clonidine has been researched along with talipexole in 82 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 63 (76.83) | 18.7374 |
1990's | 17 (20.73) | 18.2507 |
2000's | 2 (2.44) | 29.6817 |
2010's | 0 (0.00) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
---|---|
Batink, H; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B | 1 |
de Jonge, A; Lam, E; Slothorst-Grisdijk, FP; Timmermans, PB; van Meel, JC; van Zwieten, PA | 1 |
Amerini, S; Ledda, F; Mantelli, L; Rubino, A | 1 |
Piascik, MT; Pruitt, TA; Sparks, MS | 1 |
Tabrizchi, R; Triggle, CR | 2 |
Ball, SG; Ong, ML; Vaughan, PF | 1 |
Breschi, MC; Ciucci, MA; Martinotti, E; Nieri, P; Omini, C; Pani, M | 1 |
Breschi, MC; Martinotti, E; Nieri, P; Omini, C | 1 |
Cassinadri, M; Ferrari, F; Tampieri, A; Tartoni, PL | 1 |
Schott, C; Stoclet, JC; Topouzis, S | 1 |
Göthert, M; Molderings, GJ | 1 |
Arranz, A; Arribas, S; Balfagón, G; Marín, J; Sanchez-Merino, JA | 1 |
Dresse, A; Giesbers, I; Massotte, L; Scuvée-Moreau, J; Seutin, V | 1 |
de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B | 1 |
Eskinder, H; Gross, GJ | 1 |
Balfagón, G; Marín, J | 1 |
Kawasaki, H; Takasaki, K; Urabe, M | 1 |
Arrivas, S; Balfagon, G; Barrus, MT; Capilla, MI; Marin, J; Rosa de Sagarra, M | 1 |
Chernesky, CE; Chou, TC; Felsen, D; Marion, DN; Somers, WJ; Vaughan, ED | 1 |
Widdop, RE | 1 |
Bagdy, G; Fekete, MI; Kopin, IJ; Szemeredi, K; Zukowska-Grojec, Z | 1 |
File, SE; Johnston, AL | 1 |
Förstermann, U; Hohlfeld, J; Liebau, S | 1 |
Goodlett, CR; Valentino, ML | 1 |
Kulkarni, SK; Kunchandy, J | 2 |
Giesen-Crouse, E; Imbs, JL; Krieger, JP; Schmidt, M | 1 |
De Peyer, JE; Haeusler, G | 1 |
Carrier, GO; White, RE | 1 |
Cheung, DW | 1 |
Kobinger, W; Pichler, L | 3 |
Furnace, G; Hamilton, CA; Reid, JL; Sumner, DJ | 1 |
Höglund, AU; Meyerson, BJ | 1 |
Khanna, S; Kulkarni, SK; Kunchandy, J | 1 |
Cooke, JP; Flavahan, NA; Rimele, TJ; Vanhoutte, PM | 1 |
Baggio, G; Ferrari, F; Martinelli, R | 1 |
György, L; Ludvig, N; Vizi, ES | 1 |
Kulkarni, SK; Parale, MP | 2 |
Bou, J; Massingham, R | 1 |
Kannan, MS; Seip, AE | 1 |
Flores, F; Hester, RK; Satake, N; Shibata, S; Ueda, S | 1 |
Kubo, T; Misu, Y; Nagura, J | 1 |
Barrett, JA; Mann, WS; Sales, EF; Smith, RD; Van Inwegen, RG; Wolf, PS | 1 |
Korstanje, C; van Zwieten, PA | 1 |
Hester, RK; Ito, M; Kurahashi, K; Satake, N; Shibata, S | 1 |
Furuta, T | 1 |
Fondacaro, JD; Kolpak, D; McCafferty, GP | 1 |
Decker, N; Schwartz, J | 1 |
Shebuski, RJ; Zimmerman, BG | 1 |
de Jonge, A; Mathy, MJ; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B | 1 |
Kawasaki, H; Takasaki, K | 1 |
Kobinger, W | 2 |
Chapman, KL; Marwood, JF; Stokes, GS | 1 |
Baggio, G; Ferrari, W; Guarini, S | 1 |
King, KA; Pang, CC | 1 |
Kulkarni, SK; Kunchandy, J; Mehta, AK | 1 |
Ferrari, F | 1 |
De Jonge, A; Doods, HN; Korstanje, C; Thoolen, MJ; Timmermans, PB; Van Zwieten, PA; Wilffert, B | 1 |
de Jonge, A; Innemee, HC; Timmermans, PB; van Meel, JC; van Zwieten, PA | 1 |
Qian, JQ; Timmermans, PB; Van Meel, JC; Van Zwieten, PA | 1 |
Mottram, DR | 1 |
Mathy, MJ; Qian, JQ; Thoolen, MJ; Timmermans, PB; van Zwieten, PA | 1 |
Kubo, T; Su, C | 1 |
DeMarinis, RM; Lafferty, J; Macia, RA; Matthews, WD | 1 |
Mottram, DR; Thakar, Y | 1 |
Lues, I; Schümann, HJ | 1 |
Hammer, R; Kobinger, W; Pichler, L | 1 |
Kobinger, W; Lillie, C; Pichler, L | 1 |
Qian, JQ; Thoolen, MJ; Timmermans, PB; van Meel, JC; van Zwieten, PA | 1 |
Andersson, RG; Grundström, N; Visnovsky, P; Wikberg, JE | 1 |
