cocaine and vanoxerine

cocaine has been researched along with vanoxerine in 190 studies

Research

Studies (190)

TimeframeStudies, this research(%)All Research%
pre-19905 (2.63)18.7374
1990's105 (55.26)18.2507
2000's67 (35.26)29.6817
2010's12 (6.32)24.3611
2020's1 (0.53)2.80

Authors

AuthorsStudies
Boja, JW; Carroll, FI; Kuhar, MJ; Lewin, AH1
Allen, AC; George, C; Izenwasser, S; Katz, JL; Kline, RH; Newman, AH1
Allen, AC; Izenwasser, S; Katz, JL; Newman, AH1
Goodman, MM; Kabalka, GW; Kung, HF; Kung, MP; Switzer, R1
Baldessarini, RJ; Gao, Y; Kula, NS; Milius, RA; Neumeyer, JL; Tamagnan, G; Wang, S1
de Costa, BR; Dersch, CM; Glowa, JR; Matecka, D; Partilla, JS; Pert, A; Radesca, L; Rice, KC; Rothman, RB; Wojnicki, FH1
Bowen, WD; Husbands, SM; Izenwasser, S; Katz, JL; Kopajtic, T; Newman, AH; Vilner, BJ1
Beardsley, PM; Dutta, AK; Fei, XS; Newman, JL; Reith, ME1
Cao, J; Husbands, SM; Katz, JL; Kopajtic, T; Newman, AH1
Beardsley, PM; Cook, CD; Davis, MC; Dutta, AK; Fei, XS; Reith, ME1
Bradley, AL; Izenwasser, S; Klein-Stevens, C; Trudell, ML; Wade, D; Zhu, N1
Beardsley, PM; Cook, C; Davis, M; Dutta, AK; George, C; Ghorai, SK; Reith, ME; Venkataraman, SK1
Dutta, AK; Reith, ME; Zhang, S1
Dutta, AK; George, C; Ghorai, SK; Kolhatkar, RB; Reith, ME1
Bowen, WD; Cao, J; George, C; Husbands, SM; Katz, JL; Kopajtic, T; Kulkarni, SS; Newman, AH; Williams, W1
Budygin, EA; Byrd, GD; Childers, SR; Harp, JJ; Jones, SR; Lapa, AA; Lapa, GB1
Chang, LT; Dersch, CM; Hsin, LW; Jacobson, AE; Rice, KC; Rothman, RB1
Bakare, OM; Bi, GH; Bonifazi, A; Burzynski, C; Cao, J; Ellenberger, MP; He, Y; Kopajtic, T; Loland, CJ; Newman, AH; Rais, R; Slack, RD; Slusher, BS; Xi, ZX; Yano, H1
Herkenham, M; Hurd, YL1
Bergman, J; Madras, BK; Rosenzweig-Lipson, S; Spealman, RD1
Kuribara, H; Tadokoro, S; Uchihashi, Y1
Akunne, HC; de Costa, BR; Jacobson, AE; Rice, KC; Rothman, RB1
Bush, LG; Gibb, JW; Hanson, GR; Johnson, M; Midgley, L1
Carroll, FI; De Costa, BR; Grieg, N; Kim, A; Pert, A; Rice, KC; Rothman, RB1
De Montis, G; Devoto, P; Tagliamonte, A1
Borowsky, B; Kuhn, CM1
Bush, LG; Gibb, JW; Hanson, GR; Johnson, M1
Byrd, LD; Howell, LL1
Melia, KF; Spealman, RD1
Brownstein, MJ; Chen, C; Hoffman, BJ; Mezey, E; Usdin, TB1
Cox, BM; Izenwasser, S; Jacocks, HM; Werling, LL1
Akunne, H; deCosta, BR; Grieg, N; Mele, A; Pert, A; Reid, AA; Rice, KC; Rothman, RB; Thurkauf, A1
Callahan, PM; Cunningham, KA1
Baldo, BA; Kelley, AE1
Akunne, HC; de Costa, BR; Greig, N; Mele, A; Pert, A; Reid, AA; Rice, KC; Rothman, RB; Thurkauf, A1
Gale, K; Meloni, R1
Kuhar, MJ; Pögün, S; Scheffel, U1
Arroyo, J; Berger, P; Elsworth, JD; Roth, RH1
Bush, L; Gibb, JW; Hanson, GR; Johnson, M; Smiley, PL1
Bannon, MJ; Dragovic, LJ; Kapatos, G; Shibata, K; Xue, CH1
Cox, BM; Izenwasser, S; Werling, LL1
Garrett, MC; Soares-da-Silva, P1
Anthony, EW; Kleven, MS; Woolverton, WL1
Bergman, J; Johnson, SE; Madras, BK; Spealman, RD1
Andersen, PH1
Kruk, ZL; Millar, J; Stamford, JA1
Akunne, H; Greig, N; Mele, A; Pert, A; Reid, AA; Rice, KC; Rothman, RB; Thurkauf, A1
Debler, EA; Hashim, A; Lajtha, A; Sershen, H1
Spealman, RD1
Edwards, MA; Kantak, KM; Spealman, RD1
Tella, SR2
al-Tikriti, MS; Baldwin, RM; Laruelle, M; Malison, RT; Neumeyer, JL; Sybirska, EH; Wisniewski, G; Zea-Ponce, Y; Zimmermann, RC; Zoghbi, SS1
Essman, WD; Lucki, I; Singh, A1
Kling-Petersen, T; Ljung, E; Svensson, K1
Callaway, CW; Geyer, MA; Paulus, MP1
Coffey, LL; Reith, ME; Xu, C1
Goldberg, SR; Tella, SR2
Brinjak, R; Chrapusta, SJ; Hitri, A; Karoum, F; Wyatt, RJ1
Meiergerd, SM; Schenk, JO1
Coen, KM; Corrigall, WA1
Kelley, AE; Maldonado-Irizarry, CS; Stellar, JR1
Baumann, MH; Char, GU; De Costa, BR; Rice, KC; Rothman, RB1
Masserano, JM; Venable, D; Wyatt, RJ1
Dutta, AK; Madras, BK; Meltzer, PC; Reith, ME1
Erwin, VG; Jones, BC; Womer, DE1
Kameyama, T; Mori, E; Ukai, M1
Cheng, CH; Costall, B; Naylor, RJ; Rudd, JA1
Chuang, EJ; Draisci, G; Gu, J; Hoo, Y; Iadarola, MJ; Silverthorn, M; Yeung, CL1
Henry, DJ; Hu, XT; White, FJ1
Berger, P; Elsworth, JD; Roth, RH; Taylor, JR1
Skjoldager, P; Winger, G; Woods, JH1
Bergmann, JS; Gifford, AN; Johnson, KM1
Butler, T; Dobbie, JW; Duffield, R; Hjelle, JT; Ho, AK; Miller-Hjelle, MA; Reith, M; Steidley, KR1
Chen, NH; Coffey, LL; Reith, ME; Xu, C1
Dow-Edwards, DL; Frick, GS1
Sivam, SP1
Glowa, JR; Wojnicki, FH1
Glowa, JR; Koetzner, L; Riley, AL1
Brockington, A; Carrol, FI; Elmer, GI; Goldberg, SR; Gorelick, DA; Matecka, D; Rice, KC; Rothman, RB1
Andrews, AM; Cadet, JL; Goldberg, SR; Ladenheim, B; Tella, SR1
Bekavac, I; Gould, EM; Waterhouse, BD1
Fantegrossi, WE; Glowa, JR; Lewis, DB; Matecka, D; Rice, KC; Rothman, RB1
Koob, GF; Parsons, LH; Weiss, F1
Coffey, LL; Dutta, AK; Reith, ME2
Dersch, CM; DeVries, AC; Glowa, JR; Lewis, D; Matecka, D; Pert, A; Rice, KC; Rothman, RB; Wojnicki, FH1
Carroll, FI; Holmquist, CR; Kepler, JA; Kuhar, MJ; Saindane, AM; Scheffel, U; Taylor, GF; Zhan, Y1
Francis, R; Kuhn, C1
Glowa, JR; Matecka, D; Rice, KC; Rothman, RB1
Glowa, JR1
Gorelick, DA1
Gan, Q; Knuepfer, MM1
Bender, M; Drago, J; Rivkees, SA1
Izenwasser, S; Kunko, PM; Loeloff, RJ1
Dannals, RF; Liu, X; Mochizuki, T; Musachio, JL; Scheffel, U; Villemagne, VL; Wagner, HN1
Di Chiara, G; Frau, R; Pontieri, FE; Tanda, G1
Geter-Douglass, B; Tirelli, E; Witkin, JM1
Serrão, MP; Soares-Da-Silva, P; Vieira-Coelho, MA1
Gong, W; Justice, JB; Neill, DB1
Agoston, GE; Newman, AH1
Dutta, AK; Reith, ME; Xu, C1
Holtzman, SG; Waddell, AB1
Higgins, GA; Varty, GB1
Misawa, M; Mori, T; Onodera, K; Suzuki, T; Tsuji, M1
Berger, R; Brust, P; Hoepping, A; Johannsen, B; Leibnitz, P; Machill, S; Scheller, D; Spies, H1
Steketee, JD1
Booij, J; de Bruin, K; Janssen, AG; Knol, RJ; Reneman, L; van Royen, EA1
Glowa, JR; Rice, KC; Rothman, RB; Wojnicki, FH1
Gasior, M; Goldberg, SR; Jaszyna, M; Shoaib, M; Yasar, S1
Dannals, RF; Matecka, D; Rice, KC; Rothman, RB; Villemagne, VL; Wong, DF; Yokoi, F1
Dow-Edwards, D; Shi, X; Yin, R1
Carroll, FI; Damaj, MI; Martin, BR; Slemmer, JE1
Miller, DK; Nation, JR1
Binnekade, R; De Vries, TJ; Schoffelmeer, AN; Vanderschuren, LJ1
Grech, DM; Platt, DM; Rowlett, JK; Spealman, RD1
Carroll, FI; French, D; Izenwasser, S; Kunko, PM1
Besnard, JC; Chalon, S; Emond, P; Garreau, L; Guilloteau, D; Vilar, MP; Zimmer, L1
Harada, N; Kakiuchi, T; Nakanishi, S; Nishiyama, S; Ohba, H; Sato, K; Tsukada, H1
Baldessarini, RJ; Fisser, R; Kula, NS; Neumeyer, JL; Tarazi, FI; Trometer, J; Wang, S1
Besnard, JC; Bottlaender, M; Chalon, S; Coulon, C; Emond, P; Frangin, Y; Fuseau, C; Guenther, I; Guilloteau, D; Helfenbein, J; Loc'h, C; Maziere, B; Ottaviani, M1
Carrol, FI; Czoty, PW; Howell, LL; Kuhar, MJ1
Harada, N; Kakiuchi, T; Nishiyama, S; Ohba, H; Tsukada, H2
Czoty, PW; Howell, LL; Justice, JB1
Kaneda, S; Kato, B; Kawai, Y; Matsushita, H; Nishi, M; Noritake, K; Sorimachi, Y; Takeuchi, Y; Ueda, S; Yang, Y; Yasuhara, M; Yoshimoto, K1
Brezausek, C; Moore, JF; Percy, AK; Theibert, A; Zachor, DA1
Wirtshafter, D1
Davidson, C; Douglas, SB; Ellinwood, EH; Lee, TH1
Baniecki, M; Collins, HA; Hanson, RN; Hinerth, MA; Waszczak, BL1
Carboni, E; Di Chiara, G; Rolando, MT; Silvagni, A1
Brodde, OE; Leineweber, K; Seyfarth, T1
Hashim, A; Lajtha, A; Sershen, H1
Glowa, JR; Lewis, DB; Rice, KC; Stafford, D1
Glowa, JR; LeSage, MG; Rice, KC; Stafford, D1
Dutta, AK; Madras, BK; Reith, ME1
Cox, BM; D'Addario, C; Ferri, S; Izenwasser, S; Romualdi, P1
Carboni, E; Di Chiara, G; Giros, B; Nosten-Bertrand, M; Spielewoy, C; Vacca, C1
Agoston, GE; Hecht, GS; Katz, JL; Newman, AH; Woolverton, WL1
Baek, D; Bergstrom, DA; Freeman, LE; Ruskin, DN; Walters, JR1
Holtzman, SG1
Busidan, Y; Dow-Edwards, DL1
Platt, DM; Rowlett, JK; Spealman, RD2
Garland, T; Girard, I; Hosack, GR; Kelley, AE; Mitchell, GS; Rhodes, JS1
Cornish, JL; Kalivas, PW1
Brockington, A; Hope, BT; Morón, JA; Rocha, BA; Wise, RA1
Schenk, S1
Hanania, T; Zahniser, NR1
Carmona, GN; Schindler, CW1
Cadet, JL; Carroll, FI; Collins, SL; Izenwasser, S; Kunko, PM; Ladenheim, B1
Fukumoto, D; Harada, N; Kakiuchi, T; Nishiyama, S; Satoh, K; Tsukada, H1
Davidson, C; Ellinwood, EH; King, GR; Lee, TH; Yu, GZ1
Dersch, CM; Horel, R; Hsin, LW; Jacobson, AE; Prisinzano, T; Rice, KC; Rothman, RB; Wilkerson, CR1
Janak, PH; Mcgeehan, AJ; Olive, MF1
Gasior, M; Kaminski, R; Witkin, JM1
Bergman, J; Czoty, PW; Makriyannis, A1
Chen, N; Reith, ME; Zhen, J1
Hagino, Y; Hall, FS; Ikeda, K; Kobayashi, H; Lesch, KP; Murphy, DL; Shen, HW; Shinohara-Tanaka, K; Sora, I; Uhl, GR; Yamamoto, H; Yamamoto, T1
Steketee, JD; Williams, JM1
Candeletti, S; D'Addario, C; Di Benedetto, M; Feliciani, D; Izenwasser, S; Romualdi, P1
Barrett, AC; Caine, SB; Dohrmann, JM; Miller, JR1
Chen, N; Dutta, AK; Maiti, S; Reith, ME; Zhen, J1
Dutta, AK; Reith, ME; Wang, LC1
Boos, TL; Calhoun, WJ; Dersch, CM; Greiner, E; Jacobson, AE; Nightingale, B; Rice, KC; Rothman, RB1
Desai, RI; French, D; Katz, JL; Kopajtic, TA; Newman, AH1
Bronius, PF; Brueggeman, RJ; Schoffelmeer, AN; van Gaalen, MM; Vanderschuren, LJ1
Bevins, RA; Linkugel, JD; Reichel, CM1
Fagerholm, V; Grönroos, T; Haaparanta, M; Koivula, T; Lipponen, T; Marjamäki, P; Perhola, O; Solin, O; Vepsäläinen, J1
España, RA; Jones, SR; Roberts, DC1
Aksenov, MY; Aksenova, MV; Booze, RM; Mactutus, CF; Silvers, JM1
Cao, J; Katz, JL; Kopajtic, T; Newman, AH1
Chen, N; Dutta, AK; Kharkar, P; Mishra, M; Reith, ME; Schmitt, KC; Zhen, J1
Hall, FS; Jones, JD; Rice, K; Riley, AL; Uhl, GR1
Cain, SM; Dewar, D; Duncan, R; Patterson, J; Pimlott, S; Ruest, T; Sills, GJ1
Bergman, J; Desai, R; Desai, RI; Martin, J; Paronis, CA1
Aragona, BJ; Carelli, RM; Kile, BM; Park, J; Wightman, RM1
Donovan, DM; Katz, JL; Kopajtic, TA; Liu, Y; Newman, AH; Surratt, CK1
Briscione, MA; Rice, KC; Riley, AL; Serafine, KM1
Conover, K; Cossette, MP; Hernandez, G; Shizgal, P; Trujillo-Pisanty, I1
Palmiter, RD; Whiddon, BB1
Achterberg, EJ; Schoffelmeer, AN; Schrama, L; Siviy, SM; Trezza, V; Vanderschuren, LJ1
Chang, SC; Folsom, RJ; Jang, EY; Kim, HY; Kim, KJ; Kim, SH; Lee, BH; Ryu, YH; Schilaty, ND; Steffensen, SC; Yang, CH; Yeo, MJ1
Huang, X; Midde, NM; Quizon, PM; Sun, WL; Yuan, Y; Zhan, CG; Zhu, J1
Aalderink, M; Achterberg, EJ; Driel, NV; Houwing, DJ; Servadio, M; Trezza, V; van Kerkhof, LW; van Swieten, MM; Vanderschuren, LJ1
Desai, RI; Katz, JL; Slezak, JM1
Budygin, EA; Costa, F; Gerasimova, EV; Grinevich, VP; Kalueff, AV; Kolesnikova, TO; Maslov, GO; Viktorova, YA; Zabegalov, KN1
Grundt, P; Katz, JL; Kopajtic, T; Kulkarni, SS; Newman, AH1
Beardsley, PM; Cook, CD; Deschamps, J; Dutta, AK; Ghorai, SK; Kolhatkar, R; Reith, ME1

