clonidine and thiazoles

clonidine has been researched along with thiazoles in 18 studies

Research

Studies (18)

TimeframeStudies, this research(%)All Research%
pre-19905 (27.78)18.7374
1990's6 (33.33)18.2507
2000's4 (22.22)29.6817
2010's3 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Timmermans, PB; Van Zwieten, PA1
Matera, M; Mazzone, G; Mazzone, P; Mazzone, S; Panico, A; Pennisi, G; Pignatello, R; Puglisi, G; Raciti, G1
Hjorth, S; Tao, R1
Bonanno, G; Maura, G; Raiteri, M1
Kobinger, W; Pichler, L2
Hammer, R; Kobinger, W; Pichler, L1
Kobinger, W; Lillie, C; Pichler, L1
Boronat, MA; García-Sevilla, JA; Lizcano, JM; Olmos, G; Ozaita, A; Unzeta, M1
Li, G; Metz, SA; Segu, VB1
Gundlach, AL; King, PR; Louis, WJ1
Chevallet, P; Erol, K; Kiliç, FS; Turan-Zitouni, G1
Jain, NK; Kulkarni, SK; Singh, A1
Bagheri, M; Ghahremani, MH; Jorjani, M; Shafiee, A; Shekarchi, M; Vosooghi, M1
Anderson, NJ; Hudson, AL; Lupo, PA; Nutt, DJ; Robinson, ES1
Hirayama, M; Hori, Y; Inoue, N; Ito, K; Kawabata, Y; Kawachi, M; Matsunaga, Y; Nagahama, K; Ozaki, T; Takei, M; Tanaka, T; Toda, R; Yoshii, K1
Hori, Y; Ito, K; Kawachi, M; Matsunaga, Y; Nagahama, K; Oka, H; Takei, M; Tanaka, T1
Hanif, M; Shaheryar, ZA; Zaman, M1

Other Studies

18 other study(ies) available for clonidine and thiazoles

ArticleYear
Influence of structural changes in the imidazolidine ring of clonidine on hypotensive activity.
    Pharmacology, 1978, Volume: 16, Issue:2

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Drug Evaluation, Preclinical; Heart Rate; Hypotension; Imidazoles; Male; Quinazolines; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Thiazoles

1978
MAOI activity of some novel series of substituted thiazol-2-yl-hydrazines.
    Die Pharmazie, 1992, Volume: 47, Issue:12

    Topics: Amphetamine; Animals; Blood Pressure; Brain; Clonidine; Female; Hydrazines; Hydrolysis; In Vitro Techniques; Kynuramine; Lethal Dose 50; Male; Mice; Mitochondria; Monoamine Oxidase Inhibitors; Motor Activity; Rats; Rats, Sprague-Dawley; Spectrometry, Fluorescence; Thiazoles; Tyramine

1992
Alpha 2-adrenoceptor modulation of rat ventral hippocampal 5-hydroxytryptamine release in vivo.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Dioxanes; Hippocampus; Idazoxan; Male; Pindolol; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin; Thiazoles; Tyrosine 3-Monooxygenase

1992
Presynaptic alpha 2-adrenoceptors mediating inhibition of noradrenaline and 5-hydroxytryptamine release in rat cerebral cortex: further characterization as different alpha 2-adrenoceptor subtypes.
    Naunyn-Schmiedeberg's archives of pharmacology, 1992, Volume: 345, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Cerebral Cortex; Clonidine; Dioxanes; Ethylmaleimide; GTP-Binding Proteins; Idazoxan; In Vitro Techniques; Male; Mianserin; Nerve Endings; Norepinephrine; Pyridines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin; Signal Transduction; Synaptosomes; Thiazoles

1992
alpha 1-adrenoceptor blockade by alpha 2-adrenoceptor agonists in the isolated perfused hindquarter of rats.
    European journal of pharmacology, 1981, Jun-10, Volume: 72, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Clonidine; In Vitro Techniques; Male; Methoxamine; Oxazoles; Perfusion; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thiazoles; Vasoconstriction

1981
Modulation of motor activity by alpha 1- and alpha 2-adrenoceptor stimulation in mice.
    Naunyn-Schmiedeberg's archives of pharmacology, 1981, Volume: 317, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Apomorphine; Azepines; Clonidine; Exploratory Behavior; Male; Mice; Motor Activity; Thiazoles

1981
Binding of an imidazolidine (clonidine), an oxazoloazepin (B-HT 933) and a thiazoloazepin (B-HT 920) to rat brain alpha-adrenoceptors and relation to cardiovascular effects.
    European journal of pharmacology, 1980, Apr-04, Volume: 62, Issue:4

    Topics: Animals; Azepines; Binding Sites; Binding, Competitive; Blood Pressure; Brain; Clonidine; Heart Rate; Kinetics; Male; Oxazoles; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thiazoles

1980
Central cardiovascular alpha-adrenoceptors. Relation to peripheral receptors.
    Circulation research, 1980, Volume: 46, Issue:6 Pt 2