Breslin, DS; Ernsberger, P; Felsen, D; Marion, DN; May, M; Nejat, RJ; Nguyen, P; Sutaria, PM; Vaughan, ED | 1 |
Chambers, JR; Connelly, CD; Raffa, RB; Stone, DJ | 1 |
Arnsten, AF; Jentsch, DJ; Li, BM; Steere, JC | 1 |
Kubota, K; Li, BM | 1 |
Alvarez-Guerra, M; Bertholom, N; Garay, RP | 1 |
Colpaert, FC; Pauwels, PJ | 1 |
Artigues-Varin, C; Mulder, P; Richard, V; Thuillez, C; Varin, R | 1 |
1 review(s) available for clonidine and talipexole
Article | Year |
---|---|
Rudolf Buchheim lecture. Drugs as tools in research on adrenoceptors.
Topics: Angiotensin II; Animals; Azepines; Blood Pressure; Clonidine; Guanabenz; Guanfacine; Guanidines; Heart Rate; Humans; Imidazoles; Methoxamine; Oxymetazoline; Phenylacetates; Prazosin; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thiophenes; Xylazine; Yohimbine | 1986 |
81 other study(ies) available for clonidine and talipexole
Article | Year |
---|---|
Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and antagonists.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cell Membrane; Clonidine; Kinetics; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Vasoconstriction | 1984 |
Characterization of alpha-adrenoceptor populations. Quantitative relationships between cardiovascular effects initiated at central and peripheral alpha-adrenoceptors.
Topics: Animals; Blood Pressure; Blood Vessels; Brain; Hemodynamics; Male; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha | 1981 |
Alpha-adrenoceptor modulation of the efferent function of capsaicin-sensitive sensory neurones in guinea-pig isolated atria.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Calcitonin Gene-Related Peptide; Capsaicin; Clonidine; Efferent Pathways; Electric Stimulation; Guinea Pigs; Heart; In Vitro Techniques; Male; Neurons, Afferent; Norepinephrine; Receptors, Adrenergic, alpha | 1992 |
Effect of chlorethylclonidine on arterial blood pressure and heart rate in the conscious rat.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Blood Pressure; Clonidine; Heart Rate; Injections, Intraperitoneal; Male; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha | 1992 |
The interrelationship between the effects of captopril and nifedipine on pressor responses elicited by selective alpha-adrenoceptor agonists in the pithed rat preparation.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Blood Pressure; Captopril; Clonidine; Decerebrate State; Imidazoles; Male; Nifedipine; Rats; Rats, Inbred Strains | 1992 |
Regulation of noradrenaline release from rat occipital cortex tissue chops by alpha 2-adrenergic agonists.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Brimonidine Tartrate; Bucladesine; Clonidine; Colforsin; Cyclic AMP; Histological Techniques; Male; Norepinephrine; Occipital Lobe; Quinoxalines; Rats; Rats, Inbred Strains | 1991 |
Comparative study of postsynaptic alpha-adrenoceptors in aorta obtained from human and other mammalian species.
Topics: Adrenergic alpha-Agonists; Animals; Aorta; Azepines; Clonidine; Guinea Pigs; Humans; In Vitro Techniques; Male; Methoxamine; Muscle, Smooth, Vascular; Norepinephrine; Prazosin; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Species Specificity; Yohimbine | 1991 |
Differences in activity between noradrenaline and other alpha-agonists in rat vas deferens.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Clonidine; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Methoxamine; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vas Deferens | 1991 |
Effects of B-HT 920 in the tail-suspension test.