Reviews

3 review(s) available for cocaine and vanoxerine

ArticleYear
Cocaine receptor: biochemical characterization and structure-activity relationships of cocaine analogues at the dopamine transporter.
    Journal of medicinal chemistry, 1992, Mar-20, Volume: 35, Issue:6

    Topics: Animals; Binding Sites; Binding, Competitive; Carrier Proteins; Cocaine; Dopamine; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Humans; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Receptors, Drug; Stereoisomerism; Structure-Activity Relationship

1992
Dopamine, serotonin and tachykinin in self-injurious behavior.
    Life sciences, 1996, May-24, Volume: 58, Issue:26

    Topics: Animals; Cocaine; Dopamine; Humans; Lesch-Nyhan Syndrome; Piperazines; Rats; Self-Injurious Behavior; Serotonin; Tachykinins

1996
Novel benztropine [3a-(diphenylmethoxy)tropane] analogs as probes for the dopamine transporter.
    Current medicinal chemistry, 1998, Volume: 5, Issue:4

    Topics: Benztropine; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Design; Humans; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Stereoisomerism; Structure-Activity Relationship; Substance-Related Disorders

1998

Trials

1 trial(s) available for cocaine and vanoxerine

ArticleYear
Differential sensitivity to acute administration of cocaine, GBR 12909, and fluoxetine in mice selectively bred for hyperactive wheel-running behavior.
    Psychopharmacology, 2001, Volume: 158, Issue:2

    Topics: Animals; Animals, Outbred Strains; Breeding; Cocaine; Crosses, Genetic; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Female; Fluoxetine; Hyperkinesis; Injections, Intraperitoneal; Male; Mice; Mice, Inbred ICR; Piperazines

2001

Other Studies

186 other study(ies) available for cocaine and vanoxerine

ArticleYear
Novel 4'-substituted and 4',4"-disubstituted 3 alpha-(diphenylmethoxy)tropane analogs as potent and selective dopamine uptake inhibitors.
    Journal of medicinal chemistry, 1995, Sep-29, Volume: 38, Issue:20

    Topics: Animals; Cocaine; Dopamine Uptake Inhibitors; Male; Radioligand Assay; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Tropanes

1995
Novel 3 alpha-(diphenylmethoxy)tropane analogs: potent dopamine uptake inhibitors without cocaine-like behavioral profiles.
    Journal of medicinal chemistry, 1994, Jul-22, Volume: 37, Issue:15

    Topics: Animals; Behavior, Animal; Benztropine; Cocaine; Dopamine Antagonists; Mice; Rats; Structure-Activity Relationship; Tropanes

1994
Synthesis and characterization of radioiodinated N-(3-iodopropen-1-yl)-2 beta-carbomethoxy-3 beta-(4-chlorophenyl)tropanes: potential dopamine reuptake site imaging agents.
    Journal of medicinal chemistry, 1994, May-13, Volume: 37, Issue:10

    Topics: Animals; Binding, Competitive; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Iodine Radioisotopes; Isotope Labeling; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Protein Binding; Rats; Rats, Sprague-Dawley; Stereoisomerism; Tissue Distribution; Tomography, Emission-Computed, Single-Photon; Tropanes

1994
N-substituted analogs of 2 beta-carbomethoxy-3 beta- (4'-iodophenyl)tropane (beta-CIT) with selective affinity to dopamine or serotonin transporters in rat forebrain.
    Journal of medicinal chemistry, 1996, Jan-19, Volume: 39, Issue:2

    Topics: Animals; Binding Sites; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Magnetic Resonance Spectroscopy; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Probes; Nerve Tissue Proteins; Prosencephalon; Radioligand Assay; Rats; Serotonin; Serotonin Plasma Membrane Transport Proteins; Spectrometry, Mass, Fast Atom Bombardment

1996
Development of novel, potent, and selective dopamine reuptake inhibitors through alteration of the piperazine ring of 1-[2-(diphenylmethoxy)ethyl]-and 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazines (GBR 12935 and GBR 12909).
    Journal of medicinal chemistry, 1996, Nov-22, Volume: 39, Issue:24

    Topics: Animals; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Design; Magnetic Resonance Spectroscopy; Mass Spectrometry; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Conformation; Molecular Structure; Nerve Tissue Proteins; Piperazines; Rats; Receptors, Drug; Serotonin; Substance-Related Disorders

1996
Structure-activity relationships at the monoamine transporters and sigma receptors for a novel series of 9-[3-(cis-3, 5-dimethyl-1-piperazinyl)propyl]carbazole (rimcazole) analogues.
    Journal of medicinal chemistry, 1999, Oct-21, Volume: 42, Issue:21

    Topics: Aniline Compounds; Animals; Brain; Carbazoles; Carrier Proteins; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Guinea Pigs; In Vitro Techniques; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Norepinephrine Plasma Membrane Transport Proteins; Piperazines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, sigma; Serotonin Plasma Membrane Transport Proteins; Structure-Activity Relationship; Symporters

1999
Structure-activity relationship studies of 4-[2-(diphenylmethoxy)ethyl]-1-benzylpiperidine derivatives and their N-analogues: evaluation of O-and N-analogues and their binding to monoamine transporters.
    Journal of medicinal chemistry, 2001, Mar-15, Volume: 44, Issue:6

    Topics: Animals; Carrier Proteins; Cocaine; Discrimination Learning; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Motor Activity; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Piperidines; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Plasma Membrane Transport Proteins; Structure-Activity Relationship; Symporters

2001
[3-cis-3,5-Dimethyl-(1-piperazinyl)alkyl]-bis-(4'-fluorophenyl)amine analogues as novel probes for the dopamine transporter.
    Bioorganic & medicinal chemistry letters, 2001, Dec-17, Volume: 11, Issue:24

    Topics: Animals; Carbazoles; Cocaine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Probes; Nerve Tissue Proteins; Piperazines; Rats

2001
Expansion of structure-activity studies of piperidine analogues of 1-[2-(diphenylmethoxy)ethyl]-4-(3-phenylpropyl)piperazine (GBR 12935) compounds by altering substitutions in the N-benzyl moiety and behavioral pharmacology of selected molecules.
    Journal of medicinal chemistry, 2002, Jan-31, Volume: 45, Issue:3

    Topics: Animals; Binding, Competitive; Brain; Carrier Proteins; Cocaine; Discrimination Learning; Dopamine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Ligands; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Motor Activity; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Piperazines; Piperidines; Radioligand Assay; Rats; Serotonin; Serotonin Plasma Membrane Transport Proteins; Structure-Activity Relationship; Symporters

2002
Synthesis and dopamine transporter binding affinities of 3alpha-benzyl-8-(diarylmethoxyethyl)-8-azabicyclo[3.2.1]octanes.
    Bioorganic & medicinal chemistry letters, 2002, Sep-02, Volume: 12, Issue:17

    Topics: Bridged Bicyclo Compounds; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Humans; Membrane Glycoproteins; Membrane Transport Modulators; Membrane Transport Proteins; Nerve Tissue Proteins; Octanes; Protein Binding; Structure-Activity Relationship

2002
High affinity hydroxypiperidine analogues of 4-(2-benzhydryloxyethyl)-1-(4-fluorobenzyl)piperidine for the dopamine transporter: stereospecific interactions in vitro and in vivo.
    Journal of medicinal chemistry, 2003, Mar-27, Volume: 46, Issue:7

    Topics: Animals; Benzhydryl Compounds; Carrier Proteins; Cerebral Cortex; Cocaine; Corpus Striatum; Crystallography, X-Ray; Discrimination Learning; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; In Vitro Techniques; Ligands; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Molecular Structure; Motor Activity; Nerve Tissue Proteins; Norepinephrine Plasma Membrane Transport Proteins; Piperidines; Radioligand Assay; Rats; Serotonin Plasma Membrane Transport Proteins; Stereoisomerism; Structure-Activity Relationship; Symporters

2003
Design, synthesis, and activity of novel cis- and trans-3,6-disubstituted pyran biomimetics of 3,6-disubstituted piperidine as potential ligands for the dopamine transporter.
    Bioorganic & medicinal chemistry letters, 2003, May-05, Volume: 13, Issue:9

    Topics: Animals; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Ligands; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperidines; Pyrans; Rats; Stereoisomerism; Structure-Activity Relationship

2003
Interaction of cis-(6-benzhydrylpiperidin-3-yl)benzylamine analogues with monoamine transporters: structure-activity relationship study of structurally constrained 3,6-disubstituted piperidine analogues of (2,2-diphenylethyl)-[1-(4-fluorobenzyl)piperidin-
    Journal of medicinal chemistry, 2003, May-22, Volume: 46, Issue:11

    Topics: Animals; Binding, Competitive; Biogenic Monoamines; Biological Transport; Brain; Carrier Proteins; Crystallography, X-Ray; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Conformation; Nerve Tissue Proteins; Nitriles; Norepinephrine Plasma Membrane Transport Proteins; Piperazines; Piperidines; Radioligand Assay; Rats; Serotonin Plasma Membrane Transport Proteins; Stereoisomerism; Structure-Activity Relationship; Symporters

2003
Dual probes for the dopamine transporter and sigma1 receptors: novel piperazinyl alkyl-bis(4'-fluorophenyl)amine analogues as potential cocaine-abuse therapeutic agents.
    Journal of medicinal chemistry, 2003, Jun-19, Volume: 46, Issue:13

    Topics: Animals; Binding, Competitive; Brain; Cocaine-Related Disorders; Crystallography, X-Ray; Dopamine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Nerve Tissue Proteins; Piperazines; Radioligand Assay; Rats; Receptors, sigma; Structure-Activity Relationship

2003
The synthesis and biological evaluation of dopamine transporter inhibiting activity of substituted diphenylmethoxypiperidines.
    Bioorganic & medicinal chemistry letters, 2005, Nov-15, Volume: 15, Issue:22

    Topics: Dopamine Plasma Membrane Transport Proteins; Inhibitory Concentration 50; Molecular Structure; Piperidines; Structure-Activity Relationship

