clonidine has been researched along with piperidines in 81 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 38 (46.91) | 18.7374 |
1990's | 8 (9.88) | 18.2507 |
2000's | 25 (30.86) | 29.6817 |
2010's | 9 (11.11) | 24.3611 |
2020's | 1 (1.23) | 2.80 |
Authors | Studies |
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Andén, NE; Grabowska, M; Strömbom, U | 1 |
Andén, NE; Grabowska, M | 1 |
Aghajanian, GK; Cedarbaum, JM | 1 |
Kapur, H; Mottram, DR | 1 |
Bogaert, A; Bogaert, PP; DeWilde, A; Reneman, RS; Wellens, D; Wouters, L | 1 |
Franklin, KB; Herberg, LJ | 1 |
Fang, VS; Fessler, RG; Meltzer, HY | 1 |
Donabedian, RK; Gold, MS; Redmond, DE | 1 |
Kapur, H; Rouot, B; Snyder, SH | 1 |
Kobinger, W; Pichler, L | 1 |
Janssen, PA; Van Nueten, JM; Wellens, S | 1 |
Keil, LC; Nolan, PL; Reid, IA; Wolf, JA | 1 |
Buus Lassen, J | 1 |
Baran, L; Maj, J; Palider, W | 1 |
van Zwieten, PA | 2 |
De Wilde, A; Janssen, PA; Reneman, RS; van Bogaert, A; van Bogaert, PP; Wellens, D; Wouters, L | 1 |
Luo, XX; Sheng, BH; Tan, YH | 1 |
Marshall, IG; Prior, C; Wannan, G | 1 |
Chiba, S; Furukawa, Y; Nakane, T | 1 |
Brunello, N; Galimberti, R; Racagni, G; Riva, M; Rovescalli, AC | 1 |
Henderson, G; Kennedy, C | 1 |
England, CD; Smith, CF; Stillings, MR; Welbourn, AP | 1 |
Kawasaki, H; Takasaki, K | 1 |
Doğan, N; Ilhan, M; Kayaalp, SO; Tuncer, M | 1 |
Braestrup, C | 1 |
Hasselager, E; Scheel-Krüger, J | 1 |
Bolme, P; Corrodi, H; Fuxe, K; Goldstein, M; Hökfelt, T; Lidbrink, P | 1 |
Finch, L | 1 |
Anthony, M; Lance, JW | 1 |
Bolme, P; Fuxe, K; Goldstein, M; Hökfelt, T; Lidbrink, P | 1 |
Wurtman, RJ; Yehuda, S | 1 |
Beubler, E; Bukhave, K; Rask-Madsen, J | 1 |
Batink, HD; Timmermans, PB; van Kemenade, JE; van Zwieten, PA | 1 |
Timmermans, PB; Van Brummelen, P; Van Zwieten, PA | 1 |
Opie, LH | 1 |
McCall, RB; Schuette, MR | 1 |
Geyer, MA; Lee, EH | 1 |
Adelung, C; Lang, JD; Späth, L; Starke, K | 1 |
Shapiro, AK; Shapiro, E | 1 |
Bentley, GA; McLennan, PL | 1 |
Nakamura, K; Okuma, Y; Osumi, Y; Yokotani, K | 1 |
Bonanno, G; Fassio, A; Fontana, G; Marchi, M; Raiteri, M; Usai, C | 1 |
Kamato, T; Miyata, K; Nagakura, Y; Naitoh, Y; Yamano, M | 1 |
Chen, H; Cheng, L; Hsu, L; Jen, CJ; Lin, MT; Yang, C | 1 |
Benhamou, D; Mercier, FJ | 1 |
Boikova, NV; Strashnov, VI; Tomson, VV; Volchkov, VA; Zaitsev, AA | 1 |
Coruzzi, G; Poli, E; Pozzoli, C; Schunack, W; Timmerman, H; Todorov, S | 1 |
Dörges, V; Gerlach, K; Hüppe, M; Kraatz, E; Saager, L; Schmitz, A; Schmucker, P; Uhlig, T | 1 |
Alsheimer, M; Koppert, W; Scheuber, K; Schmelz, M; Schüttler, J; Sittl, R | 1 |
Choi, JI; Yoon, MH | 1 |
Dietrich, PJ; Grottke, O; Krause, TH; Müller, J; Wappler, F | 1 |
Ando, S; Harasawa, I; Honda, K; Kamiya, HO; Koga, K; Takano, Y | 1 |
Arnulf, JJ; Balarac, N; Bigeon, JY; Bonnet, F; Lena, P; Tapia, M | 1 |
Hachenberg, T; Huth, C; Kozian, A; Schilling, T; Tiede, T | 1 |
Farias-Rodríguez, VM; Gallardo-Ortíz, IA; Gómez-Zamudio, JH; Lázaro-Suárez, ML; Tanoue, A; Tsujimoto, G; Villalobos-Molina, R | 1 |
Boselli, E; Chassard, D; Duflo, F; Ryvlin, P | 1 |
Corelli, RL; Hudmon, KS | 1 |
Pityaratstian, N | 1 |
Gessa, GL; Melis, M; Muntoni, AL; Perra, S; Pillolla, G; Pistis, M | 1 |
Frishman, WH | 1 |
Arici, G; Erman, M; Ertugrul, F; Karsli, B; Kayacan, N; Nacitarhan, C; Sadan, G | 1 |
Hayashida, K; Obata, H | 1 |
Bein, B; Brand, PA; Höcker, J; Ohnesorge, H; Scholz, J; Tonner, PH; Weber, B | 1 |
Buchhalter, AR; Fant, RV; Henningfield, JE | 1 |
Liatsi, D; Matamis, D; Pampori, S; Pneumatikos, I; Tsagourias, M; Tsapas, B | 1 |
Blier, P; Haddjeri, N | 1 |
Camarini, ET; Coelho, L; de Moraes, M; Farah, GJ; Filho, LI; Pavan, AJ; Previdelli, IT | 1 |
Alfinito, PD; Cosmi, S; Deecher, DC; Pawlyk, AC; Roman, J; Zhou, T | 1 |
Deissenrieder, F; Groneberg, D; Kusma, B; Mache, S; Quarcoo, D; Welte, T | 1 |
Bains, JS; Kuzmiski, JB; Pittman, QJ | 1 |
McMahon, LR; Stewart, JL | 1 |
Bhat, A; Crain, D | 1 |
Briyal, S; Gulati, A; Lavhale, MS; Parikh, N | 1 |
Kager, HI; Likar, R; Ohner, C; Pipam, W; Schlimp, CJ; Wolrab, C | 1 |