Topics: Adrenergic alpha-Agonists; Animals; Apomorphine; Azepines; Clonidine; Depressive Disorder; Dopamine Agents; Imipramine; Male; Mice; Motor Activity; Yohimbine | 1991 |
Effects of staurosporine on the pressor responses to alpha-adrenoceptor agonists in pithed rats: a comparison with nifedipine.
Topics: Adrenergic alpha-Agonists; Alkaloids; Animals; Azepines; Blood Pressure; Clonidine; Decerebrate State; Imidazoles; Male; Muscle, Smooth, Vascular; Nifedipine; Protein Kinase C; Rats; Rats, Inbred Strains; Staurosporine | 1991 |
Participation of endothelium-derived relaxing factor and role of cyclic GMP in inhibitory effects of endothelium on contractile responses elicited by alpha-adrenoceptor agonists in rat aorta.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Arginine; Azepines; Clonidine; Cyclic GMP; Endothelium, Vascular; Female; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide; Phenylephrine; Rats; Rats, Inbred Strains | 1991 |
Mutual interaction between presynaptic alpha 2-adrenoceptors and 5-HT1B receptors on the sympathetic nerve terminals of the rat inferior vena cava.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic Fibers; Animals; Azepines; Clonidine; Dioxanes; Electric Stimulation; Idazoxan; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Neurotransmitter; Receptors, Serotonin; Serotonin; Tritium; Vena Cava, Inferior | 1990 |
Regulation of noradrenaline release in human cerebral arteries via presynaptic alpha 2-adrenoceptors.
Topics: Adrenergic alpha-Agonists; Azepines; Cerebral Arteries; Clonidine; Electric Stimulation; Humans; Methoxamine; Norepinephrine; Receptors, Adrenergic, alpha; Time Factors; Tritium; Yohimbine | 1990 |
Effect of BHT 920 on monoaminergic neurons of the rat brain: an electrophysiological in vivo and in vitro study.
Topics: Action Potentials; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Apomorphine; Azepines; Biogenic Monoamines; Brain; Clonidine; Dioxanes; Dopamine Agents; Idazoxan; In Vitro Techniques; Locus Coeruleus; Male; Neurons; Raphe Nuclei; Rats; Rats, Inbred Strains; Sulpiride; Tegmentum Mesencephali | 1990 |
Calcium dependency of vasoconstriction mediated by alpha 1- and alpha 2-adrenoceptors.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Azepines; Blood Pressure; Calcium; Calcium Channel Blockers; Clonidine; Imidazoles; Ion Channels; Nifedipine; Rats; Receptors, Adrenergic, alpha; Regional Blood Flow; Structure-Activity Relationship; Vasoconstriction | 1985 |
Sensitivity of alpha-adrenoceptor agonists to the calcium channel activator, Bay K 8644, in canine saphenous vein.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Agonists; Animals; Azepines; Clonidine; Dogs; Female; In Vitro Techniques; Ion Channels; Male; Muscle, Smooth, Vascular; Saphenous Vein | 1987 |
Modulation of noradrenaline release from cat cerebral arteries by presynaptic alpha 2-adrenoceptors. Effect of chronic treatment with desipramine and cocaine.
Topics: Animals; Azepines; Cerebral Arteries; Clonidine; Cocaine; Desipramine; Dogs; Electric Stimulation; Female; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Norepinephrine; Receptors, Adrenergic, alpha; Tetrodotoxin | 1989 |
Presynaptic alpha 2-adrenoceptor modulation of 5-hydroxytryptamine and noradrenaline release from vascular adrenergic nerves.
