP; Enzyme Activation; In Vitro Techniques; Male; Protein Kinase Inhibitors; Rats; Rats, Sprague-Dawley; Stimulation, Chemical; Synaptosomes; Thionucleotides; Tyrosine 3-Monooxygenase

1992
Volume-regulated chloride channels associated with the human multidrug-resistance P-glycoprotein.
    Nature, 1992, Feb-27, Volume: 355, Issue:6363

    Topics: 3T3 Cells; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chloride Channels; Chlorides; Colforsin; Drug Resistance; Genetic Vectors; Humans; Ion Channels; Kinetics; Membrane Glycoproteins; Membrane Potentials; Membrane Proteins; Mice; Molecular Weight; Transfection; Vaccinia virus

1992
1,9-Dideoxyforskolin does not mimic all cAMP and protein kinase A independent effects of forskolin on GABA activated ion currents in adult rat sensory neurons.
    Brain research, 1992, Jul-17, Volume: 586, Issue:1

    Topics: Animals; Colforsin; Cyclic AMP; Electric Conductivity; gamma-Aminobutyric Acid; Ion Channels; Neurons, Afferent; Protein Kinases; Rats; Rats, Inbred Strains

1992
A volume-sensitive chloride conductance revealed in cultured human keratinocytes by 36Cl- efflux and whole-cell patch clamp recording.
    Biochimica et biophysica acta, 1992, Nov-23, Volume: 1112, Issue:1

    Topics: Biological Transport; Cells, Cultured; Chlorides; Colforsin; Gluconates; Humans; Keratinocytes; Membrane Potentials; Osmolar Concentration

1992
Differential identification and localization of adenylyl cyclase and glucose transporter in brain using iodinated derivatives of forskolin.
    Brain research, 1992, May-22, Volume: 581, Issue:1

    Topics: Adenylyl Cyclases; Animals; Brain; Brain Chemistry; Cattle; Colforsin; Cytochalasin B; Glucose; Iodine Radioisotopes; Molecular Structure; Monosaccharide Transport Proteins; Radioligand Assay

1992
Participation of pertussis toxin-sensitive GTP-binding regulatory proteins in the suppression of baroreceptor reflex by neurotensin in the rat.
    Regulatory peptides, 1992, Jan-23, Volume: 37, Issue:2

    Topics: Animals; Cholera Toxin; Colforsin; Ethylmaleimide; GTP-Binding Proteins; Male; Neurotensin; Pertussis Toxin; Pressoreceptors; Rats; Rats, Inbred Strains; Reflex; Tetradecanoylphorbol Acetate; Virulence Factors, Bordetella

1992
Alteration of the functional activity of Gs protein in thyrotropin-desensitized pig thyroid cells.
    Molecular and cellular endocrinology, 1991, Volume: 75, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine Diphosphate Ribose; Adenylyl Cyclases; Animals; Cells, Cultured; Cholera Toxin; Colforsin; Cyclic AMP; Enzyme Activation; GTP-Binding Proteins; Second Messenger Systems; Swine; Thyroid Gland; Thyrotropin

1991
Regulation of islet somatostatin secretion and gene expression: selective effects of adenosine 3',5'-monophosphate and phorbol esters in normal islets of Langerhans and in a somatostatin-producing rat islet clonal cell line 1027 B2.
    Endocrinology, 1991, Volume: 128, Issue:4

    Topics: Adenoma, Islet Cell; Animals; Animals, Newborn; Bucladesine; Colforsin; Cyclic AMP; Gene Expression Regulation; Glucagon; Insulin; Insulin Secretion; Islets of Langerhans; Kinetics; Phorbol Esters; Rats; Rats, Inbred Strains; RNA, Messenger; Somatostatin; Theophylline; Tumor Cells, Cultured

1991
Interaction of forskolin with the P-glycoprotein multidrug transporter.
    Biochemistry, 1991, Aug-27, Volume: 30, Issue:34

    Topics: Affinity Labels; Amino Acid Sequence; ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Cell Line; Cell Membrane; Colforsin; Doxorubicin; Drug Interactions; Drug Resistance; Female; Humans; Membrane Glycoproteins; Molecular Sequence Data; Molecular Weight; Neoplasm Proteins; Tumor Cells, Cultured

1991
Transepithelial vinblastine secretion mediated by P-glycoprotein is inhibited by forskolin derivatives.
    Biochemical and biophysical research communications, 1991, Dec-16, Volume: 181, Issue:2

    Topics: Adenylyl Cyclases; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line; Colforsin; Dogs; Epithelium; Kidney; Membrane Glycoproteins; Verapamil; Vinblastine

1991
Reversal of doxorubicin resistance by hydrophobic, but not hydrophilic, forskolins.
    Molecular pharmacology, 1991, Volume: 40, Issue:6

    Topics: Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Chemical Phenomena; Chemistry, Physical; Colforsin; Cyclic AMP; Doxorubicin; Drug Resistance; Membrane Glycoproteins; Mice; Sarcoma, Experimental; Signal Transduction; Tumor Cells, Cultured

1991
Effects of forskolin and 1,9-dideoxy-forskolin on cochlear potentials.
    Hearing research, 1990, Volume: 45, Issue:1-2

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Bucladesine; Cochlear Microphonic Potentials; Colforsin; Evoked Potentials, Auditory; Guinea Pigs

1990
High affinity forskolin inhibition of L-type Ca2+ current in cardiac cells.
    Molecular pharmacology, 1990, Volume: 38, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium Channels; Colforsin; Cyclic AMP; In Vitro Techniques; Kinetics; Myocardium; Phosphorylation; Rana esculenta

1990
Effects of forskolin and analogues on nicotinic receptor-mediated sodium flux, voltage-dependent calcium flux, and voltage-dependent rubidium efflux in pheochromocytoma PC12 cells.
    Cellular and molecular neurobiology, 1990, Volume: 10, Issue:3

    Topics: Adrenal Gland Neoplasms; Animals; Calcium; Carbachol; Colforsin; Ion Channel Gating; Ion Channels; Neurotoxins; Pheochromocytoma; Potassium; Rats; Receptors, Nicotinic; Rubidium; Sodium; Tumor Cells, Cultured

1990
Determination of levels of cyclic AMP in the myenteric plexus of guinea-pig small intestine.
    European journal of pharmacology, 1991, Mar-25, Volume: 206, Issue:3

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Colforsin; Cyclic AMP; Electrophysiology; Enzyme Activation; Ganglia; Guinea Pigs; In Vitro Techniques; Intestine, Small; Male; Myenteric Plexus; Nerve Tissue Proteins

