cocaine and thiazoles
cocaine has been researched along with thiazoles in 62 studies
Research
Studies (62)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (3.23) | 18.7374 |
1990's | 10 (16.13) | 18.2507 |
2000's | 24 (38.71) | 29.6817 |
2010's | 25 (40.32) | 24.3611 |
2020's | 1 (1.61) | 2.80 |
Authors
Authors | Studies |
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Boudreau, NJ; Vohra, MM | 1 |
Lechat, P; Streichenberger, G | 1 |
Glatt, MM | 1 |
Acosta, D; Grant, RL | 1 |
Vanover, KE; Woolverton, WL | 1 |
Fisher, JE; Potturi, RB; Resnick, E; Zimmerman, EF | 1 |
O'Neill, WM | 1 |
Farag, M; Ho, JY; Lee, CC; Maximos, BB; Tosk, JM; Yung, HH | 1 |
Ferrari, F; Giuliani, D | 1 |
Caine, SB; Everitt, BJ; Koob, GF; Parsons, LH; Schwartz, JC; Sokoloff, P | 1 |
Misawa, M; Mori, T; Onodera, K; Suzuki, T; Tsuji, M | 1 |
Blakely, RD; Jansen, K; Richelson, E; Tatsumi, M | 1 |
Guttman, M; Houle, S; Hussey, D; Kish, S; Stewart, D; Wilson, A | 1 |
Enyedy, IJ; Johnson, KM; Wang, J; Wang, S; Zaman, WA | 1 |
Ahlskog, JE; Maraganore, DM; Uhl, GR; Uitti, RJ | 1 |
Davidson, C; Ellinwood, EH; King, GR; Lee, TH; Yu, GZ | 1 |
Bergmans, P; Booij, J; Stoof, JC; van Royen, EA; Winogrodzka, A; Wolters, EC | 1 |
Li, N; Sorg, BA; Wu, WR | 1 |
Batt, AM; Becuwe, P; Dauça, M; Ferrari, L; Lambert, H; Malaplate-Armand, C; Masson, C; Visvikis, S | 1 |
Cleveland, NJ; Dewitt, CD; Heard, K | 1 |
Clifton, PG; Hartfield, AW; Moore, NA | 1 |
Davis, J; Goeders, NE; Grajkowska, E; Iso, Y; Johnson, KM; Kozikowski, AP; Roth, BL; Sanker, S; Tueckmantel, W; Wroblewski, JT | 1 |
Bespalov, AY; Danysz, W; Dravolina, OA | 1 |
Feng, MJ; Yan, QS; Yan, SE | 1 |
Cleveland, NR; Heard, K; Krier, S | 1 |
Dey, S; Snow, DM | 1 |
Hoffman, RS; Manini, AF; Pearl-Davis, MS; Wu, S | 1 |
Fishback, JA; Green, AM; Kaushal, N; Matsumoto, RR; McCurdy, CR; Mésangeau, C; Narayanan, S; Poupaert, JH; Shaikh, J; Viard, E; Xu, YT | 1 |
Alvarez, Jdo N; Carvalho, Rde C; Frussa-Filho, R; Fukushiro, DF; Ribeiro, LT; Ricardo, VP | 1 |
Heard, K; Krier, S; Zahniser, NR | 1 |
Gass, JT; Olive, MF | 1 |
Baptista, MA; Dayas, CV; Martin-Fardon, R; Weiss, F | 1 |
Anderson, SM; Famous, KR; Kumaresan, V; Pierce, RC; Schmidt, HD; Yee, J; Yuan, M | 1 |
Di Paolo, T; Grégoire, L; Lévesque, D; Morissette, M; Ouattara, B; Rouillard, C; Samadi, P; Tamim, MK | 1 |
Hao, Y; Martin-Fardon, R; Weiss, F | 1 |
Boleij, H; Broekhoven, MH; Cousijn, J; Guitart Masip, M; Snoeren, EM; Spooren, W; Vanderschuren, LJ; Veeneman, MM | 1 |
Brown, RM; Duncan, JR; Lawrence, AJ; Ledent, C; Stagnitti, MR | 1 |
Steketee, JD; Timmer, KM | 1 |
Kalivas, PW; Knackstedt, L; Moussawi, K; Shen, H; Wang, X | 1 |
Orbach, R; Wang, F; Willner, I | 1 |
Knackstedt, LA; Schwendt, M; Trantham-Davidson, HL | 1 |
Bi, GH; Gardner, EL; Keck, TM; Newman, AH; Srivastava, R; Wang, XF; Xi, ZX; Yang, HJ; Zhang, HY; Zou, MF | 1 |
Baldaia, MA; Berro, LF; Frussa-Filho, R; Hollais, AW; Longo, BM; Marinho, EA; Oliveira-Lima, AJ; Santos, R; Wuo-Silva, R | 1 |
Arreola, AC; Kimmey, BA; Pierce, RC; Schmidt, HD | 1 |
Brown, RM; Kim, JH; Lawrence, AJ; Luikinga, S; Perry, C; Zbukvic, I | 1 |
Amato, RJ; Bubser, M; Byers, FW; Conn, PJ; Daniels, JS; Emmitte, KA; Felts, AS; Gould, RW; Joffe, ME; Jones, CK; Lindsley, CW; Morrison, RD; Nedelcovych, MT; Nickols, HH; Niswender, CM; Rodriguez, AL; Rook, JM; Thompson, AD; Yuh, JP; Zhan, X | 1 |
