clonidine and cirazoline

clonidine has been researched along with cirazoline in 63 studies

Research

Studies (63)

TimeframeStudies, this research(%)All Research%
pre-199027 (42.86)18.7374
1990's20 (31.75)18.2507
2000's13 (20.63)29.6817
2010's2 (3.17)24.3611
2020's1 (1.59)2.80

Authors

AuthorsStudies
Batink, H; de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Esbenshade, TA; Han, C; Hollinger, S; Minneman, KP; Theroux, TL1
Arrault, A; Guillaumet, G; Mérour, JY; Pfeiffer, B; Renard, P; Rettori, MC; Scalbert, E; Touzeau, F1
Agbaba, D; Filipic, S; Nikolic, K1
Elhawary, AM; Pettinger, WA; Wolff, DW1
Tabrizchi, R; Triggle, CR2
Schwietert, HR; van Zwieten, PA; Wilffert, B; Wilhelm, D1
Armah, BI; Göthert, M; Molderings, GJ1
de Jonge, A; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Dabiré, H; Mouille, P; Schmitt, H1
Horng, JS; Messick, K; Ruffolo, RR1
Kodama, CK; Menon, MK1
de Jonge, A; Qian, JQ; Thoolen, MJ; Timmermans, PB; van den Berg, G; van Zwieten, PA; Wilffert, B1
Bou, J; Massingham, R1
Herman, G; Mauduit, P; Rossignol, B1
Chiu, AT; McCall, DE; Thoolen, MJ; Timmermans, PB1
Collin, JP; Voisin, P1
Dinovo, EC; Haddox, VG; Menon, MK1
de Jonge, A; Mathy, MJ; Thoolen, MJ; Timmermans, PB; van Zwieten, PA; Wilffert, B1
Mottram, DR; Saggar, P1
Hong, KW; Jung, HO1
Cooke, JP; Flavahan, NA; Rimele, TJ; Vanhoutte, PM1
Cavero, I; Gomeni, R; Lefèvre-Borg, F; Roach, AG; Scatton, B1
Curtis-Prior, PB; Tan, S2
Aarhus, LL; Rimele, TJ; Rooke, TW; Vanhoutte, PM1
Cavero, I; Doxey, JC; Roach, AG; Strachan, DA1
de Jonge, A; Kalkman, HO; Mathy, MJ; Thoolen, MJ; Timmermans, PB; van Meel, JC; van Zwieten, PA; Wilffert, B1
Docherty, JR; McGrath, JC1
Bousquet, P; Feldman, J; Schwartz, J1
Dabiré, H; Joly, G; Lucet, B; Mouillé, P; Schmitt, H1
Lues, I; Schümann, HJ1
Dabiré, H; Joly, G; Mouillé, P; Schmitt, H1
Dubocovich, ML; Langer, SZ; Massingham, R1
Hescheler, J; Krautwurst, D; Musgrave, IF; Schultz, G1
Haque, M; Kulkarni, RN; MacDermot, J; Olmos, G1
García-Sevilla, JA; Pineda, J; Ugedo, L1
Belcourt, A; Bousquet, P; Bricca, G; Dontenwill, M; Greney, H; Stutzmann, J; Zhang, J1
Fröhlich, R; Illes, P; Szabo, B1
Beenen, OH; Pfaffendorf, M; van Zwieten, PA1
Beenen, OH; Mathy, MJ; Pfaffendorf, M; van Zwieten, PA2
Czerwiec, E; De Backer, JP; Flamez, A; Vauquelin, G1
Fink, K; Göthert, M; Kathmann, M; Molderings, GJ; Schlicker, E1
Bousquet, P; Dontenwill, M; Ehrhardt, JD; Greney, H; Molines, A; Senecheau, P1
De Backer, JP; Flamez, A; Gillard, M; Noyer, M; Vauquelin, G1
Mita, M; Walsh, MP1
Alvarez-Guerra, M; Bertholom, N; Garay, RP1
Gaivin, RJ; Gonzalez-Cabrera, P; Perez, DM; Ross, SA; Waugh, DJ; Yun, J; Zuscik, MJ1
de Vries, J; Kawahara, Y; Pudovkina, OL; Westerink, BH1
Bönisch, H; Brüss, M; Göthert, M; Hammermann, R; Molderings, GJ1
Cremers, TI; Pudovkina, OL; Westerink, BH1
Raasmaja, A; Römer, L; Savola, JM; Wurster, S1
Halaris, A; Piletz, JE; Zhu, H1
Cardin, JA; Schmidt, MF1
Kim, SH; Kim, SW; Park, WH; Rhee, KS; Yuan, K1
Bellantuono, V; Cassano, G; Lippe, C1
Centurión, D; Cobos-Puc, LE; Márquez-Conde, JA; Monroy-Ordoñez, EB; Sánchez-López, A; Villalón, CM1
Bruzzone, A; Cardinaletti, C; Del Bello, F; Ghelfi, F; Giannella, M; Mattioli, L; Paris, H; Perfumi, M; Piergentili, A; Pigini, M; Quaglia, W1
Fälting, JM; Holmström, TE; Mattsson, CL; Nedergaard, J; Wang, Y1
Bakshi, VP; Barth, KJ; Ciucci, MR; Grant, LM; Kelm-Nelson, CA; Muslu, C1
Feng, HJ; Niu, J; Tan, Z; Zhang, R1