Bloch, A; Boemke, W; Harbeck-Seu, A; Hensel, M; Meisel, C; Renius, M; Rückert, JC; Spies, C; Viviano, E; Wernecke, KD | 1 |
Guillaume, V; Lemamy, GJ; Mouecoucou, J; Ndéboko, B; Oliver, C; Renard, M | 1 |
Bahremand, A; Dehpour, AR; Moezi, L; Shafaroodi, H | 1 |
Chumas, P; Guruswamy, V; Liddington, M; Rothera, E; Russell, J | 1 |
Bernal-Sprekelsen, M; Cardesin, A; Escamilla, Y; Escobar, MJ; Marco, J; Pontes, C; Rosell, R | 1 |
Bertoglio, LJ; Troyner, F | 1 |
8 review(s) available for clonidine and piperidines
Article | Year |
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Current concepts in the pathogenesis and interval treatment of migraine.
Topics: Adrenergic beta-Antagonists; Bradykinin; Clonidine; Cycloheptanes; Cyproheptadine; Ergotamine; Histamine; Humans; Methysergide; Migraine Disorders; Norepinephrine; Piperidines; Prostaglandins; Serotonin; Serotonin Antagonists; Thiophenes; Tyramine | 1972 |
Role of alpha adrenoceptors in hypertension and in antihypertensive drug treatment.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Azepines; Blood Pressure; Calcium Channel Blockers; Clonidine; Guanfacine; Guanidines; Humans; Hypertension; Ketanserin; Methyldopa; Muscle, Smooth, Vascular; Phenylacetates; Piperazines; Piperidines; Prazosin; Radioligand Assay; Receptors, Adrenergic, alpha; Vascular Resistance | 1984 |
Promising non-narcotic analgesic techniques for labour.
Topics: Analgesia, Obstetrical; Analgesics, Non-Narcotic; Clonidine; Epinephrine; Female; Humans; Midazolam; Neostigmine; Obstetric Labor Complications; Pain; Piperidines; Pregnancy; Receptors, N-Methyl-D-Aspartate; Remifentanil | 1998 |
Pharmacologic interventions for smoking cessation.
Topics: Administration, Cutaneous; Administration, Inhalation; Antidepressive Agents, Second-Generation; Benzazepines; Bupropion; Chewing Gum; Clonidine; Critical Care; Drug Therapy, Combination; Evidence-Based Medicine; Humans; Nicotine; Nicotinic Agonists; Nortriptyline; Nurse's Role; Patient Education as Topic; Patient Selection; Phytotherapy; Piperidines; Pyrazoles; Quinoxalines; Rimonabant; Smoking Cessation; Smoking Prevention; United States; United States Food and Drug Administration; Varenicline | 2006 |
Advances in alternative pharmacotherapy of ADHD.
Topics: Adrenergic alpha-Agonists; Antidepressive Agents, Tricyclic; Attention Deficit Disorder with Hyperactivity; Bupropion; Clonidine; Donepezil; Humans; Indans; Piperidines; Treatment Outcome | 2005 |
Smoking cessation pharmacotherapy--nicotine and non-nicotine preparations.
Topics: Administration, Cutaneous; Administration, Inhalation; Benzazepines; Bupropion; Chewing Gum; Clonidine; Coronary Artery Disease; Humans; Monoamine Oxidase Inhibitors; Nicotine; Nortriptyline; Piperidines; Pyrazoles; Quinoxalines; Receptors, Nicotinic; Rimonabant; Selective Serotonin Reuptake Inhibitors; Smoking; Smoking Cessation; Substance Withdrawal Syndrome; Tobacco Use Disorder; Tobacco, Smokeless; Varenicline | 2007 |
[Alpha2-adrenergic receptors in the dorsal horn of the spinal cord--their function and the descending inhibitory systems].
Topics: Acetylcholine; Adrenergic alpha-2 Receptor Agonists; Amines; Analgesics; Animals; Brain-Derived Neurotrophic Factor; Chronic Disease; Clonidine; Cyclohexanecarboxylic Acids; Donepezil; Drug Therapy, Combination; Gabapentin; gamma-Aminobutyric Acid; Humans; Indans; Neuralgia; Norepinephrine; Piperidines; Posterior Horn Cells; Receptors, Adrenergic, alpha-2; Receptors, Muscarinic | 2007 |
Novel pharmacological approaches for treating tobacco dependence and withdrawal: current status.
Topics: Antidepressive Agents; Aryl Hydrocarbon Hydroxylases; Clonidine; Cytochrome P-450 CYP2A6; Drug Delivery Systems; GABA Modulators; Humans; Narcotic Antagonists; Nicotine; Piperidines; Pyrazoles; Receptors, Nicotinic; Rimonabant; Substance Withdrawal Syndrome; Tobacco Use Disorder; Vaccination | 2008 |
8 trial(s) available for clonidine and piperidines
Article | Year |
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Remifentanil-clonidine-propofol versus sufentanil-propofol anesthesia for coronary artery bypass surgery.