Topics: Animals; Azepines; Clonidine; Cocaine; Electric Stimulation; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Serotonin; Splanchnic Circulation; Sympathetic Nervous System; Synapses | 1989 |
Effect of phorbol esters on noradrenaline release from cerebral arteries.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Cats; Cerebral Arteries; Clonidine; Electric Stimulation; Female; Male; Norepinephrine; Phorbol Esters; Protein Kinase C; Tetradecanoylphorbol Acetate; Yohimbine | 1989 |
An in vivo evaluation of alpha adrenergic receptors in canine prostate.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Benzazepines; Clonidine; Dogs; Dose-Response Relationship, Drug; Epinephrine; Male; Prazosin; Pressure; Prostate; Receptors, Adrenergic, alpha; Yohimbine | 1989 |
The effects of B-HT 920 and St 91 on venous haemodynamics in cats.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Cats; Clonidine; Female; Hemodynamics; Male | 1989 |
Opposite effects of chronic cortisol treatment on pre- and postsynaptic actions of clonidine in pithed rats.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Blood Pressure; Body Weight; Clonidine; Decerebrate State; Drug Interactions; Epinephrine; Heart Rate; Hydrocortisone; Male; Norepinephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Sympathetic Nervous System; Time Factors | 1989 |
Yohimbine's anxiogenic action: evidence for noradrenergic and dopaminergic sites.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Adrenergic alpha-Agonists; Animals; Anxiety; Apomorphine; Azepines; Benzazepines; Clonidine; Dopamine Agents; Ergolines; Guanfacine; Guanidines; Learning; Male; Norepinephrine; Phenylacetates; Phenylephrine; Quinpirole; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Dopamine; Yohimbine | 1989 |
The inhibition of alpha 1-adrenoceptor-mediated contractions of rabbit pulmonary artery by Ca2+-withdrawal, pertussis toxin and N-ethylmaleimide is dependent on agonist intrinsic efficacy.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Calcium; Calcium Channel Blockers; Clonidine; Ethylmaleimide; Female; Gallic Acid; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Pertussis Toxin; Phenylephrine; Pulmonary Artery; Rabbits; Receptors, Adrenergic, alpha; Virulence Factors, Bordetella | 1989 |
Differential effects of clonidine, B-HT 933 and B-HT 920 in immature rat pups.
Topics: Animals; Azepines; Behavior, Animal; Clonidine; Dose-Response Relationship, Drug; Haloperidol; Motor Activity; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter | 1987 |
Modulatory effect of alpha 2 adrenoceptor agonists on Ro 5-4864-induced convulsions in rats and mice.
Topics: Animals; Anticonvulsants; Azepines; Benzodiazepinones; Brain; Clonidine; Convulsants; Guanfacine; Guanidines; Imidazoles; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Phenylacetates; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, GABA-A; Seizures | 1987 |
Characterisation of the alpha-adrenoceptors of the rat renal vascular bed.
Topics: Animals; Azepines; Clonidine; Dopamine; In Vitro Techniques; Kidney; Male; Nordefrin; Perfusion; Phenylephrine; Prazosin; Rabbits; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vascular Resistance; Yohimbine | 1987 |
Electrical membrane events in response to alpha-adrenoceptor stimulation.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Calcium; Cell Membrane; Clonidine; Female; Male; Membrane Potentials; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Potassium; Pulmonary Artery; Rabbits; Receptors, Adrenergic, alpha; Stimulation, Chemical; Strychnine | 1985 |
Enhancement of alpha-1 and alpha-2 adrenergic agonist-induced vasoconstriction by removal of endothelium in rat aorta.
Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Azepines; Calcium Chloride; Clonidine; Endothelium; In Vitro Techniques; Male; Methoxamine; Norepinephrine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Vasoconstriction; Yohimbine | 1985 |
An electrophysiological study of alpha-adrenoceptor mediated excitation-contraction coupling in the smooth muscle cells of the rat saphenous vein.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Clonidine; Electrophysiology; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Neuromuscular Junction; Norepinephrine; Phenylephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Saphenous Vein; Synaptic Transmission | 1985 |
Alpha 2-adrenoceptor blocking properties of the alpha 1-selective agonist 2-(2-chloro-5-trifluoromethylphenylimino)imidazolidine (St 587).
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Behavior, Animal; Clonidine; Dogs; Drug Interactions; Electric Stimulation; Exploratory Behavior; Female; Heart Rate; Male; Mice; Prazosin; Pressoreceptors; Rats; Spinal Cord; Vagotomy | 1985 |
Recovery of alpha-adrenoreceptor mediated responses and binding site number after intravenous benextramine in the rabbit.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Brain; Clonidine; Cystamine; Injections, Intravenous; Male; Membranes; Phenoxybenzamine; Phenylephrine; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Spleen; Time Factors | 1985 |
Increased investigative activity after presynaptic dopaminergic stimulation measured by a fixed-interval recording procedure.
Topics: Adrenergic alpha-Agonists; alpha-Methyltyrosine; Animals; Apomorphine; Azepines; Clonidine; Drug Interactions; Exploratory Behavior; Haloperidol; Male; Methyltyrosines; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Dopamine; Stimulation, Chemical; Yohimbine | 1985 |
Effect of alpha2 agonists clonidine, guanfacine and B-HT 920 on gastric acid secretion and ulcers in rats.