Buckner, RL; Hedden, T; Johnson, KA; Rieckmann, A; Sperling, RA; Younger, AP | 1 |
Bayer, S; Gomperts, SN; Growdon, JH; Johnson, KA; Locascio, JJ; Marquie, M | 1 |
Kim, JH; Lawrence, AJ; Perry, CJ; Reed, F; Zbukvic, IC | 1 |
Hasler, G; Mihov, Y | 1 |
Cannella, N; Spanagel, R; Takahashi, T; Vengeliene, V | 1 |
Baldaia, MA; Berro, LF; Frussa-Filho, R; Hollais, AW; Marinho, E; Oliveira-Lima, AJ; Ribeiro, LT; Santos-Baldaia, R; Talhati, F; Wuo-Silva, R | 1 |
Auber, A; Goldberg, SR; Justinova, Z; Panlilio, LV; Redhi, GH; Schindler, CW; Schwarcz, R; Secci, ME; Thorndike, EB | 1 |
Belin, D; Belin-Rauscent, A; Everitt, BJ; Hermine, O; Lacoste, J; Moussy, A | 1 |
Chen, T; Fu, LP; Gao, ZB; Wang, W; Wang, ZF; Xu, BX; Zhao, XL | 1 |
Hadad, NA; Hiller, H; Knackstedt, LA; Krause, EG; Namba, MD; Schwendt, M; Shallcross, J; Wu, L | 1 |
Asp, AJ; Benneyworth, MA; Ebner, SR; Hearing, MC; Ingebretson, AE; Larson, EB; Madayag, A; Schmidt, CE; Silvis, KA; Thomas, MJ | 1 |
Clement, N; Frosch, M; Gomez-Isla, T; Gomperts, SN; Growdon, JH; Johnson, KA; Katz, S; Schultz, A; Shirvan, J; Ye, R | 1 |
Gobin, C; Schwendt, M | 1 |
Bisaga, A; Danysz, W; Foltin, RW | 1 |
Reviews
1 review(s) available for cocaine and thiazoles
Article | Year |
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Negative Allosteric Modulators of Metabotropic Glutamate Receptors Subtype 5 in Addiction: a Therapeutic Window.
Topics: Allosteric Regulation; Animals; Cocaine; Drug-Seeking Behavior; Ethanol; Nicotine; Pyridines; Receptor, Metabotropic Glutamate 5; Self Administration; Substance-Related Disorders; Thiazoles | 2016 |
Trials
4 trial(s) available for cocaine and thiazoles
Article | Year |
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The cognitive and psychomotor effects of opioid drugs in cancer pain management.
Topics: Adult; Amphetamines; Analgesics, Opioid; Buprenorphine; Central Nervous System Stimulants; Chronic Disease; Cocaine; Codeine; Cognition; Dextropropoxyphene; Dopamine Uptake Inhibitors; Humans; Methylphenidate; Morphine; Neoplasms; Pain; Psychomotor Performance; Randomized Controlled Trials as Topic; Reaction Time; Thiazoles | 1994 |
Pramipexole vs levodopa as initial treatment for Parkinson disease: A randomized controlled trial. Parkinson Study Group.
Topics: Antiparkinson Agents; Benzothiazoles; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Agents; Dopamine Agonists; Dopamine Plasma Membrane Transport Proteins; Double-Blind Method; Dyskinesias; Female; Humans; Iodine Radioisotopes; Levodopa; Male; Membrane Glycoproteins; Membrane Transport Proteins; Middle Aged; Nerve Tissue Proteins; Parkinson Disease; Pramipexole; Proportional Hazards Models; Quality of Life; Radiopharmaceuticals; Thiazoles; Tomography, Emission-Computed, Single-Photon | 2000 |
Influence of L-dopa and pramipexole on striatal dopamine transporter in early PD.
Topics: Aged; Antiparkinson Agents; Benzothiazoles; Brain Chemistry; Carbon Radioisotopes; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Drug Therapy, Combination; Female; Humans; Levodopa; Male; Membrane Glycoproteins; Membrane Transport Proteins; Middle Aged; Nerve Tissue Proteins; Parkinson Disease; Pramipexole; Receptors, Dopamine; Thiazoles; Tomography, Emission-Computed | 2001 |
Dopamine transporter brain imaging to assess the effects of pramipexole vs levodopa on Parkinson disease progression.