2005
Design and synthesis of 2- and 3-substituted-3-phenylpropyl analogs of 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine and 1-[2-(diphenylmethoxy)ethyl]-4-(3-phenylpropyl)piperazine: role of amino, fluoro, hydroxyl, methoxyl, methyl, m
    Journal of medicinal chemistry, 2008, May-08, Volume: 51, Issue:9

    Topics: Dopamine Plasma Membrane Transport Proteins; Piperazines; Radioligand Assay; Serotonin Plasma Membrane Transport Proteins; Stereoisomerism; Structure-Activity Relationship

2008
Novel and High Affinity 2-[(Diphenylmethyl)sulfinyl]acetamide (Modafinil) Analogues as Atypical Dopamine Transporter Inhibitors.
    Journal of medicinal chemistry, 2016, 12-08, Volume: 59, Issue:23

    Topics: Animals; Benzhydryl Compounds; Cells, Cultured; Chlorocebus aethiops; COS Cells; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Humans; Locomotion; Male; Mice; Mice, Inbred C57BL; Microsomes, Liver; Modafinil; Molecular Structure; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship

2016
Influence of a single injection of cocaine, amphetamine or GBR 12909 on mRNA expression of striatal neuropeptides.
    Brain research. Molecular brain research, 1992, Volume: 16, Issue:1-2

    Topics: Amphetamine; Animals; Central Nervous System Stimulants; Cocaine; Corpus Striatum; Dynorphins; Enkephalins; In Situ Hybridization; Male; Neuropeptides; Neurotransmitter Uptake Inhibitors; Piperazines; Rats; Rats, Sprague-Dawley; RNA, Messenger; Substance P

1992
Stereoselective behavioral effects of Lu 19-005 in monkeys: relation to binding at cocaine recognition sites.
    Psychopharmacology, 1992, Volume: 107, Issue:2-3

    Topics: Animals; Behavior, Animal; Binding, Competitive; Carrier Proteins; Cocaine; Conditioning, Operant; Dopamine; Indans; Ligands; Male; Piperazines; Receptors, Drug; Reinforcement Schedule; Saimiri; Stereoisomerism

1992
Assessment of the ambulation-increasing effect of ketamine by coadministration with central-acting drugs in mice.
    Japanese journal of pharmacology, 1992, Volume: 60, Issue:1

    Topics: alpha-Methyltyrosine; Animals; Caffeine; Central Nervous System Agents; Central Nervous System Depressants; Ceruletide; Cocaine; Dizocilpine Maleate; Drug Synergism; Ketamine; Male; Methamphetamine; Methyltyrosines; Mice; Morphine; Motor Activity; Neurotransmitter Uptake Inhibitors; Nimodipine; Piperazines; Scopolamine

1992
[3H] cocaine labels a binding site associated with the serotonin transporter in guinea pig brain: allosteric modulation by paroxetine.
    Neurochemical research, 1992, Volume: 17, Issue:12

    Topics: Allosteric Regulation; Animals; Binding Sites; Brain; Carrier Proteins; Cell Membrane; Cocaine; Guinea Pigs; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Paroxetine; Piperazines; Serotonin; Serotonin Plasma Membrane Transport Proteins; Synaptosomes; Tritium

1992
MK-801 blocks the changes in neurotensin concentrations induced by methamphetamine, 3,4-methylenedioxymethamphetamine, cocaine, and GBR 12909.
    Annals of the New York Academy of Sciences, 1992, Volume: 668

    Topics: 3,4-Methylenedioxyamphetamine; Animals; Cocaine; Dizocilpine Maleate; Male; Methamphetamine; Neurotensin; Piperazines; Rats; Rats, Sprague-Dawley

1992
Cocaine and GBR12909 produce equivalent motoric responses at different occupancy of the dopamine transporter.
    Pharmacology, biochemistry, and behavior, 1992, Volume: 43, Issue:4

    Topics: Animals; Brain; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Male; Membrane Glycoproteins; Membrane Transport Proteins; Motor Activity; Nerve Tissue Proteins; Neurotransmitter Uptake Inhibitors; Nomifensine; Phencyclidine; Piperazines; Rats; Rats, Sprague-Dawley; Stereotyped Behavior

1992
Failure by tricyclic antidepressants to affect the increase of dopamine extracellular concentrations produced by haloperidol in the caudate and accumbens nuclei of rats.
    Biochemical pharmacology, 1992, Feb-04, Volume: 43, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Amphetamine; Animals; Antidepressive Agents, Tricyclic; Caudate Nucleus; Cocaine; Dopamine; Drug Interactions; Haloperidol; Imipramine; Male; Nucleus Accumbens; Piperazines; Rats; Rats, Inbred Strains

1992
Monoamine mediation of cocaine-induced hypothalamo-pituitary-adrenal activation.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 256, Issue:1

    Topics: Adrenocorticotropic Hormone; Animals; Biogenic Monoamines; Cocaine; Corticosterone; Dopamine; Dopamine Antagonists; Haloperidol; Hypothalamo-Hypophyseal System; Injections, Intraperitoneal; Ketanserin; Male; Neurotransmitter Agents; Neurotransmitter Uptake Inhibitors; Piperazines; Pituitary-Adrenal System; Prazosin; Propranolol; Rats; Rats, Inbred Strains; Receptors, Dopamine; Stimulation, Chemical; Time Factors

1991
Role of N-methyl-D-aspartate (NMDA) receptors in the response of extrapyramidal neurotensin and dynorphin A systems to cocaine and GBR 12909.
    Biochemical pharmacology, 1991, Feb-15, Volume: 41, Issue:4

    Topics: Animals; Cocaine; Corpus Striatum; Dizocilpine Maleate; Dynorphins; Male; Neurotensin; Neurotransmitter Uptake Inhibitors; Piperazines; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, N-Methyl-D-Aspartate; Substantia Nigra

1991
Characterization of the effects of cocaine and GBR 12909, a dopamine uptake inhibitor, on behavior in the squirrel monkey.
    The Journal of pharmacology and experimental therapeutics, 1991, Jul-01, Volume: 258, Issue:1

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Behavior, Animal; Cocaine; Dopamine Agents; Drug Interactions; Ergolines; Injections, Intravenous; Male; Neurotransmitter Uptake Inhibitors; Piperazines; Quinpirole; Saimiri; Self Administration

1991
Pharmacological characterization of the discriminative-stimulus effects of GBR 12909.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 258, Issue:2

    Topics: Animals; Cocaine; Discrimination Learning; Dopamine Agents; Male; Neurotransmitter Uptake Inhibitors; Piperazines; Receptors, Dopamine; Saimiri; Salicylamides

1991
Cloning of the cocaine-sensitive bovine dopamine transporter.
    Proceedings of the National Academy of Sciences of the United States of America, 1991, Dec-15, Volume: 88, Issue:24

    Topics: Amino Acid Sequence; Animals; Antisense Elements (Genetics); Base Sequence; Carrier Proteins; Cattle; Cell Line; Cloning, Molecular; Cocaine; Dopamine; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Gene Library; Kinetics; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Sequence Data; Nerve Tissue Proteins; Nucleic Acid Hybridization; Piperazines; RNA; RNA Probes; Sequence Homology, Nucleic Acid; Substantia Nigra; Transfection; Tyrosine 3-Monooxygenase

1991
Comparison of dopamine uptake and release in vitro in sheep and rat striatum.
    Life sciences, 1991, Volume: 49, Issue:7

    Topics: Animals; Cocaine; Corpus Striatum; Dopamine; Dopamine Antagonists; Female; Fluoxetine; In Vitro Techniques; Male; Neurotransmitter Uptake Inhibitors; Norepinephrine; Piperazines; Rats; Rats, Inbred Strains; Receptors, N-Methyl-D-Aspartate; Sheep

1991
Preliminary evidence that the high affinity dopamine reuptake inhibitor, GBR12909, antagonizes the ability of cocaine to elevate extracellular levels of dopamine.
    NIDA research monograph, 1990, Volume: 105

    Topics: Animals; Caudate Nucleus; Cocaine; Dopamine; In Vitro Techniques; Membranes; Neurotransmitter Uptake Inhibitors; Piperazines; Rats

1990
Monoamine reuptake inhibitors enhance the discriminative state induced by cocaine in the rat.
    Psychopharmacology, 1991, Volume: 104, Issue:2

    Topics: Animals; Cocaine; Desipramine; Discrimination, Psychological; Dose-Response Relationship, Drug; Fluoxetine; Male; Monoamine Oxidase Inhibitors; Neurotransmitter Uptake Inhibitors; Piperazines; Rats; Rats, Inbred Strains

1991
Cross-sensitization between cocaine and GBR 12909, a dopamine uptake inhibitor.
    Brain research bulletin, 1991, Volume: 27, Issue:1

    Topics: Analysis of Variance; Animals; Cocaine; Dopamine; Drug Administration Schedule; Drug Interactions; Male; Motor Activity; Neurotransmitter Uptake Inhibitors; Piperazines; Rats; Rats, Inbred Strains; Reference Values

1991
GBR12909 antagonizes the ability of cocaine to elevate extracellular levels of dopamine.
    Pharmacology, biochemistry, and behavior, 1991, Volume: 40, Issue:2

    Topics: Animals; Carrier Proteins; Caudate Nucleus; Chromatography, High Pressure Liquid; Cocaine; Dialysis; Dopamine; Dopamine Plasma Membrane Transport Proteins; Electrochemistry; Extracellular Space; Kinetics; Male; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurotransmitter Uptake Inhibitors; Piperazines; Radioligand Assay; Rats; Rats, Inbred Strains

1991
Cocaine-induced turning behavior in rats with 6-hydroxydopamine lesions: effect of transplants of fetal substantia nigra.
    European journal of pharmacology, 1991, Dec-10, Volume: 209, Issue:1-2

    Topics: Amphetamine; Animals; Apomorphine; Behavior, Animal; Brain Diseases; Brain Tissue Transplantation; Cocaine; Dopamine; Fetal Tissue Transplantation; Fluoxetine; Imipramine; Male; Neural Pathways; Neurotransmitter Uptake Inhibitors; Nomifensine; Oxidopamine; Piperazines; Rats; Rats, Inbred Strains; Substantia Nigra

1991
Cocaine displaces [3H]WIN 35,428 binding to dopamine uptake sites in vivo more rapidly than mazindol or GBR 12909.
    European journal of pharmacology, 1991, Jun-06, Volume: 198, Issue:2-3

    Topics: Animals; Binding Sites; Binding, Competitive; Carrier Proteins; Chromatography, High Pressure Liquid; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Injections, Intravenous; Male; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Nerve Tissue Proteins; Piperazines; Radioimmunoassay; Receptors, Drug

1991
Interaction of [3H]GBR 12935 and GBR 12909 with the dopamine uptake complex in nucleus accumbens.
    European journal of pharmacology, 1990, Feb-20, Volume: 177, Issue:1-2

    Topics: Animals; Binding, Competitive; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Kinetics; Male; Membrane Proteins; Nerve Tissue Proteins; Neurotransmitter Uptake Inhibitors; Nucleus Accumbens; Piperazines; Rats; Rats, Inbred Strains; Septal Nuclei

1990
Effects of cocaine on extrapyramidal and limbic dynorphin systems.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 253, Issue:3

    Topics: Animals; Benzazepines; Cocaine; Dopamine Antagonists; Dynorphins; Extrapyramidal Tracts; Limbic System; Male; Neurotransmitter Uptake Inhibitors; Piperazines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1990
Expression of a human cocaine-sensitive dopamine transporter in Xenopus laevis oocytes.
    Journal of neurochemistry, 1990, Volume: 54, Issue:2

    Topics: Animals; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Humans; Injections; Membrane Glycoproteins; Membrane Proteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurotransmitter Uptake Inhibitors; Oocytes; Piperazines; RNA, Messenger; Substantia Nigra; Xenopus laevis

1990
Comparison of the effects of cocaine and other inhibitors of dopamine uptake in rat striatum, nucleus accumbens, olfactory tubercle, and medial prefrontal cortex.
    Brain research, 1990, Jun-18, Volume: 520, Issue:1-2

    Topics: Animals; Cerebral Cortex; Cocaine; Corpus Striatum; Dopamine; Dopamine Antagonists; Fluoxetine; In Vitro Techniques; Kinetics; Male; Methylphenidate; Nalidixic Acid; Naphthyridines; Neurotransmitter Uptake Inhibitors; Norepinephrine; Nucleus Accumbens; Olfactory Bulb; Piperazines; Rats; Rats, Inbred Strains

1990
Overflow of endogenous dopamine and 3,4-dihydroxyphenylacetic acid from tissues of the rat brain, elicited by electrical stimulation, depolarization by potassium and activation of carrier-mediated release.
    Neuropharmacology, 1990, Volume: 29, Issue:12

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Chromatography, High Pressure Liquid; Cocaine; Corpus Striatum; Dopamine; Electric Stimulation; In Vitro Techniques; Kinetics; Male; Neurons; Neurotransmitter Uptake Inhibitors; Piperazines; Potassium; Rats; Rats, Inbred Strains

1990
Pharmacological characterization of the discriminative stimulus effects of cocaine in rhesus monkeys.
    The Journal of pharmacology and experimental therapeutics, 1990, Volume: 254, Issue:1

    Topics: Animals; Benzazepines; Cocaine; Dextroamphetamine; Discrimination Learning; Female; Haloperidol; Macaca mulatta; Male; Piperazines; Receptors, Dopamine

1990
Effects of cocaine and related drugs in nonhuman primates. III. Self-administration by squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 251, Issue:1

    Topics: Animals; Bupropion; Cocaine; Dopamine; Male; Mazindol; Methylphenidate; Neurotransmitter Uptake Inhibitors; Nomifensine; Piperazines; Propiophenones; Saimiri; Self Administration

