cocaine and rti 121

cocaine has been researched along with rti 121 in 61 studies

Research

Studies (61)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's27 (44.26)18.2507
2000's22 (36.07)29.6817
2010's12 (19.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carroll, FI; Dannals, RF; Kuhar, MJ; Scheffel, U; Wong, DF; Yokoi, F1
Boja, JW; Carroll, FI; Kuhar, MJ; Lever, SZ; Scheffel, U; Stathis, M1
Carroll, FI; Cassin, BJ; Little, KY1
al-Tikriti, MS; Baldwin, RM; Charney, DS; Giddings, SS; Hoffer, PB; Laruelle, M; Scanley, BE; Seibyl, JP; Zea-Ponce, Y; Zoghbi, SS1
al-Tikriti, MS; Baldwin, RM; Charney, DS; Gandelman, MS; Hoffer, PB; Laruelle, M; Scanley, BE; Wang, S; Zea-Ponce, Y; Zoghbi, SS1
Abraham, P; Boja, JW; Cadet, JL; Carroll, FI; Kopajtic, TA; Lever, J; Lewin, AH; Seltzman, HH; Wyrick, CD1
al-Tikriti, MS; Elsworth, JD; Innis, RB; Redmond, DE; Roth, RH; Sladek, JR; Taylor, JR1
Ali, S; Cadet, JL; Carlson, E; Epstein, C; Hirata, H; Ladenheim, B; Moran, TH; Rothman, RB1
Abraham, P; Boja, JW; Carroll, FI; Kuhar, MJ; Lever, JR; Parham, K; Scheffel, U; Seltzman, HH; Stathis, M; Thomas, BF; Wyrick, CD1
Ashworth, S; Brady, F; Brooks, DJ; Brown, DJ; Carroll, FI; Hume, SP; Kuhar, MJ; Luthra, SK; Myers, R; Opacka-Juffry, J; Osman, S1
Kuhar, MJ; Pilotte, NS; Rountree, SD; Sharpe, LG1
Abraham, P; Boja, JW; Carroll, FI; Lewin, AH; Mash, DC; Seltzman, HH; Staley, JK; Wyrick, CD1
Boja, JW; Carroll, FI; Fleckenstein, AE; Kopajtic, TA; Kuhar, MJ1
Chen, NH; Reith, ME; Wang, YL1
Cadet, JL; Ladenheim, B; Tella, SR1
Chen, NH; Ding, JH; Reith, ME; Wang, YL2
Cadet, JL; Hirata, H1
Ashworth, S; Brown, DJ; Hirani, E; Hume, SP; Lammertsma, AA; Luthra, SK1
Hume, SP; Lammertsma, AA1
Amdiss, F; Botez, MI; Hébert, C; Lalonde, R; Reader, TA; Strazielle, C1
Boja, JW; Carroll, FI; Kopajtic, T; Kuhar, MJ; Vaughan, RA1
Asanuma, M; Cadet, JL; Hirata, H1
Kreek, MJ; McEwen, BS; McKittrick, CR; Sarnyai, Z1
Chen, NH; Ding, JH; Wang, YL1
Fang, Y; Ronnekleiv, OK1
Lucas, LR; McEwen, BS; Pompei, P1
Al-Tikriti, MS; Baldwin, RM; Gandelman, MS; Hoffer, PB; Innis, RB; Laruelle, M; Neumeyer, JL; Scanley, BE; Wang, S; Zoghbi, SS1
Kim, DS; Palmiter, RD; Szczypka, MS1
Eberl, S; Fulham, MJ; Fulton, RR; Kassiou, M; Meikle, SR1
Bédard, PJ; Blanchet, PJ; Calon, F; Di Paolo, T; Goulet, M; Grondin, R; Lavertu, N; Lemieux, AM; Morissette, M1
Bohn, MC; Connor, B; Elsworth, JD; Kozlowski, DA; Schallert, T; Tillerson, JL; Unnerstall, JR1
Kulak, JM; McIntosh, JM; Polonskaya, Y; Quik, M1
Collins, SL; D'Addario, C; Izenwasser, S1
Allison, S; Angulo, JA; Cadet, JL; Ibrahim, D; Yu, J1
Boulanger, JF; Di Paolo, T; Ekue, A; Morissette, M1
Kulak, JM; McIntosh, JM; Musachio, JL; Quik, M1
Cass, WA; Guseva, M; Maragos, WF; Nath, A; Pauly, JR; Turchan, JT; Young, KL1
D'Astous, M; Di Paolo, T; Dluzen, DE; Gajjar, TM1
Desai, RI; Katz, JL; Koffarnus, M; Kopajtic, TA; Newman, AH1
Desai, RI; French, D; Katz, JL; Kopajtic, TA; Newman, AH1
Baroni, S; Betti, L; Cassano, GB; Catena, M; Dell'Osso, B; Fabbrini, L; Giannaccini, G; Italiani, P; Lucacchini, A; Marazziti, D1
Burton, NC; Guilarte, TR; Kensler, TW1
Cadet, JL; Deng, X; Jayanthi, S; Ladenheim, B1
McIntosh, JM; O'Leary, K; Parameswaran, N; Quik, M1
Alexander, M; Burton, NC; Griswold, M; Guilarte, TR; McGlothan, JL; Pham, L; Schneider, JS; Syversen, T; Verina, T; Wong, DF; Zhou, Y1
Bordia, T; Huang, LZ; Michael McIntosh, J; Parameswaran, N; Quik, M1
Calon, F; Di Paolo, T; Grégoire, L; Hornykiewicz, O; Rajput, A; Rajput, AH; Samadi, P1
Di Paolo, T; Grégoire, L; Lévesque, D; Morissette, M; Ouattara, B; Rouillard, C; Samadi, P; Tamim, MK1
Di Paolo, T; Gilbert, F; Grégoire, L; Lévesque, D; Mahmoudi, S; Morissette, M; Ouattara, B; Rouillard, C; Samadi, P1
Bordia, T; Campos, C; McIntosh, JM; Quik, M1
He, Z; Ma, T; Park, SW; Roman, RJ; Shen, X1
Crossman, AR; Kobylecki, C; Ravenscroft, P1
Daniju, Y; Davidson, C; Dawson, P; Dutta, N; Moffatt, JD; Opacka-Juffry, J; Ramsey, J1
Bornatowicz, B; Fink, C; Hacker, M; Haeusler, D; Mitterhauser, M; Nics, L; Otter, P; Rami-Mark, C; Spreitzer, H; Ungersboeck, J; Vraka, C; Wadsak, W1
Bevan, M; Davidson, C; Meintel, M; Opacka-Juffry, J; Patel, N; Pinnell, T1
Bordia, T; Drenan, RM; McGregor, M; McIntosh, JM; Quik, M1
Al Sweidi, S; Bourque, M; Caruso, D; Di Paolo, T; Melcangi, RC; Morissette, M1
Barrese, V; Davidson, C; Dutta, N; Khelashvili, G; Opacka-Juffry, J; Sahai, MA; Weinstein, H1
Bordia, T; Perez, XA; Quik, M; Zhang, D1
Di Paolo, T; Morin, N; Morissette, M; Rouillard, C1