Topics: Aged; Antiparkinson Agents; Benzothiazoles; Brain; Cocaine; Disease Progression; Dopamine; Dopamine Agents; Dopamine Plasma Membrane Transport Proteins; Female; Humans; Iodine Radioisotopes; Levodopa; Male; Membrane Glycoproteins; Membrane Transport Proteins; Middle Aged; Nerve Degeneration; Nerve Tissue Proteins; Parkinson Disease; Pramipexole; Radiopharmaceuticals; Randomized Controlled Trials as Topic; Regression Analysis; Thiazoles; Tomography, Emission-Computed, Single-Photon; Treatment Outcome | 2002 |
Other Studies
57 other study(ies) available for cocaine and thiazoles
Article | Year |
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The mechanism of [3H]noradrenaline release by histamine and its analogs from the rat vas deferens.
Topics: Animals; Cocaine; Desipramine; Histamine; Male; Methoxyhydroxyphenylglycol; Norepinephrine; Pyridines; Rats; Rats, Inbred Strains; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Tritium; Vas Deferens | 1991 |
[Application of sleep induced in the rat by sudden change in the environmental temperature to the study of antagonism between neurostimulants and hypnotics].
Topics: Amphetamine; Animals; Antidepressive Agents; Bemegride; Caffeine; Central Nervous System; Chloral Hydrate; Cocaine; Drug Antagonism; Environment; Hypnotics and Sedatives; Pentobarbital; Pentylenetetrazole; Piperidines; Pregnanediones; Rats; Secobarbital; Sleep; Strychnine; Temperature; Thiazoles | 1967 |
Chlormethiazole treatment of abstinence symptoms after drug withdrawal. Preliminary reports. II.
Topics: Adult; Cocaine; Female; Heroin; Humans; Hypnotics and Sedatives; Male; Meperidine; Substance Withdrawal Syndrome; Substance-Related Disorders; Thiazoles | 1966 |
Comparative toxicity of tetracaine, proparacaine and cocaine evaluated with primary cultures of rabbit corneal epithelial cells.
Topics: Anesthetics, Local; Animals; Cells, Cultured; Cocaine; Dose-Response Relationship, Drug; Endothelium, Corneal; L-Lactate Dehydrogenase; Mitochondria; Propoxycaine; Rabbits; Tetracaine; Tetrazolium Salts; Thiazoles; Time Factors | 1994 |
Behavioral effects of the dopamine autoreceptor agonist PD 128483 alone and in combination with cocaine.
Topics: Aminoquinolines; Animals; Behavior, Animal; Cocaine; Dopamine Agonists; Dose-Response Relationship, Drug; Drug Interactions; Feeding Behavior; Female; Macaca mulatta; Male; Milk; Self Administration; Thiazoles | 1994 |
Role of oxygen free radicals in cocaine-induced vascular disruption in mice.
Topics: Abnormalities, Drug-Induced; Animals; Antioxidants; Aorta; Blood Vessels; Cocaine; Cyclic N-Oxides; Female; Fetal Diseases; Fetal Heart; Gestational Age; Hemorrhage; Lipid Peroxidation; Maternal-Fetal Exchange; Mice; Mice, Inbred ICR; Nervous System; Nervous System Malformations; Neural Tube Defects; Nitrogen Oxides; Pregnancy; Pyrrolidonecarboxylic Acid; Reactive Oxygen Species; Thiazoles; Thiazolidines; Vasodilation; Yolk Sac | 1994 |
The effects of nerve growth factor and ganglioside GM1 on the anti-proliferative activity of cocaine in PC12 cells.
Topics: Animals; Cell Division; Cocaine; G(M1) Ganglioside; Nerve Growth Factors; PC12 Cells; Rats; Tetrazolium Salts; Thiazoles | 1996 |
Involvement of dopamine D2 receptors in the effect of cocaine on sexual behaviour and stretching-yawning of male rats.
Topics: Animals; Benzothiazoles; Cocaine; Copulation; Dopamine Agonists; Dopamine Antagonists; Lisuride; Male; Motor Activity; Pramipexole; Rats; Rats, Wistar; Receptors, Dopamine D2; Salicylamides; Sexual Behavior, Animal; Specific Pathogen-Free Organisms; Thiazoles | 1997 |
D3 receptor test in vitro predicts decreased cocaine self-administration in rats.