    Topics: Animals; Azepines; Blood Pressure; Cardiovascular System; Clonidine; Dose-Response Relationship, Drug; Heart Rate; Male; Methoxamine; Norepinephrine; Oxazoles; Perfusion; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thiazoles; Vagotomy

1980
Inhibition of monoamine oxidase A and B activities by imidazol(ine)/guanidine drugs, nature of the interaction and distinction from I2-imidazoline receptors in rat liver.
    British journal of pharmacology, 1997, Volume: 121, Issue:5

    Topics: Animals; Clonidine; Guanidines; Imidazoles; Imidazoline Receptors; Isoenzymes; Kinetics; Liver; Male; Mitochondria, Liver; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Picolinic Acids; Rats; Rats, Sprague-Dawley; Receptors, Drug; Thiazoles

1997
Use of a soluble tetrazolium compound to assay metabolic activation of intact beta cells.
    Metabolism: clinical and experimental, 1998, Volume: 47, Issue:7

    Topics: Animals; Calcium; Clonidine; Cricetinae; Cytoplasmic Granules; Glucose; Insulin; Insulin Secretion; Islets of Langerhans; Methylphenazonium Methosulfate; Mitochondria; Somatostatin; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1998
Identification of imidazoline-receptor binding sites in cortex and medulla of the bovine adrenal gland. Colocalization with MAO-A and MAO-B.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Adrenal Cortex; Adrenal Medulla; Adrenergic beta-Agonists; Animals; Autoradiography; Benzofurans; Binding Sites; Cattle; Clonidine; Imidazoles; Imidazoline Receptors; Isoenzymes; Monoamine Oxidase; Monoamine Oxidase Inhibitors; Oxazoles; Picolinic Acids; Rats; Receptors, Drug; Rilmenidine; Thiazoles; Tritium

1999
Synthesis of some thiazolyl-pyrazoline derivatives and preliminary investigation of their hypotensive activity.
    European journal of medicinal chemistry, 2000, Volume: 35, Issue:6

    Topics: Animals; Antihypertensive Agents; Clonidine; Drug Evaluation, Preclinical; Female; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Molecular Structure; Pyrazoles; Rats; Structure-Activity Relationship; Thiazoles

2000
Modulation of NSAID-induced antinociceptive and anti-inflammatory effects by alpha2-adrenoceptor agonists with gastroprotective effects.
    Life sciences, 2002, May-03, Volume: 70, Issue:24

    Topics: Adrenergic alpha-Agonists; Animals; Anti-Inflammatory Agents, Non-Steroidal; Clonidine; Drug Synergism; Drug Therapy, Combination; Meloxicam; Mice; Naproxen; Pain; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Stomach Ulcer; Sulfonamides; Thiazines; Thiazoles; Yohimbine

2002
Synthesis and antihypertensive activity of 1-(2-thiazolyl)-3, 5-disubstituted -2-pyrazolines.
    Archiv der Pharmazie, 2004, Volume: 337, Issue:1

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Clonidine; Hypotension; Injections, Intraperitoneal; Male; Molecular Structure; Pyrazoles; Quantitative Structure-Activity Relationship; Rats; Rats, Sprague-Dawley; Thiazoles

2004
Characterisation of imidazoline I2 binding sites in pig brain.
    European journal of pharmacology, 2005, Sep-05, Volume: 519, Issue:1-2

    Topics: Animals; Benzofurans; Binding Sites; Binding, Competitive; Brain; Carbolines; Clonidine; Dose-Response Relationship, Drug; Female; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Male; Monoamine Oxidase Inhibitors; Picolinic Acids; Radioligand Assay; Receptors, Drug; Swine; Thiazoles; Tritium

2005
Acotiamide hydrochloride (Z-338) enhances gastric motility and emptying by inhibiting acetylcholinesterase activity in rats.
    European journal of pharmacology, 2011, Volume: 666, Issue:1-3

    Topics: Acetylcholinesterase; Animals; Benzamides; Cholinesterase Inhibitors; Clonidine; Electric Stimulation; Gastric Emptying; Male; Muscle Contraction; Rats; Rats, Sprague-Dawley; Stomach; Thiazoles

2011
Acotiamide, a new orally active acetylcholinesterase inhibitor, stimulates gastrointestinal motor activity in conscious dogs.
    Neurogastroenterology and motility, 2012, Volume: 24, Issue:6

    Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Benzamides; Cholinesterase Inhibitors; Clonidine; Dogs; Gastric Emptying; Gastrointestinal Motility; Gastrointestinal Tract; Male; Thiazoles

2012
Development of Tizanidine HCl-Meloxicam loaded mucoadhesive buccal films: In-vitro and in-vivo evaluation.
    PloS one, 2018, Volume: 13, Issue:3

    Topics: Adhesiveness; Administration, Buccal; Animals; Biological Availability; Chemistry, Pharmaceutical; Clonidine; Cross-Over Studies; Delayed-Action Preparations; Drug Compounding; Drug Delivery Systems; Drug Evaluation, Preclinical; Drug Liberation; Half-Life; Hypromellose Derivatives; Male; Meloxicam; Mouth Mucosa; Rabbits; Solubility; Thiazines; Thiazoles; Xylans

2018