Other Studies

63 other study(ies) available for clonidine and cirazoline

ArticleYear
Quantitative relationships between alpha-adrenergic activity and binding affinity of alpha-adrenoceptor agonists and antagonists.
    Journal of medicinal chemistry, 1984, Volume: 27, Issue:4

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Blood Pressure; Brain; Cell Membrane; Clonidine; Kinetics; Prazosin; Quinazolines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship; Vasoconstriction

1984
Selectivity of agonists for cloned alpha 1-adrenergic receptor subtypes.
    Molecular pharmacology, 1994, Volume: 46, Issue:5

    Topics: Adrenergic alpha-1 Receptor Agonists; Animals; Binding, Competitive; Catecholamines; Cattle; Cell Line; Cloning, Molecular; Cricetinae; Humans; Imidazoles; Inositol Phosphates; Phenethylamines; Phenoxybenzamine; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Tetralones

1994
Synthesis and biological evaluation of new 2-(4,5-dihydro-1H-imidazol-2-yl)-3,4-dihydro-2H-1,4-benzoxazine derivatives.
    Journal of medicinal chemistry, 2003, May-08, Volume: 46, Issue:10

    Topics: Adrenal Medulla; Animals; Antihypertensive Agents; Binding Sites; Blood Pressure; Cattle; Frontal Lobe; Heart Rate; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Kidney; Oxazines; Rabbits; Radioligand Assay; Rats; Rats, Inbred SHR; Rats, Wistar; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Stereoisomerism; Structure-Activity Relationship

2003
QSAR study of imidazoline antihypertensive drugs.
    Bioorganic & medicinal chemistry, 2008, Aug-01, Volume: 16, Issue:15

    Topics: Antihypertensive Agents; Binding Sites; Imidazoline Receptors; Imidazolines; Ligands; Models, Molecular; Molecular Structure; Quantitative Structure-Activity Relationship

2008
Subtype-selective alpha-1 adrenoceptor alkylation in the rat kidney and its effect on the vascular pressor response.
    The Journal of pharmacology and experimental therapeutics, 1992, Volume: 260, Issue:2

    Topics: Adrenergic alpha-Antagonists; Alkylation; Animals; Clonidine; Imidazoles; Kidney; Male; Methoxamine; Phenylephrine; Prazosin; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Renal Artery

1992
The interrelationship between the effects of captopril and nifedipine on pressor responses elicited by selective alpha-adrenoceptor agonists in the pithed rat preparation.
    Journal of cardiovascular pharmacology, 1992, Volume: 19, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Azepines; Blood Pressure; Captopril; Clonidine; Decerebrate State; Imidazoles; Male; Nifedipine; Rats; Rats, Inbred Strains

1992
Differences between full and partial alpha-adrenoceptor agonists in eliciting phasic and tonic types of responses in the longitudinal smooth muscle of the rat portal vein.
    Naunyn-Schmiedeberg's archives of pharmacology, 1991, Volume: 344, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium; Clonidine; Imidazoles; In Vitro Techniques; Male; Muscle, Smooth, Vascular; Phenoxybenzamine; Portal Vein; Quinoxalines; Rats; Receptors, Adrenergic, alpha; Vasoconstriction

1991
Effects of staurosporine on the pressor responses to alpha-adrenoceptor agonists in pithed rats: a comparison with nifedipine.
    Pharmacology, 1991, Volume: 43, Issue:3

    Topics: Adrenergic alpha-Agonists; Alkaloids; Animals; Azepines; Blood Pressure; Clonidine; Decerebrate State; Imidazoles; Male; Muscle, Smooth, Vascular; Nifedipine; Protein Kinase C; Rats; Rats, Inbred Strains; Staurosporine