Topics: Adrenergic alpha-Agonists; Animals; Anti-Ulcer Agents; Azepines; Clonidine; Female; Gastric Acid; Gastric Acidity Determination; Guanfacine; Guanidines; Humans; Male; Phenylacetates; Pylorus; Rats; Rats, Inbred Strains; Restraint, Physical; Stomach Ulcer; Stress, Psychological; Time Factors | 1985 |
Nimodipine and inhibition of alpha adrenergic activation of the isolated canine saphenous vein.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Calcium Channel Blockers; Clonidine; Dogs; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Male; Nicotinic Acids; Nimodipine; Potassium; Receptors, Adrenergic, alpha; Saphenous Vein; Tyramine; Vasoconstriction | 1985 |
Imidazole has similar behavioural effects to yohimbine.
Topics: Adrenergic alpha-Agonists; Animals; Animals, Newborn; Azepines; Behavior, Animal; Body Temperature; Chickens; Clonidine; Haloperidol; Hypnotics and Sedatives; Imidazoles; Male; Penile Erection; Prazosin; Rats; Sexual Behavior, Animal; Sleep; Time Factors; Yohimbine | 1986 |
Evidence that serotonin receptors are involved in the anticonvulsant effect of yohimbine in mice.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Anticonvulsants; Azepines; Clonidine; Dioxanes; Electroshock; Idazoxan; Male; Metergoline; Methysergide; Mice; Quipazine; Receptors, Serotonin; Serotonin Antagonists; Yohimbine | 1986 |
Studies with alpha 2-adrenoceptor agonists and alcohol abstinence syndrome in rats.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Clonidine; Ethanol; Guanfacine; Guanidines; Male; Phenylacetates; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome | 1986 |
Effect of diltiazem upon contractile responses to phenylephrine, cirazoline, Sgd 101/75, St 587 and B-HT 920 in rabbit aorta and dog saphenous vein preparations.
Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Azepines; Benzazepines; Clonidine; Diltiazem; Dogs; Drug Interactions; Female; Imidazoles; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Rabbits; Saphenous Vein | 1986 |
Mechanisms of alpha-adrenoceptor mediated contractions of rat mesenteric artery.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Clonidine; In Vitro Techniques; Kinetics; Male; Mesenteric Arteries; Muscle, Smooth, Vascular; Nifedipine; Nitrendipine; Norepinephrine; Phenylephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vasoconstriction; Verapamil | 1986 |
Effect of nicorandil, N-(2-hydroxyethyl)nicotinamide nitrate, a new anti-anginal agent, on contractile responses to alpha-1- and alpha-2-adrenoceptor agonists in isolated rabbit aorta.
Topics: Adrenergic alpha-Agonists; Animals; Aorta; Azepines; Clonidine; Male; Methoxamine; Niacinamide; Nicorandil; Nifedipine; Rabbits; Vasodilation | 1986 |
Reversal by alpha-2 agonists of diazepam withdrawal hyperactivity in rats.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Clonidine; Diazepam; Guanfacine; Guanidines; Male; Motor Activity; Phenylacetates; Rats; Rats, Inbred Strains; Substance Withdrawal Syndrome; Yohimbine | 1986 |
Pharmacological characterization of spinal alpha adrenoceptors related to blood pressure control in rats.
Topics: Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Brain Stem; Clonidine; Dopamine; Guanabenz; Hydroxydopamines; Injections, Spinal; Male; Norepinephrine; Oxidopamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Spinal Cord; Yohimbine | 1987 |
Celiprolol, a compound possessing weak alpha 2-adrenergic antagonist properties in the dog.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Catecholamines; Celiprolol; Clonidine; Coronary Circulation; Dogs; Heart Rate; In Vitro Techniques; Methoxamine; Propanolamines; Propranolol; Saphenous Vein; Vasoconstriction; Yohimbine | 1986 |
Characterization of alpha-adrenoreceptor mediated reduction of flow in a saline-perfused constant pressure model of rat perfused hindquarters.