Topics: Adjuvants, Anesthesia; Adrenergic alpha-Agonists; Aged; Analgesics, Opioid; Anesthesia Recovery Period; Anesthetics, Combined; Anesthetics, Intravenous; Catecholamines; Clonidine; Coronary Artery Bypass; Hemodynamics; Humans; Intraoperative Complications; Male; Middle Aged; Piperidines; Propofol; Remifentanil; Sufentanil | 2002 |
Differential modulation of remifentanil-induced analgesia and postinfusion hyperalgesia by S-ketamine and clonidine in humans.
Topics: Adrenergic alpha-Agonists; Adult; Analgesics, Opioid; Anesthetics, Dissociative; Blood Pressure; Clonidine; Cross-Over Studies; Double-Blind Method; Electric Stimulation; Half-Life; Humans; Hyperalgesia; Infusions, Intravenous; Ketamine; Male; Oxygen; Pain Measurement; Physical Stimulation; Piperidines; Receptors, Opioid, mu; Remifentanil; Substance Withdrawal Syndrome | 2003 |
[Comparison of premedication with clonidine and midazolam combined with TCI for orthopaedic shoulder surgery].
Topics: Adolescent; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adult; Aged; Analgesia, Patient-Controlled; Anesthesia, Conduction; Anesthetics, Intravenous; Clonidine; Double-Blind Method; Female; Hemodynamics; Humans; Male; Midazolam; Middle Aged; Narcotics; Orthopedic Procedures; Pain, Postoperative; Piperidines; Pirinitramide; Postoperative Nausea and Vomiting; Premedication; Propofol; Prospective Studies; Remifentanil; Shoulder | 2003 |
Fast-track coronary artery bypass grafting surgery under general anesthesia with remifentanil and spinal analgesia with morphine and clonidine.
Topics: Aged; Anesthesia, General; Anesthesia, Spinal; Clonidine; Coronary Artery Bypass; Drug Therapy, Combination; Female; Humans; Male; Middle Aged; Morphine; Pain Measurement; Pain, Postoperative; Piperidines; Prospective Studies; Remifentanil | 2005 |
Induced hypotension in orthognathic surgery: a comparative study of 2 pharmacological protocols.
Topics: Adolescent; Adrenergic alpha-Agonists; Adult; Anesthesia Recovery Period; Anesthesia, Dental; Anesthesia, General; Anesthesia, Intravenous; Anesthetics, Inhalation; Anesthetics, Intravenous; Blood Pressure; Clonidine; Dexmedetomidine; Female; Heart Rate; Humans; Hypotension, Controlled; Isoflurane; Male; Oral Surgical Procedures; Piperidines; Remifentanil | 2008 |
[Clonidine for remifentanil-induced hyperalgesia: a double-blind randomized, placebo-controlled study of clonidine under intra-operative use of remifentanil in elective surgery of the shoulder].
Topics: Adult; Analgesia, Patient-Controlled; Analgesics; Analgesics, Opioid; Anesthetics, Intravenous; Arthroscopy; Austria; Clonidine; Dose-Response Relationship, Drug; Double-Blind Method; Female; Humans; Hyperalgesia; Male; Middle Aged; Morphine; Pain Measurement; Pain, Postoperative; Piperidines; Preanesthetic Medication; Remifentanil; Shoulder; Shoulder Injuries; Shoulder Pain | 2011 |
Selective neurogenic blockade and perioperative immune reactivity in patients undergoing lung resection.
Topics: Aged; Amides; Analgesics, Opioid; Anesthetics, Local; Clonidine; Female; Hemodynamics; Humans; Injections, Epidural; Injections, Intravenous; Interferon-gamma; Interleukin-4; Lung; Male; Middle Aged; Nerve Block; Pain Measurement; Perioperative Care; Piperidines; Remifentanil; Ropivacaine; Treatment Outcome | 2012 |
A randomised double blind clinical trial to compare surgical field bleeding during endoscopic sinus surgery with clonidine-based or remifentanil-based hypotensive anaesthesia.
Topics: Anesthetics, Intravenous; Antihypertensive Agents; Blood Loss, Surgical; Clonidine; Double-Blind Method; Endoscopy; Female; Hemodynamics; Humans; Male; Middle Aged; Paranasal Sinus Diseases; Piperidines; Remifentanil; Treatment Outcome | 2015 |
65 other study(ies) available for clonidine and piperidines
Article | Year |
---|---|
Different alpha-adrenoreceptors in the central nervous system mediating biochemical and functional effects of clonidine and receptor blocking agents.
Topics: Adrenergic alpha-Antagonists; Animals; Brain; Central Nervous System; Clonidine; Dihydroxyphenylalanine; Dioxanes; Dopamine; Female; Haloperidol; Male; Methyltyrosines; Mice; Motor Activity; Norepinephrine; Phenoxybenzamine; Piperidines; Rats; Receptors, Adrenergic; Reflex; Spinal Cord; Tolazoline; Yohimbine | 1976 |
Noradrenaline synthesis and utilization: control by nerve impulse flow under normal conditions and after treatment with alpha-adrenoreceptor blocking agents.
Topics: Adrenergic alpha-Antagonists; Animals; Aromatic Amino Acid Decarboxylase Inhibitors; Benzyl Compounds; Brain; Clonidine; Denervation; Dihydroxyphenylalanine; Dioxanes; Dopamine; Haloperidol; Hydrazines; Male; Methyltyrosines; Norepinephrine; Normetanephrine; Phenoxybenzamine; Piperidines; Rats; Spinal Cord; Tolazoline; Tyramine; Yohimbine | 1976 |
Noradrenergic neurons of the locus coeruleus: inhibition by epinephrine and activation by the alpha-antagonist piperoxane.