1991
Effect of temperature on alpha 2- and alpha 1-adrenoceptor-mediated responses in the pithed rat and in the rat vena cava.
    Journal of autonomic pharmacology, 1990, Volume: 10, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Clonidine; Cold Temperature; Dose-Response Relationship, Drug; Imidazoles; Male; Norepinephrine; Phenylephrine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Neurotransmitter; Temperature; Tritium; Tyramine; Vena Cava, Inferior

1990
Calcium dependency of vasoconstriction mediated by alpha 1- and alpha 2-adrenoceptors.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Azepines; Blood Pressure; Calcium; Calcium Channel Blockers; Clonidine; Imidazoles; Ion Channels; Nifedipine; Rats; Receptors, Adrenergic, alpha; Regional Blood Flow; Structure-Activity Relationship; Vasoconstriction

1985
(Imidazolinyl-2)-2-benzodioxane 1-4 (idazoxan) and its stereoisomers, new alpha 2-antagonists.
    Journal of cardiovascular pharmacology, 1985, Volume: 7 Suppl 6

    Topics: Animals; Azepines; Chickens; Clonidine; Dioxanes; Dioxins; Heart Rate; Idazoxan; Imidazoles; Male; Mice; Muscle Contraction; Rats; Receptors, Adrenergic, alpha; Stereoisomerism; Structure-Activity Relationship; Vas Deferens

1985
Interactions of dimethoxy-substituted tolazoline derivatives with alpha 1- and alpha 2-adrenoreceptors in vitro.
    Journal of autonomic pharmacology, 1985, Volume: 5, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Aorta; Brain; Brimonidine Tartrate; Clonidine; Dioxanes; Electric Stimulation; Guinea Pigs; Ileum; Imidazoles; In Vitro Techniques; Male; Muscle, Smooth; Muscle, Smooth, Vascular; Norepinephrine; Quinoxalines; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Tolazoline

1985
Antagonism of the hypnotic effect of ethanol in mice by an alpha-1 adrenoceptor agonist.
    Neuropharmacology, 1985, Volume: 24, Issue:9

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Ethanol; Hypnotics and Sedatives; Imidazoles; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL

1985
Inhibitory effect of alpha-1 adrenoceptor stimulation on cardiac sympathetic neurotransmission in pithed normotensive rats.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 236, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Decerebrate State; Ethanolamines; Heart; Heart Rate; Imidazoles; Male; Prazosin; Rats; Rats, Inbred Strains; Sympathetic Nervous System; Synaptic Transmission

1986
Effect of diltiazem upon contractile responses to phenylephrine, cirazoline, Sgd 101/75, St 587 and B-HT 920 in rabbit aorta and dog saphenous vein preparations.
    European journal of pharmacology, 1986, Mar-04, Volume: 121, Issue:3

    Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Azepines; Benzazepines; Clonidine; Diltiazem; Dogs; Drug Interactions; Female; Imidazoles; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Rabbits; Saphenous Vein

1986
Protein secretion in lacrimal gland: alpha 1-beta-adrenergic synergism.
    The American journal of physiology, 1986, Volume: 250, Issue:5 Pt 1

    Topics: Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Clonidine; Epinephrine; Imidazoles; Isoproterenol; Kinetics; Lacrimal Apparatus; Male; Norepinephrine; Phenylephrine; Prazosin; Propranolol; Proteins; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Receptors, Adrenergic, beta

1986
Ca++ utilization in the constriction of rat aorta to full and partial alpha-1 adrenoceptor agonists.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 238, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Aorta; Calcium; Clonidine; Dose-Response Relationship, Drug; Ethanolamines; Imidazoles; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Potassium; Rats; Rats, Inbred Strains; Tetrahydronaphthalenes

1986
Regulation of chicken pineal arylalkylamine-N-acetyl transferase by postsynaptic alpha 2-adrenergic receptors.
    Life sciences, 1986, Nov-24, Volume: 39, Issue:21

    Topics: Acetyltransferases; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arylamine N-Acetyltransferase; Chickens; Circadian Rhythm; Clonidine; Dose-Response Relationship, Drug; Epinephrine; Imidazoles; Norepinephrine; Organ Culture Techniques; Pineal Gland; Receptors, Adrenergic, alpha

1986
Modification of certain pharmacological effects of ethanol by lipophilic alpha-1 adrenergic agonists.
    Life sciences, 1987, Sep-28, Volume: 41, Issue:13