Topics: Animals; Benzopyrans; Benzothiazoles; Cocaine; Dopamine Agonists; Dopamine Antagonists; In Vitro Techniques; Male; Naphthalenes; Opioid-Related Disorders; Oxazines; Pramipexole; Pyrrolidines; Quinolines; Rats; Receptors, Dopamine D2; Receptors, Dopamine D3; Self Administration; Thiazoles | 1997 |
Generalization of D-, L- and DL-chlorpheniramine and zolantidine to the discriminative stimulus effects of cocaine and methamphetamine.
Topics: Animals; Antidepressive Agents, Tricyclic; Benzothiazoles; Chlorpheniramine; Clomipramine; Cocaine; Desipramine; Discrimination, Psychological; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Generalization, Stimulus; Histamine H1 Antagonists; Histamine H2 Antagonists; Humans; Male; Methamphetamine; Middle Aged; Phenoxypropanolamines; Piperazines; Piperidines; Rats; Rats, Inbred F344; Thiazoles | 1997 |
Pharmacological profile of neuroleptics at human monoamine transporters.
Topics: Antipsychotic Agents; Carrier Proteins; Cell Line; Chlorpromazine; Cocaine; Dibenzazepines; Dibenzothiepins; Dopamine Plasma Membrane Transport Proteins; Fluoxetine; Humans; Imipramine; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Norepinephrine Plasma Membrane Transport Proteins; Pimozide; Piperazines; Protein Binding; Radioligand Assay; Recombinant Fusion Proteins; Serotonin Plasma Membrane Transport Proteins; Symporters; Thiazoles; Triflupromazine; Tritium | 1999 |
Discovery of substituted 3,4-diphenyl-thiazoles as a novel class of monoamine transporter inhibitors through 3-D pharmacophore search using a new pharmacophore model derived from mazindol.
Topics: Binding Sites; Biphenyl Compounds; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Ligands; Mazindol; Membrane Glycoproteins; Membrane Transport Proteins; Models, Molecular; Nerve Tissue Proteins; Norepinephrine; Serotonin; Structure-Activity Relationship; Thiazoles | 2002 |
Brain imaging to assess the effects of dopamine agonists on progression of Parkinson disease.
Topics: Antiparkinson Agents; Benzothiazoles; Brain; Cocaine; Dopamine Agonists; Dopamine Plasma Membrane Transport Proteins; Humans; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Parkinson Disease; Pramipexole; Radiopharmaceuticals; Thiazoles; Tomography, Emission-Computed, Single-Photon | 2002 |
Effect of daily dosing duration of direct and indirect dopamine receptor agonists: cocaine cross-tolerance following chronic regimens.
Topics: Analysis of Variance; Animals; Area Under Curve; Autoreceptors; Benzothiazoles; Cocaine; Cocaine-Related Disorders; Cross-Over Studies; Dopamine Agonists; Dopamine Uptake Inhibitors; Drug Administration Schedule; Drug Interactions; Male; Motor Activity; Piperazines; Pramipexole; Psychomotor Performance; Rats; Rats, Sprague-Dawley; Thiazoles; Time Factors | 2002 |
[(123)I]beta-CIT SPECT is a useful method for monitoring dopaminergic degeneration in early stage Parkinson's disease.
Topics: Antiparkinson Agents; Benzothiazoles; Caudate Nucleus; Cocaine; Corpus Striatum; Disease Progression; Female; Humans; Male; Nerve Degeneration; Parkinson Disease; Pergolide; Pramipexole; Putamen; Radiopharmaceuticals; Receptors, Dopamine D2; Reproducibility of Results; Thiazoles; Tomography, Emission-Computed, Single-Photon; Treatment Outcome | 2003 |
Prolonged effects of repeated cocaine on medial prefrontal cortex dopamine response to cocaine and a stressful predatory odor challenge in rats.
Topics: Animals; Chromatography, High Pressure Liquid; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Extracellular Fluid; Microdialysis; Odorants; Prefrontal Cortex; Rats; Stress, Psychological; Substance Withdrawal Syndrome; Thiazoles; Time Factors | 2003 |
Effect of acute and chronic psychostimulant drugs on redox status, AP-1 activation and pro-enkephalin mRNA in the human astrocyte-like U373 MG cells.
Topics: Amino Acid Transport System X-AG; Amphetamine; Analysis of Variance; Astrocytes; Blotting, Western; Cell Line; Central Nervous System Agents; Cocaine; DNA-Binding Proteins; Dose-Response Relationship, Drug; Drug Administration Schedule; Electrophoretic Mobility Shift Assay; Enkephalins; Excitatory Amino Acid Transporter 2; Fluoresceins; Fos-Related Antigen-2; Gene Expression Regulation; Glial Fibrillary Acidic Protein; Humans; Oxidation-Reduction; Protein Precursors; Proto-Oncogene Proteins c-fos; Proto-Oncogene Proteins c-jun; Reactive Oxygen Species; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrazolium Salts; Thiazoles; Time Factors; Transcription Factor AP-1; Transcription Factors | 2005 |
Ziprasidone pretreatment attenuates the lethal effects of cocaine in a mouse model.
