cocaine has been researched along with rti 121 in 61 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 27 (44.26) | 18.2507 |
2000's | 22 (36.07) | 29.6817 |
2010's | 12 (19.67) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Carroll, FI; Dannals, RF; Kuhar, MJ; Scheffel, U; Wong, DF; Yokoi, F | 1 |
Boja, JW; Carroll, FI; Kuhar, MJ; Lever, SZ; Scheffel, U; Stathis, M | 1 |
Carroll, FI; Cassin, BJ; Little, KY | 1 |
al-Tikriti, MS; Baldwin, RM; Charney, DS; Giddings, SS; Hoffer, PB; Laruelle, M; Scanley, BE; Seibyl, JP; Zea-Ponce, Y; Zoghbi, SS | 1 |
al-Tikriti, MS; Baldwin, RM; Charney, DS; Gandelman, MS; Hoffer, PB; Laruelle, M; Scanley, BE; Wang, S; Zea-Ponce, Y; Zoghbi, SS | 1 |
Abraham, P; Boja, JW; Cadet, JL; Carroll, FI; Kopajtic, TA; Lever, J; Lewin, AH; Seltzman, HH; Wyrick, CD | 1 |
al-Tikriti, MS; Elsworth, JD; Innis, RB; Redmond, DE; Roth, RH; Sladek, JR; Taylor, JR | 1 |
Ali, S; Cadet, JL; Carlson, E; Epstein, C; Hirata, H; Ladenheim, B; Moran, TH; Rothman, RB | 1 |
Abraham, P; Boja, JW; Carroll, FI; Kuhar, MJ; Lever, JR; Parham, K; Scheffel, U; Seltzman, HH; Stathis, M; Thomas, BF; Wyrick, CD | 1 |
Ashworth, S; Brady, F; Brooks, DJ; Brown, DJ; Carroll, FI; Hume, SP; Kuhar, MJ; Luthra, SK; Myers, R; Opacka-Juffry, J; Osman, S | 1 |
Kuhar, MJ; Pilotte, NS; Rountree, SD; Sharpe, LG | 1 |
Abraham, P; Boja, JW; Carroll, FI; Lewin, AH; Mash, DC; Seltzman, HH; Staley, JK; Wyrick, CD | 1 |
Boja, JW; Carroll, FI; Fleckenstein, AE; Kopajtic, TA; Kuhar, MJ | 1 |
Chen, NH; Reith, ME; Wang, YL | 1 |
Cadet, JL; Ladenheim, B; Tella, SR | 1 |
Chen, NH; Ding, JH; Reith, ME; Wang, YL | 2 |
Cadet, JL; Hirata, H | 1 |
Ashworth, S; Brown, DJ; Hirani, E; Hume, SP; Lammertsma, AA; Luthra, SK | 1 |
Hume, SP; Lammertsma, AA | 1 |
Amdiss, F; Botez, MI; Hébert, C; Lalonde, R; Reader, TA; Strazielle, C | 1 |
Boja, JW; Carroll, FI; Kopajtic, T; Kuhar, MJ; Vaughan, RA | 1 |
Asanuma, M; Cadet, JL; Hirata, H | 1 |
Kreek, MJ; McEwen, BS; McKittrick, CR; Sarnyai, Z | 1 |
Chen, NH; Ding, JH; Wang, YL | 1 |
Fang, Y; Ronnekleiv, OK | 1 |
Lucas, LR; McEwen, BS; Pompei, P | 1 |
Al-Tikriti, MS; Baldwin, RM; Gandelman, MS; Hoffer, PB; Innis, RB; Laruelle, M; Neumeyer, JL; Scanley, BE; Wang, S; Zoghbi, SS | 1 |
Kim, DS; Palmiter, RD; Szczypka, MS | 1 |
Eberl, S; Fulham, MJ; Fulton, RR; Kassiou, M; Meikle, SR | 1 |
Bédard, PJ; Blanchet, PJ; Calon, F; Di Paolo, T; Goulet, M; Grondin, R; Lavertu, N; Lemieux, AM; Morissette, M | 1 |
Bohn, MC; Connor, B; Elsworth, JD; Kozlowski, DA; Schallert, T; Tillerson, JL; Unnerstall, JR | 1 |
Kulak, JM; McIntosh, JM; Polonskaya, Y; Quik, M | 1 |
Collins, SL; D'Addario, C; Izenwasser, S | 1 |
Allison, S; Angulo, JA; Cadet, JL; Ibrahim, D; Yu, J | 1 |
Boulanger, JF; Di Paolo, T; Ekue, A; Morissette, M | 1 |
Kulak, JM; McIntosh, JM; Musachio, JL; Quik, M | 1 |
Cass, WA; Guseva, M; Maragos, WF; Nath, A; Pauly, JR; Turchan, JT; Young, KL | 1 |
D'Astous, M; Di Paolo, T; Dluzen, DE; Gajjar, TM | 1 |
Desai, RI; Katz, JL; Koffarnus, M; Kopajtic, TA; Newman, AH | 1 |
Desai, RI; French, D; Katz, JL; Kopajtic, TA; Newman, AH | 1 |
Baroni, S; Betti, L; Cassano, GB; Catena, M; Dell'Osso, B; Fabbrini, L; Giannaccini, G; Italiani, P; Lucacchini, A; Marazziti, D | 1 |