    Topics: Adrenergic alpha-Agonists; Animals; Body Temperature; Clonidine; Drug Interactions; Ethanol; Hypnosis; Imidazoles; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred DBA; Motor Activity; Pentobarbital; Tetrahydronaphthalenes

1987
Effects of the irreversible alpha-adrenoceptor antagonists phenoxybenzamine and benextramine on the effectiveness of nifedipine in inhibiting alpha 1- and alpha 2-adrenoceptor mediated vasoconstriction in pithed rats.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 329, Issue:4

    Topics: Animals; Azepines; Clonidine; Cystamine; Decerebrate State; Diastole; Dose-Response Relationship, Drug; Imidazoles; Male; Nifedipine; Phenoxybenzamine; Rats; Rats, Inbred Strains; Receptors, Adrenergic, alpha; Vasoconstriction

1985
Cirazoline, an alpha 2-adrenoceptor antagonist in guinea-pig ileum.
    General pharmacology, 1985, Volume: 16, Issue:4

    Topics: Acetylcholine; Animals; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Female; Guinea Pigs; Ileum; Imidazoles; Male; Muscle Contraction; Nordefrin; Receptors, Adrenergic, alpha

1985
Characterization of inhibition by nifedipine and nitroprusside of the pressor responses to alpha 1-adrenoceptor agonists cirazoline and Sgd 101/75 in pithed rats.
    Yonsei medical journal, 1988, Volume: 29, Issue:2

    Topics: Animals; Blood Pressure; Clonidine; Ferricyanides; Imidazoles; Male; Nifedipine; Nitroprusside; Rats; Rats, Inbred Strains; Vasoconstriction

1988
Characterization of postjunctional alpha-1 and alpha-2 adrenoceptors activated by exogenous or nerve-released norepinephrine in the canine saphenous vein.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:3

    Topics: Animals; Clonidine; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Female; Imidazoles; Male; Methoxamine; Norepinephrine; Phenoxybenzamine; Phenylephrine; Prazosin; Receptors, Adrenergic, alpha; Saphenous Vein; Sympathetic Nervous System; Tyramine; Yohimbine

1984
Functional and biochemical evidence for the lack of cardiac presynaptic alpha-2 adrenoceptor stimulant properties of cirazoline (LD 3098), a potent alpha-1 adrenoceptor agonist in dogs and rats.
    The Journal of pharmacology and experimental therapeutics, 1982, Volume: 223, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Blood Vessels; Brimonidine Tartrate; Clonidine; Dogs; Female; Heart; Heart Rate; Imidazoles; Male; Norepinephrine; Oxymetazoline; Pentobarbital; Quinoxalines; Rats; Spinal Cord; Synapses; Tachycardia; Vagotomy

1982
Demonstration of alpha-2-adrenoceptor antagonist (yohimbine-like) activity of cirazoline using a hamster fat cell preparation.
    Pharmacological research communications, 1982, Volume: 14, Issue:9

    Topics: Adipose Tissue; Adrenergic alpha-Antagonists; Animals; Clonidine; Cricetinae; Glycerol; Imidazoles; In Vitro Techniques; Lipolysis; Male; Prazosin; Yohimbine

1982
Alpha-1 adrenoceptors and calcium in isolated canine coronary arteries.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 226, Issue:3

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Calcium; Calcium Channel Blockers; Clonidine; Coronary Vessels; Dogs; Female; Imidazoles; Male; Methoxamine; Muscle Contraction; Norepinephrine; Phenylephrine; Prazosin; Secologanin Tryptamine Alkaloids; Yohimbine

1983
Regulation of adipose tissue metabolism via adrenergic mechanisms: actions of alpha-adrenoceptor agonists on lipolysis in hamster fat cells.
    International journal of obesity, 1983, Volume: 7, Issue:4

    Topics: Adipose Tissue; Adrenergic alpha-Agonists; Animals; Clonidine; Cricetinae; Guanabenz; Imidazoles; Lipolysis; Male; Phenylephrine

1983
Sleeping times evoked by alpha adrenoceptor agonists in two-day-old chicks: an experimental model to evaluate full and partial agonists at central alpha-2 adrenoceptors.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brain; Brimonidine Tartrate; Chickens; Clonidine; Guanabenz; Guanfacine; Guanidines; Imidazoles; Phenylacetates; Quinoxalines; Receptors, Adrenergic, alpha; Sleep; Thiophenes; Time Factors; Xylazine