Topics: Acute Disease; Animals; Antipsychotic Agents; Cocaine; Cocaine-Related Disorders; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Overdose; Injections, Intraperitoneal; Mice; Piperazines; Premedication; Random Allocation; Seizures; Single-Blind Method; Survival Analysis; Thiazoles; Treatment Outcome | 2005 |
Effects of atypical antipsychotic drugs on intralipid intake and cocaine-induced hyperactivity in rats.
Topics: Animals; Antipsychotic Agents; Cocaine; Dibenzothiazepines; Dopamine Antagonists; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Eating; Fat Emulsions, Intravenous; Female; Hyperkinesis; Male; Motor Activity; Piperazines; Quetiapine Fumarate; Rats; Risperidone; Thiazoles | 2006 |
Synthesis and structure-activity relationships of 3-[(2-methyl-1,3-thiazol-4-yl)ethynyl]pyridine analogues as potent, noncompetitive metabotropic glutamate receptor subtype 5 antagonists; search for cocaine medications.
Topics: Allosteric Site; Animals; Cell Line; Cocaine; Cocaine-Related Disorders; Cricetinae; Cricetulus; Humans; Ligands; Male; Narcotics; Pyridines; Radioligand Assay; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Self Administration; Structure-Activity Relationship; Thiazoles | 2006 |
Effects of group I metabotropic glutamate receptor antagonists on the behavioral sensitization to motor effects of cocaine in rats.
Topics: Analysis of Variance; Animals; Behavior, Animal; Central Nervous System Stimulants; Cocaine; Cocaine-Related Disorders; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Motor Activity; Pyridines; Quinolines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Thiazoles; Time Factors | 2006 |
RNA interference-mediated inhibition of brain-derived neurotrophic factor expression increases cocaine's cytotoxicity in cultured cells.
Topics: Animals; Brain; Brain-Derived Neurotrophic Factor; Cell Death; Cell Line, Tumor; Cells, Cultured; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Down-Regulation; Gene Expression Regulation; Humans; Neurons; Rats; Rats, Sprague-Dawley; RNA Interference; RNA, Messenger; RNA, Small Interfering; Tetrazolium Salts; Thiazoles; Transfection | 2007 |
Ziprasidone, diazepam, or the combination for prevention of cocaine toxicity in a mouse model.
Topics: Animals; Cocaine; Cocaine-Related Disorders; Confidence Intervals; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Therapy, Combination; Male; Mice; Mice, Inbred Strains; Piperazines; Random Allocation; Reference Values; Sensitivity and Specificity; Statistics, Nonparametric; Survival Rate; Thiazoles | 2007 |
Cocaine exposure in vitro induces apoptosis in fetal locus coeruleus neurons through TNF-alpha-mediated induction of Bax and phosphorylated c-Jun NH(2)-terminal kinase.
Topics: Animals; Apoptosis; bcl-2-Associated X Protein; Blotting, Western; Caspase 3; Cell Survival; Cells, Cultured; Cocaine; Culture Media; Cyclin D1; Data Interpretation, Statistical; Enzyme-Linked Immunosorbent Assay; Female; In Situ Nick-End Labeling; JNK Mitogen-Activated Protein Kinases; Locus Coeruleus; Neurons; p38 Mitogen-Activated Protein Kinases; Phosphorylation; Pregnancy; Rats; Rats, Long-Evans; Recombinant Proteins; Signal Transduction; Tetrazolium Salts; Thiazoles; Tumor Necrosis Factor-alpha | 2007 |
Use of antipsychotics to treat cocaine toxicity?
Topics: Animals; Antipsychotic Agents; Cocaine; Cocaine-Related Disorders; Diazepam; Disease Models, Animal; Mice; Piperazines; Thiazoles; Treatment Outcome | 2008 |
Conversion of a highly selective sigma-1 receptor-ligand to sigma-2 receptor preferring ligands with anticocaine activity.
Topics: Animals; Anticonvulsants; Brain; Cocaine; Cocaine-Related Disorders; In Vitro Techniques; Ligands; Mice; Oxazoles; Piperazines; Radioligand Assay; Rats; Receptors, sigma; Seizures; Sigma-1 Receptor; Structure-Activity Relationship; Thiazoles | 2008 |
Haloperidol (but not ziprasidone) withdrawal potentiates sensitization to the hyperlocomotor effect of cocaine in mice.
Topics: Animals; Antipsychotic Agents; Behavior, Animal; Cocaine; Cocaine-Related Disorders; Haloperidol; Humans; Male; Mice; Motor Activity; Piperazines; Schizophrenia; Substance Withdrawal Syndrome; Thiazoles | 2008 |
Administration of ziprasidone for 10 days increases cocaine toxicity in mice.