Burton, NC; Guilarte, TR; Kensler, TW | 1 |
Cadet, JL; Deng, X; Jayanthi, S; Ladenheim, B | 1 |
McIntosh, JM; O'Leary, K; Parameswaran, N; Quik, M | 1 |
Alexander, M; Burton, NC; Griswold, M; Guilarte, TR; McGlothan, JL; Pham, L; Schneider, JS; Syversen, T; Verina, T; Wong, DF; Zhou, Y | 1 |
Bordia, T; Huang, LZ; Michael McIntosh, J; Parameswaran, N; Quik, M | 1 |
Calon, F; Di Paolo, T; Grégoire, L; Hornykiewicz, O; Rajput, A; Rajput, AH; Samadi, P | 1 |
Di Paolo, T; Grégoire, L; Lévesque, D; Morissette, M; Ouattara, B; Rouillard, C; Samadi, P; Tamim, MK | 1 |
Di Paolo, T; Gilbert, F; Grégoire, L; Lévesque, D; Mahmoudi, S; Morissette, M; Ouattara, B; Rouillard, C; Samadi, P | 1 |
Bordia, T; Campos, C; McIntosh, JM; Quik, M | 1 |
He, Z; Ma, T; Park, SW; Roman, RJ; Shen, X | 1 |
Crossman, AR; Kobylecki, C; Ravenscroft, P | 1 |
Daniju, Y; Davidson, C; Dawson, P; Dutta, N; Moffatt, JD; Opacka-Juffry, J; Ramsey, J | 1 |
Bornatowicz, B; Fink, C; Hacker, M; Haeusler, D; Mitterhauser, M; Nics, L; Otter, P; Rami-Mark, C; Spreitzer, H; Ungersboeck, J; Vraka, C; Wadsak, W | 1 |
Bevan, M; Davidson, C; Meintel, M; Opacka-Juffry, J; Patel, N; Pinnell, T | 1 |
Bordia, T; Drenan, RM; McGregor, M; McIntosh, JM; Quik, M | 1 |
Al Sweidi, S; Bourque, M; Caruso, D; Di Paolo, T; Melcangi, RC; Morissette, M | 1 |
Barrese, V; Davidson, C; Dutta, N; Khelashvili, G; Opacka-Juffry, J; Sahai, MA; Weinstein, H | 1 |
Bordia, T; Perez, XA; Quik, M; Zhang, D | 1 |
Di Paolo, T; Morin, N; Morissette, M; Rouillard, C | 1 |
61 other study(ies) available for cocaine and rti 121
Article | Year |
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Dopamine transporter imaging with novel, selective cocaine analogs.
Topics: Animals; Brain; Brain Chemistry; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Nerve Tissue Proteins; Papio; Protein Binding; Tomography, Emission-Computed, Single-Photon | 1992 |
Rate of binding of various inhibitors at the dopamine transporter in vivo.
Topics: Animals; Binding, Competitive; Bupropion; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred Strains; Nerve Tissue Proteins; Time Factors | 1995 |
Characterization and localization of [125I]RTI-121 binding sites in human striatum and medial temporal lobe.
Topics: Animals; Autoradiography; Binding Sites; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Guinea Pigs; Humans; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Rats; Rats, Sprague-Dawley; Temporal Lobe | 1995 |
Characterization of the dopamine transporter in nonhuman primate brain: homogenate binding, whole body imaging, and ex vivo autoradiography using [125I] and [123I]IPCIT.
Topics: Animals; Autoradiography; Brain Chemistry; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Female; Iodine Radioisotopes; Membrane Glycoproteins; Membrane Transport Proteins; Models, Biological; Nerve Tissue Proteins; Ovariectomy; Papio; Protein Binding; Tissue Distribution; Tomography, Emission-Computed, Single-Photon; Whole-Body Counting | 1995 |
Comparison of [123I]beta-CIT and [123I]IPCIT as single-photon emission tomography radiotracers for the dopamine transporter in nonhuman primates.