1989
The dopamine inhibitor GBR 12909: selectivity and molecular mechanism of action.
    European journal of pharmacology, 1989, Aug-03, Volume: 166, Issue:3

    Topics: Animals; Cocaine; Dopamine; In Vitro Techniques; Kinetics; Male; Mazindol; Methylphenidate; Neurotransmitter Uptake Inhibitors; Piperazines; Rats; Rats, Inbred Strains; Receptors, Dopamine

1989
Dissociation of the actions of uptake blockers upon dopamine overflow and uptake in the rat nucleus accumbens: in vivo voltammetric data.
    Neuropharmacology, 1989, Volume: 28, Issue:12

    Topics: Animals; Benztropine; Bupropion; Cocaine; Dopamine; Electric Stimulation; Electrochemistry; Levodopa; Male; Microelectrodes; Neurotransmitter Uptake Inhibitors; Nomifensine; Nucleus Accumbens; Piperazines; Propiophenones; Rats; Rats, Inbred Strains; Septal Nuclei

1989
Tight binding dopamine reuptake inhibitors as cocaine antagonists. A strategy for drug development.
    FEBS letters, 1989, Nov-06, Volume: 257, Issue:2

    Topics: Animals; Biological Transport; Carrier Proteins; Cell Membrane; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Extracellular Space; Kinetics; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Rats; Rats, Inbred Strains

1989
Ascorbic acid and striatal transport of [3H] 1-methyl-4-phenylpyridine (MPP+) and [3H] dopamine.
    Life sciences, 1988, Volume: 42, Issue:25

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Ascorbic Acid; Biological Transport; Cocaine; Corpus Striatum; Dopamine; Kinetics; Mazindol; Mice; Nicotine; Piperazines; Pyridines; Synaptosomes

1988
Noradrenergic involvement in the discriminative stimulus effects of cocaine in squirrel monkeys.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 275, Issue:1

    Topics: Adrenergic Agonists; Adrenergic Antagonists; Animals; Citalopram; Cocaine; Discrimination Learning; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Male; Narcotics; Neurotransmitter Uptake Inhibitors; Norepinephrine; Piperazines; Receptors, Adrenergic, alpha; Saimiri; Selective Serotonin Reuptake Inhibitors

1995
Effects of N-methyl-D-aspartate antagonists in rats discriminating different doses of cocaine: comparison with direct and indirect dopamine agonists.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 274, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Cocaine; Discrimination Learning; Dopamine Agonists; Male; N-Methylaspartate; Oxazines; Piperazines; Rats; Rats, Wistar

1995
Effects of monoamine reuptake inhibitors on cocaine self-administration in rats.
    Pharmacology, biochemistry, and behavior, 1995, Volume: 51, Issue:4

    Topics: Animals; Biogenic Monoamines; Cocaine; Desipramine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Fluoxetine; Injections, Intravenous; Male; Neurotransmitter Uptake Inhibitors; Norepinephrine; Piperazines; Rats; Rats, Sprague-Dawley; Reward; Self Administration

1995
SPECT imaging of dopamine and serotonin transporters with [123I]beta-CIT: pharmacological characterization of brain uptake in nonhuman primates.
    Synapse (New York, N.Y.), 1993, Volume: 13, Issue:4

    Topics: Animals; Brain; Brain Chemistry; Carrier Proteins; Chlorocebus aethiops; Citalopram; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Indans; Iodine Radioisotopes; Levodopa; Ligands; Maprotiline; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurotransmitter Uptake Inhibitors; Papio; Piperazines; Selective Serotonin Reuptake Inhibitors; Serotonin Plasma Membrane Transport Proteins; Tomography, Emission-Computed, Single-Photon

1993
Serotonergic properties of cocaine: effects on a 5-HT2 receptor-mediated behavior and on extracellular concentrations of serotonin and dopamine.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:1

    Topics: 5-Hydroxytryptophan; Animals; Behavior, Animal; Chromatography, High Pressure Liquid; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Electrochemistry; Extracellular Space; Ketanserin; Male; Microdialysis; Nucleus Accumbens; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists; Synaptic Transmission

1994
The preferential dopamine autoreceptor antagonist (+)-UH232 antagonizes the positive reinforcing effects of cocaine and d-amphetamine in the ICSS paradigm.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 49, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Brain; Cocaine; Dextroamphetamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Electrodes; Haloperidol; Male; Piperazines; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Stimulation

1994
Quantitative assessment of the microstructure of rat behavior: II. Distinctive effects of dopamine releasers and uptake inhibitors.
    Psychopharmacology, 1993, Volume: 113, Issue:2

    Topics: Animals; Behavior, Animal; Cocaine; Conditioning, Operant; Dextroamphetamine; Dopamine Agonists; Dopamine Uptake Inhibitors; Male; Motor Activity; Nomifensine; Piperazines; Rats; Rats, Sprague-Dawley; Serotonin Receptor Agonists

1993
Translocation of dopamine and binding of 2 beta-carbomethoxy-3 beta-(4-fluorophenyl) tropane (WIN 35,428) measured under identical conditions in rat striatal synaptosomal preparations. Inhibition by various blockers.
    Biochemical pharmacology, 1995, Jan-31, Volume: 49, Issue:3

    Topics: Animals; Binding, Competitive; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Rats; Rats, Sprague-Dawley; Synaptosomes; Tritium

1995
Monoamine uptake inhibitors alter cocaine pharmacokinetics.
    Psychopharmacology, 1993, Volume: 112, Issue:4

    Topics: Animals; Biotransformation; Cocaine; Desipramine; Dopamine Uptake Inhibitors; Drug Interactions; Fluoxetine; Male; Neurotransmitter Uptake Inhibitors; Norepinephrine; Piperazines; Rats; Rats, Sprague-Dawley

1993
Regional effects of amphetamine, cocaine, nomifensine and GBR 12909 on the dynamics of dopamine release and metabolism in the rat brain.
    British journal of pharmacology, 1994, Volume: 113, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; alpha-Methyltyrosine; Animals; Behavior, Animal; Brain Chemistry; Central Nervous System Stimulants; Cocaine; Dextroamphetamine; Dopamine; Dopamine Uptake Inhibitors; Male; Methyltyrosines; Nomifensine; Piperazines; Rats; Rats, Sprague-Dawley; Tyrosine 3-Monooxygenase

1994
Kinetic evaluation of the commonality between the site(s) of action of cocaine and some other structurally similar and dissimilar inhibitors of the striatal transporter for dopamine.
    Journal of neurochemistry, 1994, Volume: 63, Issue:5

    Topics: Animals; Benztropine; Biological Transport; Cocaine; Corpus Striatum; Dopamine; Male; Mazindol; Models, Biological; Neurotransmitter Uptake Inhibitors; Nomifensine; Piperazines; Rats; Rats, Sprague-Dawley

1994
Dopamine mechanisms play at best a small role in the nicotine discriminative stimulus.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:3

    Topics: Animals; Benzazepines; Cocaine; Cues; Discrimination Learning; Discrimination, Psychological; Dopamine; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Generalization, Stimulus; Male; Neurotransmitter Uptake Inhibitors; Nicotine; Piperazines; Rats; Receptors, Dopamine D1; Reinforcement Schedule; Spiperone

1994
Effects of cocaine and GBR-12909 on brain stimulation reward.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:4

    Topics: Animals; Brain; Cocaine; Dose-Response Relationship, Drug; Electrodes, Implanted; Male; Medial Forebrain Bundle; Motor Activity; Neurotransmitter Uptake Inhibitors; Piperazines; Rats; Rats, Sprague-Dawley; Reward; Self Stimulation

1994
GBR12909 attenuates cocaine-induced activation of mesolimbic dopamine neurons in the rat.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 271, Issue:3

    Topics: Amphetamine; Animals; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Nucleus Accumbens; Piperazines; Rats; Rats, Sprague-Dawley

1994
Effects of chronic cocaine administration on [3H]dopamine uptake in the nucleus accumbens, striatum and frontal cortex of rats.
    The Journal of pharmacology and experimental therapeutics, 1994, Volume: 270, Issue:1

    Topics: Animals; Brain; Cerebral Cortex; Cocaine; Corpus Striatum; Depression, Chemical; Dopamine; Drug Interactions; Frontal Lobe; Male; Methamphetamine; Motor Activity; Neurotransmitter Uptake Inhibitors; Nucleus Accumbens; Piperazines; Rats; Rats, Sprague-Dawley; Synaptosomes; Time Factors; Tritium

1994
O-526, a piperidine analog of GBR 12909, retains high affinity for the dopamine transporter in monkey caudate-putamen.
    European journal of pharmacology, 1994, Apr-15, Volume: 267, Issue:2

    Topics: Animals; Carrier Proteins; Caudate Nucleus; Citalopram; Cocaine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Macaca fascicularis; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurotransmitter Uptake Inhibitors; Piperazines; Piperidines; Protein Binding; Putamen; Serotonin; Serotonin Plasma Membrane Transport Proteins

1994
Characterization of dopamine transporter and locomotor effects of cocaine, GBR 12909, epidepride, and SCH 23390 in C57BL and DBA mice.
    Pharmacology, biochemistry, and behavior, 1994, Volume: 48, Issue:2

    Topics: Animals; Benzamides; Benzazepines; Binding, Competitive; Brain; Carrier Proteins; Caudate Nucleus; Cocaine; Dopamine; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Female; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Mice, Inbred DBA; Motor Activity; Nerve Tissue Proteins; Neurotransmitter Uptake Inhibitors; Nucleus Accumbens; Piperazines; Pyrrolidines; Species Specificity

1994
Discriminative stimulus properties of cocaine in the rat using a two-choice discrete-trial avoidance paradigm.
    Pharmacology, biochemistry, and behavior, 1993, Volume: 44, Issue:4

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Avoidance Learning; Benzazepines; Cocaine; Discrimination Learning; Discrimination, Psychological; Dopamine Agents; Dose-Response Relationship, Drug; Electroshock; Ergolines; Haloperidol; Male; Methamphetamine; Neurotransmitter Uptake Inhibitors; Piperazines; Quinpirole; Rats; Sulpiride

1993
The effect of 5-HT receptor ligands on the uptake of [3H]5-hydroxytryptamine into rat cortical synaptosomes.
    European journal of pharmacology, 1993, Aug-03, Volume: 239, Issue:1-3

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cerebral Cortex; Cocaine; Desipramine; Female; Fluoxetine; In Vitro Techniques; Indoles; Neurotransmitter Uptake Inhibitors; Paroxetine; Piperazines; Rats; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Synaptosomes; Tropisetron

1993
Induction and suppression of proto-oncogenes in rat striatum after single or multiple treatments with cocaine or GBR-12909.
    NIDA research monograph, 1993, Volume: 125

    Topics: Amino Acid Sequence; Animals; Benzazepines; Blotting, Northern; Blotting, Western; Cocaine; Corpus Striatum; Gene Expression; Genes, fos; Immunohistochemistry; Male; Molecular Sequence Data; Neurotransmitter Uptake Inhibitors; Piperazines; Proto-Oncogenes; Rats; Rats, Sprague-Dawley; RNA, Messenger; Sulpiride; Suppression, Genetic

1993
Electrophysiological effects of cocaine in the rat nucleus accumbens: microiontophoretic studies.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 266, Issue:2

    Topics: alpha-Methyltyrosine; Animals; Cocaine; Dopamine; Fenclonine; Fluoxetine; Iontophoresis; Male; Methyltyrosines; Nucleus Accumbens; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Serotonin

1993
Cocaine-sensitive and -insensitive dopamine uptake in prefrontal cortex, nucleus accumbens and striatum.
    Neurochemistry international, 1993, Volume: 23, Issue:1

    Topics: Analysis of Variance; Animals; Cocaine; Corpus Striatum; Dopamine; Drug Resistance; Male; Neurotransmitter Uptake Inhibitors; Nucleus Accumbens; Ouabain; Piperazines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Temperature

1993
Effects of GBR 12909 and cocaine on cocaine-maintained behavior in rhesus monkeys.
    Drug and alcohol dependence, 1993, Volume: 33, Issue:1

    Topics: Animals; Arousal; Behavior, Animal; Cocaine; Dose-Response Relationship, Drug; Female; Macaca mulatta; Male; Motivation; Motor Activity; Neurotransmitter Uptake Inhibitors; Piperazines; Self Administration; Substance-Related Disorders

1993
GBR 12909 fails to antagonize cocaine-induced elevation of dopamine in striatal slices.
    Drug and alcohol dependence, 1993, Volume: 32, Issue:1

    Topics: Animals; Cocaine; Corpus Striatum; Culture Techniques; Dopamine; Female; Male; Mazindol; Neurotransmitter Uptake Inhibitors; Piperazines; Rats; Rats, Sprague-Dawley; Synaptosomes

1993
Multiple drug classes and hyperosmolarity alter binding of muscarinic drugs to mesothelial cells in vitro.
    Advances in peritoneal dialysis. Conference on Peritoneal Dialysis, 1995, Volume: 11

    Topics: Animals; Atropine; Cells, Cultured; Cocaine; Cycloheximide; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Epithelium; Mannitol; Muscarinic Antagonists; N-Methylscopolamine; Osmolar Concentration; Parasympatholytics; Peritoneum; Piperazines; Quinuclidinyl Benzilate; Rabbits; Receptors, Muscarinic; Scopolamine Derivatives; Sodium Chloride

1995
[3H]WIN 35,428 [2 beta-carbomethoxy-3 beta-(4-fluorophenyl)tropane] binding to rat brain membranes. Comparing dopamine cell body areas with nerve terminal regions.
    Biochemical pharmacology, 1996, Feb-23, Volume: 51, Issue:4