Other Studies

61 other study(ies) available for cocaine and rti 121

ArticleYear
Dopamine transporter imaging with novel, selective cocaine analogs.
    Neuroreport, 1992, Volume: 3, Issue:11

    Topics: Animals; Brain; Brain Chemistry; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Nerve Tissue Proteins; Papio; Protein Binding; Tomography, Emission-Computed, Single-Photon

1992
Rate of binding of various inhibitors at the dopamine transporter in vivo.
    Psychopharmacology, 1995, Volume: 119, Issue:4

    Topics: Animals; Binding, Competitive; Bupropion; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred Strains; Nerve Tissue Proteins; Time Factors

1995
Characterization and localization of [125I]RTI-121 binding sites in human striatum and medial temporal lobe.
    The Journal of pharmacology and experimental therapeutics, 1995, Volume: 274, Issue:3

    Topics: Animals; Autoradiography; Binding Sites; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Guinea Pigs; Humans; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Rats; Rats, Sprague-Dawley; Temporal Lobe

1995
Characterization of the dopamine transporter in nonhuman primate brain: homogenate binding, whole body imaging, and ex vivo autoradiography using [125I] and [123I]IPCIT.
    Nuclear medicine and biology, 1995, Volume: 22, Issue:5

    Topics: Animals; Autoradiography; Brain Chemistry; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Female; Iodine Radioisotopes; Membrane Glycoproteins; Membrane Transport Proteins; Models, Biological; Nerve Tissue Proteins; Ovariectomy; Papio; Protein Binding; Tissue Distribution; Tomography, Emission-Computed, Single-Photon; Whole-Body Counting

1995
Comparison of [123I]beta-CIT and [123I]IPCIT as single-photon emission tomography radiotracers for the dopamine transporter in nonhuman primates.
    European journal of nuclear medicine, 1995, Volume: 22, Issue:1

    Topics: Animals; Brain; Brain Chemistry; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Female; Iodine Radioisotopes; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Papio; Sensitivity and Specificity; Serotonin; Serotonin Plasma Membrane Transport Proteins; Time Factors; Tomography, Emission-Computed, Single-Photon

1995
Selective labeling of the dopamine transporter by the high affinity ligand 3 beta-(4-[125I]iodophenyl)tropane-2 beta-carboxylic acid isopropyl ester.
    Molecular pharmacology, 1995, Volume: 47, Issue:4

    Topics: Animals; Brain; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Kinetics; Ligands; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Rats; Rats, Sprague-Dawley