Topics: Animals; Brain; Brain Chemistry; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Female; Iodine Radioisotopes; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Papio; Sensitivity and Specificity; Serotonin; Serotonin Plasma Membrane Transport Proteins; Time Factors; Tomography, Emission-Computed, Single-Photon | 1995 |
Selective labeling of the dopamine transporter by the high affinity ligand 3 beta-(4-[125I]iodophenyl)tropane-2 beta-carboxylic acid isopropyl ester.
Topics: Animals; Brain; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Kinetics; Ligands; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Piperazines; Rats; Rats, Sprague-Dawley | 1995 |
Novel radioligands for the dopamine transporter demonstrate the presence of intrastriatal nigral grafts in the MPTP-treated monkey: correlation with improved behavioral function.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Autoradiography; Brain Tissue Transplantation; Carrier Proteins; Chlorocebus aethiops; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Fetal Tissue Transplantation; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Parkinson Disease, Secondary; Radioligand Assay; Serotonin Plasma Membrane Transport Proteins; Substantia Nigra; Transplantation, Heterotopic; Transplantation, Homologous | 1994 |
Superoxide radicals mediate the biochemical effects of methylenedioxymethamphetamine (MDMA): evidence from using CuZn-superoxide dismutase transgenic mice.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Autoradiography; Cocaine; Corpus Striatum; Dopamine; Female; Humans; Male; Mice; Mice, Transgenic; N-Methyl-3,4-methylenedioxyamphetamine; Receptors, Dopamine; Superoxide Dismutase; Superoxides; Tissue Distribution | 1995 |
Synthesis and in vivo studies of a selective ligand for the dopamine transporter: 3 beta-(4-[125I]iodophenyl) tropan-2 beta-carboxylic acid isopropyl ester ([125I]RTI-121).
Topics: Amphetamine; Analysis of Variance; Animals; Brain; Carrier Proteins; Chromatography, High Pressure Liquid; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Isotope Labeling; Kinetics; Ligands; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred Strains; Molecular Structure; Nerve Tissue Proteins; Tissue Distribution | 1996 |
Evaluation of [11C]RTI-121 as a selective radioligand for PET studies of the dopamine transporter.
Topics: Animals; Biotransformation; Blood Proteins; Brain; Carbon Radioisotopes; Carrier Proteins; Cerebellum; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Radioligand Assay; Rats; Rats, Sprague-Dawley; Tissue Distribution; Tomography, Emission-Computed | 1996 |
Cocaine withdrawal reduces dopamine transporter binding in the shell of the nucleus accumbens.
Topics: Animals; Autoradiography; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Image Processing, Computer-Assisted; Male; Membrane Glycoproteins; Membrane Transport Proteins; Narcotics; Neostriatum; Nerve Tissue Proteins; Nucleus Accumbens; Olfactory Bulb; Rats; Rats, Inbred Lew; Substance Withdrawal Syndrome; Ventral Tegmental Area | 1996 |
Mapping dopamine transporters in the human brain with novel selective cocaine analog [125I]RTI-121.
Topics: Adult; Autoradiography; Binding Sites; Binding, Competitive; Brain; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Female; Humans; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Tissue Distribution | 1995 |
Highly potent cocaine analogs cause long-lasting increases in locomotor activity.
Topics: Analysis of Variance; Animals; Behavior, Animal; Binding, Competitive; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Mice; Motor Activity; Rats; Rats, Sprague-Dawley | 1996 |
Binding of the [125I]3 beta-(iodophenyl)tropan-2 beta-carboxylic acid isopropyl ester to the dopamine transporter at a physiologically relevant temperature: mutually exclusive binding and different ionic requirements for various uptake blockers and substr
Topics: Animals; Binding, Competitive; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Rats; Rats, Sprague-Dawley; Synaptosomes | 1997 |
Differential regulation of dopamine transporter after chronic self-administration of bupropion and nomifensine.
Topics: Animals; Bupropion; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Nomifensine; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Administration | 1997 |
Modeling of the interaction of Na+ and K+ with the binding of the cocaine analogue 3beta-(4-[125I]iodophenyl)tropane-2beta-carboxylic acid isopropyl ester to the dopamine transporter.
Topics: Animals; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Models, Biological; Nerve Tissue Proteins; Potassium; Rats; Rats, Sprague-Dawley; Sodium; Synaptosomes | 1997 |
p53-knockout mice are protected against the long-term effects of methamphetamine on dopaminergic terminals and cell bodies.
