clonidine and naphazoline

clonidine has been researched along with naphazoline in 37 studies

Research

Studies (37)

TimeframeStudies, this research(%)All Research%
pre-199027 (72.97)18.7374
1990's7 (18.92)18.2507
2000's2 (5.41)29.6817
2010's1 (2.70)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Andrews, PR; Craik, DJ; Martin, JL1
Batink, H; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
de Jonge, A; Lam, E; Slothorst-Grisdijk, FP; Timmermans, PB; van Meel, JC; van Zwieten, PA1
Timmermans, PB; van Zwieten, PA1
Agbaba, D; Filipic, S; Nikolic, K1
Kobinger, W; Pichler, L2
Bianchi, L; Florio, V; Lonogo, VG1
Endoh, M; Schümann, HJ1
Doxey, JC; Everitt, J1
Armbruster, H; Beckerhoff, R; Reck, G; Siegenthaler, W; Vetter, W1
Alexandre, JM; Chevillard, C; Duchene, N; Pasquier, R1
Rolls, ET; Shaw, SG1
Abe, K; Nishiura, T; Okina, A; Shibaike, S1
Chandranath, SI; Gokhale, SD; Sharif, SI1
Rattan, S; Yamato, S1
Booth, TF1
Hashimoto, H; Nakashima, M; Sogabe, K1
Kaliszan, R; Petrusewicz, J1
Macedo, TA; Ribeiro, CA1
Evans, PD; Reale, V; Villegas, J1
Bueno, L; Fargeas, MJ; Fioramonti, J1
Hashemzadeh, H; Hollingworth, RM; Voliva, A1
Schmitt, H; Tsoucaris-Kupfer, D1
Kobinger, W; Walland, A1
Le Douarec, JC; Petillot, N; Schmitt, H1
Jones, DJ; McKenna, LF1
Castaldi, WR; Fazio, JK; Hennig, CW; Hughes, CA; Spencer, BD1
Jarrott, B; Louis, WJ; Summers, RJ1
Agrawal, DK; Daniel, EE; Triggle, CR1
Marwaha, J1
Brown, CM; MacKinnon, AC; Olverman, HJ; Spedding, M; Stewart, M1
Belcourt, A; Bousquet, P; Bricca, G; Dontenwill, M; Greney, H; Stutzmann, J; Zhang, J1
Gorzalka, BB; Meston, CM; Moe, IV1
Chikkala, DN; Piletz, JE; Zhu, H1
Baldwin, J; Chang, CH; Ernsberger, P; Gold, G; Ivanov, TR; Jones, JC; Pickard, RT; Piletz, JE; Reis, DJ; Roth, B; Sharp, JD; Zhu, H1
Hamasaki, T; Huang, J; Ozoe, Y1

Reviews

1 review(s) available for clonidine and naphazoline

ArticleYear
alpha 2 adrenoceptors: classification, localization, mechanisms, and targets for drugs.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:12

    Topics: Adipose Tissue; Animals; Blood Platelets; Central Nervous System; Humans; Islets of Langerhans; Melanocytes; Muscle, Smooth, Vascular; Nerve Endings; Norepinephrine; Parasympathetic Nervous System; Radioligand Assay; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Serotonin; Synapses

1982

Other Studies

36 other study(ies) available for clonidine and naphazoline

ArticleYear
Functional group contributions to drug-receptor interactions.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:12

    Topics: Animals; Calorimetry; Kinetics; Models, Biological; Protein Binding; Receptors, Cell Surface; Receptors, Drug; Structure-Activity Relationship

1984
Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and antagonists.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cell Membrane; Clonidine; Kinetics; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Vasoconstriction

1984
Characterization of alpha-adrenoceptor populations. Quantitative relationships between cardiovascular effects initiated at central and peripheral alpha-adrenoceptors.
    Journal of medicinal chemistry, 1981, Volume: 24, Issue:5

    Topics: Animals; Blood Pressure; Blood Vessels; Brain; Hemodynamics; Male; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha

1981
QSAR study of imidazoline antihypertensive drugs.
    Bioorganic & medicinal chemistry, 2008, Aug-01, Volume: 16, Issue:15

    Topics: Antihypertensive Agents; Binding Sites; Imidazoline Receptors; Imidazolines; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship

2008
Investigation into some imidazoline compounds, with respect to peripheral alpha-adrenoceptor stimulation and depression of cardiovascular centers.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 291, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Atropine; Blood Pressure; Brain; Cats; Clonidine; Dogs; Female; Heart Rate; Imidazoles; Imidazolidines; Male; Naphazoline; Oxymetazoline; Pressoreceptors; Rats; Receptors, Adrenergic; Reflex; Vagotomy; Vagus Nerve; Vasomotor System; Xylazine