1995
Novel radioligands for the dopamine transporter demonstrate the presence of intrastriatal nigral grafts in the MPTP-treated monkey: correlation with improved behavioral function.
    Experimental neurology, 1994, Volume: 126, Issue:2

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Autoradiography; Brain Tissue Transplantation; Carrier Proteins; Chlorocebus aethiops; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Fetal Tissue Transplantation; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Parkinson Disease, Secondary; Radioligand Assay; Serotonin Plasma Membrane Transport Proteins; Substantia Nigra; Transplantation, Heterotopic; Transplantation, Homologous

1994
Superoxide radicals mediate the biochemical effects of methylenedioxymethamphetamine (MDMA): evidence from using CuZn-superoxide dismutase transgenic mice.
    Synapse (New York, N.Y.), 1995, Volume: 21, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Autoradiography; Cocaine; Corpus Striatum; Dopamine; Female; Humans; Male; Mice; Mice, Transgenic; N-Methyl-3,4-methylenedioxyamphetamine; Receptors, Dopamine; Superoxide Dismutase; Superoxides; Tissue Distribution

1995
Synthesis and in vivo studies of a selective ligand for the dopamine transporter: 3 beta-(4-[125I]iodophenyl) tropan-2 beta-carboxylic acid isopropyl ester ([125I]RTI-121).
    Nuclear medicine and biology, 1996, Volume: 23, Issue:3

    Topics: Amphetamine; Analysis of Variance; Animals; Brain; Carrier Proteins; Chromatography, High Pressure Liquid; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Isotope Labeling; Kinetics; Ligands; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred Strains; Molecular Structure; Nerve Tissue Proteins; Tissue Distribution

1996
Evaluation of [11C]RTI-121 as a selective radioligand for PET studies of the dopamine transporter.
    Nuclear medicine and biology, 1996, Volume: 23, Issue:3

    Topics: Animals; Biotransformation; Blood Proteins; Brain; Carbon Radioisotopes; Carrier Proteins; Cerebellum; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Radioligand Assay; Rats; Rats, Sprague-Dawley; Tissue Distribution; Tomography, Emission-Computed

1996
Cocaine withdrawal reduces dopamine transporter binding in the shell of the nucleus accumbens.
    Synapse (New York, N.Y.), 1996, Volume: 22, Issue:1

    Topics: Animals; Autoradiography; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Image Processing, Computer-Assisted; Male; Membrane Glycoproteins; Membrane Transport Proteins; Narcotics; Neostriatum; Nerve Tissue Proteins; Nucleus Accumbens; Olfactory Bulb; Rats; Rats, Inbred Lew; Substance Withdrawal Syndrome; Ventral Tegmental Area

1996
Mapping dopamine transporters in the human brain with novel selective cocaine analog [125I]RTI-121.
    Synapse (New York, N.Y.), 1995, Volume: 21, Issue:4

    Topics: Adult; Autoradiography; Binding Sites; Binding, Competitive; Brain; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Female; Humans; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Tissue Distribution

1995
Highly potent cocaine analogs cause long-lasting increases in locomotor activity.
    European journal of pharmacology, 1996, Sep-12, Volume: 311, Issue:2-3

    Topics: Analysis of Variance; Animals; Behavior, Animal; Binding, Competitive; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Mice; Motor Activity; Rats; Rats, Sprague-Dawley

1996
Binding of the [125I]3 beta-(iodophenyl)tropan-2 beta-carboxylic acid isopropyl ester to the dopamine transporter at a physiologically relevant temperature: mutually exclusive binding and different ionic requirements for various uptake blockers and substr
    Synapse (New York, N.Y.), 1997, Volume: 25, Issue:2

    Topics: Animals; Binding, Competitive; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Rats; Rats, Sprague-Dawley; Synaptosomes

1997
Differential regulation of dopamine transporter after chronic self-administration of bupropion and nomifensine.
    The Journal of pharmacology and experimental therapeutics, 1997, Volume: 281, Issue:1

    Topics: Animals; Bupropion; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Nomifensine; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Administration

1997
Modeling of the interaction of Na+ and K+ with the binding of the cocaine analogue 3beta-(4-[125I]iodophenyl)tropane-2beta-carboxylic acid isopropyl ester to the dopamine transporter.
    Journal of neurochemistry, 1997, Volume: 68, Issue:5

    Topics: Animals; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Models, Biological; Nerve Tissue Proteins; Potassium; Rats; Rats, Sprague-Dawley; Sodium; Synaptosomes

1997
p53-knockout mice are protected against the long-term effects of methamphetamine on dopaminergic terminals and cell bodies.
    Journal of neurochemistry, 1997, Volume: 69, Issue:2

    Topics: Animals; Autoradiography; Brain; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Heterozygote; Homozygote; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Methamphetamine; Mice; Mice, Knockout; Nerve Tissue Proteins; Nucleus Accumbens; RNA, Messenger; Tumor Suppressor Protein p53; Tyrosine 3-Monooxygenase