Topics: Animals; Antipsychotic Agents; Cocaine; Cocaine-Related Disorders; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug Synergism; Longevity; Male; Mice; Mice, Inbred Strains; Piperazines; Seizures; Thiazoles; Time Factors; Withholding Treatment | 2008 |
Positive allosteric modulation of mGluR5 receptors facilitates extinction of a cocaine contextual memory.
Topics: Allosteric Site; Animals; Benzamides; Cocaine; Dizocilpine Maleate; Excitatory Amino Acid Antagonists; Extinction, Psychological; Male; Memory; Pyrazoles; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Thiazoles | 2009 |
Dissociation of the effects of MTEP [3-[(2-methyl-1,3-thiazol-4-yl)ethynyl]piperidine] on conditioned reinstatement and reinforcement: comparison between cocaine and a conventional reinforcer.
Topics: Animals; Behavior, Animal; Cocaine; Conditioning, Classical; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Extinction, Psychological; Locomotion; Male; Milk; Piperidines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Reinforcement Schedule; Reinforcement, Psychology; Self Administration; Thiazoles | 2009 |
Metabotropic glutamate receptor 5 (mGluR5) antagonists attenuate cocaine priming- and cue-induced reinstatement of cocaine seeking.
Topics: Animals; Catheterization; Cocaine; Cocaine-Related Disorders; Cues; Dietary Sucrose; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Extinction, Psychological; Male; Microinjections; Nucleus Accumbens; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Reinforcement Schedule; Self Administration; Thiazoles | 2009 |
Effect of non-dopaminergic drug treatment on Levodopa induced dyskinesias in MPTP monkeys: common implication of striatal neuropeptides.
Topics: Animals; Antiparkinson Agents; Benzoxazoles; Cocaine; Corpus Striatum; Disease Models, Animal; Docosahexaenoic Acids; Dopamine; Dopamine Uptake Inhibitors; Dynorphins; Dyskinesia, Drug-Induced; Enkephalins; Female; Iodine Isotopes; Levodopa; Macaca fascicularis; Naltrexone; Neuropeptides; Ovariectomy; Parkinsonian Disorders; Piperidines; Protein Precursors; RNA, Messenger; Sulfonamides; Tachykinins; Thiazoles; Time Factors | 2010 |
Behavioral and functional evidence of metabotropic glutamate receptor 2/3 and metabotropic glutamate receptor 5 dysregulation in cocaine-escalated rats: factor in the transition to dependence.
Topics: Amino Acids; Analysis of Variance; Animals; Behavior, Addictive; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Depressants; Cocaine; Cocaine-Related Disorders; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Male; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Reinforcement Schedule; Self Administration; Thiazoles | 2010 |
Dissociable roles of mGlu5 and dopamine receptors in the rewarding and sensitizing properties of morphine and cocaine.
Topics: Animals; Behavior, Animal; Cocaine; Dopamine Antagonists; Dose-Response Relationship, Drug; Flupenthixol; Male; Morphine; Motor Activity; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Reward; Thiazoles | 2011 |
mGlu5 and adenosine A2A receptor interactions regulate the conditioned effects of cocaine.
Topics: Analysis of Variance; Animals; Autoradiography; Brain; Cocaine; Conditioning, Operant; Dopamine Uptake Inhibitors; Drug Interactions; Excitatory Amino Acid Antagonists; Iodine Isotopes; Locomotion; Male; Mice; Mice, Knockout; Protein Binding; Pyridines; Radionuclide Imaging; Receptor, Adenosine A2A; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Thiazoles; Time Factors; Triazines; Triazoles | 2012 |
Examination of a role for metabotropic glutamate receptor 5 in the medial prefrontal cortex in cocaine sensitization in rats.
Topics: 6-Cyano-7-nitroquinoxaline-2,3-dione; Animals; Benzimidazoles; Central Nervous System Sensitization; Cocaine; Drug Interactions; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Male; Microinjections; Motor Activity; Prefrontal Cortex; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, AMPA; Receptors, Metabotropic Glutamate; Resorcinols; Thiazoles; Ventral Tegmental Area | 2012 |
Role of mGluR5 neurotransmission in reinstated cocaine-seeking.
Topics: Analysis of Variance; Animals; Biotinylation; Blotting, Western; Carrier Proteins; Cocaine; Cocaine-Related Disorders; Cues; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Excitatory Amino Acid Agonists; Extinction, Psychological; Glycine; Homer Scaffolding Proteins; Male; Microinjections; Nucleus Accumbens; Phenylacetates; Protein Binding; Protein Transport; Pyridines; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Recurrence; Self Administration; Synaptic Transmission; Thiazoles | 2013 |
Detection of metal ions (Cu2+, Hg2+) and cocaine by using ligation DNAzyme machinery.