1975
A study of the central effects of sympathomimetic drugs: EEG and behavioural investigations on clonidine and naphazoline.
    Neuropharmacology, 1975, Volume: 14, Issue:10

    Topics: Adrenergic alpha-Antagonists; Amphetamine; Animals; Behavior, Animal; Cats; Clonidine; Cortical Synchronization; Electrodes, Implanted; Electroencephalography; Imidazoles; Male; Methyltyrosines; Naphazoline; Rabbits; Rats; Reserpine

1975
alpha-Adrenoceptors in the ventricular myocardium: clonidine, naphazoline and methoxamine as partial alpha-agonists exerting a competitive dualism in action to phenylephrine.
    European journal of pharmacology, 1976, Volume: 36, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Heart; Heart Ventricles; Imidazoles; In Vitro Techniques; Methoxamine; Naphazoline; Papillary Muscles; Phentolamine; Phenylephrine; Pindolol; Rabbits; Receptors, Adrenergic; Stimulation, Chemical

1976
Inhibitory effects of clonidine on responses to sympathetic nerve stimulation in the pithed rat.
    British journal of pharmacology, 1977, Volume: 61, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Eyelids; Heart Rate; Male; Muscle Contraction; Naphazoline; Phentolamine; Pressoreceptors; Rats; Sympathetic Nervous System; Synaptic Transmission; Vas Deferens

1977
Severe arterial hypertension caused by chronical abuse of a topical mineralocorticoid.
    International journal of clinical pharmacology and biopharmacy, 1975, Volume: 12, Issue:1-2

    Topics: Adult; Aldosterone; Clonidine; Drug Combinations; Drug Therapy, Combination; Female; Fluprednisolone; Humans; Hypertension; Isomerism; Methyldopa; Naphazoline; Nasal Decongestants; Potassium; Renin; Spironolactone; Substance-Related Disorders; Time Factors; Triamterene

1975
Mechanism of inhibition of renin release by clonidine in rats.
    European journal of pharmacology, 1978, Apr-15, Volume: 48, Issue:4

    Topics: Animals; Blood Pressure; Cisterna Magna; Clonidine; Injections, Intravenous; Male; Naphazoline; Rats; Renin

1978
Is the release of noradrenaline necessary for self-stimulation of the brain?
    Pharmacology, biochemistry, and behavior, 1976, Volume: 4, Issue:4

    Topics: Amphetamine; Animals; Benserazide; Bis(4-Methyl-1-Homopiperazinylthiocarbonyl)disulfide; Brain; Clonidine; Disulfiram; Levodopa; Male; Naphazoline; Nerve Endings; Norepinephrine; Oxymetazoline; Phenylephrine; Rats; Receptors, Drug; Reserpine; Self Stimulation

1976
Proceedings: Central nervous cardiovascular depression, a potential action of alpha-adrenoceptors stimulating imidazoline derivatives.
    Naunyn-Schmiedeberg's archives of pharmacology, 1975, Volume: 287 Suppl

    Topics: Animals; Cardiovascular System; Cats; Clonidine; Dogs; Imidazoles; Medulla Oblongata; Naphazoline; Oxymetazoline

1975
The effects of clonidine and three 2-imidazoline derivatives on the secretion of protein and some electrolytes by rat submandibular and parotid glands.
    Comparative biochemistry and physiology. C, Comparative pharmacology and toxicology, 1992, Volume: 101, Issue:3

    Topics: Animals; Autonomic Nervous System; Clonidine; Electrolytes; Imidazoles; Male; Naphazoline; Parotid Gland; Rats; Rats, Inbred Strains; Salivary Proteins and Peptides; Submandibular Gland

1992
Pharmacological characterization of the postjunctional alpha-adrenoceptors of the rat isolated seminal vesicle.
    Naunyn-Schmiedeberg's archives of pharmacology, 1990, Volume: 341, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Male; Naphazoline; Norepinephrine; Oxymetazoline; Phenoxybenzamine; Phentolamine; Phenylephrine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Seminal Vesicles; Yohimbine

1990
Role of alpha adrenoceptors in opossum internal anal sphincter.
    The Journal of clinical investigation, 1990, Volume: 86, Issue:2

    Topics: Anal Canal; Animals; Clonidine; Muscle Contraction; Naphazoline; Opossums; Phenylephrine; Prazosin; Receptors, Adrenergic, alpha; Yohimbine

1990
Effects of biogenic amines and adrenergic drugs on oviposition in the cattle tick Boophilus: evidence for octopaminergic innervation of the oviduct.
    Experimental & applied acarology, 1989, Volume: 7, Issue:4