1997
Potential misconceptions in dopamine transporter assays arising from the binding of [125I]RTI-121 to filters: effect of ions and cocaine.
    Journal of neuroscience methods, 1997, Aug-22, Volume: 75, Issue:2

    Topics: Animals; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Histocytochemistry; Iodine Radioisotopes; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Protein Binding; Rats; Rats, Sprague-Dawley; Sodium; Synaptosomes; Ultrafiltration

1997
In vivo saturation kinetics of two dopamine transporter probes measured using a small animal positron emission tomography scanner.
    Journal of neuroscience methods, 1997, Sep-05, Volume: 76, Issue:1

    Topics: Animals; Brain; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Male; Membrane Glycoproteins; Membrane Transport Proteins; Neostriatum; Nerve Tissue Proteins; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Tomography, Emission-Computed

1997
Simplified reference tissue model for PET receptor studies.
    NeuroImage, 1996, Volume: 4, Issue:3 Pt 1

    Topics: Animals; Benzazepines; Brain Mapping; Carrier Proteins; Cocaine; Computer Simulation; Dopamine Plasma Membrane Transport Proteins; Humans; Image Processing, Computer-Assisted; Membrane Glycoproteins; Membrane Transport Proteins; Models, Theoretical; Nerve Tissue Proteins; Raclopride; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Neurotransmitter; Reference Values; Salicylamides; Tomography, Emission-Computed

1996
Distribution of dopamine transporters in basal ganglia of cerebellar ataxic mice by [125I]RTI-121 quantitative autoradiography.
    Neurochemistry international, 1998, Volume: 32, Issue:1

    Topics: Animals; Autoradiography; Basal Ganglia; Carrier Proteins; Cerebellar Ataxia; Cocaine; Dopamine Plasma Membrane Transport Proteins; Heterozygote; Homozygote; Iodine Radioisotopes; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Neurologic Mutants; Neostriatum; Nerve Tissue Proteins; Nucleus Accumbens; Olfactory Pathways; Substantia Nigra; Tegmentum Mesencephali; Thalamus; Tissue Distribution

1998
Multiple binding sites for [125I]RTI-121 and other cocaine analogs in rat frontal cerebral cortex.
    Synapse (New York, N.Y.), 1998, Volume: 30, Issue:1

    Topics: Animals; Binding Sites; Binding, Competitive; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Frontal Lobe; Iodine Radioisotopes; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Rats; Rats, Sprague-Dawley; Regression Analysis; Serotonin; Serotonin Plasma Membrane Transport Proteins; Symporters

1998
Melatonin attenuates methamphetamine-induced toxic effects on dopamine and serotonin terminals in mouse brain.
    Synapse (New York, N.Y.), 1998, Volume: 30, Issue:2

    Topics: Animals; Antioxidants; Autoradiography; Brain Chemistry; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Iodine Radioisotopes; Male; Melatonin; Methamphetamine; Mice; Neostriatum; Nerve Endings; Nucleus Accumbens; Serotonin

1998
Selective regulation of dopamine transporter binding in the shell of the nucleus accumbens by adrenalectomy and corticosterone-replacement.
    Synapse (New York, N.Y.), 1998, Volume: 30, Issue:3

    Topics: Adrenal Glands; Adrenalectomy; Animals; Autoradiography; Brain; Carrier Proteins; Cocaine; Corticosterone; Dopamine; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Nucleus Accumbens; Organ Specificity; Rats; Rats, Sprague-Dawley

1998
Characterization of [125I]RTI-121 binding to dopamine transporter in vitro.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1997, Volume: 18, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Uptake Inhibitors; In Vitro Techniques; Male; Pergolide; Rats; Rats, Sprague-Dawley; Synaptosomes

1997
Cocaine upregulates the dopamine transporter in fetal rhesus monkey brain.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1999, Oct-15, Volume: 19, Issue:20

    Topics: Animals; Binding Sites; Brain; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Embryonic and Fetal Development; Fetus; Macaca mulatta; Membrane Glycoproteins; Membrane Transport Proteins; Mesencephalon; Nerve Tissue Proteins; Neurons; RNA, Messenger; Tissue Distribution; Tyrosine 3-Monooxygenase; Up-Regulation

1999
Correlates of deoxycorticosterone-induced salt appetite behavior and basal ganglia neurochemistry.
    Annals of the New York Academy of Sciences, 1999, Volume: 897

    Topics: Animals; Appetite; Basal Ganglia; Carrier Proteins; Cocaine; Desoxycorticosterone; Dopamine Plasma Membrane Transport Proteins; Dynorphins; Enkephalins; Gene Expression Regulation; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Nucleus Accumbens; Protein Precursors; Rats; Rats, Sprague-Dawley; RNA, Messenger; Sodium, Dietary; Transcription, Genetic; Tyrosine 3-Monooxygenase