1991
Regulation by forskolin of cyclic AMP phosphodiesterase and protein kinase C activity in LLC-PK1 cells.
    The Biochemical journal, 1991, Oct-01, Volume: 279 ( Pt 1)

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; Alkaloids; Animals; Cells, Cultured; Colforsin; Cyclic GMP; Galactose; Macaca mulatta; Pregnenolone; Protein Kinase C; Staurosporine; Tetradecanoylphorbol Acetate

1991
Effects of the adenylate cyclase activator forskolin and its inactive derivative 1,9-dideoxyforskolin on insect cytochrome P-450 dependent steroid hydroxylase activity.
    Experientia, 1992, Jan-15, Volume: 48, Issue:1

    Topics: Adenylyl Cyclases; Animals; Aryl Hydrocarbon Hydroxylases; Colforsin; Cytochrome P-450 Enzyme System; Drosophila melanogaster; Enzyme Activation; Larva; Moths; Steroid Hydroxylases

1992
Effects of dideoxyforskolin on proteoglycan synthesis and structure in embryonic chick chondrocyte cultures.
    FEBS letters, 1990, Sep-17, Volume: 270, Issue:1-2

    Topics: Animals; Biopolymers; Cartilage; Cells, Cultured; Chick Embryo; Colforsin; Culture Media; Cyclic AMP; Diterpenes; Glycosaminoglycans; Glycosides; Proteoglycans; Sulfates

1990
Induction of oligodendrocyte differentiation by activators of adenylate cyclase.
    Journal of neuroscience research, 1990, Volume: 27, Issue:1

    Topics: Adenylyl Cyclases; Animals; Bucladesine; Cell Differentiation; Cells, Cultured; Cerebral Cortex; Cholera Toxin; Colforsin; Cyclic AMP; Diterpenes; Enzyme Induction; Oligodendroglia; Rats; Second Messenger Systems; Stimulation, Chemical

1990
Forskolin but not isoprenaline increases sodium current from frog cardiac myocytes.
    Experimental physiology, 1990, Volume: 75, Issue:6

    Topics: Animals; Colforsin; Heart; In Vitro Techniques; Isoproterenol; Membrane Potentials; Rana esculenta; Sodium Channels; Tetrodotoxin

1990
Reduction of voltage-activated K+ currents by forskolin is not mediated via cAMP in pleural sensory neurons of Aplysia.
    Journal of neurophysiology, 1990, Volume: 64, Issue:5

    Topics: Adenylyl Cyclase Inhibitors; Animals; Aplysia; Colforsin; Cyclic AMP; Dimethyl Sulfoxide; Ganglia; Membrane Potentials; Neurons, Afferent; Potassium Channels

1990
Locus of inhibitory action of cAMP-dependent protein kinase in the antigen receptor-triggered cytotoxic T lymphocyte activation pathway.
    The Journal of biological chemistry, 1988, Feb-15, Volume: 263, Issue:5

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Calcimycin; Cholera Toxin; Colforsin; Cyclic AMP; Cytotoxicity, Immunologic; Exocytosis; Lymphocyte Activation; Protein Kinases; Receptors, Antigen, T-Cell; T-Lymphocytes, Cytotoxic; Tetradecanoylphorbol Acetate

1988
Effect of forskolin on voltage-gated K+ channels is independent of adenylate cyclase activation.
    Science (New York, N.Y.), 1988, Jun-17, Volume: 240, Issue:4859

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Adrenal Gland Neoplasms; Colforsin; Cyclic AMP; Electric Conductivity; Enzyme Activation; Ion Channels; Kinetics; Pheochromocytoma; Potassium; Theophylline; Tumor Cells, Cultured

1988
Forskolin alters acetylcholine receptor gating by a mechanism independent of adenylate cyclase activation.
    Molecular pharmacology, 1988, Volume: 34, Issue:4

    Topics: Adenylyl Cyclases; Anesthetics, Local; Animals; Cloning, Molecular; Colforsin; Electric Conductivity; Enzyme Activation; Ion Channels; Receptors, Nicotinic; Torpedo; Xenopus laevis

1988
Forskolin reduces a transient potassium current in lobster neurons by a cAMP-independent mechanism.
    Brain research, 1989, Jun-05, Volume: 489, Issue:1

    Topics: Animals; Colforsin; Cyclic AMP; Ganglia; Membrane Potentials; Nephropidae; Potassium Channels

1989
Activation of adenylate cyclase by forskolin prolongs calcium action potential duration in lamprey sensory neurons.
    Brain research, 1989, Apr-17, Volume: 485, Issue:1

    Topics: Action Potentials; Adenylyl Cyclases; Animals; Calcium; Colforsin; Fishes; Lampreys

1989
Partial reversal of doxorubicin resistance by forskolin and 1,9-dideoxyforskolin in murine sarcoma S180 variants.
    Cancer research, 1988, Feb-01, Volume: 48, Issue:3

    Topics: Animals; Biological Transport; Cell Survival; Colforsin; Colony-Forming Units Assay; Cyclic AMP; Dose-Response Relationship, Drug; Drug Resistance; Sarcoma, Experimental; Tumor Cells, Cultured

1988
Effect of forskolin and prostaglandin E1 on stimulus secretion coupling in cultured bovine adrenal chromaffin cells.
    Journal of neurochemistry, 1988, Volume: 50, Issue:2

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adrenal Glands; Alprostadil; Animals; Bucladesine; Calcimycin; Calcium; Cattle; Chromaffin System; Colforsin; Cyclic AMP; Drug Synergism; Nicotine; Norepinephrine; Potassium

1988
Direct anesthetic-like effects of forskolin on the nicotinic acetylcholine receptors of PC12 cells.
    The Journal of biological chemistry, 1986, Mar-05, Volume: 261, Issue:7

    Topics: Adenylyl Cyclases; Adrenal Gland Neoplasms; Anesthetics; Animals; Carbachol; Cell Line; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Pheochromocytoma; Rats; Receptors, Cholinergic; Rubidium; Time Factors

1986
Activation of adenylate cyclase and inhibition of glucose transport in rat adipocytes by forskolin analogues: structural determinants for distinct sites of action.
    Molecular pharmacology, 1988, Volume: 33, Issue:4

    Topics: Adenylyl Cyclases; Adipose Tissue; Animals; Biological Transport, Active; Colforsin; Cytochalasin B; Diterpenes; Enzyme Activation; Glucose; Male; Rats

1988
Forskolin and 3-isobutyl-1-methylxanthine increase basal and sodium nitroprusside-elevated cyclic GMP levels in adult guinea-pig cerebellar slices.
    Journal of neurochemistry, 1994, Volume: 62, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Bucladesine; Cerebellum; Colforsin; Cyclic AMP; Cyclic GMP; Ferrocyanides; Guinea Pigs; In Vitro Techniques; Nitric Oxide; Nitroprusside