Topics: Adrenergic alpha-Antagonists; Animals; Cerebral Ventricles; Clonidine; Epinephrine; gamma-Aminobutyric Acid; Iontophoresis; Isoproterenol; Male; Norepinephrine; Piperidines; Rats; Sotalol | 1976 |
A comparative study on the pre- and post-synaptic alpha blocking activity of a series of benzodioxanes.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; In Vitro Techniques; Male; Muscle Contraction; Phentolamine; Piperidines; Piperoxan; Rats; Synapses; Yohimbine | 1978 |
Proceedings: The effects of hypothalamic and reflexogenic hypertension on renal and femoral circulation.
Topics: Animals; Antihypertensive Agents; Atropine; Benzimidazoles; Blood Flow Velocity; Carotid Sinus; Clonidine; Dioxanes; Dogs; Electric Stimulation; Femoral Artery; Hypertension; Hypothalamus; Kidney; Piperidines; Pressoreceptors; Vagotomy | 1975 |
Presynaptic alpha-adenoceptors: the depression of self-stimulation by clonidine and its restoration by piperoxane but not by phentolamine or phenoxybenzamine.
Topics: Animals; Clonidine; Drug Interactions; Male; Phenoxybenzamine; Phentolamine; Piperidines; Piperoxan; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Self Stimulation; Stereotaxic Techniques; Synapses | 1977 |
Effect of piperoxane on rat plasma prolactin.
Topics: Animals; Clonidine; Dose-Response Relationship, Drug; Male; Piperidines; Piperoxan; Prolactin; Rats; Receptors, Adrenergic, alpha | 1978 |
Effect of piperoxane on serum prolactin: possible role of epinephrine-mediated synapses in the inhibition of prolactin secretion.
Topics: Animals; Clonidine; Epinephrine; Haplorhini; Male; Piperidines; Piperoxan; Prolactin; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Synapses | 1978 |
Binding to alpha-adrenergic receptors: differential pharmacological potencies and binding affinities of benzodioxanes.
Topics: Animals; Cerebral Cortex; Clonidine; Hydroxydopamines; Male; Muscle Contraction; Norepinephrine; Piperidines; Piperoxan; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Synaptosomes | 1979 |
Localization in the CNA of adrenoceptors which facilitate a cardioinhibitory reflex.
Topics: Adrenergic beta-Antagonists; Angiotensin II; Animals; Blood Pressure; Cerebellum; Clonidine; Decerebrate State; Depression, Chemical; Dioxanes; Dogs; Female; Heart; Heart Rate; Male; Medulla Oblongata; Piperidines; Propanolamines; Receptors, Adrenergic; Reflex; Vagus Nerve | 1975 |
Centrally induced hypotension unreleated to alpha-adrenergic stimulation.
Topics: Adrenergic alpha-Agonists; Animals; Arteries; Benzimidazoles; Blood Pressure; Clonidine; Depression, Chemical; Dioxanes; Dogs; Ear; Hypotension; Norepinephrine; Piperidines; Rabbits; Regional Blood Flow | 1975 |
Suppression of vasopressin secretion by clonidine: effect of alpha-adrenoceptor antagonists.
Topics: Animals; Blood Pressure; Clonidine; Dogs; Female; Heart Rate; Male; Phentolamine; Piperidines; Piperoxan; Vasopressins | 1979 |
Piperoxane reduces the effects of clonidine on aggression in mice and on noradrenaline dependent hypermotility in rats.
Topics: Aggression; Animals; Clonidine; Drug Antagonism; Female; Humans; Male; Mice; Motor Activity; Norepinephrine; Piperidines; Piperoxan; Rats; Tyramine | 1978 |
The effects of serotonergic and antiserotonergic drugs on the flexor reflex of spinal rat: a proposed model to evaluate the action on the central serotonin receptor.
Topics: 5-Hydroxytryptophan; Amphetamine; Animals; Anthracenes; Clonidine; Cyproheptadine; Decerebrate State; Fenfluramine; Hindlimb; Lysergic Acid Diethylamide; Male; Metergoline; Muscle Contraction; p-Chloroamphetamine; Piperidines; Rats; Reflex; Serotonin; Tryptophan | 1976 |
Interaction between centrally acting hypotensive drugs and tricyclic antidepressants.
Topics: Amphetamine; Animals; Antidepressive Agents, Tricyclic; Antihypertensive Agents; Benzimidazoles; Blood Pressure; Cats; Clonidine; Cocaine; Desipramine; Dioxanes; Drug Interactions; Ephedrine; Female; Male; Methyldopa; Piperidines; Reserpine | 1975 |
A benzodioxanhydroxyethylpiperidine derivative with an acute central hypotensive action, different from that of clonidine. A comparison with neuroleptic agents.
Topics: Animals; Antihypertensive Agents; Benzimidazoles; Blood Pressure; Cats; Clonidine; Dioxanes; Drug Interactions; Female; Male; Piperidines; Stellate Ganglion; Stereoisomerism; Sympathectomy; Time Factors; Tranquilizing Agents; Vagotomy; Yohimbine | 1975 |
Unusual mechanism of hypotensive activity exerted by erytrho-1-(1-[2-(1,4-benzodioxan-2-yl)-2-OH-ET-a1-4-piperidyl)-2-benzimidazolinone (R 28935).
Topics: Animals; Antihypertensive Agents; Benzimidazoles; Blood Pressure; Carotid Arteries; Clonidine; Dioxanes; Dogs; Electric Stimulation; Female; Hindlimb; Hypothalamus; Isoproterenol; Male; Norepinephrine; Piperidines; Pressoreceptors; Regional Blood Flow | 1975 |
Histamine H3-receptors inhibit sympathetic neurotransmission in guinea pig myocardium.