1999
[123I]IPCIT and [123I]beta-CIT as SPECT tracers for the dopamine transporter: a comparative analysis in nonhuman primates.
    Nuclear medicine and biology, 2000, Volume: 27, Issue:1

    Topics: Animals; Brain; Carrier Proteins; Chromatography, High Pressure Liquid; Cocaine; Dopamine Plasma Membrane Transport Proteins; Female; Half-Life; Humans; Injections, Intravenous; Iodine Radioisotopes; Ligands; Membrane Glycoproteins; Membrane Transport Proteins; Metabolic Clearance Rate; Models, Biological; Nerve Tissue Proteins; Papio; Species Specificity; Time Factors; Tissue Distribution; Tomography, Emission-Computed, Single-Photon

2000
Dopamine-deficient mice are hypersensitive to dopamine receptor agonists.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2000, Jun-15, Volume: 20, Issue:12

    Topics: Animals; Autoradiography; Benzamides; Brain; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine beta-Hydroxylase; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Levodopa; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Knockout; Mice, Transgenic; Motor Activity; Nerve Tissue Proteins; Pyrrolidines; Receptors, Dopamine; Tyrosine 3-Monooxygenase

2000
The influence of tomograph sensitivity on kinetic parameter estimation in positron emission tomography imaging studies of the rat brain.
    Nuclear medicine and biology, 2000, Volume: 27, Issue:6

    Topics: Animals; Brain; Carrier Proteins; Cerebellum; Cocaine; Computer Simulation; Corpus Striatum; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Image Processing, Computer-Assisted; Ligands; Membrane Glycoproteins; Membrane Transport Proteins; Models, Neurological; Nerve Tissue Proteins; Phantoms, Imaging; Raclopride; Radioisotopes; Rats; Reproducibility of Results; Sensitivity and Specificity; Tomography, Emission-Computed

2000
Effect of MPTP-induced denervation on basal ganglia GABA(B) receptors: correlation with dopamine concentrations and dopamine transporter.
    Synapse (New York, N.Y.), 2001, Jun-01, Volume: 40, Issue:3

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Basal Ganglia; Benzoates; Cocaine; Corpus Striatum; Disease Models, Animal; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Female; Macaca fascicularis; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Nerve Tissue Proteins; Organophosphorus Compounds; Parkinsonian Disorders; Protein Subunits; Radioligand Assay; Receptors, GABA-B; RNA, Messenger; Substantia Nigra; Subthalamic Nucleus

2001
Glial cell line-derived neurotrophic factor (GDNF) gene delivery protects dopaminergic terminals from degeneration.
    Experimental neurology, 2001, Volume: 169, Issue:1

    Topics: Aging; Animals; Autoradiography; Carrier Proteins; Cocaine; Corpus Striatum; Disease Models, Animal; Dopamine; Dopamine Plasma Membrane Transport Proteins; Genetic Therapy; Genetic Vectors; Glial Cell Line-Derived Neurotrophic Factor; Male; Membrane Glycoproteins; Membrane Transport Proteins; Microinjections; Motor Activity; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Neurotransmitter Agents; Oxidopamine; Parkinson Disease, Secondary; Presynaptic Terminals; Rats; Rats, Inbred F344; RNA, Messenger; Substantia Nigra; Tyrosine 3-Monooxygenase

2001
Vulnerability of 125I-alpha-conotoxin MII binding sites to nigrostriatal damage in monkey.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2001, Aug-01, Volume: 21, Issue:15

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Autoradiography; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Carrier Proteins; Cocaine; Conotoxins; Corpus Striatum; Disease Models, Animal; Dopamine; Dopamine Plasma Membrane Transport Proteins; Female; Habenula; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mesencephalon; Nerve Tissue Proteins; Neural Pathways; Neurons; Parkinson Disease, Secondary; Putamen; Pyridines; Receptors, Nicotinic; Saimiri; Substantia Nigra

2001
Effects of kappa-opioid receptor agonists on long-term cocaine use and dopamine neurotransmission.
    European journal of pharmacology, 2001, Aug-24, Volume: 426, Issue:1-2

    Topics: Analgesics; Animals; Autoradiography; Benzazepines; Benzeneacetamides; Benzomorphans; Binding, Competitive; Brain; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Motor Activity; Nerve Tissue Proteins; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Opioid, kappa; Sulpiride; Synaptic Transmission; Time Factors; Tyrosine 3-Monooxygenase

2001
Ontogeny of neurokinin-1 receptor mediation of methamphetamine neurotoxicity in the striatum of the mouse brain.
    Annals of the New York Academy of Sciences, 2002, Volume: 965

    Topics: Animals; Autoradiography; Binding Sites; Caudate Nucleus; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Methamphetamine; Mice; Mice, Inbred ICR; Nerve Tissue Proteins; Putamen; Receptors, Neurokinin-1; Substance P