1983
Differential effect of calcium entry blockers on alpha 1-adrenoceptor-mediated vasoconstriction in vivo.
    Naunyn-Schmiedeberg's archives of pharmacology, 1983, Volume: 324, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Blood Pressure; Calcium Channel Blockers; Catecholamines; Clonidine; Ethanolamines; Imidazoles; Imidazolines; Male; Methoxamine; Nifedipine; Phenylephrine; Rats; Rats, Inbred Strains; Vasoconstriction; Verapamil

1983
The actions of cirazoline on the rat vas deferens.
    British journal of pharmacology, 1984, Volume: 82, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Imidazoles; In Vitro Techniques; Isometric Contraction; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Prazosin; Rats; Rats, Inbred Strains; Synaptic Transmission; Vas Deferens

1984
Central cardiovascular effects of alpha adrenergic drugs: differences between catecholamines and imidazolines.
    The Journal of pharmacology and experimental therapeutics, 1984, Volume: 230, Issue:1

    Topics: Adrenergic beta-Agonists; Animals; Blood Pressure; Catecholamines; Cats; Clonidine; Female; Heart Rate; Imidazoles; Male; Microinjections; Nordefrin; Receptors, Adrenergic, alpha; Time Factors

1984
Pre- and postsynaptic alpha-adrenoceptor blocking properties of a new dihydrobenzofurane derivative (imidazolinyl-2)-2-dihydro 2,3 benzofurane (S 9871) and its stereoisomers in rats.
    Archives internationales de pharmacodynamie et de therapie, 1984, Volume: 269, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Azepines; Benzofurans; Blood Pressure; Clonidine; Drug Interactions; Electric Stimulation; Imidazoles; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Phenylephrine; Rats; Rats, Inbred Strains; Stereoisomerism; Vas Deferens

1984
Effect of removing the endothelial cells on the reactivity of rat aortic segments to different alpha-adrenoceptor agonists.
    Naunyn-Schmiedeberg's archives of pharmacology, 1984, Volume: 328, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Aorta, Thoracic; Azepines; Clonidine; Endothelium; Imidazoles; In Vitro Techniques; Male; Methoxamine; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Rats; Rats, Inbred Strains; Xylazine; Yohimbine

1984
Peripheral postsynaptic alpha-adrenoceptor blocking properties of some new dihydrobenzofurane and imidazoline derivatives in pithed rats.
    Arzneimittel-Forschung, 1984, Volume: 34, Issue:12

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Azepines; Benzofurans; Blood Pressure; Clonidine; Drug Interactions; Imidazoles; Male; Phenethylamines; Phenylephrine; Rats; Rats, Inbred Strains; Receptors, Neurotransmitter

1984
Lack of correlation between presynaptic inhibition of noradrenaline release and end organ responses during nerve stimulation.
    British journal of pharmacology, 1980, Volume: 69, Issue:1

    Topics: Animals; Blood Pressure; Cats; Clonidine; Electric Stimulation; Female; Heart Rate; Imidazoles; In Vitro Techniques; Male; Nasal Decongestants; Nervous System Physiological Phenomena; Nictitating Membrane; Norepinephrine; Receptors, Adrenergic; Receptors, Adrenergic, alpha; Spleen; Synapses

1980
Clonidine and cirazoline inhibit activation of nicotinic channels in PC-12 cells.
    Annals of the New York Academy of Sciences, 1995, Jul-12, Volume: 763

    Topics: Adrenergic alpha-Agonists; Animals; Binding Sites; Calcium; Clonidine; Imidazoles; Ion Channels; Nicotinic Antagonists; PC12 Cells; Phencyclidine; Radioligand Assay; Rats; Receptors, Nicotinic; Torpedo; Tritium

1995
Imidazolines stimulate release of insulin from RIN-5AH cells independently from imidazoline I1 and I2 receptors.
    European journal of pharmacology, 1994, Sep-01, Volume: 262, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Affinity Labels; Animals; Benzofurans; Binding, Competitive; Clonidine; Clorgyline; Diazoxide; Dioxanes; Guanidines; Idazoxan; Imidazoles; Imidazoline Receptors; Insulin; Insulinoma; Ligands; Pancreatic Neoplasms; Potassium Channels; Rats; Receptors, Drug; Regression Analysis; Software; Tumor Cells, Cultured

1994
Stimulatory effects of clonidine, cirazoline and rilmenidine on locus coeruleus noradrenergic neurones: possible involvement of imidazoline-preferring receptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1993, Volume: 348, Issue:2

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Dose-Response Relationship, Drug; Imidazoles; Imidazoline Receptors; Locus Coeruleus; Male; Membrane Potentials; Neurons; Norepinephrine; Oxazoles; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine

1993
Relevance of the use of [3H]-clonidine to identify imidazoline receptors in the rabbit brainstem.
    British journal of pharmacology, 1993, Volume: 110, Issue:4

    Topics: Animals; Binding, Competitive; Clonidine; Imidazoles; Imidazoline Receptors; Medulla Oblongata; Rabbits; Receptors, Adrenergic, alpha; Receptors, Drug

1993
No evidence for functional imidazoline receptors on locus coeruleus neurons.
    Naunyn-Schmiedeberg's archives of pharmacology, 1996, Volume: 353, Issue:5

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Benzazepines; Binding, Competitive; Clonidine; Dose-Response Relationship, Drug; Imidazoles; Imidazoline Receptors; Injections, Intravenous; Locus Coeruleus; Male; Microelectrodes; Neurons; Oxazoles; Quinolines; Rats; Rats, Wistar; Receptors, Drug; Rilmenidine

1996
Contractile responses to various inotropic agents in isolated hearts obtained from hypertensive diabetic rats.
    Blood pressure, 1995, Volume: 4, Issue:6

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Adrenergic alpha-Agonists; Animals; Calcium; Calcium Channel Agonists; Cardiotonic Agents; Clonidine; Diabetes Mellitus, Experimental; Diabetic Angiopathies; Drug Evaluation, Preclinical; Homeostasis; Hypertension; Imidazoles; In Vitro Techniques; Male; Myocardial Contraction; Rats; Rats, Inbred SHR; Rats, Inbred WKY

1995
Opposite influences of hypertension and diabetes mellitus on pressor responses induced by different alpha-adrenoceptor agonists and angiotensin II in pithed rats.
    Blood pressure, 1996, Volume: 5, Issue:1

    Topics: Adrenergic alpha-Agonists; Angiotensin II; Animals; Azepines; Blood Glucose; Blood Pressure; Brimonidine Tartrate; Clonidine; Decerebrate State; Diabetes Mellitus, Experimental; Dose-Response Relationship, Drug; Hypertension; Imidazoles; Male; Quinoxalines; Rats; Rats, Inbred SHR; Rats, Inbred WKY

1996
Influence of nifedipine on pressor responses induced by different alpha-adrenoceptor agonists and angiotensin II in pithed diabetic hypertensive rats.
    Journal of hypertension, 1996, Volume: 14, Issue:7

    Topics: Adrenergic alpha-Antagonists; Angiotensin II; Animals; Blood Pressure; Brimonidine Tartrate; Calcium; Calcium Channel Blockers; Clonidine; Diabetes Mellitus, Experimental; Hypertension; Imidazoles; Nifedipine; Quinoxalines; Rats; Rats, Inbred SHR; Rats, Inbred WKY; Streptozocin

1996
Identification and characterization of imidazoline-binding sites from calf striatum.
    European journal of pharmacology, 1996, Nov-07, Volume: 315, Issue:1

    Topics: Animals; Binding, Competitive; Cattle; Clonidine; Corpus Striatum; Guanidines; Idazoxan; Imidazoles; Imidazoline Receptors; Kinetics; Receptors, Drug

1996
Effects of imidazolines on noradrenaline release in brain: an investigation into their relationship to imidazoline, alpha 2 and H3 receptors.
    Neurochemistry international, 1997, Volume: 30, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Brain; Cerebral Cortex; Clonidine; Electric Stimulation; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Medulla Oblongata; Norepinephrine; Perfusion; Rabbits; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Drug; Receptors, Histamine H3; Tritium

1997
Binding of new cirazoline derivative to imidazoline receptors from human brain.
    Neurochemistry international, 1997, Volume: 30, Issue:1

    Topics: Adrenergic alpha-Agonists; Animals; Binding Sites; Brain; Clonidine; Humans; Idazoxan; Imidazoles; Imidazoline Receptors; Kidney; Mitochondria; Photochemistry; Rabbits; Rats; Receptors, Drug; Tritium; Ultraviolet Rays; Yohimbine

1997
The novel alpha 2-adrenoceptor agonist [3H]mivazerol binds to non-adrenergic binding sites in human striatum membranes that are distinct from imidazoline receptors.
    Neurochemistry international, 1997, Volume: 31, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Aged; Clonidine; Corpus Striatum; Female; Humans; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Membranes; Middle Aged; Radioligand Assay; Receptors, Drug; Tritium