Topics: Animals; Chlorpheniramine; Clenbuterol; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; Guinea Pigs; Heart; Heart Atria; In Vitro Techniques; Methylhistamines; Nerve Endings; Norepinephrine; Phentolamine; Piperidines; Propranolol; Ranitidine; Receptors, Histamine; Receptors, Histamine H3; Sympathetic Nervous System; Synaptic Transmission | 1991 |
Alpha-adrenoceptor blocking properties of vesamicol.
Topics: Adrenergic alpha-Antagonists; Animals; Clonidine; Corticosterone; Desipramine; Dioxanes; Electric Stimulation; Idazoxan; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Piperidines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Stereoisomerism; Vas Deferens | 1991 |
Anti-muscarinic effect of alinidine on acetylcholine-induced vasodilation in isolated and perfused dog coronary arteries.
Topics: Acetylcholine; Animals; Carbachol; Clonidine; Coronary Vessels; Dogs; Female; In Vitro Techniques; Male; Parasympatholytics; Piperidines; Pirenzepine; Vasodilation | 1991 |
Age-related changes in rat serotonergic and adrenergic systems and in receptor responsiveness to subchronic desipramine treatment.
Topics: Aging; Animals; Brain; Clonidine; Desipramine; Dihydroalprenolol; Hydroxyindoleacetic Acid; Imipramine; Ketanserin; Kinetics; Male; Paroxetine; Piperidines; Prazosin; Proteins; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Serotonin; Serotonin; Time Factors | 1988 |
An examination of the putative sigma-receptor in the mouse isolated vas deferens.
Topics: Animals; Clonidine; Electric Stimulation; In Vitro Techniques; Male; Mice; Mice, Inbred DBA; Muscle Contraction; Muscle, Smooth; Naloxone; Piperidines; Receptors, Opioid; Receptors, sigma; Vas Deferens | 1989 |
Effect of methoxy substitution on the adrenergic activity of three structurally related alpha 2-adrenoreceptor antagonists.
Topics: Adrenergic alpha-Antagonists; Animals; Chemical Phenomena; Chemistry; Clonidine; Dioxanes; Dioxins; Imidazoles; Male; Mice; Muscle Contraction; Phenylephrine; Piperidines; Piperoxan; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Structure-Activity Relationship | 1986 |
Central alpha-2 adrenoceptor-mediated hypertensive response to clonidine in conscious, normotensive rats.
Topics: Animals; Azepines; Blood Pressure; Brain; Cimetidine; Clonidine; Hydroxydopamines; Injections, Intraventricular; Ketanserin; Male; Methoxamine; Oxidopamine; Piperidines; Prazosin; Procaine; Pyrilamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine | 1986 |
Serotonin-induced contraction of canine saphenous vein: mediation by 5-HT1 receptors.
Topics: Animals; Clonidine; Dogs; Drug Interactions; Emetics; In Vitro Techniques; Ketanserin; Mianserin; Muscle Contraction; Naphthols; Piperidines; Receptors, Serotonin; Saphenous Vein; Serotonin; Yohimbine | 1985 |
Effects of phenoxybenzamine, aceperone and clonidine on the level of 3-methoxy-4-hydroxyphenylglycol (MOPEG) in rat brain.
Topics: Acetamides; Animals; Antihypertensive Agents; Brain Chemistry; Butyrophenones; Chromatography, Gas; Clonidine; Glycols; Male; Methoxyhydroxyphenylglycol; Phenoxybenzamine; Piperidines; Rats | 1974 |
Studies of various amphetamines, apomorphine and clonidine on body temperature and brain 5-hydroxytryptamine metabolism in rats.
Topics: Amphetamine; Animals; Apomorphine; Behavior, Animal; Body Temperature; Brain; Brain Chemistry; Carboxylic Acids; Chromatography, Ion Exchange; Clonidine; Fever; Hydroxyindoleacetic Acid; Male; Methylphenidate; Naphthyridines; Phenmetrazine; Piperidines; Rats; Serotonin; Spectrometry, Fluorescence; Temperature | 1974 |
Possible involvement of central adrenaline neurons in vasomotor and respiratory control. Studies with clonidine and its interactions with piperoxane and yohimbine.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Brain; Cerebral Cortex; Clonidine; Dioxins; Epinephrine; Heart Rate; Male; Methyltyrosines; Neurons; Norepinephrine; Piperidines; Rats; Receptors, Adrenergic; Reflex; Respiration; Respiratory Center; Time Factors; Vasomotor System; Yohimbine | 1974 |
The cardiovascular effects of intraventricular clonidine and Bay 1470 in conscious hypertensive cats.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Cats; Clonidine; Desipramine; Dioxanes; Dopamine Antagonists; Haloperidol; Heart Rate; Hemodynamics; Hypertension, Renal; Phentolamine; Piperidines; Thiazines; Time Factors; Xylazine | 1974 |
Effects of piperoxane on sleep and waking in the rat. Evidence for increased waking by blocking inhibitory adrenaline receptors on the locus coeruleus.
Topics: Animals; Cerebral Ventricles; Clonidine; Dioxins; Electroencephalography; Electromyography; Epinephrine; Male; Norepinephrine; Piperidines; Rats; Receptors, Drug; Sleep; Stimulation, Chemical; Time Factors; Wakefulness | 1974 |
Release of brain dopamine as the probable mechanism for the hypothermic effect of D-amphetamine.