2002
Lack of effect of testosterone and dihydrotestosterone compared to 17beta-oestradiol in 1-methyl-4-phenyl-1,2,3,6, tetrahydropyridine-mice.
    Journal of neuroendocrinology, 2002, Volume: 14, Issue:9

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Autoradiography; Cocaine; Dihydrotestosterone; Dopamine; Dopamine Plasma Membrane Transport Proteins; Estradiol; Gonadal Steroid Hormones; Homovanillic Acid; In Situ Hybridization; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; MPTP Poisoning; Nerve Tissue Proteins; Neuropeptides; RNA, Messenger; Testosterone; Tetrabenazine; Tritium; Vesicular Biogenic Amine Transport Proteins; Vesicular Monoamine Transport Proteins

2002
Declines in different beta2* nicotinic receptor populations in monkey striatum after nigrostriatal damage.
    The Journal of pharmacology and experimental therapeutics, 2002, Volume: 303, Issue:2

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Autoradiography; Azetidines; Brain Chemistry; Caudate Nucleus; Cocaine; Conotoxins; Neostriatum; Parkinson Disease, Secondary; Putamen; Radioligand Assay; Receptors, Nicotinic; Saimiri; Substantia Nigra

2002
Human immunodeficiency virus-1 Tat protein and methamphetamine interact synergistically to impair striatal dopaminergic function.
    Journal of neurochemistry, 2002, Volume: 83, Issue:4

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antioxidants; Binding, Competitive; Body Temperature; Cell Death; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Drug Synergism; Gene Products, tat; HIV-1; Homovanillic Acid; Humans; Hydroxyindoleacetic Acid; Intracellular Membranes; Male; Membrane Glycoproteins; Membrane Potentials; Membrane Transport Proteins; Methamphetamine; Mitochondria; Nerve Tissue Proteins; Neurons; Rats; Rats, Sprague-Dawley; Serotonin; tat Gene Products, Human Immunodeficiency Virus

2002
Dopamine transporter as a marker of neuroprotection in methamphetamine-lesioned mice treated acutely with estradiol.
    Neuroendocrinology, 2004, Volume: 79, Issue:6

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Autoradiography; Chromatography, High Pressure Liquid; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Interactions; Estradiol; Female; In Situ Hybridization; Iodine Isotopes; Membrane Glycoproteins; Membrane Transport Proteins; Methamphetamine; Mice; Neostriatum; Nerve Tissue Proteins; Nervous System Diseases; Neuroprotective Agents; Ovariectomy; Protein Binding; RNA, Messenger; Substantia Nigra; Time Factors

2004
Identification of a dopamine transporter ligand that blocks the stimulant effects of cocaine.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2005, Feb-23, Volume: 25, Issue:8

    Topics: Animals; Benztropine; Central Nervous System Stimulants; Cerebellum; Cocaine; Corpus Striatum; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Inhibitory Concentration 50; Ligands; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Motor Activity; Nerve Tissue Proteins; Rats

2005
Relationship between in vivo occupancy at the dopamine transporter and behavioral effects of cocaine, GBR 12909 [1-{2-[bis-(4-fluorophenyl)methoxy]ethyl}-4-(3-phenylpropyl)piperazine], and benztropine analogs.
    The Journal of pharmacology and experimental therapeutics, 2005, Volume: 315, Issue:1

    Topics: Animals; Benztropine; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Mice; Motor Activity; Piperazines

2005
Binding of 3H-WIN-35,428 and 125I-RTI-121 to human platelet membranes.
    Neurochemical research, 2006, Volume: 31, Issue:3

    Topics: Adult; Blood Platelets; Cell Membrane; Cocaine; Dopamine Plasma Membrane Transport Proteins; Female; Humans; In Vitro Techniques; Iodine Radioisotopes; Ligands; Male; Protein Binding

2006
In vivo modulation of the Parkinsonian phenotype by Nrf2.
    Neurotoxicology, 2006, Volume: 27, Issue:6

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Antineoplastic Agents; Autoradiography; Cocaine; Disease Models, Animal; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Drug Interactions; Iodine Isotopes; Male; Mice; Mice, Inbred ICR; Mice, Knockout; NF-E2-Related Factor 2; Parkinsonian Disorders; Phenotype; Thiones; Thiophenes

2006
Methamphetamine administration causes death of dopaminergic neurons in the mouse olfactory bulb.
    Biological psychiatry, 2007, Jun-01, Volume: 61, Issue:11

    Topics: Animals; Apoptosis; Autoradiography; Blotting, Western; Cell Death; Central Nervous System Stimulants; Cerebral Cortex; Chromatography, High Pressure Liquid; Cocaine; Dopamine; Immunohistochemistry; In Situ Nick-End Labeling; Male; Methamphetamine; Mice; Mice, Inbred ICR; Neostriatum; Neurons; Olfactory Bulb; Presynaptic Terminals; Tyrosine 3-Monooxygenase