Topics: Benzothiazoles; Biosensing Techniques; Cocaine; Colorimetry; Copper; DNA, Catalytic; Hemin; Hydrogen Peroxide; Ions; Ligation; Luminol; Mercury; Metals; Spectrophotometry, Ultraviolet; Sulfonic Acids; Thiazoles | 2012 |
The role of ventral and dorsal striatum mGluR5 in relapse to cocaine-seeking and extinction learning.
Topics: Allosteric Regulation; Analysis of Variance; Animals; Basal Ganglia; Biotinylation; Blotting, Western; Cocaine; Cocaine-Related Disorders; Cues; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Electrophysiological Phenomena; Extinction, Psychological; Infusions, Intravenous; Locomotion; Long-Term Synaptic Depression; Male; Microinjections; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Recurrence; Self Administration; Sucrose; Thiazoles | 2014 |
A novel mGluR5 antagonist, MFZ 10-7, inhibits cocaine-taking and cocaine-seeking behavior in rats.
Topics: Allosteric Regulation; Analysis of Variance; Animals; Binding, Competitive; Cocaine; Cues; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Enzyme-Linked Immunosorbent Assay; Excitatory Amino Acid Antagonists; HEK293 Cells; Humans; Imidazoles; In Vitro Techniques; Infusions, Intravenous; Inhibitory Concentration 50; Male; Motor Activity; Nitriles; Piperidines; Pyridines; Random Allocation; Rats; Receptor, Metabotropic Glutamate 5; Reinforcement Schedule; Reward; Secondary Prevention; Self Administration; Sucrose; Thiazoles | 2014 |
Selective action of an atypical neuroleptic on the mechanisms related to the development of cocaine addiction: a pre-clinical behavioural study.
Topics: Animals; Antipsychotic Agents; Aripiprazole; Behavior, Animal; Central Nervous System Sensitization; Cocaine; Cocaine-Related Disorders; Disease Models, Animal; Dopamine Antagonists; Dopamine Uptake Inhibitors; Haloperidol; Male; Mice; Motor Activity; Piperazines; Quinolones; Thiazoles | 2014 |
Group I metabotropic glutamate receptor-mediated activation of PKC gamma in the nucleus accumbens core promotes the reinstatement of cocaine seeking.
Topics: Animals; Benzimidazoles; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Nucleus Accumbens; Phosphorylation; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Thiazoles | 2015 |
Extinction of a cocaine-taking context that protects against drug-primed reinstatement is dependent on the metabotropic glutamate 5 receptor.
Topics: Analysis of Variance; Animals; Cocaine; Conditioning, Operant; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Extinction, Psychological; Male; Pyridines; Receptor, Metabotropic Glutamate 5; Recurrence; Reward; Self Administration; Thiazoles | 2015 |
Partial mGlu₅ Negative Allosteric Modulators Attenuate Cocaine-Mediated Behaviors and Lack Psychotomimetic-Like Effects.
Topics: Alkynes; Allosteric Regulation; Animals; Anti-Anxiety Agents; Antidepressive Agents; Brain; Cocaine; Conditioning, Classical; Conditioning, Operant; Dose-Response Relationship, Drug; Drug-Seeking Behavior; Male; Mice; Motor Activity; Phencyclidine; Pyridines; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Self Administration; Thiazoles | 2016 |
Dopamine transporter availability in clinically normal aging is associated with individual differences in white matter integrity.
Topics: Aged; Aged, 80 and over; Aging; Aniline Compounds; Benzothiazoles; Blood Pressure; Brain; Cocaine; Dopamine Plasma Membrane Transport Proteins; Female; Humans; Magnetic Resonance Imaging; Male; Multimodal Imaging; Organ Size; Positron-Emission Tomography; Radiopharmaceuticals; Regression Analysis; Thiazoles; White Matter | 2016 |
PET Radioligands Reveal the Basis of Dementia in Parkinson's Disease and Dementia with Lewy Bodies.
Topics: Alzheimer Disease; Aniline Compounds; Brain; Carbolines; Cocaine; Cognitive Dysfunction; Cross-Sectional Studies; Diagnosis, Differential; Lewy Body Disease; Magnetic Resonance Imaging; Neuropsychological Tests; Parkinson Disease; Prospective Studies; Radionuclide Imaging; Radiopharmaceuticals; Survival Analysis; Thiazoles | 2016 |
The metabotropic glutamate 5 receptor is necessary for extinction of cocaine-associated cues.
Topics: Animals; Benzamides; Cocaine; Cocaine-Related Disorders; Conditioning, Psychological; Cues; Male; Pyrazoles; Pyridines; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Thiazoles | 2016 |
Metabolic shift of the kynurenine pathway impairs alcohol and cocaine seeking and relapse.