    Topics: Animals; Brain; Cell Membrane; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Kinetics; Male; Mesencephalon; Nerve Endings; Nucleus Accumbens; Piperazines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Tritium

1996
The effects of cocaine on cerebral metabolic function in periweanling rats: the roles of serotonergic and dopaminergic uptake blockade.
    Brain research. Developmental brain research, 1995, Sep-29, Volume: 88, Issue:2

    Topics: Analysis of Variance; Animals; Brain; Cocaine; Dopamine Uptake Inhibitors; Female; Fluoxetine; Male; Pharmaceutical Vehicles; Piperazines; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Weaning

1995
Effects of drug history on the acquisition of responding maintained by GBR 12909 in rhesus monkeys.
    Psychopharmacology, 1996, Volume: 123, Issue:1

    Topics: Animals; Behavior, Animal; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Macaca mulatta; Piperazines; Reinforcement, Psychology; Self Administration; Time Factors

1996
Possible novel pharmacodynamic action of cocaine: cardiovascular and behavioral evidence.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 54, Issue:2

    Topics: Animals; Behavior, Animal; Blood Pressure; Catecholamines; Chlorisondamine; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Ganglionic Blockers; Heart Rate; Hemodynamics; Injections, Intravenous; Male; Motor Activity; Piperazines; Rats; Rats, Sprague-Dawley

1996
Discriminative stimulus effects of dopaminergic agents in rhesus monkeys.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 54, Issue:2

    Topics: Animals; Cocaine; Dextroamphetamine; Discrimination, Psychological; Dopamine Agents; Dose-Response Relationship, Drug; Macaca mulatta; Male; Narcotics; Phentermine; Piperazines; Self Administration

1996
Cocaine cross-sensitization to dopamine uptake inhibitors: unique effects of GBR12909.
    Pharmacology, biochemistry, and behavior, 1996, Volume: 53, Issue:4

    Topics: Animals; Behavior, Animal; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Mazindol; Motor Activity; Piperazines; Rats; Rats, Sprague-Dawley; Stereotyped Behavior

1996
Differential reinforcing effects of cocaine and GBR-12909: biochemical evidence for divergent neuroadaptive changes in the mesolimbic dopaminergic system.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1996, Dec-01, Volume: 16, Issue:23

    Topics: Adaptation, Physiological; Animals; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Injections, Intravenous; Limbic System; Male; Piperazines; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Administration; Water

1996
Monoaminergic substrates underlying cocaine-induced enhancement of somatosensory-evoked discharges in rat barrel field cortical neurons.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 279, Issue:2

    Topics: Animals; Cocaine; Desipramine; Dopamine; Fluoxetine; Male; Norepinephrine; Piperazines; Rats; Serotonin; Somatosensory Cortex

1996
Sustained decrease in cocaine-maintained responding in rhesus monkeys with 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-hydroxy-3-phenylpropyl) piperazinyl decanoate, a long-acting ester derivative of GBR 12909.
    Journal of medicinal chemistry, 1996, Nov-22, Volume: 39, Issue:24

    Topics: Animals; Behavior, Animal; Cocaine; Decanoates; Dopamine Uptake Inhibitors; Macaca mulatta; Male; Molecular Structure; Piperazines; Substance-Related Disorders

1996
Serotonin1b receptor stimulation enhances dopamine-mediated reinforcement.
    Psychopharmacology, 1996, Volume: 128, Issue:2

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Animals; Cocaine; Conditioning, Operant; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Narcotics; Piperazines; Quinoxalines; Rats; Rats, Wistar; Receptor, Serotonin, 5-HT1B; Receptors, Serotonin; Self Administration; Serotonin Receptor Agonists

1996
Highly selective, novel analogs of 4-[2-(diphenylmethoxy)ethyl]- 1-benzylpiperidine for the dopamine transporter: effect of different aromatic substitutions on their affinity and selectivity.
    Journal of medicinal chemistry, 1997, Jan-03, Volume: 40, Issue:1

    Topics: Animals; Carrier Proteins; Citalopram; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Rats

1997
Heteroaromatic analogs of 1-[2-(diphenylmethoxy)ethyl]- and 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazines (GBR 12935 and GBR 12909) as high-affinity dopamine reuptake inhibitors.
    Journal of medicinal chemistry, 1997, Feb-28, Volume: 40, Issue:5

    Topics: Animals; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Feeding Behavior; Ligands; Macaca mulatta; Magnetic Resonance Spectroscopy; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Structure; Motor Activity; Nerve Tissue Proteins; Pentazocine; Piperazines; Rats; Serotonin Plasma Membrane Transport Proteins; Structure-Activity Relationship

1997
RTI-352: a 3 alpha analogue of RTI-55 as an in vivo dopamine transporter binding ligand.
    Synapse (New York, N.Y.), 1997, Volume: 25, Issue:4

    Topics: Animals; Brain; Carrier Proteins; Cocaine; Desipramine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Kinetics; Ligands; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Nerve Tissue Proteins; Organ Specificity; Paroxetine; Piperazines; Tritium

1997
Gender difference in cocaine-induced HPA axis activation.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 1997, Volume: 16, Issue:6

    Topics: Adrenocorticotropic Hormone; Animals; Cocaine; Desipramine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Female; Fluoxetine; Hypothalamo-Hypophyseal System; Male; Neurotransmitter Uptake Inhibitors; Orchiectomy; Ovariectomy; Piperazines; Pituitary-Adrenal System; Rats; Sex Characteristics; Time Factors

1997
Phentermine/fenfluramine decreases cocaine self-administration in rhesus monkeys.
    Neuroreport, 1997, Apr-14, Volume: 8, Issue:6

    Topics: Analysis of Variance; Animals; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Fenfluramine; Macaca mulatta; Male; Narcotics; Phentermine; Piperazines; Reaction Time; Self Administration; Serotonin Agents

1997
Dose-response analysis in risk assessment: evaluation of behavioral specificity.
    Environmental health perspectives, 1996, Volume: 104 Suppl 2

    Topics: Animals; Behavior, Animal; Cocaine; Dose-Response Relationship, Drug; Drug Administration Schedule; Macaca mulatta; Neurotoxins; Piperazines; Probability; Risk Assessment

1996
The rate hypothesis and agonist substitution approaches to cocaine abuse treatment.
    Advances in pharmacology (San Diego, Calif.), 1998, Volume: 42

    Topics: Animals; Bupropion; Cocaine; Dopamine Uptake Inhibitors; Humans; Mazindol; Piperazines; Substance-Related Disorders

1998
Effects of proposed treatments for cocaine addiction on hemodynamic responsiveness to cocaine in conscious rats.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 283, Issue:2

    Topics: Animals; Bromocriptine; Buprenorphine; Cocaine; Desipramine; Diazepam; Dizocilpine Maleate; Hemodynamics; Male; Piperazines; Rats; Rats, Sprague-Dawley; Substance-Related Disorders

1997
D1 receptors mediate dopamine action in the fetal suprachiasmatic nuclei: studies of mice with targeted deletion of the D1 dopamine receptor gene.
    Brain research. Molecular brain research, 1997, Oct-03, Volume: 49, Issue:1-2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Autoradiography; Benzazepines; Cocaine; Crosses, Genetic; Dopamine; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Female; Fetus; Male; Mice; Mice, Knockout; Mice, Transgenic; Piperazines; Pregnancy; Proto-Oncogene Proteins c-fos; Receptors, Dopamine D1; RNA, Messenger; Signal Transduction; Suprachiasmatic Nucleus; Transcription, Genetic; Tritium

1997
Chronic administration of the selective dopamine uptake inhibitor GBR 12,909, but not cocaine, produces marked decreases in dopamine transporter density.
    Naunyn-Schmiedeberg's archives of pharmacology, 1997, Volume: 356, Issue:5

    Topics: Animals; Brain; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Male; Piperazines; Rats; Rats, Sprague-Dawley

1997
A simple probe measures the pharmacokinetics of[125I]RTI-55 in mouse brain in vivo.
    European journal of pharmacology, 1997, Oct-29, Volume: 338, Issue:1

    Topics: Absorptiometry, Photon; Animals; Brain; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Iodine Radioisotopes; Male; Mice; Paroxetine; Piperazines; Radiometry; Selective Serotonin Reuptake Inhibitors; Serotonin

1997
Contribution of blockade of the noradrenaline carrier to the increase of extracellular dopamine in the rat prefrontal cortex by amphetamine and cocaine.
    The European journal of neuroscience, 1997, Volume: 9, Issue:10

    Topics: Animals; Carrier Proteins; Cocaine; Desipramine; Dextroamphetamine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Multivariate Analysis; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Piperazines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Symporters

1997
gamma-Aminobutyric acidA agonists differentially augment gnawing induced by indirect-acting dopamine agonists in C57BL/6J mice.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 284, Issue:1

    Topics: Animals; Behavior, Animal; Benzazepines; Cocaine; Dopamine Agonists; GABA-A Receptor Agonists; Isoxazoles; Male; Mice; Mice, Inbred C57BL; Muscimol; Piperazines

1998
Apical and basolateral uptake and intracellular fate of dopamine precursor L-dopa in LLC-PK1 cells.
    The American journal of physiology, 1998, Volume: 274, Issue:2

    Topics: Animals; Aromatic Amino Acid Decarboxylase Inhibitors; Aromatic-L-Amino-Acid Decarboxylases; Benserazide; Biological Transport; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Enzyme Inhibitors; Epithelial Cells; Kidney Tubules, Proximal; Kinetics; Levodopa; LLC-PK1 Cells; Piperazines; Swine

1998
Potent and selective ligands for the dopamine transporter (DAT): structure-activity relationship studies of novel 4-[2-(diphenylmethoxy)ethyl]-1-(3-phenylpropyl)piperidine analogues.
    Journal of medicinal chemistry, 1998, Feb-26, Volume: 41, Issue:5

    Topics: Animals; Benzhydryl Compounds; Carrier Proteins; Cell Membrane; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Male; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Structure; Nerve Tissue Proteins; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship

1998
GABAergic modulation of ventral pallidal dopamine release studied by in vivo microdialysis in the freely moving rat.
    Synapse (New York, N.Y.), 1998, Volume: 29, Issue:4

    Topics: Animals; Baclofen; Cocaine; Dopamine; Dopamine Uptake Inhibitors; GABA Antagonists; gamma-Aminobutyric Acid; Globus Pallidus; Male; Microdialysis; Picrotoxin; Piperazines; Rats; Rats, Wistar

1998
Tolerance in the replacement of the benzhydrylic O atom in 4-[2-(diphenylmethoxy)ethyl]-1-benzylpiperidine derivatives by an N atom: development of new-generation potent and selective N-analogue molecules for the dopamine transporter.
    Journal of medicinal chemistry, 1998, Aug-13, Volume: 41, Issue:17

    Topics: Animals; Carrier Proteins; Cell Line; Citalopram; Cloning, Molecular; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Design; Humans; Ligands; Membrane Glycoproteins; Membrane Transport Proteins; Molecular Structure; Nerve Tissue Proteins; Piperazines; Piperidines; Rats; Rats, Sprague-Dawley; Recombinant Proteins; Serotonin; Serotonin Plasma Membrane Transport Proteins; Structure-Activity Relationship; Transfection

1998
Modulation of cocaine-induced motor activity in the rat by opioid receptor agonists.
    Behavioural pharmacology, 1998, Volume: 9, Issue:5-6

    Topics: Animals; Cisterna Magna; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Fluoxetine; Injections; Male; Motor Activity; Neurotransmitter Uptake Inhibitors; Norepinephrine; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Opioid; Selective Serotonin Reuptake Inhibitors

1998
Dopamine agonist-induced hypothermia and disruption of prepulse inhibition: evidence for a role of D3 receptors?
    Behavioural pharmacology, 1998, Volume: 9, Issue:5-6

    Topics: Animals; Body Temperature; Cocaine; Domperidone; Dopamine Agonists; Dopamine Antagonists; Dopamine Uptake Inhibitors; Hypothermia; Male; Piperazines; Raclopride; Rats; Rats, Wistar; Receptors, Dopamine D2; Receptors, Dopamine D3; Reflex, Startle; Salicylamides; Serotonin Antagonists

1998
Generalization of D-, L- and DL-chlorpheniramine and zolantidine to the discriminative stimulus effects of cocaine and methamphetamine.
    Behavioural pharmacology, 1997, Volume: 8, Issue:8

    Topics: Animals; Antidepressive Agents, Tricyclic; Benzothiazoles; Chlorpheniramine; Clomipramine; Cocaine; Desipramine; Discrimination, Psychological; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Generalization, Stimulus; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Methamphetamine; Middle Aged; Phenoxypropanolamines; Piperazines; Piperidines; Rats; Rats, Inbred F344; Thiazoles

1997
Novel rhenium complexes derived from alpha-tropanol as potential ligands for the dopamine transporter.
    Bioorganic & medicinal chemistry, 1998, Volume: 6, Issue:10

    Topics: Carrier Proteins; Chromatography, High Pressure Liquid; Cocaine; Crystallography, X-Ray; Dopamine Plasma Membrane Transport Proteins; Humans; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Rhenium; Structure-Activity Relationship; Tropanes

1998
Repeated injection of GBR 12909, but not cocaine or WIN 35,065-2, into the ventral tegmental area induces behavioral sensitization.
    Behavioural brain research, 1998, Volume: 97, Issue:1-2