1994
Antagonism by forskolin of the 5-HT3 receptor-mediated current in nodose ganglion neurons is independent of cyclic AMP.
    Brain research, 1994, Jul-04, Volume: 650, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Colforsin; Cyclic AMP; Ion Channels; Isoquinolines; Neurons; Nodose Ganglion; Piperazines; Protein Kinase Inhibitors; Rats; Second Messenger Systems; Serotonin Antagonists

1994
Transcription of the brain creatine kinase gene in glial cells is modulated by cyclic AMP-dependent protein kinase.
    Journal of neuroscience research, 1994, Sep-01, Volume: 39, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adenylyl Cyclases; Animals; Brain; Brain Neoplasms; Cloning, Molecular; Colforsin; Creatine Kinase; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Energy Metabolism; Enzyme Activation; Enzyme Induction; Glioblastoma; Glioma; HeLa Cells; Humans; Isoenzymes; Isoquinolines; Myelin Sheath; Nerve Tissue Proteins; Neuroglia; Protein Synthesis Inhibitors; Rats; Recombinant Fusion Proteins; RNA, Antisense; Sulfonamides; Transcription, Genetic; Transfection; Tumor Cells, Cultured

1994
Pathways involved in muscarinic M1 and M2 receptor stimulation in rabbit vas deferens.
    European journal of pharmacology, 1994, Sep-22, Volume: 263, Issue:1-2

    Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Adenylyl Cyclase Inhibitors; Animals; Carbachol; Colforsin; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Lithium Chloride; Male; Muscle Contraction; Muscle, Smooth; Parasympathomimetics; Phosphatidylinositols; Rabbits; Receptors, Muscarinic; Signal Transduction; Stereoisomerism; Tetradecanoylphorbol Acetate; Vas Deferens

1994
Modulatory mechanisms of cyclic AMP-stimulated steroid content in rat brain cortex.
    European journal of pharmacology, 1994, Sep-15, Volume: 269, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adrenalectomy; Animals; Benzodiazepinones; Bucladesine; Cerebral Cortex; Colforsin; Cyclic AMP; Cycloheximide; Dose-Response Relationship, Drug; In Vitro Techniques; Isoquinolines; Male; Orchiectomy; Pregnenolone; Progesterone; Rats; Rats, Sprague-Dawley; Receptors, Cytoplasmic and Nuclear

1994
Is cyclic AMP involved in excitatory amino acid-evoked adenosine release from rat cortical slices?
    European journal of pharmacology, 1994, Sep-15, Volume: 269, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Adenosine; Animals; Calcium; Chromatography, High Pressure Liquid; Colforsin; Cyclic AMP; Excitatory Amino Acids; Male; N-Methylaspartate; Parietal Lobe; Probenecid; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate

1994
Brefeldin A provokes indirect activation of cdc2 kinase (MPF) in Xenopus oocytes, resulting in meiotic cell division.
    Developmental biology, 1995, Volume: 170, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Brefeldin A; CDC2 Protein Kinase; Cell Cycle; Cholera Toxin; Colforsin; Cyclic AMP; Cycloheximide; Cyclopentanes; Enzyme Activation; Maturation-Promoting Factor; Meiosis; Oocytes; Oogenesis; Peptide Elongation Factor 1; Peptide Elongation Factors; Phosphorylation; Progesterone; Protamine Kinase; Protein Processing, Post-Translational; Signal Transduction; Xenopus laevis

1995
Isolation of small polarized bile duct units.
    Proceedings of the National Academy of Sciences of the United States of America, 1995, Jul-03, Volume: 92, Issue:14

    Topics: 1-Methyl-3-isobutylxanthine; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Animals; Bicarbonates; Bile Ducts; Bucladesine; Chlorides; Cholestasis; Colforsin; Fluoresceins; Gluconates; Hydrogen-Ion Concentration; Kinetics; Liver; Male; Microscopy, Electron; Microscopy, Video; Rats; Rats, Sprague-Dawley; Secretin; Time Factors

1995
1-Acetyl-7-deacetylforskolin: a potential non-specific inactive analog of forskolin for estimation of its specific high-affinity binding and adenylyl cyclase stimulation in vitro.
    Life sciences, 1995, Volume: 57, Issue:14

    Topics: Adenylyl Cyclases; Animals; Cell Membrane; Colforsin; Cyclic AMP; Endothelium, Vascular; Enzyme Activation; Humans; In Vitro Techniques; Prosencephalon; Rats; Umbilical Veins

1995
Thapsigargin induces IL-2 receptor alpha-chain in human peripheral and Jurkat T cells via a protein kinase C-independent mechanism.
    Immunology letters, 1995, Volume: 45, Issue:1-2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Alkaloids; Base Sequence; Calcimycin; Calcium; Calcium-Transporting ATPases; Cholera Toxin; Colforsin; Drug Synergism; Gene Expression Regulation; Gene Expression Regulation, Leukemic; Humans; Hydroquinones; Isoquinolines; Leukemia-Lymphoma, Adult T-Cell; Molecular Sequence Data; Neoplasm Proteins; NF-kappa B; Piperazines; Protein Kinase C; Receptors, Interleukin-2; RNA, Messenger; RNA, Neoplasm; Signal Transduction; Staurosporine; T-Lymphocytes; Terpenes; Tetradecanoylphorbol Acetate; Thapsigargin

1995
Cyclic adenosine-3',5'-monophosphate potentiates the synaptic potential mediated by NMDA receptors in the amygdala.
    Journal of neuroscience research, 1995, Apr-15, Volume: 40, Issue:6

    Topics: Amygdala; Animals; Bucladesine; Colforsin; Cyclic AMP; Electric Stimulation; Long-Term Potentiation; Male; Purinergic P1 Receptor Antagonists; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Synaptic Transmission; Xanthines

1995
Volume-activated chloride channels in HeLa cells are blocked by verapamil and dideoxyforskolin.
    Pflugers Archiv : European journal of physiology, 1993, Volume: 422, Issue:4

    Topics: Adenosine Triphosphate; Chloride Channels; Chlorides; Colforsin; HeLa Cells; Humans; Hypotonic Solutions; Ion Channels; Membrane Potentials; Membrane Proteins; Osmosis; Verapamil

1993
Pharmacologic properties of the swelling-induced chloride current of dog atrial myocytes.
    Journal of cardiovascular electrophysiology, 1994, Volume: 5, Issue:12

    Topics: Animals; Anthracenes; Atrial Function; Calcium; Chloride Channels; Colforsin; Dogs; Electrophysiology; Glycolates; Heart Atria; Niflumic Acid; Nitrobenzoates; Patch-Clamp Techniques; Stilbenes