Topics: Acid-Base Equilibrium; Adrenergic alpha-Agonists; Angiotensin II; Animals; Azepines; Blood Pressure; Calcium; Clonidine; Dinoprost; Gallopamil; Hindlimb; Male; Perfusion; Potassium Chloride; Prostaglandins F; Rats; Receptors, Adrenergic, alpha; Regional Blood Flow; Reserpine | 1987 |
The mode of vasoinhibitory action of a pyridazione derivative (MCI-154), a new cardiotonic agent, on contractile responses induced by alpha-adrenoceptor agonists and 45Ca influx in isolated vascular smooth muscles.
Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Azepines; Calcium; Calcium Radioisotopes; Cardiotonic Agents; Clonidine; Iliac Artery; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Pyridazines; Rabbits; Vasodilator Agents | 1988 |
Precontraction-induced contractile response of isolated canine portal vein to alpha-2 adrenoceptor agonists.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Calcimycin; Cats; Clonidine; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Portal Vein; Prazosin; Yohimbine | 1988 |
Selective alpha-2 adrenoceptor agonists alter fluid and electrolyte transport in mammalian small intestine.
Topics: 16,16-Dimethylprostaglandin E2; Adrenergic alpha-Agonists; Animals; Azepines; Clonidine; Dose-Response Relationship, Drug; Electrolytes; Intestine, Small; Male; Rabbits; Yohimbine | 1988 |
Postjunctional alpha-1 and alpha-2 adrenoceptors in the coronaries of the perfused guinea-pig heart.
Topics: Animals; Azepines; Clonidine; Coronary Vessels; Dose-Response Relationship, Drug; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Male; Myocardial Contraction; Nordefrin; Norepinephrine; Perfusion; Phenylephrine; Prazosin; Receptors, Adrenergic, alpha; Vascular Resistance; Yohimbine | 1985 |
Prejunctional alpha 2-adrenoceptor mediated inhibitory action of clonidine and B-HT 920, but not urapidil in guinea pig ileum.
Topics: Animals; Azepines; Clonidine; Electric Stimulation; Female; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Piperazines; Receptors, Adrenergic, alpha | 1985 |
Effects of the irreversible alpha-adrenoceptor antagonists phenoxybenzamine and benextramine on the effectiveness of nifedipine in inhibiting alpha 1- and alpha 2-adrenoceptor mediated vasoconstriction in pithed rats.
Topics: Animals; Azepines; Clonidine; Cystamine; Decerebrate State; Diastole; Dose-Response Relationship, Drug; Imidazoles; Male; Nifedipine; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vasoconstriction | 1985 |
Central alpha-2 adrenoceptor-mediated hypertensive response to clonidine in conscious, normotensive rats.
Topics: Animals; Azepines; Blood Pressure; Brain; Cimetidine; Clonidine; Hydroxydopamines; Injections, Intraventricular; Ketanserin; Male; Methoxamine; Oxidopamine; Piperidines; Prazosin; Procaine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine | 1986 |
Studies that question the existence of alpha-2 adrenoceptors in tail arteries of normotensive Sprague-Dawley rats.
Topics: Animals; Arteries; Azepines; Clonidine; Dose-Response Relationship, Drug; Male; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tail; Vasoconstriction; Yohimbine | 1986 |
Studies on epinephrine-induced lung edema in the rat. I. Selective alpha 1-adrenoceptor involvement.
Topics: Animals; Azepines; Blood Pressure; Clonidine; Dibenzylchlorethamine; Epinephrine; Female; Metaraminol; Norepinephrine; Phenylephrine; Practolol; Prazosin; Propranolol; Pulmonary Edema; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine | 1986 |
Clonidine--induced behavioural despair in mice: reversal by antidepressants.
Topics: Animals; Antidepressive Agents; Antidepressive Agents, Tricyclic; Azepines; Clonidine; Depression; Diazepam; Guanfacine; Guanidines; Lithium; Male; Phenylacetates; Rats; Rats, Inbred Strains; Tranylcypromine; Yohimbine | 1986 |
Differential cardiovascular effects of central clonidine and B-HT 920 in conscious rats.
Topics: Animals; Azepines; Blood Pressure; Cardiovascular System; Clonidine; Epinephrine; Heart; Injections, Intraventricular; Male; Norepinephrine; Rats; Yohimbine | 1988 |
Anti-inflammatory actions of clonidine, guanfacine and B-HT 920 against various inflammagen-induced acute paw oedema in rats.
Topics: Animals; Anti-Inflammatory Agents; Azepines; Bradykinin; Carrageenan; Clonidine; Edema; Formaldehyde; Guanfacine; Guanidines; Histamine; Injections, Intraventricular; Male; Phenylacetates; Rats; Rats, Inbred Strains; Serotonin; Time Factors | 1986 |
Behavioural pharmacology of imidazole, a potential antidepressant agent.