    Topics: Animals; Behavior, Animal; Chromatography, High Pressure Liquid; Cocaine; Dopamine Uptake Inhibitors; Injections; Male; Microdialysis; Motor Activity; Piperazines; Rats; Rats, Sprague-Dawley; Ventral Tegmental Area

1998
Iodine-123 labelled nor-beta-CIT binds to the serotonin transporter in vivo as assessed by biodistribution studies in rats.
    European journal of nuclear medicine, 1998, Volume: 25, Issue:12

    Topics: Animals; Brain; Carrier Proteins; Cocaine; Dopamine Uptake Inhibitors; Fluvoxamine; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Radionuclide Imaging; Rats; Rats, Wistar; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Plasma Membrane Transport Proteins; Tropanes

1998
Effects of phentermine on responding maintained under multiple fixed-ratio schedules of food and cocaine presentation in the rhesus monkey.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 288, Issue:2

    Topics: Animals; Behavior, Animal; Central Nervous System Stimulants; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Eating; Illicit Drugs; Macaca mulatta; Male; Phentermine; Piperazines

1999
Acquisition of nicotine discrimination and discriminative stimulus effects of nicotine in rats chronically exposed to caffeine.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 288, Issue:3

    Topics: Amphetamine; Analysis of Variance; Animals; Caffeine; Cocaine; Discrimination Learning; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Mecamylamine; Nicotine; Nicotinic Antagonists; Piperazines; Rats; Rats, Sprague-Dawley; Stimulation, Chemical; Thiazepines

1999
Doses of GBR12909 that suppress cocaine self-administration in non-human primates substantially occupy dopamine transporters as measured by [11C] WIN35,428 PET scans.
    Synapse (New York, N.Y.), 1999, Volume: 32, Issue:1

    Topics: Animals; Carbon Radioisotopes; Carrier Proteins; Cocaine; Depression, Chemical; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Infusions, Intravenous; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Papio; Piperazines; Self Administration; Tomography, Emission-Computed

1999
Chronic haloperidol alters dopamine receptors: effects of cocaine exposure during the preweaning period.
    European journal of pharmacology, 1999, Apr-16, Volume: 370, Issue:3

    Topics: Animals; Autoradiography; Basal Ganglia; Benzazepines; Cocaine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Female; Haloperidol; Male; Piperazines; Prosencephalon; Protein Binding; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Salicylamides; Sex Factors; Time Factors; Weaning

1999
Pharmacological characterization of nicotine's interaction with cocaine and cocaine analogs.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:3

    Topics: Animals; Body Temperature; Bupropion; Cocaine; Discrimination, Psychological; Female; Male; Membrane Potentials; Mice; Mice, Inbred ICR; Molecular Structure; Motor Activity; Nicotine; Oocytes; Pain; Piperazines; Psychomotor Performance; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Recombinant Proteins; Seizures; Structure-Activity Relationship; Tropanes; Xenopus laevis

1999
The effects of cadmium contamination on the discriminative stimulus properties of cocaine and related drugs.
    Experimental and clinical psychopharmacology, 1999, Volume: 7, Issue:2

    Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Animals; Apomorphine; Benzazepines; Body Weight; Cadmium Chloride; Cocaine; Dextroamphetamine; Discrimination, Psychological; Dopamine Agents; Dopamine Uptake Inhibitors; Drug Interactions; Drug Tolerance; Eating; Male; Piperazines; Procaine; Quinpirole; Rats; Rats, Sprague-Dawley

1999
Dopaminergic mechanisms mediating the incentive to seek cocaine and heroin following long-term withdrawal of IV drug self-administration.
    Psychopharmacology, 1999, Volume: 143, Issue:3

    Topics: Animals; Behavior, Addictive; Benzazepines; Cocaine; Dopamine Agonists; Dopamine Uptake Inhibitors; Heroin; Male; Narcotics; Piperazines; Quinpirole; Rats; Rats, Wistar; Receptors, Dopamine; Substance Withdrawal Syndrome

1999
Discriminative stimulus effects of morphine in squirrel monkeys: stimulants, opioids, and stimulant-opioid combinations.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 290, Issue:3

    Topics: Amphetamine; Analgesics, Opioid; Anesthetics, Local; Animals; Anti-Anxiety Agents; Cocaine; Discrimination Learning; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Combinations; Fentanyl; Male; Morphine; Naltrexone; Narcotic Antagonists; Piperazines; Receptors, Opioid; Saimiri; Selective Serotonin Reuptake Inhibitors

1999
Continuous infusion of selective dopamine uptake inhibitors or cocaine produces time-dependent changes in rat locomotor activity.
    Behavioural brain research, 1999, Volume: 99, Issue:2

    Topics: Adrenergic Uptake Inhibitors; Animals; Cocaine; Dopamine Uptake Inhibitors; Drug Tolerance; Fluoxetine; Infusion Pumps, Implantable; Male; Monoamine Oxidase Inhibitors; Motor Activity; Piperazines; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Time Factors

1999
Pharmacological characterization of (E)-N-(3-iodoprop-2-enyl)-2beta-carbomethoxy-3beta-(4'-methylphenyl)n ortropane as a selective and potent inhibitor of the neuronal dopamine transporter.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 291, Issue:2

    Topics: Animals; Autoradiography; Biological Transport, Active; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Nortropanes; Piperazines; Protein Binding; Radiopharmaceuticals; Rats; Rats, Wistar; Visual Cortex

1999
Isoflurane anesthesia enhances the inhibitory effects of cocaine and GBR12909 on dopamine transporter: PET studies in combination with microdialysis in the monkey brain.
    Brain research, 1999, Dec-04, Volume: 849, Issue:1-2

    Topics: Anesthesia, Inhalation; Animals; Brain; Carbon Radioisotopes; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Isoflurane; Kinetics; Macaca mulatta; Male; Membrane Glycoproteins; Membrane Transport Proteins; Microdialysis; Nerve Tissue Proteins; Piperazines; Receptors, Dopamine D2; Time Factors; Tomography, Emission-Computed; Wakefulness

1999
[3H]beta-CIT: a radioligand for dopamine transporters in rat brain tissue.
    European journal of pharmacology, 1999, Dec-03, Volume: 385, Issue:2-3

    Topics: Amphetamine; Animals; Autoradiography; Binding, Competitive; Brain; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Male; Membrane Glycoproteins; Membrane Transport Proteins; Methylphenidate; Nerve Tissue Proteins; Piperazines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin Plasma Membrane Transport Proteins; Stereoisomerism; Tritium

1999
A selective radiobrominated cocaine analogue for imaging of dopamine uptake sites: pharmacological evaluation and PET experiments.
    Life sciences, 1999, Volume: 65, Issue:25

    Topics: Animals; Brain; Bromine Radioisotopes; Cerebellum; Cerebral Cortex; Citalopram; Cocaine; Corpus Striatum; Dopamine; Kinetics; Male; Maprotiline; Nortropanes; Papio; Piperazines; Radiopharmaceuticals; Rats; Rats, Wistar; Thalamus; Tissue Distribution; Tomography, Emission-Computed

1999
Comparative behavioral pharmacology of cocaine and the selective dopamine uptake inhibitor RTI-113 in the squirrel monkey.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 292, Issue:2

    Topics: Animals; Behavior, Animal; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Male; Piperazines; Saimiri; Self Administration; Statistics as Topic; Time Factors

2000
Dose-response and duration effects of acute administrations of cocaine and GBR12909 on dopamine synthesis and transporter in the conscious monkey brain: PET studies combined with microdialysis.
    Brain research, 2000, Mar-31, Volume: 860, Issue:1-2

    Topics: Animals; Brain; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Administration Schedule; Macaca mulatta; Male; Membrane Glycoproteins; Membrane Transport Proteins; Microdialysis; Nerve Tissue Proteins; Piperazines; Time Factors; Tomography, Emission-Computed

2000
Cocaine-induced changes in extracellular dopamine determined by microdialysis in awake squirrel monkeys.
    Psychopharmacology, 2000, Volume: 148, Issue:3

    Topics: Animals; Cocaine; Dopamine; Dose-Response Relationship, Drug; Glial Fibrillary Acidic Protein; Immunohistochemistry; Male; Microdialysis; Piperazines; Saimiri

2000
Changes in dopamine transporter and c-Fos expression in the nucleus accumbens of alcohol-tolerant rats.
    Alcoholism, clinical and experimental research, 2000, Volume: 24, Issue:3

    Topics: Alcoholism; Animals; Carrier Proteins; Central Nervous System Depressants; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Ethanol; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Nucleus Accumbens; Piperazines; Proto-Oncogene Proteins c-fos; Rats; Rats, Wistar; Serotonin

2000
Cocaine inhibits NGF-induced PC12 cells differentiation through D(1)-type dopamine receptors.
    Brain research, 2000, Jun-30, Volume: 869, Issue:1-2

    Topics: Animals; Brain; Carrier Proteins; Cell Differentiation; Cocaine; Dopamine; Dopamine D2 Receptor Antagonists; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Embryonic and Fetal Development; Female; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Growth Factor; Nerve Tissue Proteins; Neurites; Neurons; Neurotransmitter Agents; PC12 Cells; Piperazines; Pregnancy; Prenatal Exposure Delayed Effects; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2

2000
A comparison of the patterns of striatal Fos-like immunoreactivity induced by various dopamine agonists in rats.
    Neuroscience letters, 2000, Aug-04, Volume: 289, Issue:2

    Topics: Amphetamine; Animals; Apomorphine; Cocaine; Corpus Striatum; Dopamine Agonists; Dopamine Uptake Inhibitors; Immunohistochemistry; Injections, Intraperitoneal; Male; Nalidixic Acid; Naphthyridines; Nomifensine; Piperazines; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Staining and Labeling

2000
Effect of cocaine, nomifensine, GBR 12909 and WIN 35428 on carbon fiber microelectrode sensitivity for voltammetric recording of dopamine.
    Journal of neuroscience methods, 2000, Aug-15, Volume: 101, Issue:1

    Topics: Animals; Artifacts; Calibration; Carbon; Coated Materials, Biocompatible; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Electrochemistry; Electrodes, Implanted; Equipment Failure; Fluorocarbon Polymers; Male; Microelectrodes; Nomifensine; Nucleus Accumbens; Piperazines; Rats; Rats, Sprague-Dawley; Sensitivity and Specificity

2000
Cholinergic neuronal modulation alters dopamine D2 receptor availability in vivo by regulating receptor affinity induced by facilitated synaptic dopamine turnover: positron emission tomography studies with microdialysis in the conscious monkey brain.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Sep-15, Volume: 20, Issue:18

    Topics: Animals; Brain; Carbon Radioisotopes; Carrier Proteins; Cholinergic Fibers; Cocaine; Dihydroxyphenylalanine; Dopamine; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Extracellular Space; Macaca mulatta; Male; Membrane Glycoproteins; Membrane Transport Proteins; Microdialysis; Muscarinic Antagonists; Nerve Tissue Proteins; Neurons; Piperazines; Raclopride; Receptors, Dopamine D2; Scopolamine; Synapses; Tomography, Emission-Computed; Wakefulness

2000
Novel in vivo electrophysiological assay for the effects of cocaine and putative "cocaine antagonists" on dopamine transporter activity of substantia nigra and ventral tegmental area dopamine neurons.
    Synapse (New York, N.Y.), 2000, Dec-01, Volume: 38, Issue:3

    Topics: Action Potentials; Animals; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurons; Piperazines; Rats; Rats, Sprague-Dawley; Substantia Nigra; Ventral Tegmental Area

2000
Stimulation of in vivo dopamine transmission in the bed nucleus of stria terminalis by reinforcing drugs.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Oct-15, Volume: 20, Issue:20

    Topics: Analysis of Variance; Animals; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Ethanol; Extracellular Space; Illicit Drugs; Male; Microdialysis; Morphine; Nicotine; Piperazines; Rats; Rats, Sprague-Dawley; Septal Nuclei; Synaptic Transmission

2000
Chamber-specific alterations of noradrenaline uptake (uptake(1)) in right ventricles of monocrotaline-treated rats.
    British journal of pharmacology, 2000, Volume: 131, Issue:7

    Topics: Adrenergic Uptake Inhibitors; Animals; Binding, Competitive; Cocaine; Desipramine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Fluoxetine; Heart Failure; Heart Ventricles; Hypertrophy; In Vitro Techniques; Male; Membranes; Monocrotaline; Norepinephrine; Piperazines; Rats; Rats, Wistar; Tritium

2000
Serotonin-mediated striatal dopamine release involves the dopamine uptake site and the serotonin receptor.
    Brain research bulletin, 2000, Volume: 53, Issue:3

    Topics: Animals; Bicuculline; Cocaine; Corpus Striatum; Dizocilpine Maleate; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; GABA Antagonists; Ketanserin; Male; Methiothepin; Mice; Mice, Inbred C57BL; Oxymetazoline; Piperazines; Quinoxalines; Quipazine; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists

2000
Response requirements and unit dose modify the effects of GBR 12909 on cocaine-maintained behavior.
    Experimental and clinical psychopharmacology, 2000, Volume: 8, Issue:4

    Topics: Animals; Central Nervous System Stimulants; Cocaine; Cocaine-Related Disorders; Disease Models, Animal; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Female; Macaca mulatta; Male; Piperazines

2000
A comparison of cocaine, GBR 12909, and phentermine self-administration by rhesus monkeys on a progressive-ratio schedule.
    Drug and alcohol dependence, 2001, Mar-01, Volume: 62, Issue:1

    Topics: Adrenergic Agents; Animals; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Macaca mulatta; Male; Phentermine; Piperazines; Reinforcement Schedule; Self Administration