2007
Cotinine selectively activates a subpopulation of alpha3/alpha6beta2 nicotinic receptors in monkey striatum.
    The Journal of pharmacology and experimental therapeutics, 2008, Volume: 325, Issue:2

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Azetidines; Brain; Cocaine; Conotoxins; Cotinine; Dopamine; Dopamine Agents; Female; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Receptors, Nicotinic; Saimiri

2008
Impairment of nigrostriatal dopamine neurotransmission by manganese is mediated by pre-synaptic mechanism(s): implications to manganese-induced parkinsonism.
    Journal of neurochemistry, 2008, Volume: 107, Issue:5

    Topics: Amphetamine; Animals; Cocaine; Corpus Striatum; Cyclohexanols; Disease Models, Animal; Dopamine; Dopamine Agents; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Image Processing, Computer-Assisted; Macaca fascicularis; Male; Manganese; Parkinsonian Disorders; Positron-Emission Tomography; Substantia Nigra; Synaptic Transmission; Tetrabenazine; Tyrosine 3-Monooxygenase

2008
Nicotine is neuroprotective when administered before but not after nigrostriatal damage in rats and monkeys.
    Journal of neurochemistry, 2009, Volume: 109, Issue:3

    Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Amphetamine; Analysis of Variance; Animals; Autoradiography; Cocaine; Conotoxins; Corpus Striatum; Cotinine; Disease Models, Animal; Dopamine; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Iodine Isotopes; Male; Motor Activity; Neuroprotective Agents; Neurotoxicity Syndromes; Nicotine; Oxidopamine; Protein Binding; Rats; Rats, Sprague-Dawley; Saimiri; Substantia Nigra; Time Factors

2009
Metabotropic glutamate receptor II in the brains of Parkinsonian patients.
    Journal of neuropathology and experimental neurology, 2009, Volume: 68, Issue:4

    Topics: Aged; Aged, 80 and over; Amino Acids; Antiparkinson Agents; Brain; Cocaine; Dyskinesia, Drug-Induced; Excitatory Amino Acid Antagonists; Female; Humans; Iodine Radioisotopes; Levodopa; Male; Parkinsonian Disorders; Postmortem Changes; Radioligand Assay; Receptors, Metabotropic Glutamate; Tritium; Xanthenes

2009
Effect of non-dopaminergic drug treatment on Levodopa induced dyskinesias in MPTP monkeys: common implication of striatal neuropeptides.
    Neuropharmacology, 2010, Volume: 58, Issue:1

    Topics: Animals; Antiparkinson Agents; Benzoxazoles; Cocaine; Corpus Striatum; Disease Models, Animal; Docosahexaenoic Acids; Dopamine; Dopamine Uptake Inhibitors; Dynorphins; Dyskinesia, Drug-Induced; Enkephalins; Female; Iodine Isotopes; Levodopa; Macaca fascicularis; Naltrexone; Neuropeptides; Ovariectomy; Parkinsonian Disorders; Piperidines; Protein Precursors; RNA, Messenger; Sulfonamides; Tachykinins; Thiazoles; Time Factors

2010
Nur77 mRNA levels and L-Dopa-induced dyskinesias in MPTP monkeys treated with docosahexaenoic acid.
    Neurobiology of disease, 2009, Volume: 36, Issue:1

    Topics: Acetylcholinesterase; Analysis of Variance; Animals; Antiparkinson Agents; Autoradiography; Brain; Cocaine; Disease Models, Animal; Docosahexaenoic Acids; Drug Interactions; Dyskinesia, Drug-Induced; Female; Iodine Isotopes; Levodopa; Macaca fascicularis; MPTP Poisoning; Nuclear Receptor Subfamily 4, Group A, Member 1; Protein Binding; RNA, Messenger; Statistics as Topic

2009
Nicotinic receptor-mediated reduction in L-DOPA-induced dyskinesias may occur via desensitization.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 333, Issue:3

    Topics: Amphetamine; Animals; Antiparkinson Agents; Autoradiography; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Calcium Channel Blockers; Central Nervous System Stimulants; Cocaine; Conotoxins; Dopamine Plasma Membrane Transport Proteins; Dyskinesia, Drug-Induced; Functional Laterality; Levodopa; Male; Mecamylamine; Neostriatum; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Stereotyped Behavior

2010
Differential action of methamphetamine on tyrosine hydroxylase and dopamine transport in the nigrostriatal pathway of μ-opioid receptor knockout mice.
    The International journal of neuroscience, 2012, Volume: 122, Issue:6

    Topics: Animals; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Gene Expression; Iodine Radioisotopes; Male; Methamphetamine; Mice; Mice, Inbred C57BL; Mice, Knockout; Neural Pathways; Neurons; Radionuclide Imaging; Radiopharmaceuticals; Receptors, Opioid, mu; Substantia Nigra; Tyrosine 3-Monooxygenase