1997
alpha1-Adrenoceptor-mediated phosphorylation of myosin in rat-tail arterial smooth muscle.
    The Biochemical journal, 1997, Nov-01, Volume: 327 ( Pt 3)

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Arteries; Azepines; Calcium; Clonidine; Endothelium, Vascular; Enzyme Inhibitors; Imidazoles; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myosin Light Chains; Myosin-Light-Chain Kinase; Phosphorylation; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Serine; Tail

1997
Selective blockade by nicergoline of vascular responses elicited by stimulation of alpha 1A-adrenoceptor subtype in the rat.
    Fundamental & clinical pharmacology, 1999, Volume: 13, Issue:1

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta; Azepines; Binding, Competitive; Blood Pressure; Clonidine; Decerebrate State; Dose-Response Relationship, Drug; Imidazoles; In Vitro Techniques; Male; Mesenteric Arteries; Nicergoline; Prazosin; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sensitivity and Specificity; Tritium

1999
Phe-308 and Phe-312 in transmembrane domain 7 are major sites of alpha 1-adrenergic receptor antagonist binding. Imidazoline agonists bind like antagonists.
    The Journal of biological chemistry, 2001, Jul-06, Volume: 276, Issue:27

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Amino Acid Sequence; Animals; Cell Membrane; Clonidine; Conserved Sequence; Cricetinae; Dihydropyridines; Dioxanes; Humans; Imidazoles; Models, Molecular; Molecular Sequence Data; Oxymetazoline; Phenylalanine; Piperazines; Prazosin; Protein Structure, Secondary; Rats; Receptors, Adrenergic, alpha-1; Structure-Activity Relationship

2001
The release of noradrenaline in the locus coeruleus and prefrontal cortex studied with dual-probe microdialysis.
    Brain research, 2001, Jul-06, Volume: 906, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Bicuculline; Calcium; Clonidine; Environment, Controlled; Extracellular Space; GABA Antagonists; Imidazoles; Indoles; Isoindoles; Isotonic Solutions; Locus Coeruleus; Male; Microdialysis; Neural Pathways; Neurons; Norepinephrine; Piperazines; Prefrontal Cortex; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; Receptors, Serotonin; Receptors, Serotonin, 5-HT1; Ringer's Solution; Serotonin Receptor Agonists; Stress, Physiological; Tetrodotoxin

2001
Noradrenaline release-inhibiting receptors on PC12 cells devoid of alpha(2(-)) and CB(1) receptors: similarities to presynaptic imidazoline and edg receptors.
    Neurochemistry international, 2002, Volume: 40, Issue:2

    Topics: Animals; Arachidonic Acids; Benzoxazines; Cannabinoids; Clonidine; Cyclohexanols; Endocannabinoids; Heterotrimeric GTP-Binding Proteins; Imidazoles; Imidazoline Receptors; Kinetics; Morpholines; Naphthalenes; Norepinephrine; PC12 Cells; Polyunsaturated Alkamides; Rats; Receptors, Adrenergic, alpha-2; Receptors, Cannabinoid; Receptors, Cell Surface; Receptors, Drug; Receptors, G-Protein-Coupled; Receptors, Lysophospholipid; Tritium; Veratridine

2002
Regulation of the release of serotonin in the dorsal raphe nucleus by alpha1 and alpha2 adrenoceptors.
    Synapse (New York, N.Y.), 2003, Volume: 50, Issue:1

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Imidazoles; Indoles; Isoindoles; Male; Neurons; Pons; Prazosin; Prefrontal Cortex; Raphe Nuclei; Rats; Rats, Wistar; Reaction Time; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Serotonin

2003
Identification and characterization of the imidazoline I2b-binding sites in the hamster brown adipose tissue as a study model for imidazoline receptors.
    Archives of physiology and biochemistry, 2003, Volume: 111, Issue:2

    Topics: Adipose Tissue, Brown; Amiloride; Animals; Binding Sites; Binding, Competitive; Cell Line, Tumor; Clonidine; Culture Techniques; Dose-Response Relationship, Drug; Guanabenz; Humans; Idazoxan; Imidazoles; Imidazoline Receptors; Liver; Mammary Neoplasms, Animal; Mice; Protein Binding; Rats; Receptors, Drug; Species Specificity; Yohimbine

2003
Atypical [(3)H]clonidine binding sites in human caudate and platelets on cryostat-cut sections.
    Annals of the New York Academy of Sciences, 2003, Volume: 1009