1994
Drug efflux mediated by the human multidrug resistance P-glycoprotein is inhibited by cell swelling.
    Journal of cell science, 1994, Volume: 107 ( Pt 12)

    Topics: 3T3 Cells; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Compartmentation; Cell Membrane Permeability; Chloride Channels; Colforsin; Doxorubicin; Drug Resistance, Multiple; Humans; Mice; Microscopy, Confocal; Osmotic Pressure; Recombinant Proteins; Verapamil

1994
Evaluation of cAMP involvement in cannabinoid-induced antinociception.
    Life sciences, 1995, Volume: 56, Issue:23-24

    Topics: Analgesics; Animals; Colforsin; Cyclic AMP; Cyclohexanols; Dronabinol; Injections, Intraventricular; Injections, Spinal; Male; Mice; Mice, Inbred ICR; Rats; Rats, Sprague-Dawley

1995
Lack of inhibition by dideoxy-forskolin and verapamil of DIDS-sensitive volume-activated Cl- secretion in human squamous lung carcinoma epithelial cells.
    Biochimica et biophysica acta, 1994, Dec-30, Volume: 1224, Issue:3

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Northern; Blotting, Western; Carcinoma, Squamous Cell; Cell Size; Chlorides; Colforsin; Humans; Lung Neoplasms; Osmolar Concentration; Tumor Cells, Cultured; Verapamil

1994
Distinct mechanisms for Ca2+ entry induced by OKT3 and Ca2+ depletion in Jurkat T cells.
    Experimental cell research, 1995, Volume: 216, Issue:1

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Bucladesine; Calcium; Calcium Channel Blockers; Cations, Divalent; Cholera Toxin; Colforsin; Humans; Inositol Phosphates; Ion Channel Gating; Ion Transport; Lymphocyte Activation; Muromonab-CD3; Pertussis Toxin; Receptors, Antigen, T-Cell; T-Lymphocytes; Tetradecanoylphorbol Acetate; Tumor Cells, Cultured; Virulence Factors, Bordetella

1995
Volume-activated Cl- currents in different mammalian non-excitable cell types.
    Pflugers Archiv : European journal of physiology, 1994, Volume: 428, Issue:3-4

    Topics: Animals; Anura; Cell Line; Cell Physiological Phenomena; Chlorides; Colforsin; Electric Conductivity; Endothelium, Vascular; Epithelial Cells; Epithelium; Fibroblasts; Humans; Iodides; Mammals; Neoplasms; Nitrobenzoates; Permeability; Tamoxifen

1994
Forskolin blocks the transient K current of rat cerebellar granule neurons.
    Neuroscience letters, 1994, Nov-07, Volume: 181, Issue:1-2

    Topics: Animals; Cerebellum; Colforsin; Cyclic AMP; Electric Conductivity; Electrophysiology; Neurons; Neuropeptides; Osmolar Concentration; Pituitary Adenylate Cyclase-Activating Polypeptide; Potassium; Rats; Time Factors

1994
Drug absorption limited by P-glycoprotein-mediated secretory drug transport in human intestinal epithelial Caco-2 cell layers.
    Pharmaceutical research, 1993, Volume: 10, Issue:5

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Carrier Proteins; Colforsin; Docetaxel; Epithelium; Humans; Intestinal Absorption; Intestinal Mucosa; Membrane Glycoproteins; Nifedipine; Paclitaxel; Taxoids; Tumor Cells, Cultured; Verapamil; Vinblastine

1993
NMDA receptor-mediated stimulation of rat cerebellar nitric oxide formation is modulated by cyclic AMP.
    European journal of pharmacology, 1994, Jan-01, Volume: 266, Issue:1

    Topics: Animals; Cerebellum; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Isoquinolines; Male; N-Methylaspartate; Nitric Oxide; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Sulfonamides

1994
Regulation of VLDL secretion in primary culture of rat hepatocytes: involvement of cAMP and cAMP-dependent protein kinases.
    European journal of clinical investigation, 1994, Volume: 24, Issue:2

    Topics: Animals; Apolipoproteins B; Cells, Cultured; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Lipid Metabolism; Lipoproteins, VLDL; Liver; Male; Rats; Rats, Wistar

1994
Adenosine reduces the potassium conductance of guinea pig submucosal plexus neurons by activating protein kinase A.
    Pflugers Archiv : European journal of physiology, 1993, Volume: 424, Issue:5-6

    Topics: 2-Chloroadenosine; Adenosine; Alkaloids; Animals; Cadmium; Colforsin; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Guinea Pigs; Membrane Potentials; Neurons; Phorbol 12,13-Dibutyrate; Potassium; Staurosporine; Submucous Plexus

1993
Volume-regulatory taurine release from a human lung cancer cell line. Evidence for amino acid transport via a volume-activated chloride channel.
    FEBS letters, 1993, Dec-20, Volume: 336, Issue:1

    Topics: Amino Acids; Biological Transport; Chloride Channels; Colforsin; Humans; Iodides; Lung Neoplasms; Nitrobenzoates; Osmolar Concentration; Sodium; Taurine; Tumor Cells, Cultured

1993
Forskolin inhibits platelet-activating factor binding to platelet receptors independently of adenylyl cyclase activation.
    European journal of pharmacology, 1993, Mar-15, Volume: 245, Issue:1

    Topics: Adenylyl Cyclases; Animals; Blood Platelets; Cell Membrane; Colforsin; Cyclic AMP; Dinoprostone; Enzyme Activation; GTP-Binding Proteins; In Vitro Techniques; Phosphorylation; Platelet Activating Factor; Platelet Aggregation; Rabbits

1993
Raised cyclic-AMP and a small applied electric field influence differentiation, shape, and orientation of single myoblasts.
    Developmental biology, 1993, Volume: 158, Issue:1

    Topics: Animals; Cell Differentiation; Cell Polarity; Cell Size; Cells, Cultured; Colforsin; Cyclic AMP; Electromagnetic Fields; Muscles; Xenopus

1993
Volume-sensitive chloride channels associated with human cervical carcinogenesis.
    Cancer research, 1995, Dec-15, Volume: 55, Issue:24

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; ATP Binding Cassette Transporter, Subfamily B, Member 1; Base Sequence; Carcinoma in Situ; Carcinoma, Squamous Cell; Cell Transformation, Viral; Cervix Uteri; Chloride Channels; Chlorides; Colforsin; Cyclic AMP; DNA Primers; DNA, Viral; Epithelium; Female; Humans; Ion Channel Gating; Molecular Sequence Data; Papillomaviridae; Tumor Cells, Cultured; Uterine Cervical Neoplasms; Verapamil; Water-Electrolyte Balance