2012
Alternative splicing of AMPA receptor subunits in the 6-OHDA-lesioned rat model of Parkinson's disease and L-DOPA-induced dyskinesia.
    Experimental neurology, 2013, Volume: 247

    Topics: Adamantane; Alternative Splicing; Animals; Antiparkinson Agents; Cocaine; Corpus Striatum; Disease Models, Animal; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Iodine Isotopes; Levodopa; Male; Motor Activity; Oxidopamine; Parkinson Disease; Rats; Rats, Sprague-Dawley; Receptors, AMPA; RNA, Messenger; Sympatholytics

2013
The effects of benzofury (5-APB) on the dopamine transporter and 5-HT2-dependent vasoconstriction in the rat.
    Progress in neuro-psychopharmacology & biological psychiatry, 2014, Jan-03, Volume: 48

    Topics: Animals; Aorta; Benzofurans; Brain; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; In Vitro Techniques; Iodine Isotopes; Ketanserin; Male; Muscle Contraction; N-Methyl-3,4-methylenedioxyamphetamine; Propylamines; Protein Binding; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT2; Serotonin Agents; Tritium; Vasoconstriction

2014
Synthesis, radiosynthesis and first in vitro evaluation of novel PET-tracers for the dopamine transporter: [(11)C]IPCIT and [(18)F]FE@IPCIT.
    Bioorganic & medicinal chemistry, 2013, Dec-15, Volume: 21, Issue:24

    Topics: Carbon Isotopes; Cocaine; Dopamine Plasma Membrane Transport Proteins; Fluorine Radioisotopes; Humans; Molecular Conformation; Positron-Emission Tomography; Radioactive Tracers

2013
Stimulant mechanisms of cathinones - effects of mephedrone and other cathinones on basal and electrically evoked dopamine efflux in rat accumbens brain slices.
    Progress in neuro-psychopharmacology & biological psychiatry, 2014, Oct-03, Volume: 54

    Topics: Amphetamine; Amphetamines; Animals; Bupropion; Central Nervous System Stimulants; Cocaine; Diethylpropion; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Electric Stimulation; Iodine Radioisotopes; Male; Methamphetamine; Microelectrodes; Nucleus Accumbens; Propiophenones; Radioligand Assay; Rats, Wistar; Tissue Culture Techniques

2014
Evidence for a role for α6(∗) nAChRs in l-dopa-induced dyskinesias using Parkinsonian α6(∗) nAChR gain-of-function mice.
    Neuroscience, 2015, Jun-04, Volume: 295

    Topics: Adrenergic Agents; Analysis of Variance; Animals; Antiparkinson Agents; Benserazide; Cocaine; Disease Models, Animal; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Levodopa; Male; Mice; Mice, Transgenic; Nicotine; Nicotinic Agonists; Oxidopamine; Parkinsonian Disorders; Protein Binding; Receptors, Nicotinic

2015
Neuroprotective Effect of Progesterone in MPTP-Treated Male Mice.
    Neuroendocrinology, 2016, Volume: 103, Issue:3-4

    Topics: Androstane-3,17-diol; Animals; Autoradiography; Brain; Carbon Radioisotopes; Cocaine; Dihydrotestosterone; Disease Models, Animal; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Drug Administration Schedule; Male; Mice; Mice, Inbred C57BL; MPTP Poisoning; Neuroprotective Agents; Progesterone; Testosterone; Vesicular Monoamine Transport Proteins

2016
Combined in vitro and in silico approaches to the assessment of stimulant properties of novel psychoactive substances - The case of the benzofuran 5-MAPB.
    Progress in neuro-psychopharmacology & biological psychiatry, 2017, 04-03, Volume: 75

    Topics: Animals; Benzofurans; Central Nervous System Stimulants; Cocaine; Computer Simulation; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Electrochemical Techniques; In Vitro Techniques; Iodine Isotopes; Male; Methamphetamine; Models, Molecular; Protein Binding; Psychotropic Drugs; Rats; Rats, Wistar

2017
Striatal D1 medium spiny neuron activation induces dyskinesias in parkinsonian mice.
    Movement disorders : official journal of the Movement Disorder Society, 2017, Volume: 32, Issue:4

    Topics: Animals; Antiparkinson Agents; Channelrhodopsins; Cocaine; Corpus Striatum; Disease Models, Animal; Dopamine Plasma Membrane Transport Proteins; Dyskinesias; Female; Gene Expression Regulation; Levodopa; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Neurons; Oxidopamine; Parkinsonian Disorders; Receptors, Dopamine D1; Sympatholytics

2017
Membrane cholesterol removal and replenishment affect rat and monkey brain monoamine transporters.
    Neuropharmacology, 2018, 05-01, Volume: 133

    Topics: Animals; Brain; Cell Membrane; Cholesterol; Cocaine; Cyclodextrins; Dopamine; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Iodine Radioisotopes; Macaca fascicularis; Male; Membrane Transport Proteins; Protein Binding; Rats; Rats, Sprague-Dawley

2018