Topics: Animals; Autoradiography; Brain; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Heterozygote; Homozygote; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Methamphetamine; Mice; Mice, Knockout; Nerve Tissue Proteins; Nucleus Accumbens; RNA, Messenger; Tumor Suppressor Protein p53; Tyrosine 3-Monooxygenase | 1997 |
Potential misconceptions in dopamine transporter assays arising from the binding of [125I]RTI-121 to filters: effect of ions and cocaine.
Topics: Animals; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Histocytochemistry; Iodine Radioisotopes; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Protein Binding; Rats; Rats, Sprague-Dawley; Sodium; Synaptosomes; Ultrafiltration | 1997 |
In vivo saturation kinetics of two dopamine transporter probes measured using a small animal positron emission tomography scanner.
Topics: Animals; Brain; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Male; Membrane Glycoproteins; Membrane Transport Proteins; Neostriatum; Nerve Tissue Proteins; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Tomography, Emission-Computed | 1997 |
Simplified reference tissue model for PET receptor studies.
Topics: Animals; Benzazepines; Brain Mapping; Carrier Proteins; Cocaine; Computer Simulation; Dopamine Plasma Membrane Transport Proteins; Humans; Image Processing, Computer-Assisted; Membrane Glycoproteins; Membrane Transport Proteins; Models, Theoretical; Nerve Tissue Proteins; Raclopride; Rats; Receptors, Dopamine D1; Receptors, Dopamine D2; Receptors, Neurotransmitter; Reference Values; Salicylamides; Tomography, Emission-Computed | 1996 |
Distribution of dopamine transporters in basal ganglia of cerebellar ataxic mice by [125I]RTI-121 quantitative autoradiography.
Topics: Animals; Autoradiography; Basal Ganglia; Carrier Proteins; Cerebellar Ataxia; Cocaine; Dopamine Plasma Membrane Transport Proteins; Heterozygote; Homozygote; Iodine Radioisotopes; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Neurologic Mutants; Neostriatum; Nerve Tissue Proteins; Nucleus Accumbens; Olfactory Pathways; Substantia Nigra; Tegmentum Mesencephali; Thalamus; Tissue Distribution | 1998 |
Multiple binding sites for [125I]RTI-121 and other cocaine analogs in rat frontal cerebral cortex.
Topics: Animals; Binding Sites; Binding, Competitive; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Frontal Lobe; Iodine Radioisotopes; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Norepinephrine; Norepinephrine Plasma Membrane Transport Proteins; Rats; Rats, Sprague-Dawley; Regression Analysis; Serotonin; Serotonin Plasma Membrane Transport Proteins; Symporters | 1998 |
Melatonin attenuates methamphetamine-induced toxic effects on dopamine and serotonin terminals in mouse brain.
Topics: Animals; Antioxidants; Autoradiography; Brain Chemistry; Cocaine; Dopamine; Dopamine Uptake Inhibitors; Iodine Radioisotopes; Male; Melatonin; Methamphetamine; Mice; Neostriatum; Nerve Endings; Nucleus Accumbens; Serotonin | 1998 |
Selective regulation of dopamine transporter binding in the shell of the nucleus accumbens by adrenalectomy and corticosterone-replacement.
Topics: Adrenal Glands; Adrenalectomy; Animals; Autoradiography; Brain; Carrier Proteins; Cocaine; Corticosterone; Dopamine; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Nucleus Accumbens; Organ Specificity; Rats; Rats, Sprague-Dawley | 1998 |
Characterization of [125I]RTI-121 binding to dopamine transporter in vitro.
Topics: Animals; Binding Sites; Binding, Competitive; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine Uptake Inhibitors; In Vitro Techniques; Male; Pergolide; Rats; Rats, Sprague-Dawley; Synaptosomes | 1997 |
Cocaine upregulates the dopamine transporter in fetal rhesus monkey brain.
Topics: Animals; Binding Sites; Brain; Carrier Proteins; Cocaine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Embryonic and Fetal Development; Fetus; Macaca mulatta; Membrane Glycoproteins; Membrane Transport Proteins; Mesencephalon; Nerve Tissue Proteins; Neurons; RNA, Messenger; Tissue Distribution; Tyrosine 3-Monooxygenase; Up-Regulation | 1999 |
Correlates of deoxycorticosterone-induced salt appetite behavior and basal ganglia neurochemistry.
Topics: Animals; Appetite; Basal Ganglia; Carrier Proteins; Cocaine; Desoxycorticosterone; Dopamine Plasma Membrane Transport Proteins; Dynorphins; Enkephalins; Gene Expression Regulation; Male; Membrane Glycoproteins; Membrane Transport Proteins; Nerve Tissue Proteins; Nucleus Accumbens; Protein Precursors; Rats; Rats, Sprague-Dawley; RNA, Messenger; Sodium, Dietary; Transcription, Genetic; Tyrosine 3-Monooxygenase | 1999 |
[123I]IPCIT and [123I]beta-CIT as SPECT tracers for the dopamine transporter: a comparative analysis in nonhuman primates.