Topics: Animals; Apomorphine; Brain Chemistry; Clonidine; Dextroamphetamine; Dihydroxyphenylalanine; Dopamine; Drug Combinations; Glycolates; Haloperidol; Hydroxydopamines; Hypothermia; Male; Methysergide; Phenoxybenzamine; Pimozide; Piperidines; Propranolol; Pyrrolidines; Rats; Serotonin; Tyramine | 1972 |
Colonic secretion mediated by prostaglandin E2 and 5-hydroxytryptamine may contribute to diarrhea due to morphine withdrawal in the rat.
Topics: Animals; Atropine; Clonidine; Colon; Cyclic AMP; Diarrhea; Dinoprostone; Female; Humans; Indomethacin; Ketanserin; Morphine Dependence; Naloxone; Piperidines; Prostaglandins E; Rats; Rats, Inbred Strains; Serotonin; Substance Withdrawal Syndrome | 1984 |
Selectivity of benzodioxane alpha-adrenoceptor antagonists for alpha 1- and alpha 2-adrenoceptors determined by binding affinity.
Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Clonidine; In Vitro Techniques; Male; Membranes; Piperidines; Piperoxan; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic; Receptors, Adrenergic, alpha | 1983 |
Principles of therapy for congestive heart failure.
Topics: Calcium; Calcium Channel Blockers; Calmodulin; Cardiotonic Agents; Clonidine; Cyclic AMP; Cytosol; Digitalis Glycosides; Diuretics; Heart Failure; Humans; Ketanserin; Models, Cardiovascular; Muscle, Smooth, Vascular; Myocardium; Myosins; Piperidines; Receptors, Adrenergic, alpha; Vasodilator Agents | 1983 |
Evidence for an alpha-1 receptor-mediated central sympathoinhibitory action of ketanserin.
Topics: Animals; Blood Pressure; Brain; Cats; Clonidine; Heart Rate; Ketanserin; Piperidines; Receptors, Adrenergic, alpha; Serotonin Antagonists; Sympathetic Nervous System; Sympatholytics | 1984 |
Effects of clonidine, piperoxane and locus coeruleus lesion on the serotonergic and dopaminergic systems in raphe and caudate nucleus.
Topics: Animals; Caudate Nucleus; Clonidine; Dopamine; Hydroxydopamines; Locus Coeruleus; Male; Oxidopamine; Piperidines; Piperoxan; Raphe Nuclei; Rats; Rats, Inbred Strains; Receptors, Dopamine; Receptors, Serotonin; Serotonin | 1984 |
Further functional in vitro comparison of pre- and postsynaptic dopamine receptors in the rabbit caudate nucleus.
Topics: 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine; Acetylcholine; Animals; Apomorphine; Benzazepines; Caudate Nucleus; Choline; Clonidine; Female; Male; Piperidines; Rabbits; Receptors, Dopamine | 1983 |
Clinical efficacy of haloperidol, pimozide, penfluridol, and clonidine in the treatment of tourette syndrome.
Topics: Child; Child, Preschool; Clonidine; Haloperidol; Humans; Penfluridol; Pimozide; Piperidines; Tourette Syndrome | 1982 |
Effects of prazosin and piperoxan on central cardiovascular actions of St 91 in cats.
Topics: Animals; Atropine; Blood Pressure; Brain; Cats; Clonidine; Female; Heart Rate; Hemodynamics; Injections, Intra-Arterial; Injections, Intravenous; Male; Piperidines; Piperoxan; Prazosin; Quinazolines; Vertebral Artery | 1982 |
Release of endogenous acetylcholine from a vascularly perfused rat stomach in vitro; inhibition by M3 muscarinic autoreceptors and alpha-2 adrenoceptors.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Acetylcholine; Adrenergic alpha-Antagonists; Animals; Atropine; Calcium; Clonidine; Diamines; Drug Interactions; Electric Stimulation; Gastric Mucosa; Hexamethonium; Hexamethonium Compounds; Male; Muscarinic Antagonists; Oxotremorine; Parasympatholytics; Perfusion; Phenylephrine; Piperidines; Pirenzepine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Muscarinic; Stomach; Sympathetic Nervous System; Tetrodotoxin; Vagus Nerve | 1993 |
Role of external and internal calcium on heterocarrier-mediated transmitter release.
Topics: Acetylcholine; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Carrier Proteins; Chelating Agents; Choline; Clonidine; Dopamine; Dopamine Agonists; Egtazic Acid; Ergolines; GABA Modulators; Hippocampus; Male; Muscarinic Agonists; Neostriatum; Neuromuscular Depolarizing Agents; Neurons; Neurotransmitter Agents; Norepinephrine; Oxotremorine; Piperidines; Presynaptic Terminals; Quinpirole; Rats; Rats, Sprague-Dawley; Synaptosomes; Tritium; Yohimbine | 1996 |
Compounds possessing 5-HT3 receptor antagonistic activity inhibit intestinal propulsion in mice.
Topics: Adrenergic alpha-Agonists; Animals; Benzamides; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Cholinesterase Inhibitors; Cisapride; Clonidine; Gastrointestinal Transit; Intestines; Male; Mice; Mice, Inbred C57BL; Neostigmine; Ondansetron; Piperidines; Receptors, Serotonin; Serotonin Antagonists | 1996 |
Acute exercise enhances receptor-mediated endothelium-dependent vasodilation by receptor upregulation.
Topics: Acetylcholine; Adrenergic alpha-Agonists; Animals; Clonidine; Endothelium, Vascular; In Vitro Techniques; Male; Muscarinic Antagonists; Physical Conditioning, Animal; Piperidines; Rats; Rats, Wistar; Receptor, Muscarinic M3; Receptors, Adrenergic, alpha-2; Receptors, Muscarinic; Thoracic Arteries; Tritium; Up-Regulation; Vasodilation | 1999 |
Effect of epidural injection of prosidol with clonidine on the state of spinal cord and spinal ganglion.