Topics: Aggression; Animals; Antidepressive Agents; Apomorphine; Azepines; Behavior, Animal; Body Temperature; Chickens; Clonidine; Drug Synergism; Imidazoles; Lethal Dose 50; Male; Mice; Motor Activity; Penile Erection; Rats; Rats, Inbred Strains; Sleep; Yohimbine | 1985 |
Affinity of WY 26703 for central and peripheral alpha 1- and alpha 2-adrenoreceptors in the rat; comparison with yohimbine.
Topics: Animals; Azepines; Binding, Competitive; Blood Pressure; Clonidine; In Vitro Techniques; Male; Methoxamine; Muscle, Smooth, Vascular; Myocardium; Prazosin; Quinolizines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine | 1984 |
alpha 1-adrenoceptor blockade by alpha 2-adrenoceptor agonists in the isolated perfused hindquarter of rats.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Clonidine; In Vitro Techniques; Male; Methoxamine; Oxazoles; Perfusion; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thiazoles; Vasoconstriction | 1981 |
Modulation of motor activity by alpha 1- and alpha 2-adrenoceptor stimulation in mice.
Topics: Adrenergic alpha-Agonists; Animals; Apomorphine; Azepines; Clonidine; Exploratory Behavior; Male; Mice; Motor Activity; Thiazoles | 1981 |
Differential effects of selective alpha 1- and alpha 2-adrenoceptor agonists on intraocular pressure in the conscious rabbit.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Clonidine; Female; Intraocular Pressure; Male; Phenylephrine; Procaine; Pupil; Yohimbine | 1982 |
Central blood pressure regulation. Involvement of presynaptic or postsynaptic, alpha 1- or alpha 2-adrenoceptors?
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Cats; Clonidine; Dogs; Heart Rate; Medulla Oblongata; Oxymetazoline; Piperoxan; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Synapses | 1983 |
Differential inhibition of alpha 2-adrenoceptor-mediated pressor responses by (+)- and (-)-verapamil in pithed rats.
Topics: Adrenergic alpha-Antagonists; Animals; Azepines; Blood Pressure; Clonidine; Male; Rats; Rats, Inbred Strains; Spinal Cord; Stereoisomerism; Verapamil | 1983 |
Pre-junctional alpha 2-adrenoceptor activity of B-HT920.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Clonidine; Dioxanes; Drug Interactions; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Rats; Rats, Inbred Strains; Yohimbine | 1983 |
Antihypertensive activity and interaction with alpha-adrenoceptors of tibalosine ([1-(2, 3-dihydro-5-benzo-(b)-thienyl)-2-(4-phenyl-butylamino)-1-propanol], CP 804 S) in rat and cat preparations.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Azepines; Brain; Cats; Clonidine; Female; Heart Rate; Injections, Intraventricular; Male; Membranes; Prazosin; Propanolamines; Rats; Rats, Inbred Strains; Vasopressins | 1983 |
Alpha-adrenoceptor- and prostaglandin-mediated modulation of vascular adrenergic neurotransmission in spontaneously hypertensive rats.
Topics: Animals; Autonomic Fibers, Postganglionic; Azepines; Blood Pressure; Clonidine; Dinoprostone; Electric Stimulation; Hypertension; In Vitro Techniques; Male; Mesenteric Arteries; Neurotransmitter Agents; Norepinephrine; Prostaglandins E; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vasoconstriction; Yohimbine | 1984 |
Assessment of alpha-adrenergic receptor subtypes in isolated rat aortic segments.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Azepines; Clonidine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Naphthols; Norepinephrine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine | 1984 |
The action and interaction of beta-phenethylamines and imidazolines on prejunctional alpha 2-adrenoceptors of guinea-pig ileum in the presence of the non-competitive antagonist benextramine.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Clonidine; Cystamine; Electric Stimulation; Guinea Pigs; Ileum; Imidazoles; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nordefrin; Phenethylamines; Receptors, Adrenergic, alpha | 1984 |
Effect of removing the endothelial cells on the reactivity of rat aortic segments to different alpha-adrenoceptor agonists.
Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Azepines; Clonidine; Endothelium; Imidazoles; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Rats; Rats, Inbred Strains; Xylazine; Yohimbine | 1984 |
Binding of an imidazolidine (clonidine), an oxazoloazepin (B-HT 933) and a thiazoloazepin (B-HT 920) to rat brain alpha-adrenoceptors and relation to cardiovascular effects.