    Topics: Adrenergic Agonists; Animals; Arecoline; Biogenic Amines; Cattle; Clonidine; Female; Naphazoline; Octopamine; Oviposition; Pilocarpine; Receptors, Adrenergic; Receptors, Biogenic Amine; Reserpine; Ticks; Tolazoline

1989
Affinities of adrenergic drugs for alpha 2-adrenoceptors in dog saphenous vein in comparison with those in rat brain or human platelets.
    Blood vessels, 1985, Volume: 22, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Blood Platelets; Brain; Clonidine; Dogs; Epinephrine; Guanabenz; Humans; Naphazoline; Norepinephrine; Phentolamine; Phenylephrine; Propranolol; Rats; Receptors, Adrenergic, alpha; Saphenous Vein; Tolazoline; Tritium; Yohimbine

1985
Effect of imidazoline drugs on human blood platelet aggregation.
    Thrombosis and haemostasis, 1985, Dec-17, Volume: 54, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Antazoline; Clonidine; Humans; Imidazoles; In Vitro Techniques; Naphazoline; Phentolamine; Platelet Aggregation; Tolazoline

1985
Pharmacological characterization of the postsynaptic alpha-adrenoceptors in human uterine artery.
    The Journal of pharmacy and pharmacology, 1986, Volume: 38, Issue:8

    Topics: Arteries; Clonidine; Drug Interactions; Female; Humans; Kinetics; Naphazoline; Norepinephrine; Phenylephrine; Prazosin; Receptors, Adrenergic, alpha; Uterus; Vasoconstriction; Yohimbine

1986
Octopaminergic modulation of the membrane potential of the Schwann cell of the squid giant nerve fibre.
    The Journal of experimental biology, 1986, Volume: 121

    Topics: Amines; Animals; Axons; Carbachol; Clonidine; Cyclic AMP; Decapodiformes; Membrane Potentials; Naphazoline; Octopamine; Phentolamine; Receptors, Adrenergic; Receptors, Biogenic Amine; Receptors, Nicotinic; Schwann Cells; Structure-Activity Relationship; Tyramine

1986
Central alpha 2-adrenergic control of the pattern of small intestinal motility in rats.
    Gastroenterology, 1986, Volume: 91, Issue:6

    Topics: Animals; Clonidine; Duodenum; Eating; Electromyography; Fasting; Gastrointestinal Motility; Jejunum; Male; Naphazoline; Phentolamine; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1986
Receptors for 3H-octopamine in the adult firefly light organ.
    Life sciences, 1985, Aug-05, Volume: 37, Issue:5

    Topics: Animals; Binding Sites; Binding, Competitive; Chlorphenamidine; Clonidine; Coleoptera; Guanosine Triphosphate; Male; Naphazoline; Octopamine; Phentolamine; Propranolol; Receptors, Adrenergic; Receptors, Biogenic Amine; Synephrine

1985
Hypothermic effect of alpha-sympathomimetic agents and their antagonism by adrenergic and cholinergic blocking drugs.
    Neuropharmacology, 1972, Volume: 11, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Aniline Compounds; Animals; Body Temperature; Cerebral Ventricles; Clonidine; Dose-Response Relationship, Drug; Hypothalamus; Injections; Injections, Intraperitoneal; Naphazoline; Oxazoles; Oxymetazoline; Parasympatholytics; Rats; Stereotaxic Techniques; Sympatholytics; Thiazines; Time Factors; Toluidines; Xylenes

1972
Evidence for a central activation of a vagal cardiodepressor reflex by clonidine.
    European journal of pharmacology, 1972, Volume: 19, Issue:2

    Topics: Adrenergic beta-Antagonists; Angiotensin II; Atropine; Blood Pressure; Bradycardia; Central Nervous System; Clonidine; Electrocardiography; Gallamine Triethiodide; Guanethidine; Heart Rate; Naphazoline; Neuromuscular Depolarizing Agents; Norepinephrine; Vagus Nerve

1972
Antinociceptive effects of some alpha-sympathomimetic agents.
    Neuropharmacology, 1974, Volume: 13, Issue:5

    Topics: Analgesics; Aniline Compounds; Animals; Behavior, Animal; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Escape Reaction; Imidazoles; Injections, Intraperitoneal; Naphazoline; Naphthalenes; Oxazoles; Oxymetazoline; Rats; Reaction Time; Reflex, Startle; Sympathomimetics; Tetrazoles; Thiazines; Toluidines; Vocalization, Animal

1974
Alpha adrenergic receptor mediated formation of cyclic AMP in rat spinal cord.
    Journal of cyclic nucleotide research, 1980, Volume: 6, Issue:2