Topics: Alkaline Phosphatase; Analgesics; Analgesics, Opioid; Animals; Capillaries; Clonidine; Dogs; Endothelium, Vascular; Ganglia; Nucleic Acids; Oxidation-Reduction; Piperidines; Protein Transport; Spinal Cord; Time Factors | 2001 |
Role of histamine H3 receptors in control of mouse intestinal motility in vivo and in vitro: comparison with alpha2-adrenoceptors.
Topics: Animals; Charcoal; Clonidine; Histamine Agonists; Histamine Antagonists; Idazoxan; Ileum; Imidazoles; In Vitro Techniques; Male; Methylhistamines; Mice; Peristalsis; Piperidines; Receptors, Adrenergic, alpha-2; Receptors, Histamine H3 | 2002 |
Pharmacologic interaction between cannabinoid and either clonidine or neostigmine in the rat formalin test.
Topics: Adrenergic alpha-Agonists; Analgesics; Animals; Antineoplastic Agents; Behavior, Animal; Benzoxazines; Cannabinoids; Cholinesterase Inhibitors; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Formaldehyde; Indoles; Injections, Spinal; Male; Morpholines; Naphthalenes; Neostigmine; Pain Measurement; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Receptors, Drug | 2003 |
Intrathecal clonidine inhibits mechanical allodynia via activation of the spinal muscarinic M1 receptor in streptozotocin-induced diabetic mice.
Topics: (4-(m-Chlorophenylcarbamoyloxy)-2-butynyl)trimethylammonium Chloride; Analgesics; Animals; Atropine; Blood Glucose; Clonidine; Diabetes Mellitus, Experimental; Diamines; Injections, Spinal; Male; Mice; Motor Activity; Muscarinic Agonists; Muscarinic Antagonists; Pain; Pain Threshold; Piperidines; Pirenzepine; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptor, Muscarinic M3; Spinal Cord; Streptozocin; Stress, Mechanical; Time Factors | 2004 |
[Open heart tricuspid valve replacement in a heroin addict Anaesthesiological management].
Topics: Adrenergic alpha-Agonists; Adult; Amides; Anesthesia, Epidural; Anesthesia, General; Anesthetics, Inhalation; Anesthetics, Intravenous; Anesthetics, Local; Anti-Inflammatory Agents, Non-Steroidal; Clonidine; Desflurane; Dipyrone; Female; Heart Valve Prosthesis Implantation; Heroin Dependence; Humans; Isoflurane; Pain, Postoperative; Piperidines; Propofol; Remifentanil; Ropivacaine; Tricuspid Valve | 2005 |
Chloroethylclonidine reveals that alpha (1 A)-adrenoceptors mediate contraction in aorta of alpha (1 D)-adrenoceptor knockout mice.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta; Clonidine; Dose-Response Relationship, Drug; Imines; In Vitro Techniques; Mice; Mice, Knockout; Norepinephrine; Piperazines; Piperidines; Receptors, Adrenergic, alpha-1; Vasoconstriction; Vasoconstrictor Agents | 2005 |
Spinal muscarinic and nicotinic subtypes activated by clonidine in postincisional pain.
Topics: Aconitine; Adrenergic alpha-Agonists; Animals; Behavior, Animal; Clonidine; Diamines; Dihydro-beta-Erythroidine; Injections, Spinal; Male; Muscarinic Agonists; Nicotinic Agonists; Pain; Piperidines; Rats; Rats, Sprague-Dawley; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptors, Muscarinic; Receptors, Nicotinic; Spine | 2005 |
Cannabinoids modulate spontaneous neuronal activity and evoked inhibition of locus coeruleus noradrenergic neurons.
Topics: Action Potentials; Adrenergic alpha-Agonists; Analysis of Variance; Animals; Benzoxazines; Calcium Channel Blockers; Cannabinoids; Clonidine; Dose-Response Relationship, Drug; Dronabinol; Locus Coeruleus; Male; Morpholines; Naphthalenes; Neural Inhibition; Neurons; Norepinephrine; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Rimonabant | 2006 |
The effects of opioids, local anesthetics and adjuvants on isolated pregnant rat uterine muscles.
Topics: Alfentanil; Amides; Analgesia, Obstetrical; Analgesics; Analgesics, Opioid; Anesthetics, Local; Animals; Bupivacaine; Clonidine; Dose-Response Relationship, Drug; Female; Isometric Contraction; Meperidine; Mepivacaine; Midazolam; Myometrium; Oxytocics; Oxytocin; Piperidines; Pregnancy; Rats; Rats, Wistar; Remifentanil; Ropivacaine; Uterine Contraction | 2007 |
Meperidine, remifentanil and tramadol but not sufentanil interact with alpha(2)-adrenoceptors in alpha(2A)-, alpha(2B)- and alpha(2C)-adrenoceptor knock out mice brain.
Topics: Adrenergic alpha-2 Receptor Agonists; Affinity Labels; Analgesics, Opioid; Animals; Autoradiography; Binding, Competitive; Brain; Clonidine; Drug Partial Agonism; Female; In Vitro Techniques; Male; Meperidine; Mice; Mice, Knockout; Piperidines; Radioligand Assay; Receptors, Adrenergic, alpha-2; Remifentanil; Sufentanil; Tramadol | 2008 |
Respiratory, metabolic and hemodynamic effects of clonidine in ventilated patients presenting with withdrawal syndrome.
Topics: Adrenergic alpha-Agonists; Adult; Calorimetry, Indirect; Carbon Dioxide; Clonidine; Electrocardiography; Energy Metabolism; Female; Hemodynamics; Humans; Hypertension; Hypnotics and Sedatives; Male; Oxygen Consumption; Piperidines; Propofol; Prospective Studies; Remifentanil; Respiration, Artificial; Respiratory Insufficiency; Rest; Substance Withdrawal Syndrome; Tachycardia; Ventilator Weaning | 2009 |
Neurokinin-1 receptor antagonists modulate brain noradrenaline and serotonin interactions.