Topics: Animals; Behavior, Animal; Central Nervous System Depressants; Cocaine; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Ethanol; Kynurenine; Kynurenine 3-Monooxygenase; Male; Metabolic Networks and Pathways; Rats; Rats, Wistar; Receptors, N-Methyl-D-Aspartate; Recurrence; Self Administration; Sulfonamides; Thiazoles | 2016 |
Context-dependent efficacy of a counter-conditioning strategy with atypical neuroleptic drugs in mice previously sensitized to cocaine.
Topics: Animals; Antipsychotic Agents; Aripiprazole; Cocaine; Conditioning, Operant; Dopamine Uptake Inhibitors; Exploratory Behavior; Hyperkinesis; Locomotion; Male; Mice; Piperazines; Statistics, Nonparametric; Thiazoles | 2017 |
Attenuating Nicotine Reinforcement and Relapse by Enhancing Endogenous Brain Levels of Kynurenic Acid in Rats and Squirrel Monkeys.
Topics: Animals; Cocaine; Dopamine; Isoxazoles; Kynurenic Acid; Male; Nicotine; Nucleus Accumbens; Phenylurea Compounds; Rats; Recurrence; Reinforcement, Psychology; Saimiri; Secondary Prevention; Self Administration; Sulfonamides; Thiazoles | 2017 |
Decrease of cocaine, but not heroin, self-administration and relapse by the tyrosine kinase inhibitor masitinib in male Sprague Dawley rats.
Topics: Administration, Oral; Analgesics, Opioid; Animals; Behavior, Addictive; Benzamides; Cocaine; Conditioning, Operant; Dopamine Uptake Inhibitors; Heroin; Male; Motivation; Piperidines; Protein Kinase Inhibitors; Pyridines; Rats; Rats, Sprague-Dawley; Recurrence; Reinforcement, Psychology; Self Administration; Thiazoles | 2018 |
Multi-modality molecular imaging characteristics of dementia with Lewy bodies.
Topics: Aged; Aged, 80 and over; Aniline Compounds; Cocaine; Dopamine Plasma Membrane Transport Proteins; Female; Fluorodeoxyglucose F18; Humans; Lewy Body Disease; Magnetic Resonance Imaging; Male; Middle Aged; Molecular Imaging; Multimodal Imaging; Neuroimaging; Positron-Emission Tomography; Radiopharmaceuticals; Thiazoles | 2018 |
A novel rat model of comorbid PTSD and addiction reveals intersections between stress susceptibility and enhanced cocaine seeking with a role for mGlu5 receptors.
Topics: Animals; Anxiety; Behavior, Animal; Brain; Cocaine; Cocaine-Related Disorders; Comorbidity; Disease Models, Animal; Drug-Seeking Behavior; Extinction, Psychological; Fear; Male; Phenotype; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Resilience, Psychological; Stress Disorders, Post-Traumatic; Stress, Psychological; Thiazoles | 2018 |
Synaptic Depotentiation and mGluR5 Activity in the Nucleus Accumbens Drive Cocaine-Primed Reinstatement of Place Preference.
Topics: Animals; Cocaine; Conditioning, Operant; Electrophysiological Phenomena; Long-Term Synaptic Depression; Male; Mice; Mice, Inbred C57BL; Neuronal Plasticity; Nucleus Accumbens; Optogenetics; Patch-Clamp Techniques; Piperidines; Receptors, AMPA; Receptors, Kainic Acid; Signal Transduction; Synaptic Potentials; Thiazoles | 2019 |
Neuropathologic correlates of amyloid and dopamine transporter imaging in Lewy body disease.
Topics: Aged; Aged, 80 and over; Amyloid beta-Peptides; Aniline Compounds; Autopsy; Brain; Cocaine; Contrast Media; Dopamine Plasma Membrane Transport Proteins; Female; Humans; Lewy Body Disease; Male; Middle Aged; Parkinson Disease; Positron-Emission Tomography; Thiazoles | 2019 |
The cognitive cost of reducing relapse to cocaine-seeking with mGlu5 allosteric modulators.
Topics: Animals; Benzamides; Cocaine; Cognition; Cues; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Excitatory Amino Acid Antagonists; Male; Memory, Short-Term; Pyrazoles; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Recurrence; Self Administration; Thiazoles | 2020 |
Antagonism of glutamatergic NMDA and mGluR5 receptors decreases consumption of food in baboon model of binge-eating disorder.
Topics: Animals; Appetite; Bulimia Nervosa; Candy; Conditioning, Operant; Consummatory Behavior; Dexfenfluramine; Dose-Response Relationship, Drug; Eating; Excitatory Amino Acid Antagonists; Female; Male; Memantine; Papio cynocephalus; Pyridines; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Receptors, N-Methyl-D-Aspartate; Reinforcement Schedule; Serotonin Receptor Agonists; Sex Characteristics; Thiazoles; Weight Gain | 2008 |