2001
Synthesis and preliminary characterization of a high-affinity novel radioligand for the dopamine transporter.
    Synapse (New York, N.Y.), 2001, Volume: 39, Issue:2

    Topics: Animals; Benzhydryl Compounds; Binding, Competitive; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Female; Ligands; Macaca mulatta; Male; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Neostriatum; Nerve Tissue Proteins; Piperazines; Piperidines; Radioligand Assay; Tritium

2001
Chronic GBR 12909 administration differentially alters prodynorphin gene expression compared to cocaine.
    European journal of pharmacology, 2001, Feb-16, Volume: 413, Issue:2-3

    Topics: Animals; Brain; Cocaine; Dopamine Uptake Inhibitors; Enkephalins; Gene Expression; Male; Piperazines; Protein Precursors; Rats; Rats, Sprague-Dawley; RNA, Messenger

2001
Cocaine and amphetamine increase extracellular dopamine in the nucleus accumbens of mice lacking the dopamine transporter gene.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2001, May-01, Volume: 21, Issue:9

    Topics: Adrenergic Uptake Inhibitors; Amphetamine; Animals; Carrier Proteins; Chromatography, High Pressure Liquid; Cocaine; Cocaine-Related Disorders; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Extracellular Space; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Mice, Knockout; Microdialysis; Morpholines; Nerve Tissue Proteins; Nucleus Accumbens; Piperazines; Reboxetine; Reinforcement, Psychology

2001
Further studies of the reinforcing effects of benztropine analogs in rhesus monkeys.
    Psychopharmacology, 2001, Volume: 154, Issue:4

    Topics: Animals; Benztropine; Cocaine; Dopamine Uptake Inhibitors; Female; Macaca mulatta; Male; Piperazines; Reaction Time; Reinforcement Schedule; Self Administration

2001
Subtle differences in the discriminative stimulus effects of cocaine and GBR-12909.
    Progress in neuro-psychopharmacology & biological psychiatry, 2001, Volume: 25, Issue:3

    Topics: Adrenergic Uptake Inhibitors; Animals; Carrier Proteins; Cocaine; Discrimination, Psychological; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors

2001
Cocaine or selective block of dopamine transporters influences multisecond oscillations in firing rate in the globus pallidus.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2001, Volume: 25, Issue:1

    Topics: Action Potentials; Adrenergic Uptake Inhibitors; Animals; Biogenic Monoamines; Biological Clocks; Carrier Proteins; Cocaine; Desipramine; Dizocilpine Maleate; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Excitatory Amino Acid Antagonists; Fluoxetine; Globus Pallidus; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurons; Periodicity; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, N-Methyl-D-Aspartate; Selective Serotonin Reuptake Inhibitors

2001
Differential interaction of GBR 12909, a dopamine uptake inhibitor, with cocaine and methamphetamine in rats discriminating cocaine.
    Psychopharmacology, 2001, Volume: 155, Issue:2

    Topics: Animals; Cocaine; Discrimination Learning; Discrimination, Psychological; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Synergism; Generalization, Stimulus; Male; Methamphetamine; Motor Activity; Neurons; Piperazines; Rats; Rats, Sprague-Dawley

2001
Behavioral responses to dopamine agonists in adult rats exposed to cocaine during the preweaning period.
    Pharmacology, biochemistry, and behavior, 2001, Volume: 70, Issue:1

    Topics: Animals; Cocaine; Dopamine Agonists; Dopamine Uptake Inhibitors; Female; Male; Motor Activity; Piperazines; Rats; Rats, Sprague-Dawley; Sex Factors; Weaning

2001
Similar enhancement of the discriminative stimulus effects of cocaine and GBR 12909 by heroin in squirrel monkeys.
    Psychopharmacology, 2001, Volume: 157, Issue:3

    Topics: Animals; Cocaine; Discrimination, Psychological; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Heroin; Male; Narcotics; Piperazines; Saimiri

2001
Repeated cocaine administration into the rat ventral tegmental area produces behavioral sensitization to a systemic cocaine challenge.
    Behavioural brain research, 2001, Nov-29, Volume: 126, Issue:1-2

    Topics: Animals; Arousal; Cocaine; Drug Synergism; Injections, Intraperitoneal; Male; Microinjections; Motor Activity; Piperazines; Premedication; Rats; Rats, Sprague-Dawley; Synaptic Transmission; Ventral Tegmental Area

2001
Dopamine uptake through the norepinephrine transporter in brain regions with low levels of the dopamine transporter: evidence from knock-out mouse lines.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2002, Jan-15, Volume: 22, Issue:2

    Topics: Animals; Brain; Brain Chemistry; Caudate Nucleus; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Fluoxetine; Frontal Lobe; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Knockout; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Nucleus Accumbens; Piperazines; Symporters; Synaptosomes

2002
Effects of GBR 12909, WIN 35,428 and indatraline on cocaine self-administration and cocaine seeking in rats.
    Psychopharmacology, 2002, Volume: 160, Issue:3

    Topics: Animals; Behavior, Addictive; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Indans; Male; Methylamines; Neurotransmitter Uptake Inhibitors; Piperazines; Rats; Rats, Sprague-Dawley; Self Administration

2002
Locomotor activity induced by noncompetitive NMDA receptor antagonists versus dopamine transporter inhibitors: opposite strain differences in inbred long-sleep and short-sleep mice.
    Alcoholism, clinical and experimental research, 2002, Volume: 26, Issue:4

    Topics: Amphetamine; Animals; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Excitatory Amino Acid Antagonists; Female; Male; Membrane Glycoproteins; Membrane Transport Modulators; Membrane Transport Proteins; Mice; Mice, Inbred Strains; Motor Activity; Nerve Tissue Proteins; Piperazines; Receptors, N-Methyl-D-Aspartate; Sleep; Species Specificity; Tritium

2002
Effects of dopamine agonists and antagonists on locomotor activity in male and female rats.
    Pharmacology, biochemistry, and behavior, 2002, Volume: 72, Issue:4

    Topics: Animals; Benzazepines; Cocaine; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Female; Male; Motor Activity; Piperazines; Quinpirole; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Sex Characteristics

2002
Chronic cocaine increases kappa-opioid receptor density: lack of effect by selective dopamine uptake inhibitors.
    Synapse (New York, N.Y.), 2002, Sep-01, Volume: 45, Issue:3

    Topics: Animals; Caudate Nucleus; Cocaine; Dopamine Uptake Inhibitors; Drug Administration Schedule; Infusion Pumps, Implantable; Injections, Subcutaneous; Male; Nucleus Accumbens; Piperazines; Putamen; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa

2002
Age-related changes in the striatal dopaminergic system in the living brain: a multiparametric PET study in conscious monkeys.
    Synapse (New York, N.Y.), 2002, Volume: 45, Issue:1

    Topics: Aging; Animals; Benzazepines; Cocaine; Corpus Striatum; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Extracellular Space; Levodopa; Macaca mulatta; Magnetic Resonance Imaging; Male; Microdialysis; Piperazines; Raclopride; Tomography, Emission-Computed

2002
Effect of daily dosing duration of direct and indirect dopamine receptor agonists: cocaine cross-tolerance following chronic regimens.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2002, Volume: 12, Issue:5

    Topics: Analysis of Variance; Animals; Area Under Curve; Autoreceptors; Benzothiazoles; Cocaine; Cocaine-Related Disorders; Cross-Over Studies; Dopamine Agonists; Dopamine Uptake Inhibitors; Drug Administration Schedule; Drug Interactions; Male; Motor Activity; Piperazines; Pramipexole; Psychomotor Performance; Rats; Rats, Sprague-Dawley; Thiazoles; Time Factors

2002
Synthesis and dopamine transporter affinity of chiral 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(2-hydroxypropyl)piperazines as potential cocaine abuse therapeutic agents.
    Bioorganic & medicinal chemistry letters, 2003, Feb-10, Volume: 13, Issue:3

    Topics: Animals; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Ligands; Macaca mulatta; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Protein Binding; Stereoisomerism; Structure-Activity Relationship

2003
Effect of the mGluR5 antagonist 6-methyl-2-(phenylethynyl)pyridine (MPEP) on the acute locomotor stimulant properties of cocaine, D-amphetamine, and the dopamine reuptake inhibitor GBR12909 in mice.
    Psychopharmacology, 2004, Volume: 174, Issue:2

    Topics: Amphetamine; Animals; Anti-Anxiety Agents; Cocaine; Dopamine Agents; Dopamine Uptake Inhibitors; Drug Interactions; Male; Mice; Mice, Inbred DBA; Motor Activity; Piperazines; Pyridines; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate

2004
Cocaine-like discriminative stimulus effects of heroin: modulation by selective monoamine transport inhibitors.
    The Journal of pharmacology and experimental therapeutics, 2004, Volume: 310, Issue:1

    Topics: Animals; Carrier Proteins; Citalopram; Cocaine; Discrimination, Psychological; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Interactions; Heroin; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neuropeptides; Norepinephrine Plasma Membrane Transport Proteins; Piperazines; Prazosin; Receptors, Adrenergic, alpha-1; Saimiri; Selective Serotonin Reuptake Inhibitors; Serotonin Plasma Membrane Transport Proteins; Symporters; Thiophenes; Vesicular Biogenic Amine Transport Proteins

2004
Pharmacological modulation of GABA(B) receptors affects cocaine-induced seizures in mice.
    Psychopharmacology, 2004, Volume: 174, Issue:2

    Topics: Animals; Baclofen; Cocaine; Dopamine Uptake Inhibitors; GABA-A Receptor Agonists; GABA-A Receptor Antagonists; GABA-B Receptor Agonists; GABA-B Receptor Antagonists; Kindling, Neurologic; Male; Mice; Piperazines; Receptors, GABA-A; Receptors, GABA-B; Seizures

2004
Methamphetamine discrimination and in vivo microdialysis in squirrel monkeys.
    Psychopharmacology, 2004, Volume: 175, Issue:2

    Topics: Animals; Behavior, Animal; Cocaine; Discrimination Learning; Dopamine Agents; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Male; Methamphetamine; Methylphenidate; Microdialysis; Piperazines; Saimiri

2004
Mutation of Trp84 and Asp313 of the dopamine transporter reveals similar mode of binding interaction for GBR12909 and benztropine as opposed to cocaine.
    Journal of neurochemistry, 2004, Volume: 89, Issue:4

    Topics: Amino Acid Substitution; Benztropine; Binding, Competitive; Cell Line; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Humans; Kidney; Ligands; Membrane Glycoproteins; Membrane Transport Proteins; Muscarinic Antagonists; Mutagenesis, Site-Directed; Nerve Tissue Proteins; Piperazines; Protein Binding; Sodium; Structure-Activity Relationship; Zinc

2004
Regional differences in extracellular dopamine and serotonin assessed by in vivo microdialysis in mice lacking dopamine and/or serotonin transporters.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2004, Volume: 29, Issue:10

    Topics: Animals; Caudate Nucleus; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Extracellular Space; Fluoxetine; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Mice, Knockout; Microdialysis; Nerve Tissue Proteins; Nucleus Accumbens; Piperazines; Prefrontal Cortex; Putamen; Reverse Transcriptase Polymerase Chain Reaction; Serotonin; Serotonin Plasma Membrane Transport Proteins; Stereotaxic Techniques

2004
Characterization of dopamine transport in crude synaptosomes prepared from rat medial prefrontal cortex.
    Journal of neuroscience methods, 2004, Aug-30, Volume: 137, Issue:2

    Topics: Animals; Biological Transport; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Fluoxetine; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Norepinephrine; Piperazines; Prefrontal Cortex; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Sensitivity and Specificity; Synaptosomes; Time Factors; Tritium

2004
Effects of the selective norepinephrine uptake inhibitor nisoxetine on prodynorphin gene expression in rat CNS.
    Brain research. Molecular brain research, 2004, Aug-23, Volume: 127, Issue:1-2

    Topics: Adrenergic Uptake Inhibitors; Animals; Blotting, Northern; Central Nervous System; Cocaine; Dopamine Uptake Inhibitors; Enkephalins; Fluoxetine; Gene Expression; Male; Piperazines; Protein Precursors; Rats; Rats, Sprague-Dawley; RNA, Messenger; Selective Serotonin Reuptake Inhibitors

2004
Effects of dopamine indirect agonists and selective D1-like and D2-like agonists and antagonists on cocaine self-administration and food maintained responding in rats.
    Neuropharmacology, 2004, Volume: 47 Suppl 1

    Topics: Animals; Benzazepines; Cocaine; Conditioning, Operant; Dopamine Agonists; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Food; Male; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine D1; Receptors, Dopamine D2; Reinforcement, Psychology; Salicylamides; Self Administration; Tetrahydronaphthalenes

2004
Interaction between a hydroxypiperidine analogue of 4-(2-benzhydryloxy-ethyl)-1-(4-fluorobenzyl)piperidine and Aspartate 68 in the human dopamine transporter.
    European journal of pharmacology, 2004, Dec-03, Volume: 506, Issue:1

    Topics: Animals; Aspartic Acid; Benzhydryl Compounds; Binding Sites; Binding, Competitive; Biological Transport; Cell Line; Cell Membrane; Cerebral Cortex; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Humans; Male; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Mutation; Nerve Tissue Proteins; Norepinephrine; Piperazines; Piperidines; Protein Binding; Rats; Rats, Sprague-Dawley; Serotonin; Stereoisomerism; Synaptosomes; Tritium

2004
Pharmacological profile of radioligand binding to the norepinephrine transporter: instances of poor indication of functional activity.
    Journal of neuroscience methods, 2005, Apr-15, Volume: 143, Issue:1