Topics: Adrenergic alpha-Agonists; Animals; Biphenyl Compounds; Clonidine; Drug Administration Schedule; Electrophysiology; Hypnotics and Sedatives; Locus Coeruleus; Male; Neurokinin-1 Receptor Antagonists; Neurons; Norepinephrine; Piperidines; Raphe Nuclei; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT1A; Serotonin | 2008 |
Simultaneous telemetric monitoring of tail-skin and core body temperature in a rat model of thermoregulatory dysfunction.
Topics: Adrenergic alpha-Agonists; Animals; Body Temperature; Body Temperature Regulation; Clonidine; Disease Models, Animal; Estradiol; Estrogens; Female; Fluorobenzenes; Monitoring, Physiologic; Ovariectomy; Piperidines; Rats; Rats, Sprague-Dawley; Serotonin Antagonists; Skin Temperature; Tail; Telemetry; Time Factors | 2009 |
[Current and future medical drugs for smoking cessation].
Topics: Adrenergic alpha-Agonists; Antidepressive Agents; Behavior Therapy; Benzazepines; Bupropion; Cannabinoid Receptor Antagonists; Clinical Trials as Topic; Clonidine; Combined Modality Therapy; Counseling; Humans; Nicotine; Nicotinic Agonists; Nortriptyline; Piperidines; Pyrazoles; Quinoxalines; Rimonabant; Smoking Cessation; Tobacco Use Disorder; Vaccines; Varenicline | 2009 |
Metaplasticity of hypothalamic synapses following in vivo challenge.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Animals, Newborn; Biophysics; Carbolines; Clonidine; Down-Regulation; Drug Interactions; Egtazic Acid; Electric Stimulation; Excitatory Amino Acid Agents; Excitatory Postsynaptic Potentials; Glutamic Acid; Guanosine Diphosphate; Hypothalamus; In Vitro Techniques; Intracranial Hemorrhages; Long-Term Synaptic Depression; Male; Microinjections; Neurons; Patch-Clamp Techniques; Piperidines; Pyrazoles; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Receptors, Metabotropic Glutamate; Synapses; Thionucleotides; Yohimbine | 2009 |
Rimonabant-induced Delta9-tetrahydrocannabinol withdrawal in rhesus monkeys: discriminative stimulus effects and other withdrawal signs.
Topics: Adrenergic Agonists; Animals; Behavior, Animal; Benzoxazines; Cannabinoid Receptor Agonists; Cannabinoid Receptor Antagonists; Clonidine; Cyclohexanols; Discrimination, Psychological; Dronabinol; Female; Heart Rate; Macaca mulatta; Male; Morpholines; Motor Activity; Naphthalenes; Piperidines; Pyrazoles; Rimonabant; Substance Withdrawal Syndrome | 2010 |
Current treatment options in smoking cessation.
Topics: Adrenergic alpha-Agonists; Antidepressive Agents; Behavior Therapy; Benzazepines; Bupropion; Clonidine; Combined Modality Therapy; Counseling; Humans; Nicotine; Nicotinic Agonists; Nortriptyline; Patient Selection; Piperidines; Practice Guidelines as Topic; Pyrazoles; Quinoxalines; Rimonabant; Self-Help Groups; Smoking Cessation; Tobacco Use Disorder; United States; Vaccines; Varenicline | 2010 |
Endothelin modulates the cardiovascular effects of clonidine in the rat.
Topics: Adrenergic alpha-2 Receptor Agonists; Animals; Antihypertensive Agents; Aorta, Abdominal; Blood Gas Analysis; Blood Pressure; Brain; Clonidine; Endothelins; Heart Rate; Male; Oligopeptides; Peptide Fragments; Piperidines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Endothelin; Vasoconstriction | 2010 |
Clonidine-induced growth hormone and growth-hormone-releasing hormone release is mediated by tachykinin NK2 receptors in sheep.
Topics: Adrenergic alpha-Agonists; Animals; Benzamides; Clonidine; Growth Hormone; Growth Hormone-Releasing Hormone; Male; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Sheep | 2012 |
The role of α₂-adrenoceptors in the anti-convulsant effects of cannabinoids on pentylenetetrazole-induced seizure threshold in mice.
Topics: Animals; Anticonvulsants; Arachidonic Acids; Cannabinoids; Clonidine; Dose-Response Relationship, Drug; Drug Interactions; Male; Mice; Pentylenetetrazole; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Receptors, Adrenergic, alpha-2; Seizures; Yohimbine | 2013 |
Scalp blocks in nonsyndromic craniosynostosis surgery - a retrospective case series review.
Topics: Analgesics; Anesthetics, Inhalation; Anesthetics, Intravenous; Anesthetics, Local; Bupivacaine; Child; Child, Preschool; Clonidine; Craniosynostoses; Female; Humans; Infant; Male; Methyl Ethers; Nerve Block; Nitrous Oxide; Piperidines; Propofol; Remifentanil; Retrospective Studies; Scalp; Sevoflurane | 2014 |
Thalamic nucleus reuniens regulates fear memory destabilization upon retrieval.
Topics: Amygdala; Animals; Anisomycin; CA1 Region, Hippocampal; Clonidine; Cognition; Cysteine Proteinase Inhibitors; Early Growth Response Protein 1; Excitatory Amino Acid Antagonists; Fear; GABA-A Receptor Agonists; Lactones; Memory; Midline Thalamic Nuclei; Muscimol; Neurons; Piperidines; Prefrontal Cortex; Rats; Receptors, N-Methyl-D-Aspartate | 2020 |