Topics: Animals; Brain; Carrier Proteins; Chromatography, High Pressure Liquid; Cocaine; Dopamine Plasma Membrane Transport Proteins; Female; Half-Life; Humans; Injections, Intravenous; Iodine Radioisotopes; Ligands; Membrane Glycoproteins; Membrane Transport Proteins; Metabolic Clearance Rate; Models, Biological; Nerve Tissue Proteins; Papio; Species Specificity; Time Factors; Tissue Distribution; Tomography, Emission-Computed, Single-Photon | 2000 |
Dopamine-deficient mice are hypersensitive to dopamine receptor agonists.
Topics: Animals; Autoradiography; Benzamides; Brain; Carrier Proteins; Cocaine; Corpus Striatum; Dopamine; Dopamine Agonists; Dopamine beta-Hydroxylase; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Levodopa; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Knockout; Mice, Transgenic; Motor Activity; Nerve Tissue Proteins; Pyrrolidines; Receptors, Dopamine; Tyrosine 3-Monooxygenase | 2000 |
The influence of tomograph sensitivity on kinetic parameter estimation in positron emission tomography imaging studies of the rat brain.
Topics: Animals; Brain; Carrier Proteins; Cerebellum; Cocaine; Computer Simulation; Corpus Striatum; Dopamine Antagonists; Dopamine D2 Receptor Antagonists; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Image Processing, Computer-Assisted; Ligands; Membrane Glycoproteins; Membrane Transport Proteins; Models, Neurological; Nerve Tissue Proteins; Phantoms, Imaging; Raclopride; Radioisotopes; Rats; Reproducibility of Results; Sensitivity and Specificity; Tomography, Emission-Computed | 2000 |
Effect of MPTP-induced denervation on basal ganglia GABA(B) receptors: correlation with dopamine concentrations and dopamine transporter.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Basal Ganglia; Benzoates; Cocaine; Corpus Striatum; Disease Models, Animal; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Female; Macaca fascicularis; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; Nerve Tissue Proteins; Organophosphorus Compounds; Parkinsonian Disorders; Protein Subunits; Radioligand Assay; Receptors, GABA-B; RNA, Messenger; Substantia Nigra; Subthalamic Nucleus | 2001 |
Glial cell line-derived neurotrophic factor (GDNF) gene delivery protects dopaminergic terminals from degeneration.
Topics: Aging; Animals; Autoradiography; Carrier Proteins; Cocaine; Corpus Striatum; Disease Models, Animal; Dopamine; Dopamine Plasma Membrane Transport Proteins; Genetic Therapy; Genetic Vectors; Glial Cell Line-Derived Neurotrophic Factor; Male; Membrane Glycoproteins; Membrane Transport Proteins; Microinjections; Motor Activity; Nerve Growth Factors; Nerve Tissue Proteins; Neurons; Neurotransmitter Agents; Oxidopamine; Parkinson Disease, Secondary; Presynaptic Terminals; Rats; Rats, Inbred F344; RNA, Messenger; Substantia Nigra; Tyrosine 3-Monooxygenase | 2001 |
Vulnerability of 125I-alpha-conotoxin MII binding sites to nigrostriatal damage in monkey.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Autoradiography; Binding Sites; Binding, Competitive; Bridged Bicyclo Compounds, Heterocyclic; Carrier Proteins; Cocaine; Conotoxins; Corpus Striatum; Disease Models, Animal; Dopamine; Dopamine Plasma Membrane Transport Proteins; Female; Habenula; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mesencephalon; Nerve Tissue Proteins; Neural Pathways; Neurons; Parkinson Disease, Secondary; Putamen; Pyridines; Receptors, Nicotinic; Saimiri; Substantia Nigra | 2001 |
Effects of kappa-opioid receptor agonists on long-term cocaine use and dopamine neurotransmission.
Topics: Analgesics; Animals; Autoradiography; Benzazepines; Benzeneacetamides; Benzomorphans; Binding, Competitive; Brain; Carrier Proteins; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Motor Activity; Nerve Tissue Proteins; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Opioid, kappa; Sulpiride; Synaptic Transmission; Time Factors; Tyrosine 3-Monooxygenase | 2001 |
Ontogeny of neurokinin-1 receptor mediation of methamphetamine neurotoxicity in the striatum of the mouse brain.