Topics: Animals; Azepines; Binding Sites; Binding, Competitive; Blood Pressure; Brain; Clonidine; Heart Rate; Kinetics; Male; Oxazoles; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thiazoles | 1980 |
Central cardiovascular alpha-adrenoceptors. Relation to peripheral receptors.
Topics: Animals; Azepines; Blood Pressure; Cardiovascular System; Clonidine; Dose-Response Relationship, Drug; Heart Rate; Male; Methoxamine; Norepinephrine; Oxazoles; Perfusion; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Thiazoles; Vagotomy | 1980 |
Hypotensive activity of tetrandrine in rats. Investigation into its mode of action.
Topics: Alkaloids; Anesthesia; Animals; Antihypertensive Agents; Azepines; Benzylisoquinolines; Blood Pressure; Brain; Clonidine; Heart Rate; Hypertension; Male; Methoxamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vasopressins | 1983 |
Pharmacology of B-HT 920 in some isolated smooth muscles of the guinea-pig.
Topics: Animals; Aorta; Azepines; Clonidine; Dogs; Drug Interactions; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Trachea; Vas Deferens; Yohimbine | 1982 |
Identification, localization and functional analysis of imidazoline and alpha adrenergic receptors in canine prostate.
Topics: Animals; Autoradiography; Azepines; Binding Sites; Clonidine; Dogs; Guanylyl Imidodiphosphate; Imidazoles; Imidazoline Receptors; Male; Prostate; Prostatic Hyperplasia; Receptors, Adrenergic, alpha; Receptors, Drug | 1994 |
Alpha-subunit G-protein antisense oligodeoxynucleotide effects on supraspinal (i.c.v.) alpha2-adrenoceptor antinociception in mice.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Base Sequence; Cerebral Ventricles; Clonidine; GTP-Binding Proteins; Injections, Intraventricular; Male; Mice; Mice, Inbred Strains; Molecular Sequence Data; Oligonucleotide Probes; Oligonucleotides, Antisense; Pain; Receptors, Adrenergic, alpha-2 | 1996 |
Noradrenergic influences on prefrontal cortical cognitive function: opposing actions at postjunctional alpha 1 versus alpha 2-adrenergic receptors.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Animals; Azepines; Brimonidine Tartrate; Clonidine; Cognition; Discrimination, Psychological; Guanfacine; Haplorhini; Memory; Norepinephrine; Quinoxalines; Reaction Time; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Visual Perception | 1998 |
Alpha-2 adrenergic modulation of prefrontal cortical neuronal activity related to a visual discrimination task with GO and NO-GO performances in monkeys.
Topics: Adrenergic alpha-Agonists; Animals; Azepines; Clonidine; Discrimination, Psychological; Female; Macaca mulatta; Neurons; Prefrontal Cortex; Receptors, Adrenergic, alpha-2; Visual Perception | 1998 |
Selective blockade by nicergoline of vascular responses elicited by stimulation of alpha 1A-adrenoceptor subtype in the rat.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta; Azepines; Binding, Competitive; Blood Pressure; Clonidine; Decerebrate State; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Male; Mesenteric Arteries; Nicergoline; Prazosin; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sensitivity and Specificity; Tritium | 1999 |
Partial to complete antagonism by putative antagonists at the wild-type alpha(2C)-adrenoceptor based on kinetic analyses of agonist:antagonist interactions.
Topics: Adrenergic Agonists; Adrenergic Antagonists; Animals; Azepines; Brimonidine Tartrate; Calcium; CHO Cells; Clonidine; Cricetinae; DNA, Recombinant; Dose-Response Relationship, Drug; Drug Interactions; Epinephrine; GTP-Binding Protein alpha Subunits, Gi-Go; GTP-Binding Protein alpha Subunits, Gq-G11; Heterotrimeric GTP-Binding Proteins; Idazoxan; Kinetics; Medetomidine; Mice; Oxymetazoline; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Recombinant Fusion Proteins; Transfection | 2000 |
Alpha2-adrenoceptor ligands inhibit alpha1-adrenoceptor-mediated contraction of isolated rat arteries.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Arteries; Azepines; Brimonidine Tartrate; Clonidine; Idazoxan; In Vitro Techniques; Ligands; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Oxazoles; Prostaglandins; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Rilmenidine; Yohimbine | 2002 |