1995
Cyclic AMP-independent inhibition of voltage-sensitive calcium channels by forskolin in PC12 cells.
    Journal of neurochemistry, 1996, Volume: 66, Issue:1

    Topics: Adenylyl Cyclase Inhibitors; Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Colforsin; Cyclic AMP; Ion Channel Gating; Nerve Tissue Proteins; PC12 Cells; Rats

1996
Volume-sensitive chloride currents in primary cultures of human fetal vas deferens epithelial cells.
    Pflugers Archiv : European journal of physiology, 1996, Volume: 432, Issue:4

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Bromides; Calcium; Cells, Cultured; Chloride Channels; Colforsin; Cyclic AMP; Epithelial Cells; Epithelium; Gluconates; Humans; Male; Tamoxifen; Time Factors; Vas Deferens

1996
Regulation of 5-hydroxytryptamine-induced calcium mobilization by cAMP-elevating agents in cultured canine tracheal smooth muscle cells.
    Pflugers Archiv : European journal of physiology, 1996, Volume: 432, Issue:4

    Topics: Adenine; Aluminum Compounds; Animals; Bucladesine; Calcium; Cholera Toxin; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Diterpenes; Dogs; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Fluorides; GTP-Binding Proteins; Isoquinolines; Male; Muscle, Smooth; PC12 Cells; Rats; Serotonin; Serotonin Antagonists; Sulfonamides; Trachea

1996
Forskolin's structural analogue 1,9-dideoxyforskolin has Ca2+ channel blocker-like action in rat cerebellar granule cells.
    European journal of pharmacology, 1996, May-06, Volume: 303, Issue:1-2

    Topics: Animals; Barium; Calcium; Calcium Channel Blockers; Cells, Cultured; Cerebellum; Colforsin; Dose-Response Relationship, Drug; Fura-2; Membrane Potentials; Patch-Clamp Techniques; Rats

1996
Adenylate cyclase in striatal cholinergic interneurons regulates acetylcholine release.
    Brain research, 1996, Oct-07, Volume: 735, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Acetylcholine; Adenylyl Cyclases; Animals; Colforsin; Corpus Striatum; Cyclic AMP; Interneurons; Male; Parasympathetic Nervous System; Rats

1996
Cyclic AMP-independent inhibition of cardiac calcium current by forskolin.
    Molecular pharmacology, 1996, Volume: 50, Issue:5

    Topics: Animals; Binding Sites; Calcium; Calcium Channels; Chlorides; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Electrophysiology; Guinea Pigs; Heart; Heart Ventricles; Membrane Potentials; Stimulation, Chemical; Ventricular Function

1996
Doxorubicin selection for MDR1/P-glycoprotein reduces swelling-activated K+ and Cl- currents in MES-SA cells.
    The American journal of physiology, 1996, Volume: 270, Issue:4 Pt 1

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Body Fluids; Chlorides; Colforsin; Doxorubicin; Drug Resistance, Multiple; Electric Conductivity; Female; Humans; Patch-Clamp Techniques; Potassium; RNA, Messenger; Stilbenes; Tumor Cells, Cultured; Verapamil

1996
Effects of 1, 9-dideoxy forskolin on delayed rectifier potassium current of bullfrog dorsal root ganglion cells.
    The Tokai journal of experimental and clinical medicine, 1995, Volume: 20, Issue:4-6

    Topics: Animals; Cells, Cultured; Colforsin; Delayed Rectifier Potassium Channels; Ganglia, Spinal; Potassium Channel Blockers; Potassium Channels; Potassium Channels, Voltage-Gated; Rana catesbeiana

1995
Essential role of adenosine triphosphate in activation of 17beta-hydroxysteroid dehydrogenase in the rat Leydig cell.
    Endocrinology, 1997, Volume: 138, Issue:4

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenosine Triphosphate; Aminoglutethimide; Animals; Chorionic Gonadotropin; Colforsin; Enzyme Activation; Hydroxysteroid Dehydrogenases; Leydig Cells; Male; Monosaccharide Transport Proteins; Rats; Rats, Sprague-Dawley; Testosterone

1997
Cl- currents activated by extracellular nucleotides in human bronchial cells.
    The Journal of membrane biology, 1997, Apr-01, Volume: 156, Issue:3

    Topics: Adenosine Triphosphate; Bronchi; Calcium; Cells, Cultured; Chelating Agents; Chlorides; Colforsin; Cystic Fibrosis; Egtazic Acid; Epithelial Cells; Epithelium; Extracellular Space; Humans; Intracellular Fluid; Ion Transport; Membrane Potentials; Niflumic Acid; Patch-Clamp Techniques; Uridine Triphosphate

1997
Biglycan gene promoter activity in osteosarcoma cells is regulated by cyclic AMP.
    Biochemical and biophysical research communications, 1997, Jun-18, Volume: 235, Issue:2

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Biglycan; Carbazoles; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Extracellular Matrix Proteins; Gene Expression Regulation, Neoplastic; Genes, Reporter; Humans; Indoles; Osteosarcoma; Plasmids; Promoter Regions, Genetic; Proteoglycans; Pyrroles; RNA, Messenger; Sequence Deletion; Tetradecanoylphorbol Acetate; Transcription, Genetic; Transfection; Tumor Cells, Cultured

1997
Inhibition of [Ca2+]i transients in rat adrenal chromaffin cells by neuropeptide Y: role for a cGMP-dependent protein kinase-activated K+ conductance.
    The European journal of neuroscience, 1997, Volume: 9, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenal Glands; Animals; Calcium Channel Agonists; Calcium Channel Blockers; Calcium Channels; Cells, Cultured; Cholinergic Agonists; Chromaffin Cells; Colforsin; Cyclic AMP; Cyclic GMP; Electrophysiology; In Vitro Techniques; Ion Channel Gating; Male; Neuropeptide Y; Potassium; Potassium Channels; Rats; Rats, Wistar

1997
Differential effects of forskolin and 1,9-dideoxy-forskolin on nicotinic receptor- and K+-induced responses in chromaffin cells.
    European journal of pharmacology, 1997, Jun-25, Volume: 329, Issue:2-3

    Topics: Actins; Animals; Calcium; Calcium Channel Blockers; Catecholamines; Cattle; Cells, Cultured; Chromaffin Cells; Colforsin; Gelsolin; Membrane Potentials; Microfilament Proteins; Microscopy, Fluorescence; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Patch-Clamp Techniques; Potassium

1997
Volume regulation in NIH/3T3 cells not expressing P-glycoprotein. I. Regulatory volume decrease.
    The American journal of physiology, 1997, Volume: 272, Issue:6 Pt 1

