Page last updated: 2024-09-05

clorazepate dipotassium and gamma-aminobutyric acid

clorazepate dipotassium has been researched along with gamma-aminobutyric acid in 5 studies

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

*gamma-Aminobutyric Acid: The most common inhibitory neurotransmitter in the central nervous system. [MeSH]

Compound Research Comparison

Studies
(clorazepate dipotassium)
Trials
(clorazepate dipotassium)
Recent Studies (post-2010)
(clorazepate dipotassium)
Studies
(gamma-aminobutyric acid)
Trials
(gamma-aminobutyric acid)
Recent Studies (post-2010) (gamma-aminobutyric acid)
325901140,2151,4239,631

Protein Interaction Comparison

ProteinTaxonomyclorazepate dipotassium (IC50)gamma-aminobutyric acid (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid type B receptor subunit 2Rattus norvegicus (Norway rat)0.0292
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0332
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0323
Sodium- and chloride-dependent GABA transporter 1Rattus norvegicus (Norway rat)2.152
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0333
Sodium- and chloride-dependent GABA transporter 1Homo sapiens (human)5.2623
Sodium- and chloride-dependent taurine transporterHomo sapiens (human)354
Sodium- and chloride-dependent GABA transporter 2Rattus norvegicus (Norway rat)2.51
Sodium- and chloride-dependent GABA transporter 3Rattus norvegicus (Norway rat)0.02
Sodium- and chloride-dependent GABA transporter 1Mus musculus (house mouse)6.349
Sodium- and chloride-dependent GABA transporter 2Mus musculus (house mouse)7.0795
Sodium- and chloride-dependent GABA transporter 3Mus musculus (house mouse)8.1283
Sodium- and chloride-dependent betaine transporterRattus norvegicus (Norway rat)0.02
Sodium- and chloride-dependent betaine transporterHomo sapiens (human)6.4082
Sodium- and chloride-dependent GABA transporter 3Homo sapiens (human)3.9953
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0333
GABA theta subunitRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0333
Gamma-aminobutyric acid type B receptor subunit 1Rattus norvegicus (Norway rat)0.0292

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19903 (60.00)18.7374
1990's2 (40.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Baur, R; Sigel, E1
Corradetti, R; Moroni, F; Pepeu, G1
Barnard, EA; Mamalaki, C; Sigel, E1
Gitter, AH; Möhler, H; Plinkert, PK; Zenner, HP1
Boothe, DM1

Reviews

1 review(s) available for clorazepate dipotassium and gamma-aminobutyric acid

ArticleYear
Anticonvulsant therapy in small animals.
    The Veterinary clinics of North America. Small animal practice, 1998, Volume: 28, Issue:2

    Topics: Acetates; Amines; Animals; Anticonvulsants; Bromides; Clonazepam; Clorazepate Dipotassium; Cyclohexanecarboxylic Acids; Diazepam; Felbamate; Gabapentin; gamma-Aminobutyric Acid; Mephenytoin; Pentobarbital; Phenobarbital; Phenylcarbamates; Phenytoin; Primidone; Propylene Glycols; Seizures; Valproic Acid

1998

Other Studies

4 other study(ies) available for clorazepate dipotassium and gamma-aminobutyric acid

ArticleYear
Allosteric modulation by benzodiazepine receptor ligands of the GABAA receptor channel expressed in Xenopus oocytes.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1988, Volume: 8, Issue:1

    Topics: Animals; Benzodiazepines; Clorazepate Dipotassium; Electrophysiology; Flumazenil; gamma-Aminobutyric Acid; Ion Channels; Ligands; Oocytes; Osmolar Concentration; Receptors, GABA-A; Xenopus

1988
Pharmacological effects of benzodiazepines in the leech; benzodiazepine and GABA receptors and GABA level.
    Pharmacological research communications, 1980, Volume: 12, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Clorazepate Dipotassium; Flurazepam; gamma-Aminobutyric Acid; Glutamates; Glutamine; Leeches; Lidocaine; Proteins; Receptors, Drug

1980
Isolation of a GABA receptor from bovine brain using a benzodiazepine affinity column.
    FEBS letters, 1982, Oct-04, Volume: 147, Issue:1

    Topics: Animals; Cattle; Cell Membrane; Cerebral Cortex; Chromatography, Affinity; Clorazepate Dipotassium; Flunitrazepam; gamma-Aminobutyric Acid; Muscimol; Receptors, Cell Surface; Receptors, GABA-A

1982
Structure, pharmacology and function of GABA-A receptors in cochlear outer hair cells.
    European archives of oto-rhino-laryngology : official journal of the European Federation of Oto-Rhino-Laryngological Societies (EUFOS) : affiliated with the German Society for Oto-Rhino-Laryngology - Head and Neck Surgery, 1993, Volume: 250, Issue:6

    Topics: Animals; Clorazepate Dipotassium; Dose-Response Relationship, Drug; Electrophysiology; gamma-Aminobutyric Acid; Guinea Pigs; Hair Cells, Auditory, Outer; In Vitro Techniques; Membrane Potentials; Pentobarbital; Picrotoxin; Receptors, GABA-A

1993