Topics: Animals; Autoradiography; Binding Sites; Caudate Nucleus; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Iodine Radioisotopes; Kinetics; Male; Membrane Glycoproteins; Membrane Transport Proteins; Methamphetamine; Mice; Mice, Inbred ICR; Nerve Tissue Proteins; Putamen; Receptors, Neurokinin-1; Substance P | 2002 |
Lack of effect of testosterone and dihydrotestosterone compared to 17beta-oestradiol in 1-methyl-4-phenyl-1,2,3,6, tetrahydropyridine-mice.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Autoradiography; Cocaine; Dihydrotestosterone; Dopamine; Dopamine Plasma Membrane Transport Proteins; Estradiol; Gonadal Steroid Hormones; Homovanillic Acid; In Situ Hybridization; Iodine Radioisotopes; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Mice, Inbred C57BL; MPTP Poisoning; Nerve Tissue Proteins; Neuropeptides; RNA, Messenger; Testosterone; Tetrabenazine; Tritium; Vesicular Biogenic Amine Transport Proteins; Vesicular Monoamine Transport Proteins | 2002 |
Declines in different beta2* nicotinic receptor populations in monkey striatum after nigrostriatal damage.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Autoradiography; Azetidines; Brain Chemistry; Caudate Nucleus; Cocaine; Conotoxins; Neostriatum; Parkinson Disease, Secondary; Putamen; Radioligand Assay; Receptors, Nicotinic; Saimiri; Substantia Nigra | 2002 |
Human immunodeficiency virus-1 Tat protein and methamphetamine interact synergistically to impair striatal dopaminergic function.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antioxidants; Binding, Competitive; Body Temperature; Cell Death; Cocaine; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Drug Synergism; Gene Products, tat; HIV-1; Homovanillic Acid; Humans; Hydroxyindoleacetic Acid; Intracellular Membranes; Male; Membrane Glycoproteins; Membrane Potentials; Membrane Transport Proteins; Methamphetamine; Mitochondria; Nerve Tissue Proteins; Neurons; Rats; Rats, Sprague-Dawley; Serotonin; tat Gene Products, Human Immunodeficiency Virus | 2002 |
Dopamine transporter as a marker of neuroprotection in methamphetamine-lesioned mice treated acutely with estradiol.
Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Autoradiography; Chromatography, High Pressure Liquid; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Drug Interactions; Estradiol; Female; In Situ Hybridization; Iodine Isotopes; Membrane Glycoproteins; Membrane Transport Proteins; Methamphetamine; Mice; Neostriatum; Nerve Tissue Proteins; Nervous System Diseases; Neuroprotective Agents; Ovariectomy; Protein Binding; RNA, Messenger; Substantia Nigra; Time Factors | 2004 |
Identification of a dopamine transporter ligand that blocks the stimulant effects of cocaine.
Topics: Animals; Benztropine; Central Nervous System Stimulants; Cerebellum; Cocaine; Corpus Striatum; Dopamine Antagonists; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Inhibitory Concentration 50; Ligands; Male; Membrane Glycoproteins; Membrane Transport Proteins; Mice; Motor Activity; Nerve Tissue Proteins; Rats | 2005 |
Relationship between in vivo occupancy at the dopamine transporter and behavioral effects of cocaine, GBR 12909 [1-{2-[bis-(4-fluorophenyl)methoxy]ethyl}-4-(3-phenylpropyl)piperazine], and benztropine analogs.
Topics: Animals; Benztropine; Cocaine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Male; Mice; Motor Activity; Piperazines | 2005 |
Binding of 3H-WIN-35,428 and 125I-RTI-121 to human platelet membranes.
Topics: Adult; Blood Platelets; Cell Membrane; Cocaine; Dopamine Plasma Membrane Transport Proteins; Female; Humans; In Vitro Techniques; Iodine Radioisotopes; Ligands; Male; Protein Binding | 2006 |
In vivo modulation of the Parkinsonian phenotype by Nrf2.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Antineoplastic Agents; Autoradiography; Cocaine; Disease Models, Animal; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Drug Interactions; Iodine Isotopes; Male; Mice; Mice, Inbred ICR; Mice, Knockout; NF-E2-Related Factor 2; Parkinsonian Disorders; Phenotype; Thiones; Thiophenes | 2006 |
Methamphetamine administration causes death of dopaminergic neurons in the mouse olfactory bulb.