    Topics: 3T3 Cells; 4-Aminopyridine; Animals; Anions; ATP Binding Cassette Transporter, Subfamily B, Member 1; Barium; Cell Membrane Permeability; Chloride Channels; Chlorides; Colchicine; Colforsin; Dipyridamole; Gramicidin; Kinetics; Mice; Niflumic Acid; Nitrobenzoates; Potassium Channel Blockers; Potassium Channels; Quinidine; Tetraethylammonium; Tetraethylammonium Compounds; Time Factors; Water-Electrolyte Balance

1997
Volume regulation in NIH/3T3 cells not expressing P-glycoprotein. II. Chloride and amino acid fluxes.
    The American journal of physiology, 1997, Volume: 272, Issue:6 Pt 1

    Topics: 3T3 Cells; 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Amino Acids; Animals; ATP Binding Cassette Transporter, Subfamily B, Member 1; Calcium Channel Blockers; Calcium Channels; Chloride Channels; Chlorides; Colforsin; Dipyridamole; Fatty Acids, Nonesterified; Intracellular Fluid; Iodine Radioisotopes; Kinetics; Mice; Niflumic Acid; Nitrobenzoates; Osmolar Concentration; Taurine; Water-Electrolyte Balance

1997
cAMP and forskolin inhibit potassium currents in rat taste receptor cells by different mechanisms.
    The American journal of physiology, 1997, Volume: 272, Issue:6 Pt 1

    Topics: 1-Methyl-3-isobutylxanthine; Action Potentials; Animals; Bucladesine; Colforsin; Cyclic AMP; Female; In Vitro Techniques; Kinetics; Male; Patch-Clamp Techniques; Phosphorylation; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Taste Buds; Thionucleotides

1997
Contribution of osmotic changes to disintegrative globulization of single cortical fibers isolated from rat lens.
    Experimental eye research, 1997, Volume: 65, Issue:2

    Topics: Animals; Calcium; Cataract; Cells, Cultured; Chloride Channels; Colforsin; Edetic Acid; HEPES; Hypotonic Solutions; Lens Cortex, Crystalline; Nitrobenzoates; Osmosis; Rats; Sucrose

1997
Activation of phosphodiesterase IV during desensitization of the A2A adenosine receptor-mediated cyclic AMP response in rat pheochromocytoma (PC12) cells.
    Journal of neurochemistry, 1997, Volume: 69, Issue:3

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adenosine; Adrenal Gland Neoplasms; Animals; Blotting, Western; Caffeine; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cyclic Nucleotide Phosphodiesterases, Type 4; Enzyme Activation; Enzyme Inhibitors; Isoquinolines; Kinetics; PC12 Cells; Phenethylamines; Pheochromocytoma; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Polymerase Chain Reaction; Purinergic P1 Receptor Agonists; Rats; Receptor, Adenosine A2A; Receptors, Purinergic P1; Recombinant Proteins; Sulfonamides

1997
Modulation by extracellular Cl- of volume-activated organic osmolyte and halide permeabilities in HeLa cells.
    The American journal of physiology, 1997, Volume: 273, Issue:3 Pt 1

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Cell Membrane Permeability; Chloride Channels; Chlorides; Colforsin; HeLa Cells; Humans; Kinetics; Osmolar Concentration; Radioisotope Dilution Technique; Tamoxifen; Taurine; Tritium; Water-Electrolyte Balance

1997
Inhibitory effect of dideoxyforskolin on cell death induced by ricin, modeccin, diphtheria toxin, and Pseudomonas toxin in MDCK cells.
    Cell structure and function, 1997, Volume: 22, Issue:5

    Topics: Animals; Apoptosis; Bacterial Toxins; Brefeldin A; Calcium; Cell Death; Cell Line; Colforsin; Cyclopentanes; Diphtheria; DNA Fragmentation; Dogs; Kidney; Lectins; Plant Lectins; Protein Biosynthesis; Protein Synthesis Inhibitors; Proteins; Pseudomonas; Ribosome Inactivating Proteins, Type 2; Ricin

1997
Therapy for X-adrenoleukodystrophy: normalization of very long chain fatty acids and inhibition of induction of cytokines by cAMP.
    Journal of lipid research, 1998, Volume: 39, Issue:5

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenoleukodystrophy; Animals; Astrocytes; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Cytokines; Enzyme Inhibitors; Fatty Acids; Genetic Linkage; Interleukin-1; Isoquinolines; Neuroglia; Oxidation-Reduction; Protein Kinase Inhibitors; Pyrrolidinones; Rats; Rolipram; Sulfonamides; Tumor Necrosis Factor-alpha; X Chromosome

1998
Osmosensitive C1- currents and their relevance to regulatory volume decrease in human intestinal T84 cells: outwardly vs. inwardly rectifying currents.
    The Journal of physiology, 1998, Aug-15, Volume: 511 ( Pt 1)

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Cadmium; Cell Line; Chloride Channels; CLC-2 Chloride Channels; Colforsin; Colonic Neoplasms; Humans; Hypertonic Solutions; Hypotonic Solutions; Intestinal Mucosa; Membrane Potentials; Nerve Tissue Proteins; Osmolar Concentration; Tamoxifen; Tumor Cells, Cultured

1998
Regulation of cyclic AMP level by progesterone in ovariectomized rat neocortex.
    Brain research, 1999, Apr-10, Volume: 824, Issue:2

    Topics: Animals; Colforsin; Cyclic AMP; Dose-Response Relationship, Drug; Female; Neocortex; Ovariectomy; Ovary; Progesterone; Rats; Rats, Sprague-Dawley

1999
FlCRhR/cyclic AMP signaling in myenteric ganglia and calbindin-D28 intrinsic primary afferent neurons involves adenylyl cyclases I, III and IV.
    Brain research, 1999, May-01, Volume: 826, Issue:2

    Topics: Action Potentials; Adenylyl Cyclases; Amidohydrolases; Animals; Antibody Specificity; Blotting, Western; Calbindins; Colforsin; Cyclic AMP; Cyclic AMP-Dependent Protein Kinases; Duodenum; Electrophysiology; Ethylmaleimide; Fluorescent Antibody Technique; Fluorescent Dyes; Ganglia, Autonomic; Guinea Pigs; Isoenzymes; Jejunum; Microscopy, Confocal; Myenteric Plexus; Neuroglia; Neurons; Neurons, Afferent; Peptide-N4-(N-acetyl-beta-glucosaminyl) Asparagine Amidase; S100 Calcium Binding Protein G; Signal Transduction