    Topics: 4-(3-Butoxy-4-methoxybenzyl)-2-imidazolidinone; Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Clonidine; Cyclic AMP; Male; Methoxamine; Naphazoline; Oxymetazoline; Phenylephrine; Rats; Spinal Cord

1980
Duration of tonic immobility in chickens as a function of alpha-adrenergic receptor stimulation and blockade.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 20, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Behavior, Animal; Chickens; Clonidine; Guanfacine; Guanidines; Methoxamine; Naphazoline; Phenylacetates; Phenylephrine; Prazosin; Restraint, Physical; Time Factors; Yohimbine

1984
Selectivity of a series of clonidine-like drugs for alpha 1 and alpha 2 adrenoceptors in rat brain.
    Neuroscience letters, 1980, Volume: 20, Issue:3

    Topics: Aniline Compounds; Animals; Cerebral Cortex; Clonidine; Guanabenz; Guanfacine; Guanidines; Imidazoles; In Vitro Techniques; Indoramin; Naphazoline; Oxazoles; Phenylacetates; Prazosin; Rats; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Thiophenes; Toluidines

1980
Pharmacological characterization of the postsynaptic alpha adrenoceptors in vascular smooth muscle from canine and rat mesenteric vascular beds.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 229, Issue:3

    Topics: Animals; Clonidine; Dose-Response Relationship, Drug; Hydroxydopamines; Muscle, Smooth, Vascular; Naphazoline; Oxidopamine; Phenylephrine; Prazosin; Receptors, Adrenergic, alpha; Splanchnic Circulation; Yohimbine

1984
Supersensitivity of analgesic responses to alpha 2-adrenergic agonists in genetically hypertensive rats.
    Brain research, 1984, Jun-25, Volume: 304, Issue:2

    Topics: Animals; Clonidine; Hypertension; Male; Naphazoline; Pain; Prazosin; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Yohimbine

1984
[3H]p-aminoclonidine and [3H]idazoxan label different populations of imidazoline sites on rat kidney.
    European journal of pharmacology, 1993, Feb-23, Volume: 232, Issue:1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Dioxanes; Guanosine Triphosphate; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isoquinolines; Kidney; Male; Naphazoline; Naphthyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Drug; Tritium

1993
Human brain imidazoline receptors: further characterization with [3H]clonidine.
    European journal of pharmacology, 1994, Jan-01, Volume: 266, Issue:1

    Topics: Binding, Competitive; Brain Stem; Clonidine; Guanylyl Imidodiphosphate; Humans; Imidazoline Receptors; In Vitro Techniques; Naphazoline; Receptors, Adrenergic, alpha; Receptors, Drug

1994
Effects of sympathetic inhibition on receptive, proceptive, and rejection behaviors in the female rat.
    Physiology & behavior, 1996, Volume: 59, Issue:3

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Animals; Clonidine; Female; Guanethidine; Male; Naphazoline; Norepinephrine; Ovariectomy; Posture; Rats; Sexual Behavior, Animal; Sympathetic Nervous System; Sympatholytics

1996
Comparison of ligand binding affinities at human I1-imidazoline binding sites and the high affinity state of alpha-2 adrenoceptor subtypes.
    The Journal of pharmacology and experimental therapeutics, 1996, Volume: 279, Issue:2

    Topics: Animals; Binding Sites; Binding, Competitive; Blood Platelets; CHO Cells; Clonidine; Cricetinae; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Imidazoline Receptors; Naphazoline; Radioligand Assay; Receptors, Adrenergic, alpha-2; Receptors, Drug

1996
Imidazoline receptor antisera-selected (IRAS) cDNA: cloning and characterization.
    DNA and cell biology, 2000, Volume: 19, Issue:6

    Topics: Amino Acid Motifs; Amino Acid Sequence; Animals; Blotting, Western; CHO Cells; Clonidine; Cloning, Molecular; COS Cells; Cricetinae; DNA, Complementary; Epinephrine; Humans; Idazoxan; Imidazoles; Imidazoline Receptors; Immune Sera; Iodine Radioisotopes; Molecular Sequence Data; Naphazoline; Receptors, Drug; Ruthenium Red; Sequence Tagged Sites; Staining and Labeling; Transfection; Yohimbine

2000
Pharmacological characterization of a Bombyx mori alpha-adrenergic-like octopamine receptor stably expressed in a mammalian cell line.
    Archives of insect biochemistry and physiology, 2010, Volume: 73, Issue:2

    Topics: Amidines; Animals; Bombyx; Calcium; Cell Line; Chlorpromazine; Clonidine; Cyclic AMP; Imidazolidines; Insect Proteins; Insecticides; Mammals; Naphazoline; Receptors, Adrenergic, alpha; Receptors, Biogenic Amine; Tolazoline; Yohimbine

2010