Topics: Animals; Apoptosis; Autoradiography; Blotting, Western; Cell Death; Central Nervous System Stimulants; Cerebral Cortex; Chromatography, High Pressure Liquid; Cocaine; Dopamine; Immunohistochemistry; In Situ Nick-End Labeling; Male; Methamphetamine; Mice; Mice, Inbred ICR; Neostriatum; Neurons; Olfactory Bulb; Presynaptic Terminals; Tyrosine 3-Monooxygenase | 2007 |
Cotinine selectively activates a subpopulation of alpha3/alpha6beta2 nicotinic receptors in monkey striatum.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Animals; Azetidines; Brain; Cocaine; Conotoxins; Cotinine; Dopamine; Dopamine Agents; Female; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Receptors, Nicotinic; Saimiri | 2008 |
Impairment of nigrostriatal dopamine neurotransmission by manganese is mediated by pre-synaptic mechanism(s): implications to manganese-induced parkinsonism.
Topics: Amphetamine; Animals; Cocaine; Corpus Striatum; Cyclohexanols; Disease Models, Animal; Dopamine; Dopamine Agents; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Image Processing, Computer-Assisted; Macaca fascicularis; Male; Manganese; Parkinsonian Disorders; Positron-Emission Tomography; Substantia Nigra; Synaptic Transmission; Tetrabenazine; Tyrosine 3-Monooxygenase | 2008 |
Nicotine is neuroprotective when administered before but not after nigrostriatal damage in rats and monkeys.
Topics: 1-Methyl-4-phenyl-1,2,3,6-tetrahydropyridine; Amphetamine; Analysis of Variance; Animals; Autoradiography; Cocaine; Conotoxins; Corpus Striatum; Cotinine; Disease Models, Animal; Dopamine; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Iodine Isotopes; Male; Motor Activity; Neuroprotective Agents; Neurotoxicity Syndromes; Nicotine; Oxidopamine; Protein Binding; Rats; Rats, Sprague-Dawley; Saimiri; Substantia Nigra; Time Factors | 2009 |
Metabotropic glutamate receptor II in the brains of Parkinsonian patients.
Topics: Aged; Aged, 80 and over; Amino Acids; Antiparkinson Agents; Brain; Cocaine; Dyskinesia, Drug-Induced; Excitatory Amino Acid Antagonists; Female; Humans; Iodine Radioisotopes; Levodopa; Male; Parkinsonian Disorders; Postmortem Changes; Radioligand Assay; Receptors, Metabotropic Glutamate; Tritium; Xanthenes | 2009 |
Effect of non-dopaminergic drug treatment on Levodopa induced dyskinesias in MPTP monkeys: common implication of striatal neuropeptides.
Topics: Animals; Antiparkinson Agents; Benzoxazoles; Cocaine; Corpus Striatum; Disease Models, Animal; Docosahexaenoic Acids; Dopamine; Dopamine Uptake Inhibitors; Dynorphins; Dyskinesia, Drug-Induced; Enkephalins; Female; Iodine Isotopes; Levodopa; Macaca fascicularis; Naltrexone; Neuropeptides; Ovariectomy; Parkinsonian Disorders; Piperidines; Protein Precursors; RNA, Messenger; Sulfonamides; Tachykinins; Thiazoles; Time Factors | 2010 |
Nur77 mRNA levels and L-Dopa-induced dyskinesias in MPTP monkeys treated with docosahexaenoic acid.
Topics: Acetylcholinesterase; Analysis of Variance; Animals; Antiparkinson Agents; Autoradiography; Brain; Cocaine; Disease Models, Animal; Docosahexaenoic Acids; Drug Interactions; Dyskinesia, Drug-Induced; Female; Iodine Isotopes; Levodopa; Macaca fascicularis; MPTP Poisoning; Nuclear Receptor Subfamily 4, Group A, Member 1; Protein Binding; RNA, Messenger; Statistics as Topic | 2009 |
Nicotinic receptor-mediated reduction in L-DOPA-induced dyskinesias may occur via desensitization.
Topics: Amphetamine; Animals; Antiparkinson Agents; Autoradiography; Behavior, Animal; Bridged Bicyclo Compounds, Heterocyclic; Calcium Channel Blockers; Central Nervous System Stimulants; Cocaine; Conotoxins; Dopamine Plasma Membrane Transport Proteins; Dyskinesia, Drug-Induced; Functional Laterality; Levodopa; Male; Mecamylamine; Neostriatum; Nicotine; Nicotinic Agonists; Nicotinic Antagonists; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Stereotyped Behavior | 2010 |
Differential action of methamphetamine on tyrosine hydroxylase and dopamine transport in the nigrostriatal pathway of μ-opioid receptor knockout mice.
Topics: Animals; Cocaine; Corpus Striatum; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Gene Expression; Iodine Radioisotopes; Male; Methamphetamine; Mice; Mice, Inbred C57BL; Mice, Knockout; Neural Pathways; Neurons; Radionuclide Imaging; Radiopharmaceuticals; Receptors, Opioid, mu; Substantia Nigra; Tyrosine 3-Monooxygenase | 2012 |
Alternative splicing of AMPA receptor subunits in the 6-OHDA-lesioned rat model of Parkinson's disease and L-DOPA-induced dyskinesia.