1999
Voltage-activated K+ channels and membrane depolarization regulate accumulation of the cyclin-dependent kinase inhibitors p27(Kip1) and p21(CIP1) in glial progenitor cells.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Jul-01, Volume: 19, Issue:13

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Cell Cycle Proteins; Cell Division; Cell Lineage; Cerebellum; Colforsin; Cyclin D; Cyclin-Dependent Kinase Inhibitor p21; Cyclin-Dependent Kinase Inhibitor p27; Cyclins; Deferoxamine; Ion Channel Gating; Isoproterenol; Membrane Potentials; Mice; Microtubule-Associated Proteins; Oligodendroglia; Potassium; Potassium Channel Blockers; Potassium Channels; Rats; Rats, Sprague-Dawley; Sirolimus; Stem Cells; Tetraethylammonium; Tumor Suppressor Proteins; Veratridine

1999
Effect of protein kinase A-induced phosphorylation on the gating mechanism of the brain Na+ channel: model fitting to whole-cell current traces.
    Biophysical journal, 1999, Volume: 77, Issue:1

    Topics: Animals; Brain; Cells, Cultured; Colforsin; Computer Simulation; Cyclic AMP-Dependent Protein Kinases; Dopamine and cAMP-Regulated Phosphoprotein 32; Electrophysiology; Enzyme Inhibitors; Ion Channel Gating; Kinetics; Nerve Tissue Proteins; Patch-Clamp Techniques; Phosphoprotein Phosphatases; Phosphoproteins; Phosphorylation; Rats; Rats, Wistar; Sodium Channels

1999
Anion channel blockers differentially affect T-type Ca(2+) currents of mouse spermatogenic cells, alpha1E currents expressed in Xenopus oocytes and the sperm acrosome reaction.
    Developmental genetics, 1999, Volume: 25, Issue:2

    Topics: Acrosome Reaction; Animals; Base Sequence; Calcium Channels; Colforsin; DNA Primers; DNA, Complementary; Female; In Vitro Techniques; Ion Channels; Male; Mice; Molecular Sequence Data; Niflumic Acid; Nitrobenzoates; Oocytes; Rats; Sequence Homology, Nucleic Acid; Spermatozoa; Xenopus laevis; Zona Pellucida

1999
Adenylate cyclase and potassium channels are involved in forskolin- and 1,9-dideoxyforskolin-induced inhibition of pregnant rat uterus contractility.
    American journal of obstetrics and gynecology, 2000, Volume: 182, Issue:3

    Topics: Adenylyl Cyclases; Animals; Colforsin; Female; In Vitro Techniques; Potassium Channels; Pregnancy; Quaternary Ammonium Compounds; Rats; Rats, Sprague-Dawley; Uterine Contraction; Uterus

2000
Volume sensitive efflux of taurine in HEK293 cells overexpressing phospholemman.
    Biochimica et biophysica acta, 2000, Apr-17, Volume: 1496, Issue:2-3

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Cell Line; Cell Size; Colforsin; Down-Regulation; Humans; Iodine Radioisotopes; Ion Channels; Membrane Proteins; Nitrobenzoates; Osmolar Concentration; Phosphoproteins; Taurine; Transfection; Tritium

2000
Interaction of cyclic AMP modulating agents with levcromakalim in the relaxation of rat isolated mesenteric artery.
    European journal of pharmacology, 2000, Jul-28, Volume: 401, Issue:1

    Topics: Adenosine-5'-(N-ethylcarboxamide); Animals; Bucladesine; Colforsin; Cromakalim; Cyclic AMP; Dose-Response Relationship, Drug; Drug Interactions; Glyburide; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; Rats; Rats, Wistar; Thionucleotides; Vasoconstrictor Agents; Vasodilation; Vasodilator Agents

2000
Pharmacological characterization of volume-sensitive, taurine permeable anion channels in rat supraoptic glial cells.
    British journal of pharmacology, 2000, Volume: 130, Issue:8

    Topics: 4,4'-Diisothiocyanostilbene-2,2'-Disulfonic Acid; Acetophenones; Adenosine Triphosphate; Animals; Calcium Channel Blockers; Chloride Channels; Colforsin; Diffusion; Dose-Response Relationship, Drug; Gene Expression; In Situ Hybridization; Ion Channels; Male; Mibefradil; Neuroglia; Niflumic Acid; Nitrobenzoates; ortho-Aminobenzoates; Osmotic Pressure; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Supraoptic Nucleus; Tamoxifen; Taurine

2000
Contribution of the IsK (MinK) potassium channel subunit to regulatory volume decrease in murine tracheal epithelial cells.
    The Journal of biological chemistry, 2000, Nov-10, Volume: 275, Issue:45

    Topics: Animals; Anti-Arrhythmia Agents; Apamin; Barium; Calcium Channels; Cells, Cultured; Cilia; Colforsin; Electrophysiology; Epithelial Cells; Mice; Mice, Knockout; Potassium Channels; Potassium Channels, Voltage-Gated; Quaternary Ammonium Compounds; Tamoxifen; Tetraethylammonium; Time Factors; Trachea

2000
Differential actions of PKA and PKC in the regulation of glutamate release by group III mGluRs in the entorhinal cortex.
    Journal of neurophysiology, 2001, Volume: 85, Issue:2

    Topics: Adenine; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Cyclopentanes; Entorhinal Cortex; Enzyme Activation; Enzyme Inhibitors; Excitatory Amino Acid Antagonists; Excitatory Postsynaptic Potentials; Glutamic Acid; Glycine; In Vitro Techniques; Indoles; Isoquinolines; Male; Maleimides; Presynaptic Terminals; Protein Kinase C; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Sulfonamides; Tricarboxylic Acids

2001
Effect of forskolin on acetylcholine-induced current in rat pheochromocytoma cells.
    Acta pharmacologica Sinica, 2000, Volume: 21, Issue:3

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Acetylcholine; Animals; Colforsin; Cyclic AMP-Dependent Protein Kinases; Membrane Potentials; Patch-Clamp Techniques; PC12 Cells; Pheochromocytoma; Rats; Receptors, Nicotinic

2000
The expression and regulation of depolarization-activated K+ channels in the insulin-secreting cell line INS-1.
    Pflugers Archiv : European journal of physiology, 2001, Volume: 442, Issue:1

    Topics: 1-Methyl-3-isobutylxanthine; 4-Aminopyridine; 8-Bromo Cyclic Adenosine Monophosphate; Action Potentials; Animals; Calcium; Colforsin; Electric Conductivity; Gene Expression Regulation; Insulin; Insulin Secretion; Insulinoma; Pancreatic Neoplasms; Potassium Channel Blockers; Potassium Channels; Quaternary Ammonium Compounds; Rats; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetraethylammonium; Tolbutamide; Tumor Cells, Cultured

