Page last updated: 2024-09-05

clorazepate dipotassium and flumazenil

clorazepate dipotassium has been researched along with flumazenil in 8 studies

Compound Research Comparison

Studies
(clorazepate dipotassium)
Trials
(clorazepate dipotassium)
Recent Studies (post-2010)
(clorazepate dipotassium)
Studies
(flumazenil)
Trials
(flumazenil)
Recent Studies (post-2010) (flumazenil)
32590114,673426981

Protein Interaction Comparison

ProteinTaxonomyclorazepate dipotassium (IC50)flumazenil (IC50)
Gamma-aminobutyric acid receptor subunit piRattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-1Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit beta-1Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit alpha-2Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit alpha-3Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit beta-1Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit deltaRattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit gamma-2Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-5Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-3Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-4Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit gamma-2Bos taurus (cattle)0.0005
Gamma-aminobutyric acid receptor subunit gamma-1Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-2Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-4Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit gamma-3Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-6Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit alpha-1Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit beta-3Rattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit beta-2Rattus norvegicus (Norway rat)0.0038
GABA theta subunitRattus norvegicus (Norway rat)0.0038
Gamma-aminobutyric acid receptor subunit epsilonRattus norvegicus (Norway rat)0.0038

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19905 (62.50)18.7374
1990's2 (25.00)18.2507
2000's1 (12.50)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beauvoir, C; Biboulet, P; Passeron, D1
Baur, R; Sigel, E1
Belzung, C; Chapouthier, G; Dodd, RH; Misslin, R; Vogel, E1
Mormède, P1
Dantzer, R; Mormede, P; Perio, A1
Dantzer, R; Pério, A1
Alzieu, M; Becquemont, L; Delhotal Landes, B; Guglielminotti, J; Guidet, B; Maury, E; Offenstadt, G1
Capasso, A; Cavallo, F; Raffa, RB1

Reviews

1 review(s) available for clorazepate dipotassium and flumazenil

ArticleYear
[Neuroendocrine effects of benzodiazepines].
    L'Encephale, 1983, Volume: 9, Issue:4 Suppl 2

    Topics: Adrenal Cortex Hormones; Anti-Anxiety Agents; Benzodiazepinones; Chlordiazepoxide; Clorazepate Dipotassium; Flumazenil; Growth Hormone; Humans; Hypothalamo-Hypophyseal System; Male; Pituitary-Adrenal System; Prolactin; Stress, Psychological; Sympathetic Nervous System

1983

Other Studies

7 other study(ies) available for clorazepate dipotassium and flumazenil

ArticleYear
[Difficulties in antagonizing dipotassium chlorazepate using flumazenil in cases of acute poisoning].
    Cahiers d'anesthesiologie, 1991, Volume: 39, Issue:1

    Topics: Adult; Clorazepate Dipotassium; Drug Overdose; Female; Flumazenil; Humans; Male; Middle Aged

1991
Allosteric modulation by benzodiazepine receptor ligands of the GABAA receptor channel expressed in Xenopus oocytes.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 1988, Volume: 8, Issue:1

    Topics: Animals; Benzodiazepines; Clorazepate Dipotassium; Electrophysiology; Flumazenil; gamma-Aminobutyric Acid; Ion Channels; Ligands; Oocytes; Osmolar Concentration; Receptors, GABA-A; Xenopus

1988
Anxiogenic effects of methyl-beta-carboline-3-carboxylate in a light/dark choice situation.
    Pharmacology, biochemistry, and behavior, 1987, Volume: 28, Issue:1

    Topics: Animals; Anxiety; Benzodiazepines; Carbolines; Choice Behavior; Clorazepate Dipotassium; Darkness; Dose-Response Relationship, Drug; Flumazenil; Light; Male; Mice

1987
Relationship of the effects of the benzodiazepine derivative clorazepate on corticosterone secretion with its behavioural actions. Antagonism by Ro 15-1788.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 21, Issue:6

    Topics: Adrenal Cortex; Animals; Anti-Anxiety Agents; Benzodiazepinones; Brain; Clorazepate Dipotassium; Corticosterone; Flumazenil; Humans; Male; Pituitary-Adrenal System; Rats; Rats, Inbred Strains; Receptors, GABA-A; Stress, Psychological

1984
Behavioural evidence for partial agonist properties of RO 15-1788, a benzodiazepine receptor antagonist.
    European journal of pharmacology, 1982, Jul-30, Volume: 81, Issue:4

    Topics: Animals; Behavior, Animal; Benzodiazepinones; Clorazepate Dipotassium; Conflict, Psychological; Cues; Discrimination, Psychological; Flumazenil; Male; Pentylenetetrazole; Rats

1982
Prolonged sedation requiring mechanical ventilation and continuous flumazenil infusion after routine doses of clorazepam for alcohol withdrawal syndrome.
    Intensive care medicine, 1999, Volume: 25, Issue:12

    Topics: Aged; Alcohol Withdrawal Seizures; Anticonvulsants; Antidotes; Bronchitis; Clorazepate Dipotassium; Coma; Fatal Outcome; Flumazenil; Humans; Infusions, Intravenous; Liver Diseases; Male; Middle Aged; Nordazepam; Pneumonia; Respiration, Artificial

1999
Flumazenil-sensitive dose-related physical dependence in planarians produced by two benzodiazepine and one non-benzodiazepine benzodiazepine-receptor agonists.
    European journal of pharmacology, 2007, Jun-14, Volume: 564, Issue:1-3

    Topics: Analysis of Variance; Animals; Benzodiazepines; Clorazepate Dipotassium; Dose-Response Relationship, Drug; Flumazenil; GABA Agonists; GABA Modulators; Locomotion; Midazolam; Planarians; Pyridines; Receptors, GABA-A; Reproducibility of Results; Substance Withdrawal Syndrome; Substance-Related Disorders; Zolpidem

2007