Topics: Adamantane; Alternative Splicing; Animals; Antiparkinson Agents; Cocaine; Corpus Striatum; Disease Models, Animal; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Excitatory Amino Acid Antagonists; Gene Expression Regulation; Iodine Isotopes; Levodopa; Male; Motor Activity; Oxidopamine; Parkinson Disease; Rats; Rats, Sprague-Dawley; Receptors, AMPA; RNA, Messenger; Sympatholytics | 2013 |
The effects of benzofury (5-APB) on the dopamine transporter and 5-HT2-dependent vasoconstriction in the rat.
Topics: Animals; Aorta; Benzofurans; Brain; Cocaine; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; In Vitro Techniques; Iodine Isotopes; Ketanserin; Male; Muscle Contraction; N-Methyl-3,4-methylenedioxyamphetamine; Propylamines; Protein Binding; Rats; Rats, Wistar; Receptors, Serotonin, 5-HT2; Serotonin Agents; Tritium; Vasoconstriction | 2014 |
Synthesis, radiosynthesis and first in vitro evaluation of novel PET-tracers for the dopamine transporter: [(11)C]IPCIT and [(18)F]FE@IPCIT.
Topics: Carbon Isotopes; Cocaine; Dopamine Plasma Membrane Transport Proteins; Fluorine Radioisotopes; Humans; Molecular Conformation; Positron-Emission Tomography; Radioactive Tracers | 2013 |
Stimulant mechanisms of cathinones - effects of mephedrone and other cathinones on basal and electrically evoked dopamine efflux in rat accumbens brain slices.
Topics: Amphetamine; Amphetamines; Animals; Bupropion; Central Nervous System Stimulants; Cocaine; Diethylpropion; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Electric Stimulation; Iodine Radioisotopes; Male; Methamphetamine; Microelectrodes; Nucleus Accumbens; Propiophenones; Radioligand Assay; Rats, Wistar; Tissue Culture Techniques | 2014 |
Evidence for a role for α6(∗) nAChRs in l-dopa-induced dyskinesias using Parkinsonian α6(∗) nAChR gain-of-function mice.
Topics: Adrenergic Agents; Analysis of Variance; Animals; Antiparkinson Agents; Benserazide; Cocaine; Disease Models, Animal; Dose-Response Relationship, Drug; Dyskinesia, Drug-Induced; Levodopa; Male; Mice; Mice, Transgenic; Nicotine; Nicotinic Agonists; Oxidopamine; Parkinsonian Disorders; Protein Binding; Receptors, Nicotinic | 2015 |
Neuroprotective Effect of Progesterone in MPTP-Treated Male Mice.
Topics: Androstane-3,17-diol; Animals; Autoradiography; Brain; Carbon Radioisotopes; Cocaine; Dihydrotestosterone; Disease Models, Animal; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dose-Response Relationship, Drug; Drug Administration Schedule; Male; Mice; Mice, Inbred C57BL; MPTP Poisoning; Neuroprotective Agents; Progesterone; Testosterone; Vesicular Monoamine Transport Proteins | 2016 |
Combined in vitro and in silico approaches to the assessment of stimulant properties of novel psychoactive substances - The case of the benzofuran 5-MAPB.
Topics: Animals; Benzofurans; Central Nervous System Stimulants; Cocaine; Computer Simulation; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Electrochemical Techniques; In Vitro Techniques; Iodine Isotopes; Male; Methamphetamine; Models, Molecular; Protein Binding; Psychotropic Drugs; Rats; Rats, Wistar | 2017 |
Striatal D1 medium spiny neuron activation induces dyskinesias in parkinsonian mice.
Topics: Animals; Antiparkinson Agents; Channelrhodopsins; Cocaine; Corpus Striatum; Disease Models, Animal; Dopamine Plasma Membrane Transport Proteins; Dyskinesias; Female; Gene Expression Regulation; Levodopa; Male; Mice; Mice, Inbred C57BL; Mice, Transgenic; Neurons; Oxidopamine; Parkinsonian Disorders; Receptors, Dopamine D1; Sympatholytics | 2017 |
Membrane cholesterol removal and replenishment affect rat and monkey brain monoamine transporters.
Topics: Animals; Brain; Cell Membrane; Cholesterol; Cocaine; Cyclodextrins; Dopamine; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Iodine Radioisotopes; Macaca fascicularis; Male; Membrane Transport Proteins; Protein Binding; Rats; Rats, Sprague-Dawley | 2018 |