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Animals; Binding Sites; Blood Platelets; Brain Chemistry; Caudate Nucleus; Clonidine; Female; Harmine; Humans; Imidazoles; Imidazoline Receptors; Male; Middle Aged; Radioligand Assay; Receptors, Adrenergic, alpha-2; Receptors, Drug

2003
Noradrenergic inputs mediate state dependence of auditory responses in the avian song system.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2004, Sep-01, Volume: 24, Issue:35

    Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Adrenergic Fibers; Animals; Arousal; Auditory Perception; Clonidine; Dose-Response Relationship, Drug; Finches; Guanabenz; Idazoxan; Imidazoles; Isoproterenol; Male; Norepinephrine; Oxathiins; Phenylephrine; Propanolamines; Prosencephalon; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Adrenergic, beta-2; Vocalization, Animal; Yohimbine

2004
Different response of ANP secretion to adrenoceptor stimulation in renal hypertensive rat atria.
    Peptides, 2008, Volume: 29, Issue:7

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Animals; Atrial Natriuretic Factor; Clonidine; Cyclic AMP; Dose-Response Relationship, Drug; Guanabenz; Heart Atria; Hypertension, Renal; Imidazoles; Isoproterenol; Male; Phenylephrine; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic; RNA, Messenger; Time Factors

2008
The adrenergic receptor subtypes present in frog (Rana esculenta) skin.
    Comparative biochemistry and physiology. Toxicology & pharmacology : CBP, 2008, Volume: 148, Issue:2

    Topics: Adrenergic alpha-Agonists; Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Amphibian Proteins; Animals; Calmodulin; Chlorides; Clonidine; Cyclic AMP; Dose-Response Relationship, Drug; Ethanolamines; Formoterol Fumarate; Imidazoles; Membrane Potentials; Propanolamines; Rana esculenta; Receptors, Adrenergic; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, beta-2; Receptors, Adrenergic, beta-3; Signal Transduction; Skin; Sodium; Xamoterol

2008
Evidence that some imidazoline derivatives inhibit peripherally the vasopressor sympathetic outflow in pithed rats.
    Autonomic neuroscience : basic & clinical, 2008, Dec-05, Volume: 143, Issue:1-2

    Topics: Adrenergic alpha-Agonists; Agmatine; Animals; Antihypertensive Agents; Azepines; Blood Pressure; Blood Vessels; Clonidine; Decerebrate State; Dose-Response Relationship, Drug; Electric Stimulation; Heart Rate; Imidazoles; Imidazoline Receptors; Imidazolines; Injections, Intravenous; Male; Methoxamine; Rats; Rats, Wistar; Sympathetic Nervous System; Vasomotor System

2008
Might adrenergic alpha2C-agonists/alpha2A-antagonists become novel therapeutic tools for pain treatment with morphine?
    Journal of medicinal chemistry, 2009, Nov-26, Volume: 52, Issue:22

    Topics: Adjuvants, Pharmaceutic; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analgesics; Animals; CHO Cells; Clonidine; Cricetinae; Cricetulus; Drug Discovery; Humans; Imidazoles; Morphine; Pain; Receptors, Adrenergic, alpha-2

2009
In brown adipocytes, adrenergically induced β₁-/β₃-(Gs)-, α₂-(Gi)- and α₁-(Gq)-signalling to Erk1/2 activation is not mediated via EGF receptor transactivation.
    Experimental cell research, 2013, Oct-15, Volume: 319, Issue:17

    Topics: Adipocytes, Brown; Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic Antagonists; Adrenergic beta-1 Receptor Agonists; Adrenergic beta-3 Receptor Agonists; Animals; Clonidine; Dioxoles; Dose-Response Relationship, Drug; Drug Synergism; ErbB Receptors; Imidazoles; Male; MAP Kinase Signaling System; Mice; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Norepinephrine; Phosphorylation; Quinazolines; Receptors, Adrenergic; Tyrphostins

2013
Noradrenergic receptor modulation influences the acoustic parameters of pro-social rat ultrasonic vocalizations.
    Behavioral neuroscience, 2018, Volume: 132, Issue:4

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Imidazoles; Male; Models, Animal; Norepinephrine; Propranolol; Rats; Rats, Long-Evans; Receptors, Adrenergic; Ultrasonics; Vocalization, Animal

2018
Adrenergic α2 receptors are implicated in seizure-induced respiratory arrest in DBA/1 mice.
    Life sciences, 2021, Nov-01, Volume: 284

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Antagonists; Animals; Atomoxetine Hydrochloride; Clonidine; Imidazoles; Mice, Inbred DBA; Receptors, Adrenergic, alpha-2; Respiration; Seizures

2021