2001
PKA modulation of Kv4.2-encoded A-type potassium channels requires formation of a supramolecular complex.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Dec-01, Volume: 22, Issue:23

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Amino Acid Substitution; Animals; Binding Sites; Calcium-Binding Proteins; Colforsin; COS Cells; Cyclic AMP-Dependent Protein Kinases; Enzyme Activation; Enzyme Inhibitors; Kv Channel-Interacting Proteins; Macromolecular Substances; Mutagenesis, Site-Directed; Oocytes; Patch-Clamp Techniques; Phosphopeptides; Phosphorylation; Potassium Channels; Potassium Channels, Voltage-Gated; Protein Subunits; Repressor Proteins; Shal Potassium Channels; Structure-Activity Relationship; Transfection; Xenopus laevis

2002
Apoptosis to necrosis switching downstream of apoptosome formation requires inhibition of both glycolysis and oxidative phosphorylation in a BCL-X(L)- and PKB/AKT-independent fashion.
    Cell death and differentiation, 2004, Volume: 11, Issue:3

    Topics: Adenosine Triphosphate; Apoptosis; bcl-X Protein; Blotting, Western; Caspases; Cell Fractionation; Colforsin; Colorimetry; Dose-Response Relationship, Drug; Enzyme Activation; Flow Cytometry; Fluorescent Dyes; Glucose; Glycolysis; Green Fluorescent Proteins; Humans; Jurkat Cells; Kinetics; Lactic Acid; Luminescent Proteins; Microscopy, Confocal; Mitochondria; Necrosis; Oxidative Phosphorylation; Protein Serine-Threonine Kinases; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-akt; Proto-Oncogene Proteins c-bcl-2; Rhodamines

2004
Induction of drug metabolism by forskolin: the role of the pregnane X receptor and the protein kinase a signal transduction pathway.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 312, Issue:2

    Topics: Animals; Blotting, Northern; Cells, Cultured; Colforsin; Cyclic AMP-Dependent Protein Kinases; Hepatocytes; Mice; Pharmaceutical Preparations; Phosphorylation; Plant Extracts; Plasmids; Pregnane X Receptor; Receptors, Cytoplasmic and Nuclear; Receptors, Steroid; Reverse Transcriptase Polymerase Chain Reaction; RNA; Signal Transduction; Transfection; Xenobiotics

2005
Analysis of glycoproteins in human colon cancers, normal tissues and in human colon carcinoma cells reactive with monoclonal antibody NCL-19-9.
    Oncology reports, 2005, Volume: 14, Issue:3

    Topics: Aged; Antibodies, Monoclonal; CA-19-9 Antigen; Cell Line, Tumor; Cell Proliferation; Colforsin; Colon; Colonic Neoplasms; Female; Glycoproteins; Humans; Immunoblotting; Male; Middle Aged; Molecular Weight

2005
Block of spontaneous termination of paroxysmal depolarizations by forskolin (buccal ganglia, Helix pomatia).
    Neuroscience letters, 2006, Jan-09, Volume: 392, Issue:1-2

    Topics: Action Potentials; Animals; Colforsin; Drug Interactions; Electric Stimulation; Epilepsy; Ganglia, Invertebrate; Helix, Snails; Models, Neurological; Neurons; Pentylenetetrazole; Time Factors

2006
Synthetic transformation of ptychantin into forskolin and 1,9-dideoxyforskolin.
    The Journal of organic chemistry, 2006, Jun-09, Volume: 71, Issue:12

    Topics: Adenylyl Cyclases; Colforsin; Diterpenes; Glucose Transport Proteins, Facilitative

2006
Tamoxifen does not inhibit the swell activated chloride channel in human neutrophils during the respiratory burst.
    Biochemical and biophysical research communications, 2008, Oct-31, Volume: 375, Issue:4

    Topics: Cells, Cultured; Chloride Channels; Colforsin; Humans; N-Formylmethionine Leucyl-Phenylalanine; NADPH Oxidases; Neutrophils; Phloretin; Respiratory Burst; Superoxides; Tamoxifen; Tetradecanoylphorbol Acetate; Trialkyltin Compounds

2008
The adenylyl cyclase-cAMP system suppresses TARC/CCL17 and MDC/CCL22 production through p38 MAPK and NF-kappaB in HaCaT keratinocytes.
    Molecular immunology, 2009, Volume: 46, Issue:10

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adenine; Adenylyl Cyclases; Bucladesine; Chemokine CCL17; Chemokine CCL22; Colforsin; Cyclic AMP; Enzyme Activation; Humans; Interferon-gamma; Keratinocytes; Models, Immunological; NF-kappa B; p38 Mitogen-Activated Protein Kinases; STAT1 Transcription Factor; Thionucleotides; Tumor Necrosis Factor-alpha

2009
Extracellular osmolarity modulates G protein-coupled receptor-dependent ATP release from 1321N1 astrocytoma cells.
    American journal of physiology. Cell physiology, 2010, Volume: 298, Issue:2

    Topics: Adenosine Triphosphate; Anions; Astrocytoma; Calcium Signaling; Carbenoxolone; Cell Line, Tumor; Chelating Agents; Colforsin; Dose-Response Relationship, Drug; Egtazic Acid; Enzyme Activation; Extracellular Fluid; Humans; Hypertonic Solutions; Hypotonic Solutions; Ion Channels; Kinetics; Osmolar Concentration; Probenecid; Receptor, PAR-1; rho GTP-Binding Proteins; Tetanus Toxin; Thrombin

2010
Suppression of GLUT1; a new strategy to prevent diabetic complications.
    Journal of cellular physiology, 2013, Volume: 228, Issue:2

    Topics: Animals; beta-Crystallin B Chain; Blood Glucose; Brain; Brain Chemistry; Colforsin; Diabetes Mellitus, Experimental; Diabetic Retinopathy; Erythrocytes; Gene Knockdown Techniques; Gene Silencing; Genistein; Glucose; Glucose Transporter Type 1; Male; Mice; Protein Kinase Inhibitors; Retina; Superoxides; Vascular Endothelial Growth Factor A

2013
Forskolin suppresses delayed-rectifier K+ currents and enhances spike frequency-dependent adaptation of sympathetic neurons.
    PloS one, 2015, Volume: 10, Issue:5

    Topics: Adaptation, Physiological; Animals; Cells, Cultured; Colforsin; Cyclic AMP; Delayed Rectifier Potassium Channels; Dose-Response Relationship, Drug; HEK293 Cells; Humans; Male; Membrane Potentials; Neurons; Rats; Shab Potassium Channels; Signal Transduction; Superior Cervical Ganglion

2015