    Topics: Binding Sites; Binding, Competitive; Brain Chemistry; Buffers; Cell Line; Cell Membrane; Cocaine; Dopamine Uptake Inhibitors; Fluoxetine; Humans; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Piperazines; Radioligand Assay; Reproducibility of Results; Symporters; Temperature

2005
Studies of the biogenic amine transporters. XI. Identification of a 1-[2-[bis(4-fluorophenyl)methoxy]ethyl]-4-(3-phenylpropyl)piperazine (GBR12909) analog that allosterically modulates the serotonin transporter.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 314, Issue:2

    Topics: Animals; Benzhydryl Compounds; Binding, Competitive; Brain; Cell Line; Cocaine; Dopamine; Humans; In Vitro Techniques; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Neurotransmitter Agents; Piperazines; Piperidines; Protein Binding; Rats; Rats, Sprague-Dawley; Selective Serotonin Reuptake Inhibitors; Serotonin; Serotonin Plasma Membrane Transport Proteins

2005
Relationship between in vivo occupancy at the dopamine transporter and behavioral effects of cocaine, GBR 12909 [1-{2-[bis-(4-fluorophenyl)methoxy]ethyl}-4-(3-phenylpropyl)piperazine], and benztropine analogs.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 315, Issue:1

    Topics: Animals; Benztropine; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Mice; Motor Activity; Piperazines

2005
Behavioral disinhibition requires dopamine receptor activation.
    Psychopharmacology, 2006, Volume: 187, Issue:1

    Topics: Amphetamine; Animals; Behavior, Animal; Benzazepines; Cocaine; Desipramine; Dose-Response Relationship, Drug; Impulsive Behavior; Male; Nicotine; Piperazines; Rats; Rats, Wistar; Receptors, Dopamine; Serotonin

2006
Nicotine as a conditioned stimulus: impact of attention-deficit/hyperactivity disorder medications.
    Experimental and clinical psychopharmacology, 2007, Volume: 15, Issue:5

    Topics: Animals; Atomoxetine Hydrochloride; Attention Deficit Disorder with Hyperactivity; Behavior, Animal; Bupropion; Cocaine; Conditioning, Operant; Conditioning, Psychological; Discrimination Learning; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Generalization, Psychological; Male; Methylphenidate; Nicotine; Nicotinic Antagonists; Piperazines; Propylamines; Rats; Rats, Sprague-Dawley

2007
Ex vivo evaluation of N-(3-[18F]fluoropropyl)-2 beta-carbomethoxy-3 beta-(4-fluorophenyl)nortropane in rats.
    Nuclear medicine and biology, 2008, Volume: 35, Issue:2

    Topics: Animals; Binding, Competitive; Bone and Bones; Cerebellum; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Fluorine Radioisotopes; Limbic System; Male; Nortropanes; Piperazines; Radioligand Assay; Radionuclide Imaging; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Tissue Distribution

2008
Short-acting cocaine and long-acting GBR-12909 both elicit rapid dopamine uptake inhibition following intravenous delivery.
    Neuroscience, 2008, Jul-31, Volume: 155, Issue:1

    Topics: Analysis of Variance; Animals; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Interactions; Electric Stimulation; Injections, Intravenous; Male; Piperazines; Rats; Rats, Sprague-Dawley; Time Factors; Ventral Tegmental Area

2008
Different effects of selective dopamine uptake inhibitors, GBR 12909 and WIN 35428, on HIV-1 Tat toxicity in rat fetal midbrain neurons.
    Neurotoxicology, 2008, Volume: 29, Issue:6

    Topics: Animals; Cell Survival; Cells, Cultured; Cocaine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Interactions; Embryo, Mammalian; HIV Envelope Protein gp120; Mesencephalon; Neurons; Piperazines; Protein Binding; Rats; Serotonin Plasma Membrane Transport Proteins; tat Gene Products, Human Immunodeficiency Virus

2008
Dual DAT/sigma1 receptor ligands based on 3-(4-(3-(bis(4-fluorophenyl)amino)propyl)piperazin-1-yl)-1-phenylpropan-1-ol.
    Bioorganic & medicinal chemistry letters, 2008, Oct-01, Volume: 18, Issue:19

    Topics: Animals; Carbazoles; Cocaine; Combinatorial Chemistry Techniques; Dopamine Plasma Membrane Transport Proteins; Molecular Structure; Piperazines; Protein Binding; Rats; Receptors, sigma; Stereoisomerism; Structure-Activity Relationship

2008
Interaction of cocaine-, benztropine-, and GBR12909-like compounds with wild-type and mutant human dopamine transporters: molecular features that differentially determine antagonist-binding properties.
    Journal of neurochemistry, 2008, Volume: 107, Issue:4

    Topics: Animals; Asparagine; Aspartic Acid; Benztropine; Binding, Competitive; Cell Line, Transformed; Cocaine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Interactions; Humans; Leucine; Models, Molecular; Mutation; Piperazines; Protein Binding; Protein Structure, Tertiary; Sodium; Structure-Activity Relationship; Transfection; Tritium; Tryptophan

2008
Differential involvement of the norepinephrine, serotonin and dopamine reuptake transporter proteins in cocaine-induced taste aversion.
    Pharmacology, biochemistry, and behavior, 2009, Volume: 93, Issue:1

    Topics: Animals; Cocaine; Cocaine-Related Disorders; Conditioning, Psychological; Dopamine; Dopamine Uptake Inhibitors; Fluoxetine; Male; Mice; Norepinephrine; Piperazines; Selective Serotonin Reuptake Inhibitors; Serotonin; Taste

2009
High resolution micro-SPECT scanning in rats using 125I beta-CIT: effects of chronic treatment with carbamazepine.
    Epilepsia, 2009, Volume: 50, Issue:8

    Topics: Animals; Anticonvulsants; Autoradiography; Brain; Brain Mapping; Carbamazepine; Cocaine; Dopamine Uptake Inhibitors; Iodine Radioisotopes; Male; Piperazines; Protein Binding; Radiopharmaceuticals; Rats; Rats, Sprague-Dawley; Tomography, Emission-Computed, Single-Photon

2009
Monoaminergic psychomotor stimulants: discriminative stimulus effects and dopamine efflux.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 333, Issue:3

    Topics: Animals; Avoidance Learning; Biogenic Monoamines; Central Nervous System Stimulants; Cocaine; Conditioning, Operant; Discrimination, Psychological; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Extracellular Space; Male; Methamphetamine; Methylphenidate; Microdialysis; Motor Activity; Nucleus Accumbens; Piperazines; Rats; Rats, Sprague-Dawley; Reinforcement Schedule

2010
In vivo voltammetric monitoring of catecholamine release in subterritories of the nucleus accumbens shell.
    Neuroscience, 2010, Aug-11, Volume: 169, Issue:1

    Topics: Animals; Chromatography, High Pressure Liquid; Cocaine; Desipramine; Dopamine; Electric Stimulation; Male; Medial Forebrain Bundle; Microelectrodes; Neural Pathways; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Nucleus Accumbens; Piperazines; Raclopride; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic; Substantia Nigra; Synaptic Transmission; Ventral Tegmental Area

2010
Dopamine transporter-dependent and -independent striatal binding of the benztropine analog JHW 007, a cocaine antagonist with low abuse liability.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 335, Issue:3

    Topics: Adrenergic Uptake Inhibitors; Animals; Benztropine; Binding, Competitive; Cell Line, Tumor; Cell Membrane; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Female; Histamine H1 Antagonists; Humans; Kinetics; Male; Mice; Mice, 129 Strain; Mice, Inbred Strains; Mice, Knockout; Neuroblastoma; Piperazines; Pirenzepine; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Selective Serotonin Reuptake Inhibitors; Sodium; Triprolidine

2010
Dopamine mediates cocaine-induced conditioned taste aversions as demonstrated with cross-drug preexposure to GBR 12909.
    Pharmacology, biochemistry, and behavior, 2012, Volume: 102, Issue:2

    Topics: Animals; Avoidance Learning; Cocaine; Conditioning, Classical; Dopamine; Dopamine Uptake Inhibitors; Male; Piperazines; Rats; Rats, Sprague-Dawley; Taste

2012
Role of dopamine tone in the pursuit of brain stimulation reward.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Aug-08, Volume: 32, Issue:32

    Topics: Analysis of Variance; Animals; Brain; Cocaine; Conditioning, Operant; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Electric Stimulation; Male; Microdialysis; Models, Biological; Piperazines; Rats; Rats, Long-Evans; Reward; Self Stimulation; Time Factors

2012
Ablation of neurons expressing melanin-concentrating hormone (MCH) in adult mice improves glucose tolerance independent of MCH signaling.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2013, Jan-30, Volume: 33, Issue:5

    Topics: Animals; Behavior, Animal; Cocaine; Dopamine Uptake Inhibitors; Eating; Glucose; Glucose Tolerance Test; Hypothalamic Hormones; Melanins; Mice; Motor Activity; Neurons; Piperazines; Pituitary Hormones; Signal Transduction

2013
Amphetamine and cocaine suppress social play behavior in rats through distinct mechanisms.
    Psychopharmacology, 2014, Volume: 231, Issue:8

    Topics: Adrenergic Agents; Adrenergic alpha-2 Receptor Antagonists; Adrenergic Uptake Inhibitors; Amphetamine; Animals; Atomoxetine Hydrochloride; Behavior, Animal; Cocaine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Exploratory Behavior; Fluoxetine; Flupenthixol; Idazoxan; Male; Motor Activity; Piperazines; Play and Playthings; Propylamines; Rats, Wistar; Selective Serotonin Reuptake Inhibitors; Serotonin Antagonists; Social Behavior

2014
Involvement of reactive oxygen species in cocaine-taking behaviors in rats.
    Addiction biology, 2015, Volume: 20, Issue:4

    Topics: Animals; Antioxidants; Cocaine; Cocaine-Related Disorders; Conditioning, Operant; Cyclic N-Oxides; Dopamine; Dopamine Uptake Inhibitors; Dopaminergic Neurons; Male; Neuroprotective Agents; Nucleus Accumbens; Oxidative Stress; Piperazines; Rats, Sprague-Dawley; Reactive Oxygen Species; Reinforcement Schedule; Self Administration; Spin Labels

2015
Mutations at tyrosine 88, lysine 92 and tyrosine 470 of human dopamine transporter result in an attenuation of HIV-1 Tat-induced inhibition of dopamine transport.
    Journal of neuroimmune pharmacology : the official journal of the Society on NeuroImmune Pharmacology, 2015, Volume: 10, Issue:1

    Topics: Animals; Binding Sites; CHO Cells; Cocaine; Cricetinae; Cricetulus; Dopamine; Dopamine Plasma Membrane Transport Proteins; Humans; Lysine; Models, Molecular; Mutation; Piperazines; Protein Binding; Protein Conformation; tat Gene Products, Human Immunodeficiency Virus; Tyrosine

2015
Contrasting Roles of Dopamine and Noradrenaline in the Motivational Properties of Social Play Behavior in Rats.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2016, Volume: 41, Issue:3

    Topics: Adrenergic alpha-2 Receptor Antagonists; Adrenergic Uptake Inhibitors; Animals; Atomoxetine Hydrochloride; Cocaine; Conditioning, Operant; Dopamine; Dopamine Antagonists; Dopamine Uptake Inhibitors; Flupenthixol; Idazoxan; Male; Methylphenidate; Motivation; Neuropsychological Tests; Norepinephrine; Piperazines; Random Allocation; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Dopamine; Social Behavior

2016
Further delineation between typical and atypical dopamine uptake inhibitors: effects on food-maintained behavior and food consumption.
    Behavioural pharmacology, 2017, Volume: 28, Issue:1

    Topics: Animals; Behavior, Animal; Benztropine; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Eating; Feeding Behavior; Male; Piperazines; Rats; Rats, Sprague-Dawley; Reinforcement Schedule

2017
Behavioral profile of adult zebrafish acutely exposed to a selective dopamine uptake inhibitor, GBR 12909.
    Journal of psychopharmacology (Oxford, England), 2023, Volume: 37, Issue:6

    Topics: Animals; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Zebrafish

2023
Structure-activity relationships at monoamine transporters for a series of N-substituted 3alpha-(bis[4-fluorophenyl]methoxy)tropanes: comparative molecular field analysis, synthesis, and pharmacological evaluation.
    Journal of medicinal chemistry, 2004, Jun-17, Volume: 47, Issue:13

    Topics: Animals; Brain; Carrier Proteins; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; In Vitro Techniques; Male; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Nerve Tissue Proteins; Norepinephrine Plasma Membrane Transport Proteins; Protein Binding; Quantitative Structure-Activity Relationship; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Serotonin Plasma Membrane Transport Proteins; Symporters; Tropanes

2004
Further structurally constrained analogues of cis-(6-benzhydrylpiperidin-3-yl)benzylamine with elucidation of bioactive conformation: discovery of 1,4-diazabicyclo[3.3.1]nonane derivatives and evaluation of their biological properties for the monoamine tr
    Journal of medicinal chemistry, 2004, Oct-07, Volume: 47, Issue:21

    Topics: Animals; Benzhydryl Compounds; Biological Transport; Bridged Bicyclo Compounds, Heterocyclic; Carrier Proteins; Cocaine; Corpus Striatum; Crystallography, X-Ray; Discrimination Learning; Dopamine; Dopamine Plasma Membrane Transport Proteins; In Vitro Techniques; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Models, Molecular; Molecular Conformation; Motor Activity; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Piperidines; Radioligand Assay; Rats; Serotonin; Serotonin Plasma Membrane Transport Proteins; Stereoisomerism; Structure-Activity Relationship; Symporters

2004